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VU041 is an inhibitor of Anopheles gambiae and Aedes aegypti inward rectifier potassium 1 channels (IC50: 2.5 μM and 1.7 μM, respectively). VU041 inhibits appreciably is mammalian Kir2.1 (IC50: 12.7 μM) and has less inhibitory effect on mammalian Kir1.1, Kir4.1, Kir6.2/SUR1, and Kir7.1.
VU041 is an inhibitor of Anopheles gambiae and Aedes aegypti inward rectifier potassium 1 channels (IC50: 2.5 μM and 1.7 μM, respectively). VU041 inhibits appreciably is mammalian Kir2.1 (IC50: 12.7 μM) and has less inhibitory effect on mammalian Kir1.1, Kir4.1, Kir6.2/SUR1, and Kir7.1.
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 484 | 5日内发货 | |
5 mg | ¥ 792 | 5日内发货 | |
1 mL x 10 mM (in DMSO) | ¥ 793 | 5日内发货 |
产品描述 | VU041 is an inhibitor of Anopheles gambiae and Aedes aegypti inward rectifier potassium 1 channels (IC50: 2.5 μM and 1.7 μM, respectively). VU041 inhibits appreciably is mammalian Kir2.1 (IC50: 12.7 μM) and has less inhibitory effect on mammalian Kir1.1, Kir4.1, Kir6.2/SUR1, and Kir7.1. |
靶点活性 | Kir1 channel (Anopheles An. gambiae):2.5 μM, Kir1 channel (aedes Ae. aegypti):1.7 μM, Kir2.1 (mammalian):12.7 μM |
分子量 | 363.38 |
分子式 | C19H20F3N3O |
CAS No. | 332943-64-3 |
密度 | no data available |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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