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RR-49是一种新型双氟化类似物。该化合物在pH 6.5相比pH 7.4时,在MOR cAMP测定中显示出对DAMGO具有相同的有效性,但其功效(IC50)提高了19倍,表现出卓越的pH敏感性。RR-49作为一种治疗炎症疼痛的镇痛剂,具有较低的滥用潜力,显示出显著的应用前景。
RR-49是一种新型双氟化类似物。该化合物在pH 6.5相比pH 7.4时,在MOR cAMP测定中显示出对DAMGO具有相同的有效性,但其功效(IC50)提高了19倍,表现出卓越的pH敏感性。RR-49作为一种治疗炎症疼痛的镇痛剂,具有较低的滥用潜力,显示出显著的应用前景。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
10 mg | 询价 | 10-14周 | |
50 mg | 询价 | 10-14周 |
产品描述 | RR-49 is an innovative difluorinated analogue. This compound demonstrates exceptional pH sensitivity, showing the same efficacy for DAMGO in MOR cAMP assays at pH 6.5 as it does at pH 7.4, but with a 19-fold increase in potency (IC50). It holds significant promise as an analgesic for treating inflammatory pain with a lower potential for abuse. |
别名 | RR49, RR 49 |
分子量 | 372.45 |
分子式 | C22H26F2N2O |
CAS No. | 2376328-79-7 |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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