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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 813 | 现货 | |
5 mg | ¥ 1,980 | 现货 | |
10 mg | ¥ 3,230 | 现货 | |
25 mg | ¥ 5,930 | 现货 | |
50 mg | ¥ 8,180 | 现货 | |
100 mg | ¥ 10,800 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 2,320 | 现货 |
产品描述 | CDK4/6-IN-6 is a potent CDK4/CDK6 inhibitor with Ki of 0.6 nM and 13.9 nM for CDK4/Cyclin D1 and CDK6/Cyclin D3, respectively. |
靶点活性 | CDK6-CyclinD3:13.9 nM (Ki), CDK4-CyclinD1:0.6 nM (Ki) |
体外活性 | 在JEKO-1细胞中,通过使用磷酸化的Rb S795 ELISA测定法,CDK4/6-IN-6的IC50分别针对CDK4/Cyclin D1和CDK6/Cyclin D3为38.5 nM和144.9 nM [1]。 |
分子量 | 463.93 |
分子式 | C22H27ClFN5O3 |
CAS No. | 2380321-51-5 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 55 mg/mL (118.55 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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