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Butabindide (UCL-1397) 是三肽肽酶II (TPP II)的选择性抑制剂,对 TPP I 和TPP II 的Ki 值分别为 10 μM 和 7 nM。Butabindide 抑制 TPP II 以保护 CCK-8 免于失活。
Butabindide (UCL-1397) 是三肽肽酶II (TPP II)的选择性抑制剂,对 TPP I 和TPP II 的Ki 值分别为 10 μM 和 7 nM。Butabindide 抑制 TPP II 以保护 CCK-8 免于失活。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
25 mg | ¥ 10,600 | 6-8周 | |
50 mg | ¥ 13,800 | 6-8周 | |
100 mg | ¥ 17,500 | 6-8周 |
产品描述 | Butabindide (UCL-1397) is a potent, selective inhibitor of tripeptidvl peptidase II (TPP II) with Ki values of 10 μM and 7 nM for TPP I and TPP II, respectively. Butabindide inhibits TPP II in order to protect CCK-8 against inactivation [1] [2]. |
体外活性 | Butabindide (UCL-1397; 0-24 nM; membranes of rat cerebral cortex) inhibits TPP II activity of cerebral membranes [2]. |
体内活性 | Butabindide (UCL-1397; 10 mg/kg; i.v.; for 20 min) inhibits the breakdown of CCK-8 in the gastrointestinal tract and increases satiety in mice [2]. Animal Model: Mice (25-30 g) Dosage: 10 mg/kg Administration: Intravenous injection; for 20 minutes Result: Reduces food intake and elicits other behavioral concomitants of satiation. |
分子量 | 303.4 |
分子式 | C17H25N3O2 |
CAS No. | 175553-48-7 |
存储 | Shipping with blue ice. |
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