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BRK inhibitor P21d hydrochloride
还可以产品编号 T39772Cas号 2250025-98-8
别名 BRK inhibitor P21d hydrochloride
BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM. Additionally, it effectively suppresses p-SAM68 with an IC50 value of 52 nM. This compound, BRK inhibitor P21d hydrochloride, serves as a valuable tool for evaluating the efficacy of BRK inhibitors in xenograft breast tumor models, enabling the assessment of their in vivo activity.
BRK inhibitor P21d hydrochloride
还可以产品编号 T39772 别名 BRK inhibitor P21d hydrochlorideCas号 2250025-98-8
BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM. Additionally, it effectively suppresses p-SAM68 with an IC50 value of 52 nM. This compound, BRK inhibitor P21d hydrochloride, serves as a valuable tool for evaluating the efficacy of BRK inhibitors in xenograft breast tumor models, enabling the assessment of their in vivo activity.
| 规格 | 价格 | 库存 | 数量 |
|---|---|---|---|
| 25 mg | ¥ 16,700 | 8-10周 | |
| 50 mg | ¥ 25,300 | 8-10周 | |
| 100 mg | ¥ 38,300 | 8-10周 |
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| 产品描述 | BRK inhibitor P21d hydrochloride is a highly potent inhibitor of breast tumor kinase (BRK/PTK6), displaying an IC50 of 30 nM. Additionally, it effectively suppresses p-SAM68 with an IC50 value of 52 nM. This compound, BRK inhibitor P21d hydrochloride, serves as a valuable tool for evaluating the efficacy of BRK inhibitors in xenograft breast tumor models, enabling the assessment of their in vivo activity. |
| 靶点活性 | Aurora B:>20 μM (IC50), Brk:30 nM (IC50), pSAM68:52 nM (IC50), Lck:>20 μM (IC50) |
| 体外活性 | BRK inhibitor P21d hydrochloride (compound 21d) inhibits Aurora B (IC 50 >20 μM) and Lck (IC 50 >20 μM)[1]. |
| 体内活性 | BRK inhibitor P21d hydrochloride (compound 21d) has much better permeability (CACO-2:314 nm/s) and PK profile (rat, po, 10 mpk, AUC 0–6h =31.1 μM?h,C 6h =3.5 μM)[1]. |
| 别名 | BRK inhibitor P21d hydrochloride |
| 分子量 | 483.93 |
| 分子式 | C23H23ClFN7O2 |
| CAS No. | 2250025-98-8 |
| 密度 | no data available |
储存&溶解度
| 存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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