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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 497 | 现货 | |
5 mg | ¥ 1,180 | 现货 | |
10 mg | ¥ 1,930 | 现货 | |
25 mg | ¥ 3,170 | 现货 | |
50 mg | ¥ 4,490 | 现货 | |
100 mg | ¥ 5,920 | 现货 | |
200 mg | ¥ 7,990 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 1,250 | 现货 |
产品描述 | SIRT-IN-1 is a potent SIRT1/2/3 inhibitor(IC50s of 15, 10, 33 μM, respectively). |
靶点活性 | SIRT1:15 nM, SIRT3:33 nM, SIRT2:10 nM |
体外活性 | SIRT-IN-1是一种SIRT1/2/3的强效抑制剂,其IC50值分别为0.015、0.010、0.033 μM。SIRT-IN-1在催化活性位点具有一致的结合模式(RMS=0.29 Å),通过占据了烟酰胺C-口袋和乙酰化赖氨酸底物通道。 |
分子量 | 389.52 |
分子式 | C19H27N5O2S |
CAS No. | 1431411-60-7 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
溶解度信息 | DMSO: 3.89 mg/mL (10 mM), Sonication is recommended. | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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