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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 2,650 | 现货 | |
5 mg | ¥ 6,630 | 现货 | |
10 mg | ¥ 8,930 | 现货 | |
25 mg | ¥ 13,200 | 现货 | |
50 mg | ¥ 17,900 | 现货 | |
100 mg | ¥ 23,900 | 现货 |
产品描述 | KDM2A/7A-IN-1 is a cell-permeable and selective inhibitor of the histone lysine demethylase KDM2A/7A with potential antitumor activity for the study of duodenal adenomas and ossifying fibromucoid tumors. |
靶点活性 | KDM2A:0.16 μM |
体外活性 | KDM2A/7A-IN-1 是 KDM2A/7A 的高效细胞渗透性抑制剂,其 IC50 为 0.16 μM 。KDM2A/7A-IN-1 (0.4,3.1,6.2 μM)能够增加异位表达催化活性 KDM2A 的 HeLa 细胞中的 H3K36me2 水平[1]。 |
分子量 | 506.68 |
分子式 | C33H38N4O |
CAS No. | 2169272-46-0 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 120 mg/mL (236.84 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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