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TargetMol | Compound Library

细胞凋亡化合物库现货

Apoptosis Compound Library

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产品编号 L9000

细胞凋亡是一种发生在多细胞生物中的程序性细胞死亡。相对于细胞坏死,细胞凋亡是受基因调控的主动过程,细胞凋亡时会发生特征性的形态学变化,产生称为凋亡小体的细胞碎片被吞噬细胞吞噬。细胞凋亡受到促凋亡因子(Fas 受体和 caspases)和抑凋亡因子(Bcl-2蛋白和 IAP)的调控,异常凋亡过程牵涉到多种疾病中,细胞凋亡的抑制可导致癌症、自身免疫性疾病、炎性疾病和病毒感染。另一方面,过度的细胞凋亡可能导致神经退行性疾病、血液疾病和组织损伤。目前在细胞凋亡与癌症发生和自身免疫性疾病之间的关系有着很多研究,人们希望激发癌细胞的细胞凋亡,以达到治疗癌症的目的。“细胞凋亡在神经退化性疾病中所扮演的角色(如阿兹海默氏症、亨丁顿舞蹈症、帕金森病、肌肉萎缩性侧索硬化症),是目前热门的研究领域。” TargetMol 细胞凋亡化合物库精选 2394 种与凋亡相关的生物活性小分子化合物,适用于癌症和神经退行性疾病相关研究。

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产品编号 L9000

细胞凋亡化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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产品描述 产品描述

  • 2394种与凋亡相关的生物活性小分子化合物的特有集合,多用于研究肿瘤发生发展机制和抗癌药物筛选等。可用于高通量筛选和高内涵筛选;
  • 靶点含Bcl-2、Caspase、p53、TNF-α和survivin等;
  • 通过前期临床研究和临床实验,生物活性和安全性已经得到验证;
  • 其中一些活性化合物已得到FDA批准上市;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR和HPLC检测技术保证产品高纯度和高质量;
  • 所有化合物现货供应。

Packaging And Storage | TargetMol 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。

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Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
EGFR
TNF
Endogenous Metabolite
NF-κB
Ferroptosis
Antibacterial
Caspase
Bcl-2 Family
JAK
CDK
STAT
COX
Reactive Oxygen Species
PI3K
ERK
p38 MAPK
Akt
VEGFR
DNA/RNA Synthesis
p53
Raf
Antibiotic
Antioxidant
IL Receptor
HDAC
FLT
Src
Antifungal
Microtubule Associated
c-RET
JNK
Parasite
mTOR
MEK
Mitophagy
RIP kinase
HIV Protease
PDGFR
AMPK
FGFR
c-Kit
Mdm2
Dehydrogenase
PERK
PARP
Aurora Kinase
E1/E2/E3 Enzyme
Epigenetic Reader Domain
Influenza Virus
Tyrosine Kinases
Bcr-Abl
HER
PKC
MAPK
Topoisomerase
HSP
Interleukin
Nrf2
PD-1/PD-L1
c-Met/HGFR
Phosphatase
PPAR
Wnt/beta-catenin
Pim
Ras
Proteasome
GSK-3
Nucleoside Antimetabolite/Analog
Potassium Channel
Histone Methyltransferase
IAP
ROS
MMP
NO Synthase
Mitochondrial Metabolism
Lipoxygenase
Sirtuin
Virus Protease
IκB/IKK
Cytochromes P450
ADC Cytotoxin
Calcium Channel
HSV
IGF-1R
AChR
RAAS
PDE
DNA-PK
Estrogen/progestogen Receptor
Chk
P-gp
Syk
FAK
ATPase
DUB
Beta Amyloid
S6 Kinase
DNA Alkylator/Crosslinker
Histone Demethylase
PKA
Estrogen Receptor/ERR
Gamma-secretase
Cholinesterase (ChE)
PDK
5-HT Receptor
HMG-CoA Reductase
HIF/HIF Prolyl-Hydroxylase
PROTACs
Dopamine Receptor
Rho
TRP/TRPV Channel
TGF-beta/Smad
Antiviral
Prostaglandin Receptor
TLR
Trk receptor
ALK
Retinoid Receptor
c-Fms
Phospholipase
HIF
Tyrosinase
Histamine Receptor
Histone Acetyltransferase
ASK
Casein Kinase
ATM/ATR
PLK
Anti-infection
S1P Receptor
NOS
HBV
Adrenergic Receptor
Immunology/Inflammation related
Drug Metabolite
BTK
DNA Alkylation
CaMK
SARS-CoV
Reverse Transcriptase
Ligand for E3 Ligase
GPR
Sodium Channel
TAM Receptor
Transferase
HCV Protease
Integrin
NADPH
Glutathione Peroxidase
MAO
UGT
Molecular Glues
Fatty Acid Synthase
GluR
Survivin
Kras
GABA Receptor
DAPK
DNA Methyltransferase
Kinesin
MRP
Antifolate
Cysteine Protease
iGluR
Antifection
Opioid Receptor
Pyroptosis
MLK
Monoamine Oxidase
Proton pump
LPL Receptor
Adenosine Receptor
Reductase
c-Myc
Serine Protease
Cell Cycle Arrest
ROCK
CSF-1R
IRE1
DPP-4
PTEN
DNA
Androgen Receptor
Telomerase
MNK
GPX
NOD-like Receptor (NLR)
DHFR
ROR
CRM1
Ligands for Target Protein for PROTAC
LTR
BACE
IFNAR
DYRK
Necroptosis
TOPK
Cholecystokinin Receptor
Hck
Serine/threonin kinase
FXR
Leukotriene Receptor
Aryl Hydrocarbon Receptor
LDL
P2X Receptor
Hexokinase
PAK
Hedgehog/Smoothened
Xanthine Oxidase
Transketolase
Wee1
Lipid
OXPHOS
PGE Synthase
Free radical scavengers
transporter
PAI-1
CRISPR/Cas9
Cuproptosis
SGK
NADPH-oxidase
NOD
Carbonic Anhydrase
Amino Acids and Derivatives
YAP
Tie-2
OCT
VDAC
Liver X Receptor
PYK2
NAMPT
Glucokinase
FOXO1
Glucocorticoid Receptor
FLAP
PAFR
Fas/FasL
NMDAR
ABC Transporter
Glucosidase
Smo
CXCR
Endothelin Receptor
PAD
KSP
cAMP
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Beta-Secretase
Acyltransferase
STING
LRRK2
Aminopeptidase
Hippo pathway
GST
Aromatase
BMI-1
IRAK
Sigma receptor
ROS Kinase
Apelin receptor
Chloride channel
Hydrogenase
MALT
NEDD8
Dynamin
P2Y Receptor
Na+/Ca2+ Exchanger
RAR/RXR 
Lipase
gp120/CD4
GTPase
VDA
Progesterone Receptor
Melatonin Receptor
GNRH Receptor
RANKL/RANK
Amylase
IDO
SIK
Myosin
MTH1
DNA gyrase
Monoamine Transporter
Guanylate cyclase
PROTAC Linker
Thioredoxin
FAAH
Stearoyl-CoA Desaturase (SCD)
CCR
ACK1
Somatostatin
Norepinephrine
Glutathione reductase
Ephrin Receptor
AIM2
hCE
HuR
MELK
RSV
Neprilysin
FKBP
Protease
LPA Receptor
Melanocortin Receptor
KLF
PI4K
Adenosine Deaminase
Cannabinoid Receptor
Platelet aggregation
APC/C
Thrombin
Protease-activated Receptor
Lysosomal Autophagy
p97
CFTR
Imidazoline Receptor
PKM