购物车
- 全部删除
- 您的购物车当前为空
CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 1,355 | 期货 | |
5 mg | ¥ 2,010 | 期货 | |
10 mg | ¥ 3,040 | 期货 | |
50 mg | ¥ 7,150 | 期货 | |
100 mg | ¥ 11,100 | 期货 | |
200 mg | 询价 | 期货 | |
500 mg | 询价 | 期货 |
产品描述 | CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1). |
体外活性 | CBB1007 efficiently can block LSD1-mediated demethylation of H3K4Me2 and H3K4Me (IC50 ≤ 5 μM) with no effect on H3K4Me3 and H3K9Me2, and LSD2 and JARID1A activities. Increases H3K4Me2 and H3K4Me contents (IC50 ≤ 5 μM), and causes activation of epigenetically suppressed CHRM4/M4-ArchR and SCN3A genes in F9 cells (IC50 ≤ 3.74 μM). |
别名 | CBB1007 hydrochloride |
分子量 | 716.91 |
分子式 | C27H39Cl5N8O4 |
密度 | no data available |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
版权所有©2015-2024 TargetMol Chemicals Inc.保留所有权利.
评论内容