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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
5 mg | ¥ 12,600 | 期货 | |
1 mL x 10 mM (in DMSO) | ¥ 15,000 | 期货 |
产品描述 | 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone showed strong anti-proliferation effect on ER-positive breast cancer MCF-7 cells in vitro, with an IC50 value of 4.41 uM. 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone can significantly down-regulate the expression of estrogen receptor-α (ER-α) and inhibit tumor growth in human breast cancer cell line BCAP-37 xenograft model. |
体外活性 | 我们发现5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone在体外对ER阳性乳腺癌MCF-7细胞展现出强大的抑制增殖效果(IC50为4.41 μM)。[1] |
体内活性 | 我们发现5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone显著降低了雌激素受体-α (ER-α) 的表达浓度,并能够在人乳腺癌细胞系BCAP-37的异种移植模型中抑制肿瘤生长。[1] |
分子量 | 452.5 |
分子式 | C26H28O7 |
CAS No. | 1353676-65-9 |
存储 | store at low temperature,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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