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Search Results for " peripheral antinociceptive "
Targets Recommended: Others

1

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T61850 Adenosine receptor inhibitor 1

Others Others
Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties. Therefore, Adenosine receptor inhibitor 1 holds great promise for investigating cancer and neurodegenerative diseases [1].

化合物

Adenosine receptor inhibitor 1
Cat.No: T61850
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T7907 7-Methoxyflavone

Others Others
7-Methoxyflavone 是一种分离自 Zornia brasiliensis 的化合物。它能够抑制福尔马林疼痛反应神经源期的舔爪时间 (65.6%),有外周镇痛活性,但不影响炎症期的伤害性反映。
T2786 Oxysophocarpine

氧化槐树碱,氧卡地平

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Oxysophocarpine 是提取自海藻的生物碱。它对中枢神经系统和周围神经系统具有神经保护作用和抗伤害感受作用。

天然产物

7-Methoxyflavone
Cat.No: T7907
Synonym:
Target: Others
Oxysophocarpine
Cat.No: T2786
Synonym: 氧化槐树碱,氧卡地平
Target: Prostaglandin Receptor
TargetMol Loading
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