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TAK-448 acetate (MVT-602 acetate) 是一种小分子 KISS1R 激动剂,是一种和 kisspeptin 类似的合成肽。TAK-448 acetate 具有抗肿瘤活性,抑制 VCaP 细胞增殖,可用于研究前列腺癌。
TAK-448 acetate (MVT-602 acetate) 是一种小分子 KISS1R 激动剂,是一种和 kisspeptin 类似的合成肽。TAK-448 acetate 具有抗肿瘤活性,抑制 VCaP 细胞增殖,可用于研究前列腺癌。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 993 | 现货 | |
5 mg | ¥ 2,480 | 现货 | |
10 mg | ¥ 3,980 | 现货 | |
25 mg | ¥ 6,270 | 现货 | |
50 mg | ¥ 8,460 | 现货 | |
100 mg | ¥ 11,300 | 现货 |
产品描述 | TAK-448 acetate (MVT-602 acetate) is a small molecule KISS1R agonist, a synthetic peptide similar to kisspeptin.TAK-448 acetate has antitumor activity, inhibits the proliferation of VCaP cells, and can be used in prostate cancer research.TAK-448 acetate is a small molecule KISS1R agonist. |
靶点活性 | KISS1R:632 pM, KISS1R:460 pM |
体内活性 | 单次注射 TAK-448 可显著提高雄性大鼠和雄性血浆促性腺激素和睾酮(T)水平。在雄性大鼠 VCaP 异种移植雄激素敏感前列腺癌模型中,TAK-448 (0.01, 0.03, 0.3, 3 mg/kg;i.h.;0,28天) 显示出更强的抗肿瘤效果[1]。 |
别名 | TAK-448 acetate (1234319-68-6 Free base), MVT-602 acetate |
分子量 | 1285.41 |
分子式 | C60H84N16O16 |
CAS No. | 1470374-22-1 |
存储 | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 80 mg/mL (62.24 mM), Sonication is recommended. H2O: 30 mg/mL (23.34 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
H2O/DMSO
DMSO
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