购物车
  • TargetMol
    您的购物车当前为空
TargetMol | Compound Library

抗癌活性化合物库现货

Anti-Cancer Active Compound Library
Rating icon 很棒
货号 L2160

尽管在过去的几十年中癌症的研究和治疗取得了巨大的成功,但癌症仍然是人类面临的巨大挑战,给患者身心健康带来巨大的痛苦。癌细胞具有许多显著不同的生物学特征,表现出无限的增殖潜能,维持自身生长信号的持续稳定,逃避应激信号诱导的细胞凋亡,刺激血管生长,为肿瘤提供营养,同时逃避免疫系统防御和诱导局部慢性炎症,发挥其侵袭和转移能力;并且表现出异常的代谢活动,并通过突变和表观遗传机制显著改变全基因组的稳定性。

根据文献报道和有关公开资料,我们挑选了 4270 个具有已知抗癌活性的化合物组成抗癌活性库,可用于具体癌症的阳性对照及癌症机理的研究。希望我们在抗癌研究的路上,助您一臂之力!

TargetMol 的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
资源下载
化合物库相关信息
Excel
SDF
联系我们获取更多批次信息

货号 L2160

抗癌活性化合物库

规格

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
询价 & 定制

产品描述 产品描述

  • 4270种具有抗肿瘤活性的化合物的特有集合,用于高通量、高内涵筛选;
  • 是肿瘤发生机理研究、抗肿瘤药物筛选的有效工具;
  • 靶点含PI3K、HDAC、mTOR、CDK、Aurora Kinase、JAK等;
  • 结构多样,药效显著,可渗透细胞;
  • 详细的说明书,化合物结构、靶点信息、IC50值、活性描述等;
  • NMR、HPLC/LCMS检测技术保证产品高纯度和高质量,减少假阳性发生概率。

包装和储存 包装和储存

  • 可选用DMSO耐受的96/384孔板或2D 条形码编码管;
  • 干粉蓝冰运输,DMSO溶液干冰运输;
  • 排布:96孔板:1st & 12th 空白对照,384孔板:1st & 2nd & 23th & 24th空白对照。
  • 本化合物库通常以 DMSO 10 mM 浓度提供。少量产品可能因溶解性或稳定性需求,采用其他溶剂或浓度包装,具体以实际产品信息为准。

使用TargetMol产品
发表顶级期刊文献

引用更多关于TargetMol产品的科学文献吧!

查看更多

Library Customization | TargetMol 化合物库定制

Compound Library | TargetMol
您可以通过点击按钮
定制您专属的化合物!
联系专属定制

Library Customization | TargetMol 化合物库组成

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Microtubule Associated
Parasite
Topoisomerase
mTOR
Epigenetic Reader Domain
Caspase
Antifungal
Reactive Oxygen Species
Bcl-2 Family
ERK
FLT
Dehydrogenase
Nucleoside Antimetabolite/Analog
PDGFR
COX
STAT
Histone Methyltransferase
PARP
p38 MAPK
HDAC
FGFR
c-Met/HGFR
Estrogen Receptor/ERR
TNF
Wnt/beta-catenin
Cytochromes P450
HIV Protease
c-Kit
Ferroptosis
Src
Raf
Interleukin
Phosphatase
JAK
MDM-2/p53
HSP
Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
Bcr-Abl
AMPK
NO Synthase
ALK
Aurora Kinase
Androgen Receptor
PPAR
JNK
Nrf2
Calcium Channel
E1/E2/E3 Enzyme
P-gp
SARS-CoV
MEK
GSK-3
DUB
FAK
HIF/HIF Prolyl-Hydroxylase
IL Receptor
MAPK
TLR
PROTACs
p53
DNA Alkylator/Crosslinker
HSV
IGF-1R
TGF-beta/Smad
Mitophagy
Antiviral
Drug Metabolite
Mitochondrial Metabolism
c-RET
AChR
Histone Demethylase
PDE
Chk
Sirtuin
ATM/ATR
Proteasome
Gamma-secretase
Lipoxygenase
Potassium Channel
TAM Receptor
Tyrosine Kinases
HER
Trk receptor
Histone Acetyltransferase
c-Fms
DNA-PK
Pim
Adrenergic Receptor
Molecular Glues
Cholinesterase (ChE)
Sodium Channel
S6 Kinase
PERK
Casein Kinase
Retinoid Receptor
5-HT Receptor
Mdm2
Transferase
Hedgehog/Smoothened
HIF
ROS Kinase
Integrin
Reductase
Smo
PLK
DNA Methyltransferase
PD-1/PD-L1
ADC Cytotoxin
Serine Protease
IAP
Fatty Acid Synthase
CXCR
GABA Receptor
Anti-infection
Kinesin
YAP
Histamine Receptor
HBV
Aryl Hydrocarbon Receptor
HCV Protease
Glutathione Peroxidase
PKA
TRP/TRPV Channel
DNA Alkylation
PDK
Tyrosinase
LPL Receptor
c-Myc
Antifolate
Beta Amyloid
Phospholipase
Dopamine Receptor
Serine/threonin kinase
IDO
Antifection
Isocitrate Dehydrogenase (IDH)
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
S1P Receptor
BTK
GPCR
Carbonic Anhydrase
DNA
transporter
IκB/IKK
Aromatase
DHFR
MAO
Immunology/Inflammation related
CSF-1R
Prostaglandin Receptor
Syk
IKZF
ATPase
NOS
Adenosine Receptor
DYRK
Rho
ROCK
CaMK
OXPHOS
Monocarboxylate transporter
NADPH
Cell Cycle Arrest
Cysteine Protease
Glutaminase
glycosidase
Survivin
AhR
Monoamine Oxidase
IFNAR
Progesterone Receptor
Photosensitizer
RIP kinase
Glucosidase
Telomerase
BCRP
STING
Ephrin Receptor
Reverse Transcriptase
NOD
Proton pump
Amino Acids and Derivatives
Tie-2
Cholecystokinin Receptor
RANKL/RANK
Glucocorticoid Receptor
iGluR
Opioid Receptor
PAK
CCR
Wee1
MNK
Acyltransferase
PAI-1
Methionine Adenosyltransferase (MAT)
GPX
IRAK
NOD-like Receptor (NLR)
Chloride channel
MicroRNA
Bcl-6
GNRH Receptor
NAMPT
IRE1
P2X Receptor
ABC Transporter
Somatostatin
Lipid
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
ROR
Ligands for Target Protein for PROTAC
RAAS
Necroptosis
ATG
Liver X Receptor
Leukotriene Receptor
Glucokinase
PYK2
UGT
Endothelin Receptor
Angiotensin-converting Enzyme (ACE)
GluR
Orphan Receptor
PSMA
Aminopeptidase
Pyroptosis
LPA Receptor
BMI-1
HMG-CoA Reductase
Thrombin
p97
PKM
MALT
GTPase
Galectin
Myosin
MTH1
NMDAR
Hexokinase
FAAH
PTEN
cAMP
MELK
p62
Hydroxylase
FOXO
Complement System
Neurokinin receptor
DAPK
NEDD8
CRM1
MyD88
LTR
Arrestin
Lipase
TOPK
Factor Xa
MRP
Serotonin Transporter
FXR
NR4A
GRK
Bombesin Receptor
ACK1
Xanthine Oxidase
PAD
KSP
Cadherin
Porcupine
CD73
Decarboxylase
ASK
GST
ribosome
KLF
CRISPR/Cas9
Adenosine Deaminase
SGK
Platelet aggregation
APC/C
Protease-activated Receptor
MLK
FOXO3
Thyroid hormone receptor(THR)
RAR/RXR
Factor VIIa
MIF
CaSR
Hck
Neurotensin Receptor
Vitamin
Adenylate cyclase
Annexin A
FLAP
Adiponectin Receptor
PAFR
Haspin Kinase
Arp2/3 Complex
DNA gyrase
Stearoyl-CoA Desaturase (SCD)
Thrombopoietin Receptor
ATP Citrate Lyase
GPCR19
E3 Ligase Ligand-Linker Conjugates
HuR
RSV
Drug-Linker Conjugates for ADC
Hippo pathway
Acetyl-CoA Carboxylase
FKBP
Protease
PI4K
Cuproptosis
Gap Junction Protein
Sigma receptor
Lysosomal Autophagy
CFTR
PARG(Poly(ADP-ribose) Glycohydrolase)
Apelin receptor
Advanced Glycation End Products
CAT
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
Dynamin
Y Box Binding Protein 1
Arginase
P2Y Receptor
Na+/Ca2+ Exchanger
gp120/CD4
VDA
Melatonin Receptor
OCT
Kisspeptin
AAK1
B7
Target Protein Ligand-Linker Conjugates
LIM Kinase
Stemness kinase
LDLR
Amylase
LAG-3
SIK
Prolyl Endopeptidase (PREP)
FABP
LDL
GlyT
Na-K-Cl cotransporter
PROTAC Linker
DPP-4
Neuropeptide Y Receptor
Thioredoxin
Vasopressin Receptor
HCAR
Epoxide Hydrolase
Transketolase
SGLT
Beta-Secretase
PGE Synthase
Glutathione reductase
LRRK2
Free radical scavengers
Urea Transporter
GluCls
NEDD4-1
Carboxypeptidase
TMV
Melanocortin Receptor
GHSR
Aquaporin
RXFP receptor
NADPH-oxidase
Tight Junction Protein
Liposome
Glyoxalase
Ferroportin
ADC Linker
Poly(ADP-ribose) Glycohydrolase (PARG)

Keywords