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KOR agonist 3 (Compound 5) 是 κ 阿片受体 (κOR) 的激动剂,EC50为 0.88 nM,并对 μOR 展示一定激活效应,EC50 为 720 nM。在浓度小于 1 μM 时,KOR agonist 3 对 δOR 无激动活性。相比 U50488,KOR agonist 3 诱导 β-Arrestin-2 的募集能力较低。
KOR agonist 3 (Compound 5) 是 κ 阿片受体 (κOR) 的激动剂,EC50为 0.88 nM,并对 μOR 展示一定激活效应,EC50 为 720 nM。在浓度小于 1 μM 时,KOR agonist 3 对 δOR 无激动活性。相比 U50488,KOR agonist 3 诱导 β-Arrestin-2 的募集能力较低。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
10 mg | 询价 | 期货 | |
50 mg | 询价 | 期货 |
产品描述 | KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488. |
靶点活性 | κ Opioid Receptor:0.88 nM (EC50) |
分子量 | 388.46 |
分子式 | C24H24N2O3 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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