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KH-CB19
还可以产品编号 T15657Cas号 1354037-26-5
KH-CB19 is an effective and highly specific inhibitor of the CDC2-like kinase isoforms 1 and 4 (CLK1/CLK4).
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KH-CB19
还可以产品编号 T15657Cas号 1354037-26-5
KH-CB19 is an effective and highly specific inhibitor of the CDC2-like kinase isoforms 1 and 4 (CLK1/CLK4).
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 2 mg | ¥ 1,590 | 5日内发货 | |
| 5 mg | 询价 | 5日内发货 | |
| 25 mg | 询价 | 6-8周 | |
| 50 mg | 询价 | 6-8周 | |
| 100 mg | 询价 | 6-8周 | |
| 1 mL x 10 mM (in DMSO) | 询价 | 5日内发货 |
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产品介绍
生物活性
化学信息
| 产品描述 | KH-CB19 is an effective and highly specific inhibitor of the CDC2-like kinase isoforms 1 and 4 (CLK1/CLK4). |
| 靶点活性 | CLK1:19.7 nM, DYRK1A:55.2 nM, CLK3:530 nM |
| 体外活性 | KH-CB19 showed potent inhibition of CLK1 (IC50: 20 nM), and for the pure isomer KH-CB19, almost 100-fold selectivity against the CLK3 isoform. Treatment of resting cells with 10 μM KH-CB19 significantly reduced the basal expression of flTF as well as HTF. Pretreatment of cells with KH-CB19 or TG003 led to a reduction of the TNF-α-induced increase in phosphorylation of all analyzed SR proteins compared with TNF-α-stimulated controls [1]. |
| 分子量 | 338.19 |
| 分子式 | C15H13Cl2N3O2 |
| CAS No. | 1354037-26-5 |
| 密度 | 1.39 g/cm3 (Predicted) |
储存&溶解度
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
| 溶解度信息 | DMSO: 50 mg/mL (147.85 mM) | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
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计算器
体内实验配液计算器
请在以下方框中输入您的动物实验信息后点击计算，可以得到母液配置方法和体内配方的制备方法：
比如您的给药剂量是 10 mg/kg ，每只动物体重 20 g ，给药体积 100 μL ， 
剂量转换
对于不同动物的给药剂量换算，您也可以参考 更多
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