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EPZ011989是一种高选择性可口服的 EZH2抑制剂,对wt EZH2以及EZH2突变型Ki 值<3nM。
EPZ011989是一种高选择性可口服的 EZH2抑制剂,对wt EZH2以及EZH2突变型Ki 值<3nM。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 237 | 现货 | |
2 mg | ¥ 336 | 现货 | |
5 mg | ¥ 546 | 现货 | |
10 mg | ¥ 818 | 现货 | |
25 mg | ¥ 1,550 | 现货 | |
50 mg | ¥ 2,550 | 现货 | |
100 mg | ¥ 3,970 | 现货 |
产品描述 | EPZ011989 is a effective, specific orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 Y646 and EZH2 wt; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. |
靶点活性 | EZH2:<3 nM(Ki), EZH1:103 nM |
分子量 | 605.81 |
分子式 | C35H51N5O4 |
CAS No. | 1598383-40-4 |
Smiles | CCN([C@H]1CC[C@@H](CC1)N(C)CCOC)c1cc(cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C#CCN1CCOCC1 |
密度 | 1.17 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 1 mg/mL Ethanol: 100 mg/mL (155.7 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
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