Ipamorelin

Name: Ipamorelin
Brand: TargetMol
SKU: T7809
Price: 198 USD
Availability: InStock
Rating: 4.5 (1 reviews)

还可以

产品编号 T7809Cas号 170851-70-4

别名 伊帕瑞林, NNC-26-0161

Ipamorelin (NNC-26-0161) 是一种生长激素释放肽，可诱导大鼠纵向骨生长。

还可以

产品编号 T7809 别名 伊帕瑞林, NNC-26-0161Cas号 170851-70-4

Ipamorelin (NNC-26-0161) 是一种生长激素释放肽，可诱导大鼠纵向骨生长。

大包装 & 定制

加入购物车

实验操作小课堂

选择批次:

联系我们获取更多批次信息

资源下载

凭借在化合物合成方面的丰富经验，我们可以根据您的研究需求为该产品提供快速定制合成服务.

产品介绍

生物活性

产品描述	Ipamorelin (NNC-26-0161) is a growth-hormone-releasing peptide, induces longitudinal bone growth in rats.
体外活性	In vitro, ipamorelin released GH from primary rat pituitary cells with a potency and efficacy similar to GHRP-6 (ECs) = 1.3+/-0.4nmol/l and Emax = 85+/-5% vs 2.2+/-0.3nmol/l and 100%).?A pharmacological profiling using GHRP and growth hormone-releasing hormone (GHRH) antagonists clearly demonstrated that ipamorelin, like GHRP-6, stimulates GH release via a GHRP-like receptor[1]
体内活性	In pentobarbital anaesthetised rats, ipamorelin released GH with a potency and efficacy comparable to GHRP-6 (ED50 = 80+/-42nmol/kg and Emax = 1545+/-250ng GH/ml vs 115+/-36nmol/kg and 1167+/-120ng GH/ml).?In conscious swine, ipamorelin released GH with an ED50 = 2.3+/-0.03 nmol/kg and an Emax = 65+/-0.2 ng GH/ml plasma.?Again, this was very similar to GHRP-6 (ED50 = 3.9+/-1.4 nmol/kg and Emax = 74+/-7ng GH/ml plasma)[1].
别名	伊帕瑞林, NNC-26-0161

化学信息

分子量	711.85
分子式	C₃₈H₄₉N₉O₅
CAS No.	170851-70-4
Smiles	C([C@@H](NC([C@H](CC1=CN=CN1)NC(C(C)(C)N)=O)=O)C(N[C@H](CC2=CC=CC=C2)C(N[C@@H](CCCCN)C(N)=O)=O)=O)C3=CC4=C(C=C3)C=CC=C4
密度	1.264g/cm3