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TEAD-IN-2是 一种高效和双功能的TEAD 抑制剂,能够同时结合 TEAD 蛋白和 E3 泛素连接酶或降解诱导基团,通过泛素化途径诱导 TEAD 蛋白的降解,具有抗癌和抗增殖的潜力。
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TEAD-IN-2是 一种高效和双功能的TEAD 抑制剂,能够同时结合 TEAD 蛋白和 E3 泛素连接酶或降解诱导基团,通过泛素化途径诱导 TEAD 蛋白的降解,具有抗癌和抗增殖的潜力。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 1,540 | 现货 | |
5 mg | ¥ 2,610 | 5日内发货 | |
25 mg | ¥ 9,160 | 6-8周 | |
50 mg | ¥ 11,900 | 6-8周 | |
100 mg | ¥ 17,634 | 6-8周 |
产品描述 | TEAD-IN-2 is a potent and bifunctional TEAD inhibitor that binds to both TEAD proteins and E3 ubiquitin ligases or degradation-inducing motifs to induce TEAD protein degradation via the ubiquitination pathway, with anticancer and antiproliferative potential. |
分子量 | 391.23 |
分子式 | C16H18BrF3N2O |
CAS No. | 2563849-97-6 |
Smiles | FC(F)(F)C1=CC=C(C=C1)CN2CCC(CC2)C3ON=C(Br)C3 |
存储 | keep away from moisture,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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