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CSV0C018875 是基于喹啉的EHMT2/G9a 抑制剂,其细胞毒性低于 BIX-01294。
CSV0C018875 是基于喹啉的EHMT2/G9a 抑制剂,其细胞毒性低于 BIX-01294。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 10,600 | 6-8周 | |
50 mg | ¥ 13,800 | 6-8周 | |
100 mg | ¥ 17,500 | 6-8周 |
产品描述 | CSV0C018875 is a quinoline-based EHMT2/G9a inhibitor with lower cytotoxicity than BIX-01294 [1]. |
体外活性 | CSV0C018875 (2.5-20 μM; 48 hours) inhibits the levels of H3K9me2 modifications in the histones [1]. Western Blot Analysis [1] Cell Line: HEK293 cells Concentration: 2.5 μM, 10 μM, 20 μM Incubation Time: 48 hours Result: Inhibited the enzymatic activity of G9a in a dose-dependent manner in HEK293 cells. |
分子量 | 312.79 |
分子式 | C18H17ClN2O |
CAS No. | 442150-41-6 |
存储 | Shipping with blue ice. |
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