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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 239 | 现货 | |
5 mg | ¥ 696 | 现货 | |
10 mg | ¥ 987 | 现货 | |
25 mg | ¥ 1,750 | 现货 | |
50 mg | ¥ 2,590 | 现货 | |
100 mg | ¥ 3,690 | 现货 | |
200 mg | ¥ 4,970 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 798 | 现货 |
产品描述 | Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase. Ibiglustat (L-Malic acid) can be used in studies about PD Parkinson’s disease, SRT in Fabry’s and Gaucher’s. |
体外活性 | Ibiglustat (L-Malic acid) (1 μM)处理的Fabry病细胞中的GL-3含量接近未处理野生型细胞的生理水平。Ibiglustat (L-Malic acid) 可阻止GL-3的进一步积聚,并改善FD心肌细胞中丰富的GL-3含量[4]。 |
别名 | Ibiglustat L-Malic acid, GZ402671 (L-Malic acid), Venglustat (L-Malic acid), SAR402671 (L-Malic acid) |
分子量 | 523.57 |
分子式 | C24H30FN3O7S |
CAS No. | 1629063-78-0 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 90 mg/mL (171.9 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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