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GNE-6468 is a potent and selective agonist of RORγ(RORc) (EC50: 13 nM for HEK-293 cell).
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GNE-6468 is a potent and selective agonist of RORγ(RORc) (EC50: 13 nM for HEK-293 cell).
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
2 mg | ¥ 2,650 | 5日内发货 | |
5 mg | ¥ 3,730 | 5日内发货 | |
25 mg | ¥ 10,800 | 8-10周 | |
50 mg | ¥ 16,800 | 8-10周 | |
100 mg | ¥ 21,500 | 8-10周 | |
1 mL x 10 mM (in DMSO) | ¥ 3,570 | 5日内发货 |
产品描述 | GNE-6468 is a potent and selective agonist of RORγ(RORc) (EC50: 13 nM for HEK-293 cell). |
靶点活性 | RORγ:2 nM (EC50) |
分子量 | 433.84 |
分子式 | C23H16ClN3O4 |
CAS No. | 1677668-27-7 |
密度 | 1.55 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
溶解度信息 | DMSO: 5 mg/mL (11.52 mM), Sonication is recommended. | ||||||||||||||||||||
溶液配制表 | |||||||||||||||||||||
DMSO
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