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TargetMol | Compound Library

抗癌活性化合物库现货

Anti-Cancer Active Compound Library
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货号 L2160

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

根据文献报道和有关公开资料,我们挑选了 4270 个具有已知抗癌活性的化合物组成抗癌活性库,可用于具体癌症的阳性对照及癌症机理的研究。希望我们在抗癌研究的路上,助您一臂之力!

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
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货号 L2160

抗癌活性化合物库

规格

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 4270种具有抗肿瘤活性的化合物的特有集合,用于高通量、高内涵筛选;
  • 是肿瘤发生机理研究、抗肿瘤药物筛选的有效工具;
  • 靶点含PI3K、HDAC、mTOR、CDK、Aurora Kinase、JAK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Parasite
Microtubule Associated
Topoisomerase
mTOR
Epigenetic Reader Domain
Caspase
Antifungal
Reactive Oxygen Species
Bcl-2 Family
ERK
Dehydrogenase
COX
FLT
Nucleoside Antimetabolite/Analog
STAT
PDGFR
PARP
p38 MAPK
Histone Methyltransferase
HDAC
FGFR
Estrogen Receptor/ERR
TNF
Wnt/beta-catenin
c-Met/HGFR
Cytochromes P450
c-Kit
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Ferroptosis
Src
Raf
Interleukin
MDM-2/p53
JAK
HSP
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Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
AMPK
NO Synthase
Bcr-Abl
ALK
Aurora Kinase
Androgen Receptor
PPAR
JNK
Nrf2
MEK
Calcium Channel
SARS-CoV
P-gp
E1/E2/E3 Enzyme
DUB
HIF/HIF Prolyl-Hydroxylase
GSK-3
FAK
IL Receptor
MAPK
TLR
p53
PROTACs
Mitophagy
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DNA Alkylator/Crosslinker
HSV
IGF-1R
Antiviral
Mitochondrial Metabolism
c-RET
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Chk
PDE
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HER
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Pim
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5-HT Receptor
Retinoid Receptor
PERK
Casein Kinase
Transferase
Hedgehog/Smoothened
Mdm2
HIF
ROS Kinase
DNA Methyltransferase
PLK
Reductase
Smo
GABA Receptor
PD-1/PD-L1
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Integrin
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transporter
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FKBP
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CD38
VDA
Target Protein Ligand-Linker Conjugates
LAG-3
Monoamine Transporter
PROTAC Linker
Transketolase
CAT
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
Vasopressin Receptor
Carboxypeptidase
Melanocortin Receptor
GHSR
Poly(ADP-ribose) Glycohydrolase (PARG)
ADC Linker
Ferroportin

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