JWH 302, a cannabimimetic indole, exhibits 5-fold selectivity for the central cannabinoid (CB1) receptor, evidenced by a Ki value of 17 nM, versus the peripheral cannabinoid (CB2) receptor, which has a Ki value of 89 nM. Additionally, JWH 302 stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 nM and 24.4 nM, respectively.
JWH 302
JWH 302
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产品编号 T84498Cas号 864445-45-4
JWH 302, a cannabimimetic indole, exhibits 5-fold selectivity for the central cannabinoid (CB1) receptor, evidenced by a Ki value of 17 nM, versus the peripheral cannabinoid (CB2) receptor, which has a Ki value of 89 nM. Additionally, JWH 302 stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 nM and 24.4 nM, respectively.
JWH 302, a cannabimimetic indole, exhibits 5-fold selectivity for the central cannabinoid (CB1) receptor, evidenced by a Ki value of 17 nM, versus the peripheral cannabinoid (CB2) receptor, which has a Ki value of 89 nM. Additionally, JWH 302 stimulates GTPγS binding of CB1 and CB2 receptors with EC50 values of 29.3 nM and 24.4 nM, respectively.
化学信息
分子量
335.447
分子式
C22H25NO2
CAS No.
864445-45-4
储存&溶解度
存储
Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
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