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ERAP1-in-1 是一种内质网氨基肽酶 1 (ERAP1) 抑制剂,能竞争性地抑制 ERAP1 对代表性生物底物九聚物肽的作用。
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ERAP1-in-1 是一种内质网氨基肽酶 1 (ERAP1) 抑制剂,能竞争性地抑制 ERAP1 对代表性生物底物九聚物肽的作用。
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
1 mg | ¥ 598 | 现货 | |
5 mg | ¥ 1,730 | 现货 | |
10 mg | ¥ 2,560 | 现货 | |
25 mg | ¥ 3,970 | 现货 | |
50 mg | ¥ 5,560 | 现货 | |
100 mg | ¥ 7,380 | 现货 | |
200 mg | ¥ 9,980 | 现货 | |
1 mL x 10 mM (in DMSO) | ¥ 1,750 | 现货 |
产品描述 | ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activity toward a nonamer peptide representative of physiological substrates. |
体外活性 | ERAP1-IN-1(50 μM)在细胞环境中展示出对ERAP1的特异性抑制效果。同时,ERAP1-IN-1能通过变构方式激活ERAP1对荧光和显色氨基酸底物的水解作用。 |
分子量 | 458.45 |
分子式 | C20H21F3N2O5S |
CAS No. | 865273-97-8 |
Smiles | COc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O |
密度 | 1.428 g/cm3 (Predicted) |
存储 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||||||||||||
溶解度信息 | DMSO: 250 mg/mL (545.32 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
溶液配制表 | ||||||||||||||||||||||||||||||||||||
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