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规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 892 | 现货 | |
5 mg | ¥ 2,320 | 现货 | |
10 mg | ¥ 3,290 | 现货 | |
25 mg | ¥ 5,550 | 现货 | |
50 mg | ¥ 7,460 | 现货 | |
100 mg | ¥ 9,860 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 2,560 | 现货 |
产品描述 | CDK8-IN-1 is a selective CDK8 inhibitor (IC50: 3 nM). |
靶点活性 | CDK8:3 nM |
体内活性 | CDK8-IN-1展现出低系统性清除率,良好的化合物接触度和口服生物利用度。口服给药后,tmax为0.25小时。静脉注射和口服给药的AUC值分别为9378和25952。其平均Cmax值分别为静脉注射9940 μg/L和口服12740 μg/L[1]。 |
分子量 | 255.2 |
分子式 | C11H8F3N3O |
CAS No. | 1629633-48-2 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 90 mg/mL (352.7 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
DMSO
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