首页工具

登录

搜索结果

Search Results for " spasms "

Targets Recommended: 5-HT Receptor

16

抑制剂 & 化合物

3

同位素标记化合物

如果没找到您满意的产品或者您对产品有其他要求，可以联系我们专业顾问为您提供针对性的合理建议。 QQ咨询网站留言咨询

Cat. No.	Product Name	Target	Signaling Pathways
T1092	Zolmitriptan 佐米曲普坦,311C90,BW-311C90	5-HT Receptor	GPCR/G Protein; Neuroscience
	Zolmitriptan (311C90) 是一种5-HT1B/1D 受体部分激动剂，可用于偏头痛的研究，对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。
T33846	Oxyphenonium bromide Spasmophen,Oxifenon,奥芬溴铵,Oxyfenon,Atrenyl,Oxyphenon	Others	Others
	Oxyphenonium bromide (Oxyfenon) 具有抗胆碱能活性，可用于治疗胃和十二指肠溃疡以及缓解内脏痉挛的研究。
T21447	Tolazoline Priscol,妥拉苏林,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Tolazoline (Benzalolin) 是一种竞争性的α-肾上腺素受体拮抗剂。
T1065	Baclofen 巴氯芬,Lioresal	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Baclofen (Lioresal) 是 γ-氨基丁酸 (GABA) 的亲脂性衍生物，是可口服的选择性代谢型 GABA-B 受体激动剂，具有高血脑屏障渗透率，用于治疗因脊髓损伤和多发性硬化引起的痉挛。
T1475	Fesoterodine fumarate Toviaz,SPM 907,富马酸非索罗定	AChR	Neuroscience
	Fesoterodine fumarate (Toviaz) 是可口服的，非亚型选择性的竞争性毒蕈碱受体拮抗剂，用于膀胱过度活动症，对 M1、M2、M3、M4 和 M5 受体的pKi 值分别为 8.0、7.7、7.4、7.3 和 7.5。
T0786	Clidinium bromide 克利溴铵,Ro 2-3773	AChR	Neuroscience
	Clidinium bromide (Ro 2-3773) 是季胺抗毒蕈碱剂，可通过减少胃酸和减慢肠道速度，缓解痉挛和腹部疼痛的症状。
T34121	Pramiverine EMD 9806,HSP 2986,EMD9806,HSP2986,EMD-9806	Others	Others
	Pramiverine is a long-acting choline dissolving agent used for gastrointestinal spasms.
T33314	Methantheline Bromide Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide	Others	Others
	Methantheline Bromide is a synthetic spasmolytic used to relieve cramps or spasms of the stomach, bowel, and bladder. It is also useful for intestinal or gastric ulcers (peptic ulcer disease), intestinal problems, pancreatitis, gastritis, biliary dysmotil
T21376	Chlorphenesin Carbamate Kolpicortin-sine,Rinlaxer,Chlorphensin carbamate,Maolate,氯苯氨酸甘油酯,laChlorphenesin Carbamate	Others	Others
	Chlorphenesin Carbamate is a centrally acting muscle relaxant used to treat muscle pain and spasms and also an antifungal agent.
T25654	Leiopyrrole Leioplegil,DV 714,Leiopyrrolum,DV714,DV-714	Others	Others
	Leiopyrrole 是一种抗胆碱能化合物，能够用于解痉挛。
T70153	Pipoxolan hydrochloride	Others	Others
	Pipoxolan (HCl) is an antispasmodic drug. In vivo, the drug inhibited the contractions of intestines caused by neostigmine, barium chloride or injection of acetylcholine. The drug possesses ganglioplegic action and inhibited the decrease in blood pressure caused by stimulation of the vagus nerve. The drug is marketed under tradename Rowapraxin worldwide for the treatment of spasms and colics in the gastrointestinal tract, gallbladder and urogenital area, bronchial spasms, spastic menstrual cramp...
T61453	Propantheline	Others	Others
	Propantheline is an orally active antagonist of muscarinic acetylcholine receptors (mAChRs), commonly employed to investigate smooth muscle dysfunction, hyperhidrosis, smooth muscle spasms or cramps in the stomach, intestines, or bladder, as well as involuntary urination [1] [2] [3].
T29000	Tralomethrin EPA Pesticide Chemical Code 121501,SAGA,HAG-107,HAG 107,Scout	Others	Others
	Tralomethrin is used as a pyrethroid insecticide. It modifies the gating kinetics of the sodium channels in neurons, increases the length of time the channel remains open after a stimulus, thereby depolarizing the neuron for a longer period of time. This leads to uncontrolled spasms, paralysis, and eventual death.
T69661	Pipoxolan (free base)	Others	Others
	Pipoxolan (free base) is an antispasmodic drug. In vivo, the drug inhibited the contractions of intestines caused by neostigmine, barium chloride or injection of acetylcholine. The drug possesses ganglioplegic action and inhibited the decrease in blood pressure caused by stimulation of the vagus nerve. The drug is marketed under tradename Rowapraxin worldwide for the treatment of spasms and colics in the gastrointestinal tract, gallbladder and urogenital area, bronchial spasms, spastic menstrual...
T25325	Dicyclonon LAB 145-138H,BAS 145-138	Others	Others
	Dicyclonon is a muscarinic antagonist utilized as an antispasmodic and in urinary incontinence. It has little effect on glandular secretion or the cardiovascular system. It has some local anesthetic properties and is utilized in biliary, gastrointestinal,
T37950	2-(Isopentylamino)naphthalene-1,4-dione	Others	Others
	2-(Isopentylamino)naphthalene-1,4-dione is a vitamin K analog.1It inhibits spasms induced by pentylenetetrazole and tonic hindlimb extension induced by maximal electroshock (MES) in mice (ED50s = 349.2 and 108.1 mg/kg, respectively). It also protects mice against seizures in the 6 Hz psychomotor seizure test (ED50s = 152.7 and 263.7 mg/kg at stimulus intensities of 32 and 44 mA, respectively). 1.Li, X., Himes, R.A., Prosser, L.C., et al.Discovery of the first vitamin K analogue as a potential tr...

化合物

Cat.No: T1092

Synonym: 佐米曲普坦,311C90,BW-311C90

Target: 5-HT Receptor

Oxyphenonium bromide

Cat.No: T33846

Synonym: Spasmophen,Oxifenon,奥芬溴铵,Oxyfenon,Atrenyl,Oxyphenon

Target: Others

Cat.No: T21447

Synonym: Priscol,妥拉苏林,Priscoline,Pridazole,Divascol,Vasimid,Benzalolin

Target: Adrenergic Receptor

Cat.No: T1065

Synonym: 巴氯芬,Lioresal

Target: GABA Receptor

Fesoterodine fumarate

Cat.No: T1475

Synonym: Toviaz,SPM 907,富马酸非索罗定

Target: AChR

Clidinium bromide

Cat.No: T0786

Synonym: 克利溴铵,Ro 2-3773

Target: AChR

Cat.No: T34121

Synonym: EMD 9806,HSP 2986,EMD9806,HSP2986,EMD-9806

Target: Others

Methantheline Bromide

Cat.No: T33314

Synonym: Frenogastrico,Dixamone bromide,Banthine,Asabaine,Methanthelinium bromide

Target: Others

Chlorphenesin Carbamate

Cat.No: T21376

Synonym: Kolpicortin-sine,Rinlaxer,Chlorphensin carbamate,Maolate,氯苯氨酸甘油酯,laChlorphenesin Carbamate

Target: Others

Cat.No: T25654

Synonym: Leioplegil,DV 714,Leiopyrrolum,DV714,DV-714

Target: Others

Pipoxolan hydrochloride

Cat.No: T70153

Target: Others

Cat.No: T61453

Target: Others

Cat.No: T29000

Synonym: EPA Pesticide Chemical Code 121501,SAGA,HAG-107,HAG 107,Scout

Target: Others

Pipoxolan (free base)

Cat.No: T69661

Target: Others

Cat.No: T25325

Synonym: LAB 145-138H,BAS 145-138

Target: Others

2-(Isopentylamino)naphthalene-1,4-dione

Cat.No: T37950

Target: Others

Cat. No.	Product Name	Target	Signaling Pathways
TMID-0252	Diazepam-d5
	Diazepam-d5 是 Diazepam 的氘代化合物。Diazepam 的 CAS 号为 439-14-5。
TMIH-0163	Clidinium Bromide-d5
	Clidinium Bromide-d5 是 Clidinium Bromide 的氘代化合物。Clidinium Bromide 的 CAS 号为 3485-62-9。Clidinium bromide 是季胺抗毒蕈碱剂，可通过减少胃酸和减慢肠道速度，缓解痉挛和腹部疼痛的症状。
TMIJ-0314	Baclofen-d4
	Baclofen-d4 是 Baclofen 的氘代化合物。Baclofen 的 CAS 号为 1134-47-0。Baclofen 是 γ-氨基丁酸 (GABA) 的亲脂性衍生物，是可口服的选择性代谢型 GABA-B 受体激动剂，具有高血脑屏障渗透率，用于治疗因脊髓损伤和多发性硬化引起的痉挛。

同位素标记化合物

Cat.No: TMID-0252

Clidinium Bromide-d5

Cat.No: TMIH-0163

Cat.No: TMIJ-0314

我们的所有产品和服务仅用于科学研究，不能被用于人体，我们也不向个人提供产品和服务。

Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved. 沪ICP备20019793号-4

沪公网安备 31010602006700号

沪公网安备 31010602006700号

TargetMol Loading

联系我们

电话：

400-820-0310

邮箱：

service@tsbiochem.com

QQ：

2881945090（终端用户）

2885109491（经销商）

经销：

终端：

地址：

上海市静安区江场三路238号8楼