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Targets Recommended: Adrenergic Receptor

1503

抑制剂 & 化合物

171

天然产物

130

化合物库

14

TargetMol 试剂盒

465

重组蛋白

20

同位素标记化合物

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Cat. No. Product Name
L7800 高溶解性片段库

2728 compounds
2728 种片段分子合集,数量适中,是 FBDD 方法新药筛选的有力工具。
L7820 高溶解性微型片段化合物库

1081 compounds
高溶解性微型片段化合物库由 1081 个低分子量片段组成。
L7830 高溶解性片段药效团化合物库

985 compounds
高溶解性片段药效团库包含985 个片段小分子。
L7840 高溶解性卤化片段化合物库

796 compounds
高溶解性卤化片段库包含796 个卤化片段化合物。
L7850 高溶解性3D结构多样性片段化合物库

1079 compounds
高溶解性3D 结构多样性片段库包含1079 个化合物。
L7810 高溶解性多官能团片段化合物库

1159 compounds
高溶解性多官能团片段库包含1159 种片段分子
LF1030 LC高溶解性片段化合物库

9600 compounds
L2010 高选择性抑制剂库

575 compounds
575种具有高选择性的抑制剂集合
L6900 稀有天然产物库

693 compounds
693 种稀有天然产物的集合,可以用于高通量和高内涵筛选;
LF1000 多样性核心预制库

50000 compounds
For your convenience, there are Diversity Sets of 5,000, 10,000, 15,000, and 20,000 compounds with no structure overlap.
L9610 环肽库

80 compounds
80 种环肽分子,可用于高通量和高内涵筛选;
L3410 临床前化合物库

701 compounds
701 种临床前小分子化合物的特有集合,用于高通量、高内涵筛选;
L3900 DNA 损伤和修复分子库

910 compounds
910 个与 DNA 损伤和修复紧密相关的化合物集合,是高通量筛选,高内涵筛选的良好载体;
L6100 天然多酚类化合物库

635 compounds
635 个天然多酚化合物的独特集合,可用于高通量、高内涵筛选;
L2000 抑制剂库

8328 compounds
8328 个小分子抑制剂的独特集合,主要用于细胞信号研究、新药筛选、高通量筛选和高内涵筛选;
L6230 苗药化合物库

534 compounds
534种苗族特色药材的天然产物分子,可用于高通量和高内涵筛选
L6010 天然产物库

3840 compounds
3840 种天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L1510 核受体化合物库

531 compounds
531 个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2400 内分泌激素分子库

784 compounds
784 种与内分泌系统相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L8400 血液病分子库

514 compounds
514 种造血系统疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L1200 表观遗传库

953 compounds
953 种表观遗传学研究相关的生物活性小分子的特有集合,用于表观遗传学研究及其相关的检测和高通量、高内涵筛选;
L5400 抗心血管疾病化合物库

1408 compounds
1408 种心血管疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L6220 蒙药化合物库

950 compounds
950 种蒙药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L3600 细胞因子抑制剂库

604 compounds
604 个与细胞因子紧密相关的化合物集合,是高通量、高内涵筛选的良好载体;
L2120 抗癌临床化合物库

2545 compounds
2545 个具有抗癌活性小分子的独特集合,可用于高通量高内涵筛选。
L7000 活性脂质化合物库

385 compounds
385 种生物活性小分子化合物,用于高通量、高内涵筛选;
L6300 药食同源库

1290 compounds
1290 个药食同源化合物的独特集合,可用于高通量筛选和高内涵筛选;
L3700 JAK-STAT 化合物库

252 compounds
252 个 JAK/STAT 靶点相关的小分子化合物的独特集合,用于高通量、高内涵筛选;
L9200 药物功能重定位化合物库

4630 compounds
4630 种全球上市药物和临床药物的独特集合,可用于高通量筛选和高内涵筛选,是老药新用、新的药物靶点筛选和细胞诱导的有效工具。
L5500 毒性化合物库

262 compounds
262 个细胞毒性化合物的特有集合,可用于高通量、高内涵筛选。
L8300 染色质修饰分子库

250 compounds
250 种染色质化学修饰相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L2800 5-羟色胺分子库

268 compounds
268 种生物活性小分子化合物,用于高通量、高内涵筛选;
L4100 TGF-β/Smad靶点化合物库

184 compounds
184 个 TGF-β/Smad 靶点相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L9850 口服活性化合物库

2427 compounds
2427 种口服活性化合物独特集合,可用于高通量筛选和高内涵筛选
L2910 抗氧化化合物库

1314 compounds
氧化应激(Oxidative Stress,OS)是指体内氧化与抗氧化作用失衡的一种状态。氧化应激导致活性氧(ROS)大量积累,氧化程度超出抗氧化物的清除能力,从而引起氧化损伤,氧化应激损伤是许多疾病发生的基础,不同程度的氧化应激造成的细胞效应与心脑血管疾病、神经退行性病变、炎症和肿瘤密切相关。抗氧化剂是一类能够对抗氧化应激,降低氧化损伤的一类化合物。 TargetMol 抗氧化化合物库是1314 种对氧化应激具有抑制作用的小分子特有集合,是研究氧化应激的有用工具,可以用于高通量筛选和高内涵筛选。
L6610 抗感染天然产物库

1060 compounds
1060 个抗感染相关的天然产物集合,是药物开发、药理研究的有效工具;
L8000 干细胞分化化合物库

1197 compounds
1197 种干细胞分化信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选;
L1000 上市药物库

2808 compounds
2808 个上市药物化合物集合,可用于高通量筛选和高内涵筛选;
L2600 神经信号分子库

2540 compounds
2540 种CNS 相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L2152 靶向治疗药物库

119 compounds
119 个肿瘤靶向治疗药物,可以用于高通量和高内涵筛选;
L2140 癌细胞分化化合物库

406 compounds
406 个诱导肿瘤细胞分化化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2130 抗癌细胞代谢库

1268 compounds
1268 种癌细胞代谢相关的生物活性小分子化合物的特有集合,用于肿瘤相关的研究以及抗肿瘤药物的筛选,用于高通量、高内涵筛选;
L1010 FDA上市及药典收录分子库

3158 compounds
3158 个上市及药典分子集合,可用于高通量筛选和高内涵筛选;
L9240 农药化合物库

270 compounds
270种农药相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L3980 DNA损伤/修复库Plus

667 compounds
667 种 DNA 损伤/修复靶向、结构新颖的化合物;
L1600 激酶抑制剂库

2720 compounds
2720 种激酶抑制剂/调节剂的独特集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
L9410 共价抑制剂库

1920 compounds
1920 种小分子的独特集合,包含已发现的共价抑制剂以及包含某些共价反应基团常见弹头的分子,如氯乙酰基,2-氯丙酰基,丙烯酰基,1-丙-2-炔基,1-丁-2-炔基,酮羰基,二硫键等,可以用于共价抑制剂药物研发;
L2300 离子通道库

931 compounds
931 种与离子通道相关的生物活性小分子化合物的特有集合,用于离子通道相关的疾病和药物研究,可用于高通量筛选和高内涵筛选;
L4300 Wnt/Hedgehog/Notch 通路化合物库

237 compounds
237 个Wnt & Hedgehog & Notch 靶点相关的生物活性小分子化合物的特有集合,用于相关通路的研究及药物的筛选,可用于高通量、高内涵筛选。
L1610 FDA 上市激酶抑制剂库

263 compounds
263种靶向激酶的上市药物集合,用于特定靶向激酶,可用于高通量筛选和高内涵筛选;
L8600 泛素化化合物库

210 compounds
210 种泛素化相关的小分子,用于高通量和高内涵筛选;
L1500 GPCR靶点分子库

1940 compounds
1940 种与 G 蛋白及其耦联受体相关的生物活性小分子化合物,所有小分子都具有良好的生物和药理活性,部分是 FDA 批准的上市药物;
L3800 NF-κB 通路分子库

729 compounds
729 个 NF-κB 信号通路相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L6210 藏药化合物库

747 compounds
747 种藏药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L2195 抗前列腺癌化合物库

2070 compounds
2070 种与前列腺癌相关的化合物,可以用于高通量和高内涵筛选
L2900 氧化还原化合物库

1264 compounds
1264 个活性化合物,已经验证具有一定的抗氧化活性,包括 ROS 清除剂、iNOS、eNOS、及抗氧化的天然产物,是研究疾病机理以及药物研究的优良载体
L4200 FDA 上市药物库

1729 compounds
1729 个FDA 批准药物的独特集合,可用于高通量筛选和高内涵筛选;
L7870 可溶性羧酸片段化合物库

1806 compounds
可溶性羧酸片段库包含 1806 个化合物
L5200 抗代谢疾病化合物库

1544 compounds
1544 个代谢疾病相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L1300 PI3K/Akt/mTOR 化合物库

420 compounds
420 种与PI3K/Akt/mTOR 相关的生物活性小分子化合物的特有集合,用于PI3K/Akt/mTOR 相关研究以及高通量、高内涵筛选;
L6200 瑶药化合物库

221 compounds
221 种瑶药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L6700 抗癌天然产物库

1772 compounds
1772 种已知活性天然产物的独特集合,是肿瘤药物开发、抗癌先导化合物筛选等领域的有力工具,可用于HTS 和HCS。
L2191 抗乳腺癌化合物库

1939 compounds
1939 种与乳腺癌相关的化合物,可以用于抗乳腺癌药物研发和药理研究;
L1800 抗感染化合物库

2938 compounds
2938 种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
L3400 临床期小分子药物库

3404 compounds
3404 个临床期化合物集合,可用于高通量筛选和高内涵筛选;
L4510 抗寄生虫库

419 compounds
419 种具有抗寄生虫活性的小分子化合物;
L3100 造血毒性小分子库

101 compounds
101 种生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L2521 糖酵解化合物库

555 compounds
555 种糖酵解相关的活性化合物,可用于高通量和高内涵筛选
L2570 人代谢物化合物库

4454 compounds
4454 种人代谢物的独特集合,用于高通量、高内涵筛选;
L1700 抗病毒库

1040 compounds
1040 种具有抗病毒活性的化合物的特有集合,是筛选新型抗病毒药的有效工具;可用于高通量筛选和高内涵筛选;
L2151 化疗药物库

48 compounds
48 个肿瘤化疗药物,可以用于高通量和高内涵筛选;
L5800 药物代谢杂质库

197 compounds
197 种药物异构体/代谢产物的特有集合,可用于高通量、高内涵筛选;
L9230 ReFRAME 相关化合物库

3210 compounds
3210 化合物的独特集合,可用于高通量筛选和高内涵筛选
L9210 儿童药物库

972 compounds
972 种儿童药物的独特集合,可用于高通量筛选和高内涵筛选
L7300 钾通道分子库

152 compounds
152 种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L4710 非甾体类抗炎化合物库

530 compounds
530 种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
L6001 Mini真菌代谢天然产物筛选库

Inquiry
L4020 NO PAINS 化合物库

9384 compounds
TargetMol NO PAINS 化合物库包含 9384 个剔除了PAINS 的小分子活性化合物,可用于新药研发,信号通路研究,老药新用等研究。
L6030 天然产物衍生物虚筛化合物库

163000 compounds
16.3万种天然产物衍生物,并且在持续增加中;
L2194 抗结直肠癌化合物库

1545 compounds
1545 种与结直肠癌相关的化合物,可以用于高通量和高内涵筛选;
L3500 组蛋白修饰化合物库

469 compounds
469 个组蛋白修饰相关的小分子化合物的特有集合,用于高通量、高内涵筛选;
L3200 自噬库

1248 compounds
1248 种细胞自噬相关的生物活性小分子化合物的特有集合,用于自噬相关的研究,用于高通量、高内涵筛选;
L2200 酪氨酸激酶分子库

1016 compounds
1016 种酪氨酸激酶抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
L6400 海洋天然产物库

144 compounds
144 种海洋来源的单体化合物,是药物开发、药理研究等领域的有力工具;
L2150 抗癌药物库

3080 compounds
3080 个具有抗癌活性小分子的独特集合,生物活性已经临床前实验证实,可用于高通量、高内涵筛选;
L8720 细胞焦亡化合物库

1066 compounds
1066 种细胞焦亡相关的化合物,可以用于细胞焦亡相关研究。
L2560 代谢化合物库

2320 compounds
2320 种代谢途径相关的化合物,可用于高通量和高内涵筛选。
L2160 抗癌活性化合物库

3188 compounds
3188 种具有抗肿瘤活性的化合物的特有集合,用于高通量、高内涵筛选;
L6130 萜类天然产物库

622 compounds
622 种萜类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L6620 抗寄生虫天然产物库

253 compounds
253 个抗寄生虫相关的天然产物集合,是药物开发、药理研究的有效工具;
L6000 高通量筛选天然产物库

4533 compounds
4533 种天然产物的独特集合,是药物开发、药理研究、干细胞分化、指纹图谱研究、质量研究等领域的有力工具,可用于HTS 和HCS;
L2100 抗癌化合物库

7234 compounds
7234 种肿瘤相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L8100 细胞周期化合物库

677 compounds
677 种细胞周期相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L6600 胃肠炎天然产物库

219 compounds
219 种胃肠炎相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L4800 血管生成库

1353 compounds
1353 个高潜力的抑制或促进血管生成的小分子集合,可用于药物靶点开发、血管生成机理研究的高通量筛选,高内涵筛选;
L8200 抗衰老化合物库

3279 compounds
3279 个抗衰老化合物的独特集合,可用于高通量筛选和高内涵筛选;
L4000 经典已知活性库

14439 compounds
14439 个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
L5900 血脑屏障通透化合物库

509 compounds
509 个 CNS-Penetrant 生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L8110 细胞重编程化合物库

1813 compounds
1813 种重编程信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选
L2110 抗癌上市药物库

1779 compounds
1779 个具有抗癌活性小分子的独特集合,所有化合物都经过了严格的临床前研究和临床试验,由FDA、EMA 或NMPA 批准上市,可用于高通量、高内涵筛选。
L8110 细胞重编程化合物库

1813 compounds
1813 种重编程信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选
L9860 抗抑郁症化合物库

1163 compounds
1163 种与抑郁症相关的化合物,可以用于高通量和高内涵筛选
L3510 甲基化化合物库

128 compounds
128 种甲基化相关的化合物,可以用于高通量和高内涵筛选;
L6110 生物碱类天然产物库

500 compounds
500 种生物碱类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L7500 凝血与抗凝化合物库

144 compounds
144 个化合物的独特集合,可用于高通量筛选和高内涵筛选;
L4010 已知活性化合物库

22555 compounds
22555 个已知活性化合物的集合,可用于高通量筛选、高内涵筛选、细胞诱导和靶点确认;
L3300 组胺&褪黑色素化合物库

153 compounds
153 种生物活性小分子化合物,用于高通量、高内涵筛选;
L7400 钠通道分子库

118 compounds
118 种钠通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2500 人内源代谢化合物库

499 compounds
499 种内源性生物活性化合物的独特集合,用于高通量、高内涵筛选;
L7200 钙通道分子库

140 compounds
140 种钙通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7900 成骨分子库

317 compounds
317 种成骨相关的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L7700 神经再生化合物库

524 compounds
524 种神经再生相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L4700 免疫/炎症分子化合物库

4720 compounds
4720 种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选;
L4600 植物来源化合物库

3048 compounds
3048 个植物来源天然产物的独特集合,来自277类植物的精心之选;
L2510 脂代谢化合物库

492 compounds
492 个脂代谢相关的化合物集合,可用于高通量和高内涵筛选;
L5100 含氟化合物库

574 compounds
574 个含氟化合物的独特集合,可用于高通量筛选和高内涵筛选;
L2550 谷氨酰胺代谢化合物库

565 compounds
565 种谷氨酰胺代谢相关的分子,可以用于高通量和高内涵筛选;
L9500 表型筛选靶点鉴定库

1796 compounds
1796 种靶点明确的已知活性化合物,适合表型筛选;
L6820 烟草单体化合物库

747 compounds
747种烟草单体化合物的独特集合,可用于高通量筛选和高内涵筛选
L9700 内质网应激化合物库

193 compounds
193 个内质网应激相关的化合物集合,可用于高通量和高内涵筛选;
L6120 黄酮类天然产物库

514 compounds
514 种黄酮类天然产物的独特集合,可用于高通量筛选和高内涵筛选;
L9420 外泌体相关化合物库

76 compounds
76 种外泌体相关的化合物,可以用于高通量和高内涵筛选;
L7100 抗肥胖化合物库

2247 compounds
2247 个抗肥胖化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7600 趋化因子抑制剂库

59 compounds
59 种趋化因子或其受体抑制剂的独特集合,可用于高通量筛选和高内涵筛选;
L1710 抗COVID-19化合物库

1133 compounds
1133 种对SARS-CoV-2有抑制作用或潜在抑制作用的化合物集合,可用于高通量和高内涵筛选;
L2170 肿瘤免疫治疗小分子化合物库

449 compounds
449 种靶向肿瘤免疫治疗靶点的小分子,可用于高通量和高内涵筛选,是研究肿瘤免疫治疗的有力工具;
L6500 微生物天然产物库

685 compounds
685 种微生物来源的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;
L9300 大环化合物库

210 compounds
210 种活性已知的大环化合物,用于高通量、高内涵筛选;
DO1200 药物靶点库

53200 compounds
数量多,含53200种小分子化合物,是高通量筛选的有力工具;
L7110 抗高血压化合物库

678 compounds
678 种高血压相关的小分子,用于高通量和高内涵筛选;

化合物库

高溶解性片段库
Cat.No: L7800
Compounds: 2728
高溶解性微型片段化合物库
Cat.No: L7820
Compounds: 1081
高溶解性片段药效团化合物库
Cat.No: L7830
Compounds: 985
高溶解性卤化片段化合物库
Cat.No: L7840
Compounds: 796
高溶解性3D结构多样性片段化合物库
Cat.No: L7850
Compounds: 1079
高溶解性多官能团片段化合物库
Cat.No: L7810
Compounds: 1159
LC高溶解性片段化合物库
Cat.No: LF1030
Compounds: 9600
高选择性抑制剂库
Cat.No: L2010
Compounds: 575
稀有天然产物库
Cat.No: L6900
Compounds: 693
多样性核心预制库
Cat.No: LF1000
Compounds: 50000
环肽库
Cat.No: L9610
Compounds: 80
临床前化合物库
Cat.No: L3410
Compounds: 701
DNA 损伤和修复分子库
Cat.No: L3900
Compounds: 910
天然多酚类化合物库
Cat.No: L6100
Compounds: 635
抑制剂库
Cat.No: L2000
Compounds: 8328
苗药化合物库
Cat.No: L6230
Compounds: 534
天然产物库
Cat.No: L6010
Compounds: 3840
核受体化合物库
Cat.No: L1510
Compounds: 531
内分泌激素分子库
Cat.No: L2400
Compounds: 784
血液病分子库
Cat.No: L8400
Compounds: 514
表观遗传库
Cat.No: L1200
Compounds: 953
抗心血管疾病化合物库
Cat.No: L5400
Compounds: 1408
蒙药化合物库
Cat.No: L6220
Compounds: 950
细胞因子抑制剂库
Cat.No: L3600
Compounds: 604
抗癌临床化合物库
Cat.No: L2120
Compounds: 2545
活性脂质化合物库
Cat.No: L7000
Compounds: 385
药食同源库
Cat.No: L6300
Compounds: 1290
JAK-STAT 化合物库
Cat.No: L3700
Compounds: 252
药物功能重定位化合物库
Cat.No: L9200
Compounds: 4630
毒性化合物库
Cat.No: L5500
Compounds: 262
染色质修饰分子库
Cat.No: L8300
Compounds: 250
5-羟色胺分子库
Cat.No: L2800
Compounds: 268
TGF-β/Smad靶点化合物库
Cat.No: L4100
Compounds: 184
口服活性化合物库
Cat.No: L9850
Compounds: 2427
抗氧化化合物库
Cat.No: L2910
Compounds: 1314
抗感染天然产物库
Cat.No: L6610
Compounds: 1060
干细胞分化化合物库
Cat.No: L8000
Compounds: 1197
上市药物库
Cat.No: L1000
Compounds: 2808
神经信号分子库
Cat.No: L2600
Compounds: 2540
靶向治疗药物库
Cat.No: L2152
Compounds: 119
癌细胞分化化合物库
Cat.No: L2140
Compounds: 406
抗癌细胞代谢库
Cat.No: L2130
Compounds: 1268
FDA上市及药典收录分子库
Cat.No: L1010
Compounds: 3158
农药化合物库
Cat.No: L9240
Compounds: 270
DNA损伤/修复库Plus
Cat.No: L3980
Compounds: 667
激酶抑制剂库
Cat.No: L1600
Compounds: 2720
共价抑制剂库
Cat.No: L9410
Compounds: 1920
离子通道库
Cat.No: L2300
Compounds: 931
Wnt/Hedgehog/Notch 通路化合物库
Cat.No: L4300
Compounds: 237
FDA 上市激酶抑制剂库
Cat.No: L1610
Compounds: 263
泛素化化合物库
Cat.No: L8600
Compounds: 210
GPCR靶点分子库
Cat.No: L1500
Compounds: 1940
NF-κB 通路分子库
Cat.No: L3800
Compounds: 729
藏药化合物库
Cat.No: L6210
Compounds: 747
抗前列腺癌化合物库
Cat.No: L2195
Compounds: 2070
氧化还原化合物库
Cat.No: L2900
Compounds: 1264
FDA 上市药物库
Cat.No: L4200
Compounds: 1729
可溶性羧酸片段化合物库
Cat.No: L7870
Compounds: 1806
抗代谢疾病化合物库
Cat.No: L5200
Compounds: 1544
PI3K/Akt/mTOR 化合物库
Cat.No: L1300
Compounds: 420
瑶药化合物库
Cat.No: L6200
Compounds: 221
抗癌天然产物库
Cat.No: L6700
Compounds: 1772
抗乳腺癌化合物库
Cat.No: L2191
Compounds: 1939
抗感染化合物库
Cat.No: L1800
Compounds: 2938
临床期小分子药物库
Cat.No: L3400
Compounds: 3404
抗寄生虫库
Cat.No: L4510
Compounds: 419
造血毒性小分子库
Cat.No: L3100
Compounds: 101
糖酵解化合物库
Cat.No: L2521
Compounds: 555
人代谢物化合物库
Cat.No: L2570
Compounds: 4454
抗病毒库
Cat.No: L1700
Compounds: 1040
化疗药物库
Cat.No: L2151
Compounds: 48
药物代谢杂质库
Cat.No: L5800
Compounds: 197
ReFRAME 相关化合物库
Cat.No: L9230
Compounds: 3210
儿童药物库
Cat.No: L9210
Compounds: 972
钾通道分子库
Cat.No: L7300
Compounds: 152
非甾体类抗炎化合物库
Cat.No: L4710
Compounds: 530
Mini真菌代谢天然产物筛选库
Cat.No: L6001
Compounds: Inquiry
NO PAINS 化合物库
Cat.No: L4020
Compounds: 9384
天然产物衍生物虚筛化合物库
Cat.No: L6030
Compounds: 163000
抗结直肠癌化合物库
Cat.No: L2194
Compounds: 1545
组蛋白修饰化合物库
Cat.No: L3500
Compounds: 469
自噬库
Cat.No: L3200
Compounds: 1248
酪氨酸激酶分子库
Cat.No: L2200
Compounds: 1016
海洋天然产物库
Cat.No: L6400
Compounds: 144
抗癌药物库
Cat.No: L2150
Compounds: 3080
细胞焦亡化合物库
Cat.No: L8720
Compounds: 1066
代谢化合物库
Cat.No: L2560
Compounds: 2320
抗癌活性化合物库
Cat.No: L2160
Compounds: 3188
萜类天然产物库
Cat.No: L6130
Compounds: 622
抗寄生虫天然产物库
Cat.No: L6620
Compounds: 253
高通量筛选天然产物库
Cat.No: L6000
Compounds: 4533
抗癌化合物库
Cat.No: L2100
Compounds: 7234
细胞周期化合物库
Cat.No: L8100
Compounds: 677
胃肠炎天然产物库
Cat.No: L6600
Compounds: 219
血管生成库
Cat.No: L4800
Compounds: 1353
抗衰老化合物库
Cat.No: L8200
Compounds: 3279
经典已知活性库
Cat.No: L4000
Compounds: 14439
血脑屏障通透化合物库
Cat.No: L5900
Compounds: 509
细胞重编程化合物库
Cat.No: L8110
Compounds: 1813
抗癌上市药物库
Cat.No: L2110
Compounds: 1779
细胞重编程化合物库
Cat.No: L8110
Compounds: 1813
抗抑郁症化合物库
Cat.No: L9860
Compounds: 1163
甲基化化合物库
Cat.No: L3510
Compounds: 128
生物碱类天然产物库
Cat.No: L6110
Compounds: 500
凝血与抗凝化合物库
Cat.No: L7500
Compounds: 144
已知活性化合物库
Cat.No: L4010
Compounds: 22555
组胺&褪黑色素化合物库
Cat.No: L3300
Compounds: 153
钠通道分子库
Cat.No: L7400
Compounds: 118
人内源代谢化合物库
Cat.No: L2500
Compounds: 499
钙通道分子库
Cat.No: L7200
Compounds: 140
成骨分子库
Cat.No: L7900
Compounds: 317
神经再生化合物库
Cat.No: L7700
Compounds: 524
免疫/炎症分子化合物库
Cat.No: L4700
Compounds: 4720
植物来源化合物库
Cat.No: L4600
Compounds: 3048
脂代谢化合物库
Cat.No: L2510
Compounds: 492
含氟化合物库
Cat.No: L5100
Compounds: 574
谷氨酰胺代谢化合物库
Cat.No: L2550
Compounds: 565
表型筛选靶点鉴定库
Cat.No: L9500
Compounds: 1796
烟草单体化合物库
Cat.No: L6820
Compounds: 747
内质网应激化合物库
Cat.No: L9700
Compounds: 193
黄酮类天然产物库
Cat.No: L6120
Compounds: 514
外泌体相关化合物库
Cat.No: L9420
Compounds: 76
抗肥胖化合物库
Cat.No: L7100
Compounds: 2247
趋化因子抑制剂库
Cat.No: L7600
Compounds: 59
抗COVID-19化合物库
Cat.No: L1710
Compounds: 1133
肿瘤免疫治疗小分子化合物库
Cat.No: L2170
Compounds: 449
微生物天然产物库
Cat.No: L6500
Compounds: 685
大环化合物库
Cat.No: L9300
Compounds: 210
药物靶点库
Cat.No: DO1200
Compounds: 53200
抗高血压化合物库
Cat.No: L7110
Compounds: 678
Cat. No. Product Name Form Specificity Of Inhibition
C0007 SYBR Green qPCR Master Mix (High ROX)

SYBR Green qPCR Master Mix (High ROX)

Solution in bottle
C0074 Mag Beads COOH High capacity (2.8 μm)

羧基磁珠 (2.8 μm)

Suspension in bottle 蛋白纯化、免疫检测、细胞分选、特异性核酸分离、生物传感器、药物筛选和输送
C0090 Mag Beads Streptavidin (1 μm)

链霉亲和素磁珠 (1 μm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0104B Protein A/G Immunomagnetic Beads

Protein A/G 免疫沉淀磁珠

Suspension in bottle IP, Co-IP, ChIP
C0109 Magrose Beads IDA-Nickel

His-tag 蛋白纯化磁珠 IDA-Ni

Suspension in bottle 蛋白纯化
C0089 Mag Beads Streptavidin (300 nm)

链霉亲和素磁珠 (300 nm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0093 Mag Beads Streptavidin (3 μm)

链霉亲和素磁珠 (3 μm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0094 Mag Beads Streptavidin (5 μm)

链霉亲和素磁珠 (5 μm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0092 Mag Beads Streptavidin (2.8 μm)

链霉亲和素磁珠 (2.8 μm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0091 Mag Beads Streptavidin (2 μm)

链霉亲和素磁珠 (2 μm)

Suspension in bottle 免疫检测、分离蛋白;分离核酸、制备核酸探针;DNA-蛋白质相互作用研究;细胞分选与激活
C0105 Protein A Immunoprecipitation Kit

Protein A 免疫沉淀试剂盒

Suspension in bottle IP, Co-IP, ChIP
C0104 Protein A/G Immunoprecipitation Kit

Protein A/G 免疫沉淀试剂盒

Suspension in bottle IP, Co-IP, ChIP
C0110 Magrose Beads IDA-Cobalt

His-tag 蛋白纯化磁珠 IDA-Co

Suspension in bottle 蛋白纯化
C0111 Magrose Beads NTA-Nickel (Ultra-suspension)

His-tag 蛋白纯化磁珠 NTA-Ni

Suspension in bottle 蛋白纯化

TargetMol 试剂盒

SYBR Green qPCR Master Mix (High ROX)
Cat.No: C0007
羧基磁珠 (2.8 μm)
Cat.No: C0074
链霉亲和素磁珠 (1 μm)
Cat.No: C0090
Protein A/G 免疫沉淀磁珠
Cat.No: C0104B
His-tag 蛋白纯化磁珠 IDA-Ni
Cat.No: C0109
链霉亲和素磁珠 (300 nm)
Cat.No: C0089
链霉亲和素磁珠 (3 μm)
Cat.No: C0093
链霉亲和素磁珠 (5 μm)
Cat.No: C0094
链霉亲和素磁珠 (2.8 μm)
Cat.No: C0092
链霉亲和素磁珠 (2 μm)
Cat.No: C0091
Protein A 免疫沉淀试剂盒
Cat.No: C0105
Protein A/G 免疫沉淀试剂盒
Cat.No: C0104
His-tag 蛋白纯化磁珠 IDA-Co
Cat.No: C0110
His-tag 蛋白纯化磁珠 NTA-Ni
Cat.No: C0111
Cat. No. Product Name Target Signaling Pathways
T5471 GUANABENZ

Adrenergic Receptor GPCR/G Protein; Neuroscience
GUANABENZ 是一种中枢 alpha-2 肾上腺素能激动剂。它的作用机制是作为肾上腺素能 α2-激动剂。
T2086 ELN-441958

ELN 441958

Bradykinin Receptor GPCR/G Protein
ELN-441958是一种B1受体拮抗剂,能够抑制B1激动剂配体[3H] DAKD 与IMR-90细胞结合(Ki:0.26 nM),相较于B2受体,它对B1受体的抑制作用具有更高的选择性,且比抑制μ阿片受体选择性高500多倍,比抑制δ阿片受体选择性高2000多倍。
T6054 GSK256066

PDE Metabolism
GSK256066 是高亲和力的、选择性的PDE4抑制剂,IC50=3.2 pM,被开发用于慢性阻塞性肺病的研究。
T13884 Shield-1

Others Others
Shield-1 是 FK506 结合蛋白 12 (FKBP) 的特异性、高亲和力和细胞渗透性配体,通过与突变的 FKBP (mtFKBP) 结合来逆转不稳定性,允许 mtFKBP 融合蛋白的条件表达。它可以稳定整个融合蛋白。
T11344 G150

DNA; cGAS DNA Damage/DNA Repair; Immunology/Inflammation
G150 是高选择性h-cGAS 抑制剂,IC50值为 10.2 nM,用于抑制 dsDNA 引发的干扰素表达。
T21957 Guanabenz hydrochloride

NE56490

Adrenergic Receptor GPCR/G Protein; Neuroscience
Guanabenz hydrochloride (NE56490) 是一种具有降血压作用的口服活性 α2-肾上腺素受体激动剂。
T7686 Ramiprilat

RAAS Endocrinology/Hormones
Ramiprilat 是 Ramipril 的活性代谢物,是一种口服有活力的血管紧张素转换酶 (ACE) 抑制剂,其 Ki=7 pM。它可用于研究心力衰竭以及高血压。
T33639 Neotame

NC 00723,HSDB 7965,NC-00723,NC00723,纽甜

Others Others
Neotame (HSDB 7965) 是阿斯巴甜的衍生物,是低热量、高效的人造甜味剂,非营养性甜味剂和增味剂,其甜度是糖的 7000-13,000 倍,可用于多种食品。
T6581 Methyclothiazide

Duretic,Enduron,甲氯噻嗪,Aquatensen

Others; Carbonic Anhydrase Metabolism; Others
Methyclothiazide (Aquatensen) 是一种具有口服活性的利尿剂,也是一种降压剂。它能够拮抗体外的电压依赖性钙通道的 (VDCC) 活性,也可以抑制内源性血管收缩刺激导致的血管反应。
T4524 SBC-110736

SBC110736

Others; Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism; Others
SBC-110736 是一种蛋白转化酶枯草杆菌蛋白酶 9 型 (PCSK9) 抑制剂。
T3283 Cetilistat

新利司他,ATL-962

Lipid Metabolism
Cetilistat (ATL-962) 是胰腺脂肪酶 (pancreatic lipase) 抑制剂,能够抑制大鼠脂肪酶(IC50:54.8 nM)和人胰脂肪酶(IC50:5.95 nM)的活性,可用作有效的抗肥胖药。
T14667 BLT-1

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
BLT-1 是一种氨基硫脲铜螯合剂,是一种选择性清除受体 B1 型 (SR-BI) 抑制剂,抑制高密度脂蛋白 (HDL) 和 SR-BI 介导的细胞之间的脂质转移。
T2499 Torcetrapib

CP-529414,托彻普

CETP Metabolism
是胆固醇酯转移蛋白 (CETP) 选择性抑制剂。根据人血浆的抑制曲线,Torcetrapib (CP-529414) 对CETP 的最有效浓度为 37 nM。
T0197 Terazosin hydrochloride

盐酸特拉唑嗪,Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic

Adrenergic Receptor GPCR/G Protein; Neuroscience
Terazosin hydrochloride (Hytrin) 是一种竞争性和口服活性的 α1-肾上腺素受体拮抗剂,是一种喹唑啉衍生物。它通过舒张血管和打开膀胱来起作用。它可用于良性前列腺增生和高血压的研究。
T1050 Prazosin hydrochloride

Prazosin hydrochloride,哌唑嗪盐酸盐,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,盐酸哌唑嗪,Minipress

Potassium Channel; MRP; Adrenergic Receptor; ABC; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Prazosin hydrochloride (Vasoflex) 是一种选择性肾上腺素能 α-1 拮抗剂,可降低外周阻力并放松血管平滑肌。 它可用于研究高血压和酒精使用障碍。 它是一种合成哌嗪衍生物,具有降压抗肾上腺素能特性。它抑制有机阳离子转运蛋白 OCT-1 和 OCT-3,IC50分别为 1.8 和 13 μM 。
T20656 Verapamil

NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil (CP-16533-1) 是一种非二氢吡啶类钙通道阻滞剂,一种 P-gp 抑制剂,也是一种 CYP3A4 抑制剂,具有口服活性。Verapamil 可以用于治疗高血压、心绞痛、心肌梗塞等。
T1010 Verapamil hydrochloride

Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil hydrochloride (Verapamil HCl) 是一种钙通道阻滞剂,是一种可口服的 P 糖蛋白 (P-gp) 抑制剂,可抑制CYP3A4,用于高血压、心律不齐和心绞痛的研究。
T6701 Terazosin hydrochloride dihydrate

Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate,盐酸特拉唑嗪(二水合物)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Terazosin hydrochloride dihydrate (Heitrin dihydrate) 是一种竞争性和口服活性的 α1-肾上腺素受体(α1-adrenoceptor) 拮抗剂,是一种喹唑啉衍生物,通过舒张血管和打开膀胱的方式起作用。它可用于研究良性前列腺增生 (BPH) 和高血压。
T1203 Nadolol

Anabet,Corgard,Solgol,苯甲丁氮酮,纳多洛尔,SQ11725

Adrenergic Receptor GPCR/G Protein; Neuroscience
Nadolol 是一种有机阴离子转运多肽 1A2 (OATP1A2) 的底物,是一种非选择性的、具有口服活性的 β-肾上腺素受体 (β-adrenergic receptors) 阻滞剂,可用于高血压,心绞痛和血管性头痛的研究。
T10477 BAY-985

IκB/IKK NF-κB
BAY-985 是高效的、ATP 竞争性的、有口服活性的、选择性的TBK1和IKKε双重抑制剂,对 TBK1 (在低/高 ATP 实验中) 和 IKKε 的IC50分别为 2/30 和 2 nM。它具有抗肿瘤作用。
T12140 N-Acetyl-Calicheamicin

N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin

Antibacterial; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Microbiology/Virology
N-Acetyl-Calicheamicin (N-Acetyl-γ-calicheamicin)是一种具有很高抗肿瘤活性的的抗生素。
T34383L 2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv

Others Others
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv在Sprague Dawley大鼠上进行测试时显示出高局部抗炎效力和高肺选择性。
T2229 Tetraethylenepentamine Pentahydrochloride

Others Others
Tetraethylenepentamine Pentahydrochloride 是一种高亲和力的铜和锌螯合剂。
T20761 RU 59063

RU-59063,RU59063

Androgen Receptor Endocrinology/Hormones
RU 59063 是一类新型高亲和力非甾体雄激素受体 (AR) 配体的原型。
T11864 Iptacopan

LNP023

Others Others
Iptacopan (LNP023) 是一种与factor B 亲和力较高的抑制剂。
T34994 Uk-390957

Uk390957,Uk 390957

Others Others
Uk-390957 是一种磺酰胺化合物,由于与碳酸酐酶结合而具有高BPR。
T9058 Bisphenoxyethanolfluorene

Others Others
Bisphenoxyethanolfluorene 是一种高稳定性的新型有机化工原料,主要用于合成耐热、透明性和高折射率的高分子单体。
T15581 Inolitazone

RS5444,Efatutazone,CS-7017,伊诺他酮

PPAR DNA Damage/DNA Repair; Metabolism
Inolitazone (RS5444) 是一种高亲和力PPARγ激动剂。在体外,Inotazone 显示生长抑制的IC50约为0.8 nM。
T31362 Deferitazole

SPD602,FBS 0701,SPD-602,FBS0701,FBS-0701,SPD 602

Others Others
Deferitazole (FBS 0701) 是一种新型且具有口服活性、选择性和高亲和力的铁螯合剂。
T34383 Rofleponide

Glucocorticoid Receptor Endocrinology/Hormones
Rofleponide 是一种人工合成的糖皮质激素,与大鼠胸腺糖皮质激素受体有很高的亲和力。
T26085 Rilapine

Rilapinum

5-HT Receptor GPCR/G Protein; Neuroscience
Rilapine (Rilapinum) 是一种抗精神病化合物,对 5-HT6 受体显示出较高亲和力,可以用于研究神经系统疾病。
TP1044L Pancreatic Polypeptide, rat acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Pancreatic Polypeptide, rat acetate 是 NPY 受体的激动剂,对 NPYR4 具有高亲和力。
T9501 Enterobactin

Enterochelin

Others Others
Enterobactin (Enterochelin) 是一种高亲和力铁载体,可为微生物系统获取铁。
T9989 AChE-IN-27

Others Others
AChE-IN-27是一种用于高通量测定的小分子。
T11349 GABAA receptor agent 1

GABA Receptor Membrane transporter/Ion channel; Neuroscience
GABAA receptor agent 1 是GABAA 受体的高亲和力配体,有抗惊厥活性。
T15364 G-1

Estrogen Receptor/ERR; GPR Endocrinology/Hormones; GPCR/G Protein
G-1 是一种高亲和力的、非甾体的、有选择性的 GPR30激动剂(Ki:11 nM)。
T7021 ZM241385

Adenosine Receptor GPCR/G Protein; Neuroscience
ZM241385 是一种高亲和力的,选择性的腺苷A2AR 拮抗剂,Ki 值为 1.4 nM。
T7716 TNCA

(S)-2,3,4,9-四氢-1H-吡啶[3,4-B]吲哚-3-羧酸,Lycoperodine-1

Others Others
TNCA (Lycoperodine-1) 是一种具有共激动剂活性的高亲和力 CaSR 配体 (CaSRL)。
T6333 MM-102

MM102,HMTase Inhibitor IX

Histone Methyltransferase Chromatin/Epigenetic
MM-102 (HMTase Inhibitor IX) 是一种有效的 WDR5/MLL 相互作用抑制剂,在 WDR5 结合检测中,IC50为 2.4 nM,Ki 小于 1 nM。
T9995 Antituberculosis agent-5

Others Others
Antituberculosis agent-5是一种用于高通量测定的小分子。
T3497 Ocaperidone

奥卡哌酮,Ocaperidona,R79598

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Ocaperidone (Ocaperidona) 是5-HT2和多巴胺D2的拮抗剂,也是5-HT1A 的激动剂,有安定作用。
T9994 WAY-620521

Others Others
WAY-620521是一种用于细胞的高通量测定小分子。
T23312 SB 204741

5-HT Receptor GPCR/G Protein; Neuroscience
SB 204741 是一种选择性的5-HT2B 拮抗剂,具有高亲和性,pKi 值为7.1。
T0107 Halcinonide

Halcimat,Halciderm,哈西奈德,Halcinonida,氯氟舒松,SQ-18566

Glucocorticoid Receptor; Smo Endocrinology/Hormones; Stem Cells
Halcinonide (Halciderm) 是一种糖皮质激素,可用于局部皮肤感染的研究。
T4531 GSK2200150A

Antibacterial Microbiology/Virology
GSK2200150A 是一种通过高通量筛选活动确定的抗结核剂,对 H37Rv 的 MIC 是 0.38 μM。
T21246 Metsulfuron-methyl

Others Others
Metsulfuron-methyl 是一种内吸传导选择性麦田高效磺酰脲类除草剂,主要防治麦田大多数阔叶杂草和禾本科杂草。
T39573 GSK251

PI3K PI3K/Akt/mTOR signaling
GSK251是一种新型的,口服生物利用度高的PI3Kδ抑制剂,具有高效性和高选择性,且具有独特的结合模式。
T9755 MRTX0902

UNII-CRG69FR93G

Raf MAPK
MRTX0902 是一种有效且高选择性的 SOS1 抑制剂,IC50 为 46 nM,Ki 为 2 nM。
T68134 Ro-3201195

p38 MAPK MAPK
Ro-3201195是一种新型可口服的p38 MAPK 抑制剂,具有很高的选择性。
TP1957L PKI (5-24) Acetate(99534-03-9 free base)

PKA Tyrosine Kinase/Adaptors
PKI (5-24) Acetate(99534-03-9 free base) 是一种高亲和力 PKA 抑制剂 (Ki = 2.3 nM)。

化合物

GUANABENZ
Cat.No: T5471
Synonym:
Target: Adrenergic Receptor
ELN-441958
Cat.No: T2086
Synonym: ELN 441958
Target: Bradykinin Receptor
GSK256066
Cat.No: T6054
Synonym:
Target: PDE
Shield-1
Cat.No: T13884
Synonym:
Target: Others
G150
Cat.No: T11344
Synonym:
Target: DNA, cGAS
Guanabenz hydrochloride
Cat.No: T21957
Synonym: NE56490
Target: Adrenergic Receptor
Ramiprilat
Cat.No: T7686
Synonym:
Target: RAAS
Neotame
Cat.No: T33639
Synonym: NC 00723,HSDB 7965,NC-00723,NC00723,纽甜
Target: Others
Methyclothiazide
Cat.No: T6581
Synonym: Duretic,Enduron,甲氯噻嗪,Aquatensen
Target: Others, Carbonic Anhydrase
SBC-110736
Cat.No: T4524
Synonym: SBC110736
Target: Others, Serine/threonin kinase
Cetilistat
Cat.No: T3283
Synonym: 新利司他,ATL-962
Target: Lipid
BLT-1
Cat.No: T14667
Synonym:
Target: Others, HCV Protease
Torcetrapib
Cat.No: T2499
Synonym: CP-529414,托彻普
Target: CETP
Terazosin hydrochloride
Cat.No: T0197
Synonym: 盐酸特拉唑嗪,Terazosin HCl,Terazosine,Blavin,Hytrin,Zayasel,Fosfomic
Target: Adrenergic Receptor
Prazosin hydrochloride
Cat.No: T1050
Synonym: Prazosin hydrochloride,哌唑嗪盐酸盐,Prazosin HCl,cp-12299-1,Peripress,Vasoflex,盐酸哌唑嗪,Minipress
Target: Potassium Channel, MRP, Adrenergic Receptor, ABC, Autophagy
Verapamil
Cat.No: T20656
Synonym: NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil
Target: P450, Calcium Channel, P-gp
Verapamil hydrochloride
Cat.No: T1010
Synonym: Manidon,盐酸维拉帕米,(±)-Verapamil hydrochlorid,Verapamil HCl,Calcan hydrochloride
Target: P450, Calcium Channel, P-gp
Terazosin hydrochloride dihydrate
Cat.No: T6701
Synonym: Flotrin dihydrate,Terazosin HCl Dihydrate,Dysalfa dihydrate,Heitrin dihydrate,盐酸特拉唑嗪(二水合物)
Target: Adrenergic Receptor
Nadolol
Cat.No: T1203
Synonym: Anabet,Corgard,Solgol,苯甲丁氮酮,纳多洛尔,SQ11725
Target: Adrenergic Receptor
BAY-985
Cat.No: T10477
Synonym:
Target: IκB/IKK
N-Acetyl-Calicheamicin
Cat.No: T12140
Synonym: N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin
Target: Antibacterial, ADC Cytotoxin
2H-Naphth[2′,1′:4,5]indeno[1,2-d][1,3]dioxole, pregn-4-ene-3,20-dione deriv
Cat.No: T34383L
Synonym:
Target: Others
Tetraethylenepentamine Pentahydrochloride
Cat.No: T2229
Synonym:
Target: Others
RU 59063
Cat.No: T20761
Synonym: RU-59063,RU59063
Target: Androgen Receptor
Iptacopan
Cat.No: T11864
Synonym: LNP023
Target: Others
Uk-390957
Cat.No: T34994
Synonym: Uk390957,Uk 390957
Target: Others
Bisphenoxyethanolfluorene
Cat.No: T9058
Synonym:
Target: Others
Inolitazone
Cat.No: T15581
Synonym: RS5444,Efatutazone,CS-7017,伊诺他酮
Target: PPAR
Deferitazole
Cat.No: T31362
Synonym: SPD602,FBS 0701,SPD-602,FBS0701,FBS-0701,SPD 602
Target: Others
Rofleponide
Cat.No: T34383
Synonym:
Target: Glucocorticoid Receptor
Rilapine
Cat.No: T26085
Synonym: Rilapinum
Target: 5-HT Receptor
Pancreatic Polypeptide, rat acetate
Cat.No: TP1044L
Synonym:
Target: Neuropeptide Y Receptor
Enterobactin
Cat.No: T9501
Synonym: Enterochelin
Target: Others
AChE-IN-27
Cat.No: T9989
Synonym:
Target: Others
GABAA receptor agent 1
Cat.No: T11349
Synonym:
Target: GABA Receptor
G-1
Cat.No: T15364
Synonym:
Target: Estrogen Receptor/ERR, GPR
ZM241385
Cat.No: T7021
Synonym:
Target: Adenosine Receptor
TNCA
Cat.No: T7716
Synonym: (S)-2,3,4,9-四氢-1H-吡啶[3,4-B]吲哚-3-羧酸,Lycoperodine-1
Target: Others
MM-102
Cat.No: T6333
Synonym: MM102,HMTase Inhibitor IX
Target: Histone Methyltransferase
Antituberculosis agent-5
Cat.No: T9995
Synonym:
Target: Others
Ocaperidone
Cat.No: T3497
Synonym: 奥卡哌酮,Ocaperidona,R79598
Target: Dopamine Receptor, 5-HT Receptor
WAY-620521
Cat.No: T9994
Synonym:
Target: Others
SB 204741
Cat.No: T23312
Synonym:
Target: 5-HT Receptor
Halcinonide
Cat.No: T0107
Synonym: Halcimat,Halciderm,哈西奈德,Halcinonida,氯氟舒松,SQ-18566
Target: Glucocorticoid Receptor, Smo
GSK2200150A
Cat.No: T4531
Synonym:
Target: Antibacterial
Metsulfuron-methyl
Cat.No: T21246
Synonym:
Target: Others
GSK251
Cat.No: T39573
Synonym:
Target: PI3K
MRTX0902
Cat.No: T9755
Synonym: UNII-CRG69FR93G
Target: Raf
Ro-3201195
Cat.No: T68134
Synonym:
Target: p38 MAPK
PKI (5-24) Acetate(99534-03-9 free base)
Cat.No: TP1957L
Synonym:
Target: PKA
Cat. No. Product Name Target Signaling Pathways
T8465 28-high brassinolide

Others Others
28-high brassinolide 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T8465,CAS号为 82373-95-3。
T3804 Neomangiferin

Mangiferin 7-glucoside,新芒果苷

Phosphatase Metabolism
Neomangiferin (Mangiferin 7-glucoside) 是一种天然的 C-glucosyl xanthone,分离自干燥的Anemarrhena asphodeloides 的根茎中。它能够减轻大鼠高脂饮食诱导的非酒精性脂肪性肝病 (NAFLD)。
TN1624 Ethyl cinnamate

Calcium Channel; ROS; NO Synthase Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Ethyl cinnamate 是食品香料和化妆品添加剂,也是哺乳动物组织的优良清除剂。
TN1117 Veraguensin

p38 MAPK; NF-κB; Antibiotic; Parasite; Antifection MAPK; Microbiology/Virology; NF-κB
Veraguensin 来源于 Magnolia sp.。 Veraguensin 抑制骨吸收并显示出高抗寄生虫活性。
T14961 Chrysene

䓛,屈

Others Others
Chrysene 是高分子量 (HMW) 多环芳烃,有极强的顽固性和致癌性。
T12296 Oleoylethanolamide

油酰单乙醇胺,N-Oleoylethanolamide,Oleamide MEA,Oleic acid monoethanolamide

Endogenous Metabolite; PPAR DNA Damage/DNA Repair; Metabolism
Oleoylethanolamide (N-Oleoylethanolamide) 是一种PPAR-α 的高亲和力内源性激动剂,可用于肥胖和动脉硬化的相关研究。
T4S1951 10-Methoxycamptothecin

Others; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Others
10-Methoxycamptothecin 是分离自喜树的喜树碱衍生物,具有高抗癌特性。通过对 2774 细胞系的抗肿瘤活性测定,发现它比 10-羟基喜树碱的细胞毒性更高。
TMA2386 4,4'-Methylenediphenol

Others Others
4,4'-Methylenediphenol 首次从 Galeola Faberi 的根茎中分离出来,具有抗氧化活性。
T0532 5,6-Dihydro-5-methyluracil

5, 6-Dihydrothymine,二氢朐腺嘧啶,Dihydrothymine

Nucleoside Antimetabolite/Analog; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Dihydrothymine 是胸腺嘧啶的中间代谢产物之一,来源于动植物,浓度过高时会产生毒性。
TQ0027 Transcrocetinate disodium

Disodium trans-crocetinate,藏红花,藏红花酸二钠盐

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Transcrocetinate disodium (Disodium trans-crocetinate) 从藏红花中提取的一种天然产物,是高亲和力NMDA 受体拮抗剂。
T22300 Creatine monohydrate

Methylguanidoacetic acid monohydrate,一水肌酸

Others; Endogenous Metabolite Metabolism; Others
Creatine monohydrate (Methylguanidoacetic acid monohydrate) 是磷酸原能量系统的关键参与者,尤其是在肌肉和大脑中。 Creatine monohydrate 是高强度、短期活动中 ATP 的主要来源。
TMA1570 Sappanone A

NF-κB; Nrf2 Immunology/Inflammation; NF-κB
Sappanone A 是一种高异黄烷酮,通过调节 Nrf2 和 NF-κB 表现出抗炎作用。Sappanone A 可以减轻卵清蛋白引起的哮喘中的过敏性气道炎症。
T0344L Miconazole nitrate

NSC 169434 Nitrate,硝酸咪康唑,R18134 nitrate

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Miconazole nitrate (R18134 nitrate) 是咪唑类可抗菌的抗真菌剂。
T19608 Zinc sulfate heptahydrate

Others Others
Zinc sulfate heptahydrate 是七水合形式的硫酸锌,是一种膳食补充剂,可用于锌缺乏症和预防高危人群的锌缺乏症。
T1424 Ethynyl estradiol

乙炔基雌二醇,17α-Ethynylestradiol,Ethinyl Estradiol,炔雌醇

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Ethynyl estradio 是一种高效的生物活性雌激素。
TP1232L Amylin, amide, rat acetate(124447-81-0,free base)

Amylin Receptor GPCR/G Protein
Amylin, amide, rat acetate(124447-81-0,free base) 是 AMY1 和 AMY3 受体以及 AMY2 受体的强效和高亲和力配体。
TN1048 Cnidilin

Knidilin

Cnidilin (Knidilin) 存在与Angelica dahurica 根中,具有高BBB 通透性,在治疗中枢神经系统疾病方面具有药代动力学潜力。
T3878 Raddeanin A

NSC382873,竹节香附素A,Anemodeanin A,Raddeanin R3

Apoptosis; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Raddeanin A (NSC-382873) 是竹节香附中的一种天然三萜皂苷,可抑制组蛋白去乙酰化酶,具有很强的抗血管生成能力和抗肿瘤活性。
T19344 Glycogen, Mussel

α-1,6 葡聚糖,Glycogen

Endogenous Metabolite Metabolism
Glycogen, Mussel 是一种糖酵解的中间产物和高能磷酸盐,它是人类、动物、真菌和细菌的一种能量储存形式。
T2975 2,3-Dimethoxybenzaldehyde

5,6-Dimethoxybenzaldehyde,邻藜芦醛,o-Veratraldehyde

Antifungal Microbiology/Virology
2,3-Dimethoxybenzaldehyde (5,6-Dimethoxybenzaldehyde) 是苯甲酸类似物,具有高抗真菌活性(MIC=2.5 mM)。2,3-Dimethoxybenzaldehyde 可用于合成小檗碱。
T39887 (S)-3-(4-Hydroxyphenyl)lactic acid

(S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid

Others; Antioxidant Others; oxidation-reduction
(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid 是分离自间肠隐球菌培养基的代谢物,具有高的 DPPH 清除自由基活性和抗氧化活性。
TN1049 Ingenol-5,20-acetonide

Others Others
Ingenol-5,20-acetonide 是一种天然化合物,Ingenol 3-Angelate的类似物,当局部用于治疗光化性角化病时具有抗肿瘤活性。
TN7241 Annatto

T4831 α,α-Dimethylglycine

2-Aminoisobutyric acid,α-Aminoisobutanoic acid,2-甲基丙氨酸

Others; Endogenous Metabolite Metabolism; Others
NSC-16590 (2-Aminoisobutyric acid) 对苍耳子叶中内源性乙烯(ethylene)的产生具有抑制作用。
TN1012 Febrifugine

IL Receptor; Anti-infection; Parasite Immunology/Inflammation; Microbiology/Virology
Febrifugine 是存在于常山的根和叶中的一种喹唑啉酮类生物碱,有抗疟活性。它是一种有效的抗球虫药,具有杀灭裂殖体的作用。
TN1860 Licoflavone B

甘草黄酮 B,甘草黄酮B

ATPase; Anti-infection; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Licoflavone B 是从甘草中得到的一种类黄酮,抑制曼氏血吸虫 ATPase 和 ADPase 的活性,IC50值分别为 23.78 µM 和 31.50 µM。
T3S0872 Paederoside

Antiviral; HBV Immunology/Inflammation; Microbiology/Virology
Paederoside 是从Paederia pertomentosa 分离的一种单萜 S-甲基硫代碳酸酯。它抑制 Epstein-Barr 病毒的激活,有抗肿瘤促进作用。
T3262 Phosphocreatine disodium

Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium (Phosphocreatine disodium salt) 是一种磷酸化的肌酸分子,在肌肉、骨骼和大脑中作为一种可快速动员的高能磷酸盐储备。
T19924 Rhododendrol

Betuligenol,Frambinol,杜鹃醇

Others Others
Rhododendrol (Frambinol) 是一种黑色素合成物,防止雄性小鼠高脂饮食引起的体重升高和增加雄性小鼠白色脂肪细胞的脂肪分解。Rhododendrol 可用作美白/美白化妆品抑制剂。
T3976 Cytosporone B

Csn-B,Dothiorelone G

Others Others
Cytosporone B (Dothiorelone G) 是一种天然存在的核孤儿受体Nur77/NR4A1激动剂(EC50=0.278 nM)。
T3S1692 Octahydrocurcumin

Anti-infection; NF-κB; Reactive Oxygen Species; ROS Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Octahydrocurcumin 是一种姜黄素的氢化衍生物,是姜黄素的代谢物。
TN3831 (-)-Denudatin B

Denudatin B

ATPase; Potassium Channel; Calcium Channel; PAFR GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
(-)-Denudatin B (Denudatin B) 源自 Magnolia fargesii。 (-)-Denudatin B 通过抑制胶原蛋白和凝血酶诱导的磷酸肌醇分解,在高浓度下具有非特异性抗血小板作用。
T3313 D-Luciferin

Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin

Others Others
D-Luciferin (D-(-)-Luciferin) 是一种萤光素酶的底物,能够催化生物发光昆虫产生典型的黄绿光。
T21205 Ponasterone A

坡那甾酮A,AI3-44686

Others Others
Ponasterone A 是一种蜕皮激素,能够高度亲和蜕皮激素受体。它能够使报告基因能够快速打开和关闭,是细胞和转基因动物中基因表达的有效调节剂。
T5545 Maltol

Veltol,Larixinic acid,麦芽酚,Palatone

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
Maltol 是一种在红参中高浓度存在的芳香化合物的类型,是一种有效的抗氧化剂,用于增强味道和保藏食品。
T3382 Wilforlide A

Abruslactone A,雷公藤内酯甲,3-Epiabruslactone A,Regelide

Tyrosinase Proteases/Proteasome
Wilforlide A (3-Epiabruslactone A) 是一种具有生物活性的三萜,从雷公藤中分离得到,具有抗炎和免疫抑制活性。
T21418 Lisinopril

Linopril,赖诺普利,Zestril,Prinivil,Lisipril

RAAS Endocrinology/Hormones
Lisinopril (Prinivil) 是一种血管紧张素转化酶抑制剂,能够作用于高血压,充血性心力衰竭和心脏病等。
TN1150 Procyanidin B3

原花青素B3,原花青素 B3

Histone Acetyltransferase Chromatin/Epigenetic
Procyanidin B3 是从葡萄中提取的一种黄酮类天然产物,是组蛋白乙酰转移酶特异性抑制剂,可与 p300的其他位点而非活性位点结合,选择性抑制 p300 介导的 androgen 受体乙酰化。
TN1035 Irisolidone

尼泊尔鸢尾异黄酮,葛花苷元

IL Receptor; NF-κB; Chloride channel Immunology/Inflammation; Membrane transporter/Ion channel; NF-κB
Irisolidone 是葛根花中的一种异黄酮,具有较强的保肝活性。它是一种有效的体积调节阴离子通道 (VRAC) 电流抑制剂,有高效阻断作用,IC50 为 5-13 μM。
T3666 Atractylodin

苍术素,Atractydin

Lipid Metabolism
Atractylodin (Atractydin) 是一种Atractylodes lancea 和A. chinensis 的根茎中所含精油的活性成分。它是天然杀虫剂,能够抑制Tribolium castaneum 的活性。
T5081 Adenine monohydrochloride hemihydrate

腺嘌呤盐酸盐,Adenine hydrochloride hydrate,6-Aminopurine hydrochloride hydrate

Endogenous Metabolite; Adenosine Receptor GPCR/G Protein; Metabolism; Neuroscience
Adenine monohydrochloride hemihydrate 是内源性代谢产物的一种。
T13795 Nicotinamide riboside

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Nicotinamide riboside 是维生素 B3 的来源,可以增强氧化代谢并防止高脂肪饮食诱导的代谢异常。它是具有口服活性的 NAD+的前体,增加 NAD+水平并激活SIRT1和SIRT3,可用于研究阿尔茨海默氏病的认知退化。
T8148 Mupirocin calcium hydrate

莫匹罗星钙,Mupirocin calcium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Mupirocin calcium hydrate 是从Pseudomonas fluorescens 中分离得到的,一种有口服活性的抗生素。它可逆地抑制异亮氨酸转移RNA,并抑制细菌蛋白和RNA 的合成起到抗菌作用。
TN1146 8-​Prenylnaringenin

8-Prenylnaringenin,8-异戊烯基柚皮素

Apoptosis; ROS Apoptosis; Immunology/Inflammation
8-prenylnaringenin 是一种从啤酒花穗中分离到的异戊烯类黄酮,具有细胞毒性。它能通过激活小鼠 Akt 磷酸化途径,使其从静止诱导的停用性肌肉萎缩中恢复。它能通过诱导内源性和外源性通路介导的凋亡,对 HCT-116 结肠癌细胞产生抗增殖活性。
TN2031 γ-Terpinene

Moslene,p-Mentha-1,4-diene,Crithmene

Antioxidant oxidation-reduction
γ-Terpinene (p-Mentha-1,4-diene) 是一种单萜化合物,具有高抗氧化属性,适合口服。它展示了直接的自由基清除能力,并且已知是一种有效的抗痛剂。
TN2158 Robinetin

3,3',4',5',7-Pentahydroxyflavone,洋槐黄素

Anti-infection; HIV Protease; Antibacterial Microbiology/Virology; Proteases/Proteasome
Robinetin (3,3',4',5',7-Pentahydroxyflavone) 是一种天然黄酮,具有显著的“两种颜色”固有荧光特性。它具有抗真菌、抗病毒、抗菌、抗突变、抗氧化和抗自由基活性,高效抑制 EYPC 膜脂质过氧化和 HbA 糖基化。
T4726 D-Glucose 6-phosphate sodium

G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate

Others; Endogenous Metabolite Metabolism; Others
D-Glucose 6-phosphate sodium (G6P sodium salt) 是内源性代谢产物的一种。
T5251 Phenylpyruvic acid

2-Oxo-3-phenylpropanoic acid,3-Phenylpyruvic acid,苯丙酮酸

Others; Endogenous Metabolite Metabolism; Others
Phenylpyruvic acid (3-Phenylpyruvic acid) 可以通过乳酸脱氢酶合成3-苯基乳酸 (PLA)。
T4785 Oxfenicine

4-羟基-L-苯甘氨酸,4-Hydroxy-L-phenylglycine

Others Others
Oxfenicine (4-Hydroxy-L-phenylglycine) 是具有口服活性的肉碱棕榈酰转移酶-1 抑制剂。它在缺血期间保护心脏免受坏死组织的损害。它可抑制心脏中脂肪酸的氧化。
T0775 Coumarin

Factor Xa; Influenza Virus Metabolism; Microbiology/Virology
Coumarin 是中国北沙参中的一种主要生物活性成分,具有抗癌、抗炎和抗病毒等活性。它作为几种抗凝剂的前体具有临床价值,尤其是华法林。
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天然产物

28-high brassinolide
Cat.No: T8465
Synonym:
Target: Others
Neomangiferin
Cat.No: T3804
Synonym: Mangiferin 7-glucoside,新芒果苷
Target: Phosphatase
Ethyl cinnamate
Cat.No: TN1624
Synonym:
Target: Calcium Channel, ROS, NO Synthase
Veraguensin
Cat.No: TN1117
Synonym:
Target: p38 MAPK, NF-κB, Antibiotic, Parasite, Antifection
Chrysene
Cat.No: T14961
Synonym: 䓛,屈
Target: Others
Oleoylethanolamide
Cat.No: T12296
Synonym: 油酰单乙醇胺,N-Oleoylethanolamide,Oleamide MEA,Oleic acid monoethanolamide
Target: Endogenous Metabolite, PPAR
10-Methoxycamptothecin
Cat.No: T4S1951
Synonym:
Target: Others, ADC Cytotoxin
4,4'-Methylenediphenol
Cat.No: TMA2386
Synonym:
Target: Others
5,6-Dihydro-5-methyluracil
Cat.No: T0532
Synonym: 5, 6-Dihydrothymine,二氢朐腺嘧啶,Dihydrothymine
Target: Nucleoside Antimetabolite/Analog, Endogenous Metabolite
Transcrocetinate disodium
Cat.No: TQ0027
Synonym: Disodium trans-crocetinate,藏红花,藏红花酸二钠盐
Target: NMDAR, iGluR
Creatine monohydrate
Cat.No: T22300
Synonym: Methylguanidoacetic acid monohydrate,一水肌酸
Target: Others, Endogenous Metabolite
Sappanone A
Cat.No: TMA1570
Synonym:
Target: NF-κB, Nrf2
Miconazole nitrate
Cat.No: T0344L
Synonym: NSC 169434 Nitrate,硝酸咪康唑,R18134 nitrate
Target: Antibacterial, Antibiotic, Antifungal
Zinc sulfate heptahydrate
Cat.No: T19608
Synonym:
Target: Others
Ethynyl estradiol
Cat.No: T1424
Synonym: 乙炔基雌二醇,17α-Ethynylestradiol,Ethinyl Estradiol,炔雌醇
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Amylin, amide, rat acetate(124447-81-0,free base)
Cat.No: TP1232L
Synonym:
Target: Amylin Receptor
Cnidilin
Cat.No: TN1048
Synonym: Knidilin
Target:
Raddeanin A
Cat.No: T3878
Synonym: NSC382873,竹节香附素A,Anemodeanin A,Raddeanin R3
Target: Apoptosis, HDAC
Glycogen, Mussel
Cat.No: T19344
Synonym: α-1,6 葡聚糖,Glycogen
Target: Endogenous Metabolite
2,3-Dimethoxybenzaldehyde
Cat.No: T2975
Synonym: 5,6-Dimethoxybenzaldehyde,邻藜芦醛,o-Veratraldehyde
Target: Antifungal
(S)-3-(4-Hydroxyphenyl)lactic acid
Cat.No: T39887
Synonym: (S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid
Target: Others, Antioxidant
Ingenol-5,20-acetonide
Cat.No: TN1049
Synonym:
Target: Others
Annatto
Cat.No: TN7241
Synonym:
Target:
α,α-Dimethylglycine
Cat.No: T4831
Synonym: 2-Aminoisobutyric acid,α-Aminoisobutanoic acid,2-甲基丙氨酸
Target: Others, Endogenous Metabolite
Febrifugine
Cat.No: TN1012
Synonym:
Target: IL Receptor, Anti-infection, Parasite
Licoflavone B
Cat.No: TN1860
Synonym: 甘草黄酮 B,甘草黄酮B
Target: ATPase, Anti-infection, Parasite
Paederoside
Cat.No: T3S0872
Synonym:
Target: Antiviral, HBV
Phosphocreatine disodium
Cat.No: T3262
Synonym: Disodium phosphocreatine,Phosphocreatine disodium salt,Creatine phosphate disodium salt,磷酸肌酸钠
Target: Others, Endogenous Metabolite
Rhododendrol
Cat.No: T19924
Synonym: Betuligenol,Frambinol,杜鹃醇
Target: Others
Cytosporone B
Cat.No: T3976
Synonym: Csn-B,Dothiorelone G
Target: Others
Octahydrocurcumin
Cat.No: T3S1692
Synonym:
Target: Anti-infection, NF-κB, Reactive Oxygen Species, ROS
(-)-Denudatin B
Cat.No: TN3831
Synonym: Denudatin B
Target: ATPase, Potassium Channel, Calcium Channel, PAFR
D-Luciferin
Cat.No: T3313
Synonym: Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin
Target: Others
Ponasterone A
Cat.No: T21205
Synonym: 坡那甾酮A,AI3-44686
Target: Others
Maltol
Cat.No: T5545
Synonym: Veltol,Larixinic acid,麦芽酚,Palatone
Target: Antioxidant, Endogenous Metabolite
Wilforlide A
Cat.No: T3382
Synonym: Abruslactone A,雷公藤内酯甲,3-Epiabruslactone A,Regelide
Target: Tyrosinase
Lisinopril
Cat.No: T21418
Synonym: Linopril,赖诺普利,Zestril,Prinivil,Lisipril
Target: RAAS
Procyanidin B3
Cat.No: TN1150
Synonym: 原花青素B3,原花青素 B3
Target: Histone Acetyltransferase
Irisolidone
Cat.No: TN1035
Synonym: 尼泊尔鸢尾异黄酮,葛花苷元
Target: IL Receptor, NF-κB, Chloride channel
Atractylodin
Cat.No: T3666
Synonym: 苍术素,Atractydin
Target: Lipid
Adenine monohydrochloride hemihydrate
Cat.No: T5081
Synonym: 腺嘌呤盐酸盐,Adenine hydrochloride hydrate,6-Aminopurine hydrochloride hydrate
Target: Endogenous Metabolite, Adenosine Receptor
Nicotinamide riboside
Cat.No: T13795
Synonym:
Target: Sirtuin
Mupirocin calcium hydrate
Cat.No: T8148
Synonym: 莫匹罗星钙,Mupirocin calcium
Target: Others, Antibacterial, Antibiotic
8-​Prenylnaringenin
Cat.No: TN1146
Synonym: 8-Prenylnaringenin,8-异戊烯基柚皮素
Target: Apoptosis, ROS
γ-Terpinene
Cat.No: TN2031
Synonym: Moslene,p-Mentha-1,4-diene,Crithmene
Target: Antioxidant
Robinetin
Cat.No: TN2158
Synonym: 3,3',4',5',7-Pentahydroxyflavone,洋槐黄素
Target: Anti-infection, HIV Protease, Antibacterial
D-Glucose 6-phosphate sodium
Cat.No: T4726
Synonym: G6P sodium salt,D-Glucose 6-phosphate sodium salt,D-葡萄糖-6-磷酸钠盐,Sodium Glucose-6-Phosphate
Target: Others, Endogenous Metabolite
Phenylpyruvic acid
Cat.No: T5251
Synonym: 2-Oxo-3-phenylpropanoic acid,3-Phenylpyruvic acid,苯丙酮酸
Target: Others, Endogenous Metabolite
Oxfenicine
Cat.No: T4785
Synonym: 4-羟基-L-苯甘氨酸,4-Hydroxy-L-phenylglycine
Target: Others
Coumarin
Cat.No: T0775
Synonym:
Target: Factor Xa, Influenza Virus
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Cat. No. Product Name Species Expression System
TMPY-04261 CD64 Protein, Human, Recombinant (His)

Fc γ RI,Fc receptor, IgG, high affinity I,Fc gamma ...

Human HEK293 Cells
CD64 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32 kDa and the accession number is P12314-1.
TMPY-01848 HMGB1 Protein, Human, Recombinant (aa 1-215, His)

SBP-1,high mobility group box 1,HMG-1,HMG3,HMG1

Human HEK293 Cells
HMGB1 Protein, Human, Recombinant (aa 1-215, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26.3 kDa and the accession number is A0A024RDR0.
TMPY-01205 CD64 Protein, Mouse, Recombinant (His)

Fc receptor, IgG, high affinity I,IGGHAFC,AI323638,...

Mouse HEK293 Cells
CD64 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32 kDa and the accession number is P26151.
TMPY-02590 HMGB1 Protein, Mouse, Recombinant (hFc)

HMG-1,SBP-1,high mobility group box 1,p30,Hmg1,DEF,...

Mouse HEK293 Cells
HMGB1 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 53.3 kDa and the accession number is P63158.
TMPY-03054 Fc epsilon RI Protein, Human, Recombinant (His)

Fc ε RI,α polypeptide,Fc fragment of IgE, high affi...

Human HEK293 Cells
Fc epsilon RI Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 22.5 kDa and the accession number is P12319.
TMPY-05084 Fc epsilon RI Protein, Human, Recombinant

alpha polypeptide,FcERI,α polypeptide,Fc fragment of IgE,

Human HEK293 Cells
Fc epsilon RI Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 21 kDa and the accession number is P12319.
TMPH-02707 HMGB1 Protein, Mouse, Recombinant (His)

High mobility group protein 1,Hmgb1,High m...

Mouse E. coli
HMGB1 Protein, Mouse, Recombinant (His) is expressed in E. coli.
TMPJ-00918 HMGB2 Protein, Human, Recombinant (His)

High Mobility Group Protein B2,HMG2,High M...

Human HEK293 Cells
High Mobility Group Protein B2 (HMGB2) belongs to the non-histone chromosomal high-mobility group protein family. Members of this family are chromatin-associated and widely spread in the nucleus of higher eukaryotic cells. HMGB2 contains 2 HMG box DNA-binding domains. It is associated with chromatin and has the ability to bend DNA, preferentially single-stranded DNA. It is shown that HMGB2 is able to efficiently bend DNA and form DNA circles. In addition, HMGB2 is involved in the final ligation ...
TMPJ-00668 HMGB3 Protein, Human, Recombinant (His)

HMG4,High Mobility Group Protein 2a,HMG-2a,High...

Human HEK293 Cells
High Mobility Group Protein B3 (HMGB3) belongs to the HMGB family. Members of the HMG box subfamily are thought to be have an important role in DNA replication, nucleosome assembly and transcription. HMGB3 binds preferentiallly single-stranded DNA and unwinds double stranded DNA. HMGB3 consists of 200 amino acids and is localized to the cell nucleus. It contains two HMG box DNA-binding domain. HMGB3 binds preferentially single-stranded DNA and unwinds double stranded DNA.
TMPY-05257 FCAMR/CD351 Protein, Mouse, Recombinant (His)

Fc receptor, IgA, IgM, high affinity

Mouse HEK293 Cells
FCAMR/CD351 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.4 kDa and the accession number is Q2TB54-2.
TMPJ-00095 HMGB1 Protein, Human, Recombinant (Truncated)

HMG1,HMG-1,High Mobility Group Protein B1,High<...

Human E. coli
HMGB1 Protein, Human, Recombinant (Truncated) is expressed in E. coli expression system. The predicted molecular weight is 13 KDa and the accession number is P09429.
TMPJ-00094 HMGB1 Protein, Human, Recombinant (N-teminal)

HMG1,HMGB1,High Mobility Group Protein B1,HMG-1,

Human E. coli
HMGB1 Protein, Human, Recombinant (N-teminal) is expressed in E. coli expression system. The predicted molecular weight is 14 KDa and the accession number is P09429.
TMPY-02015 CD64 Protein, Rat, Recombinant (His)

Fc receptor, IgG, high affinity I

Rat HEK293 Cells
CD64 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31.6 kDa and the accession number is A0A0B4J2J0.
TMPH-03313 HMGB1 Protein, Rat, Recombinant (His)

High mobility group protein 1,Amphoterin,High

Rat E. coli
HMGB1 Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 30.8 kDa and the accession number is P63159.
TMPY-02146 CD64 Protein, Human, Recombinant (His & Avi), Biotinylated

Fc γ RI,Fc receptor, IgG, high affinity I,CD64,Fc g...

Human HEK293 Cells
CD64 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 34.4 kDa and the accession number is P12314-1.
TMPH-02706 PDE9A Protein, Mouse, Recombinant (His)

High affinity cGMP-specific 3',5'-cyclic phosphodie...

Mouse E. coli
PDE9A Protein, Mouse, Recombinant (His) is expressed in E. coli.
TMPY-00559 GPIHBP1 Protein, Human, Recombinant (His)

GPI-HBP1,HYPL1D,glycosylphosphatidylinositol anchored hi...

Human HEK293 Cells
GPIHBP1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 16.9 kDa and the accession number is Q8IV16.
TMPY-00822 HMGB1 Protein, Human, Recombinant (hFc)

HMG1,SBP-1,high mobility group box 1,HMG3,HMG-1

Human HEK293 Cells
HMGB1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 51.5 kDa and the accession number is A0A024RDR0.
TMPJ-01004 HDGF Protein, Human, Recombinant (His)

HDGF,Hepatoma-Derived Growth Factor,HMG1L2,High Mob...

Human E. coli
Hepatoma-Derived Growth Factor is a original member of the HDGF family. HDGF is a cytoplasmic protein and contains one PWWP domain. HDGF expression levels are high in the nucleus and cytoplasm of smooth muscle and endothelial cells. HDGF has proliferative, angiogenic and neurotrophic activity. HDGF was initially characterized as a secreted mitogen from the Huh-7 human hepatoma cell line. As a heparin-binding protein, which is highly expressed in tumor cells where it stimulates proliferation. HDG...
TMPH-01467 PDE9A Protein, Human, Recombinant (His & Myc)

PDE9A,High affinity cGMP-specific 3',5'-cyclic phos...

Human E. coli
PDE9A Protein, Human, Recombinant (His & Myc) is expressed in E. coli.
TMPY-00557 GPIHBP1 Protein, Human, Recombinant (hFc)

glycosylphosphatidylinositol anchored high density ...

Human HEK293 Cells
GPIHBP1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.2 kDa and the accession number is Q8IV16.
TMPY-02979 HMGN3 Protein, Human, Recombinant (His)

PNAS-24,TRIP7,PNAS-25,high mobility group nucleosom...

Human E. coli
HMGN3 belongs to the HMGN family and is expressed in the kidney, lung, pancreas, testis, skeletal muscle, heart, thyroid gland, pituitary gland, prostate, and uterus. Members of the HMGN family bind to nucleosomes without any specificity for the underlying DNA sequence. They affect the global and local structure of chromatin, as well as the levels of histone modifications, and thus play a role in epigenetic regulation of gene expression. HMGN3 regulates the expression of the glucose transporter ...
TMPY-03427 HMGB1 Protein, Human, Recombinant (aa 57-158, His)

SBP-1,HMG3,high mobility group box 1,HMG1,HMG-1

Human E. coli
HMGB1 Protein, Human, Recombinant (aa 57-158, His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 13.6 kDa and the accession number is P09429.
TMPH-00189 HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO)

Chaperone protein HtpG,Heat shock protein HtpG,htpG,High...

Bacteroides fragilis E. coli
Molecular chaperone. Has ATPase activity. HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 57.0 kDa and the accession number is Q5LCH4.
TMPH-02939 TFAM Protein, Mouse, Recombinant (His & Myc)

Testis-specific high mobility group protein,Transcr...

Mouse E. coli
TFAM Protein, Mouse, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 30.9 kDa and the accession number is P40630.
TMPH-03027 HMW1 Protein, Mycoplasma pneumoniae, Recombinant (His & Myc)

Cytadherence accessory protein 1,Cytadherence high ...

Mycoplasma pneumoniae E. coli
Component of the cytoskeleton-like structure which stabilizes the shape of the wall-less Mycoplasma. This cytoskeleton-like network of accessory proteins containing HMW proteins 1 to 5 allows the proper anchoring of cytadhesin proteins in the mycoplasmal membrane at the attachment organelle.
TMPY-01988 CD64 Protein, Mouse, Recombinant (His & Avi), Biotinylated

Fc receptor, IgG, high affinity I,FcgammaRI,CD64,IG...

Mouse HEK293 Cells
CD64 Protein, Mouse, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 34.3 kDa and the accession number is P26151.
TMPH-03028 HMW3 Protein, Mycoplasma pneumoniae, Recombinant (His & Myc)

hmw3,Accessory adhesin protein 3,Cytadherence accessory prot...

Mycoplasma pneumoniae E. coli
Component of the cytoskeleton-like structure which stabilizes the shape of the wall-less mycoplasma. This cytoskeleton-like network of accessory proteins containing HMW proteins 1 to 5 allows the proper anchoring of cytadhesin proteins in the mycoplasmal membrane at the attachment organelle. Essential for successful surface parasitism. HMW3 Protein, Mycoplasma pneumoniae, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight...
TMPH-00594 HtpG Protein, E. coli, Recombinant (His)

Chaperone protein HtpG,Heat shock protein C62.5,Heat shock p...

E. coli E. coli
Molecular chaperone. Has ATPase activity.
TMPH-02894 HTRA1 Protein, Mouse, Recombinant (His)

Serine protease 11,Serine protease HTRA1,Htra1,High...

Mouse E. coli
HTRA1 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with C-6xHis tag. The predicted molecular weight is 39.0 kDa and the accession number is Q9R118.
TMPH-02081 HTRA1 Protein, Human, Recombinant (His & SUMO)

Serine protease HTRA1,HTRA1,Serine protease 11,L56,High<...

Human E. coli
HTRA1 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli.
TMPH-01776 HMGN2 Protein, Human, Recombinant (GST)

Non-histone chromosomal protein HMG-17,HMGN2,High m...

Human E. coli
Binds to the inner side of the nucleosomal DNA thus altering the interaction between the DNA and the histone octamer. May be involved in the process which maintains transcribable genes in a unique chromatin conformation. HMGN2 Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 36.4 kDa and the accession number is P05204.
TMPH-01468 SLC31A1 Protein, Human, Recombinant (His & SUMO)

Copper transporter 1,SLC31A1,High affinity copper u...

Human E. coli
SLC31A1 Protein, Human, Recombinant (His & SUMO) is expressed in in vitro E. coli expression system.
TMPH-00595 HtpG Protein, E. coli, Recombinant

High temperature protein G,Heat shock protein C62.5...

E. coli E. coli
Molecular chaperone. Has ATPase activity.
TMPY-03064 Fc epsilon RI Protein, Mouse, Recombinant (hFc)

α polypeptide,FcERI,Fc ε RI,Fcr-5,alpha polypeptide,Fce1a,Fc...

Mouse HEK293 Cells
Fc epsilon RI Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 48 kDa and the accession number is P20489.
TMPJ-00326 CD122/IL2RB Protein, Human, Recombinant (aa 27-239, His & Avi), Biotinylated

IL-2R subunit beta,High affinity IL-2 receptor subu...

Human HEK293 Cells
Human IL-2RB, also known asinterleukin-2 receptor subunit beta,is the receptor for interleukin-2. IL2 receptor complex is involved in receptor mediated endocytosis and transduces the mitogenic signals of IL2. IL2 receptor complex has three forms with respect to ability to bind IL2. IL-2RB is belonged to a type I membrane protein,and has a 26 residue signal peptide, a 214 residue extracellular region, a 25 residue transmembrane region and a 286 residue cytoplasmic domain. IL-2RB is the subunit c...
TMPJ-00734 KNG1 Protein, Human, Recombinant (His)

KNG1,High Molecular Weight Kininogen,BDK,HMWK,KNG,W...

Human HEK293 Cells
Kininogen-1 is a secreted protein which contains three cystatin domains. There are two alternatively spliced forms, designated as the high molecular weight (HMW) and low MW (LMW) forms. Kininogen-1 plays a critical role in blood coagulation and inflammatory response. Kininogens are inhibitors of thiol proteases. Kininogen-1 participates in blood coagulation by helping to position optimally prekallikrein and factor XI next to factor XII, also inhibits the thrombin- and plasmin-induced aggregation...
TMPH-01709 Mucin-5B/MUC5B Protein, Human, Recombinant (His & Myc)

Mucin-5 subtype B, tracheobronchial,Mucin-5B,Sublingual glan...

Human E. coli
Gel-forming mucin that is thought to contribute to the lubricating and viscoelastic properties of whole saliva and cervical mucus. Mucin-5B/MUC5B Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 18.9 kDa and the accession number is Q9HC84.
TMPJ-00617 IL-33 Protein, Rhesus macaque, Recombinant (His)

Interleukin-33,IL1F11,IL33,白介素,白细胞介素,IL-1F11,Interleukin-1 F...

Rhesus E. coli
Interleukin-33 (IL-33) belongs to the IL-1 superfamily. IL33 is highly expressed in endothelial venules found in tonsils, Peyer patches and mesenteric lymph nodes, but almost undetectable in placenta. IL33 induces the production of T helper-2 (Th2)-associated cytokines. IL-33 is a cytokine that mediates its biological effects by binding to and signals through IL1RL1/ST2 and IL-1 Receptor Accessory Protein (IL1RAP), activating intracellular molecules in the NF-κB and MAP kinase signaling pathways...
TMPJ-01019 NHP2L1 Protein, Human, Recombinant (His)

High Mobility Group-Like Nuclear Protein 2 Homolog ...

Human E. coli
NHP2-Like Protein 1 (NHP2L1) is a member of the ribosomal protein L7Ae family. NHP2L1 proteinis limited to the nucleus, primarily focused in the dense fibrillar component of the nucleolus. NHP2L1 has been shown to interact with RAD17and PRPF31. The protein undergoes a conformational change upon RNA-binding. NHP2L1 binds to the 5-stem-loop of U4 snRNA and may play a role in the late stage of spliceosome assembly, prior to step I of splicing catalysis.
TMPY-05033 5T4/TPBG Protein, Human, Recombinant (aa 60-345, His)

5T4AG,trophoblast glycoprotein,WAIF1,M6P1,5T4

Human HEK293 Cells
Trophoblast glycoprotein (TPBG), also known as 5T4, is the therapeutic target of several anticancer agents currently in clinical development, largely due to its high expression in tumors and low expression in normal adult tissues. 5T4/TPBG Protein, Human, Recombinant (aa 60-345, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 33.1 kDa and the accession number is Q13641.
TMPY-00021 PADI4 Protein, Human, Recombinant (His)

PADI5,PAD4,PDI4,peptidyl arginine deiminase, type IV,PAD,PDI...

Human Baculovirus Insect Cells
Protein-arginine deiminase type-4, also known as HL-6 PAD, Peptidylarginine deiminase IV, Protein-arginine deiminase type I V and PADI4, is a cytoplasm and nucleus protein that belongs to the protein arginine deiminase family. PADI4 is expressed in CD34+stem cells in normal tissues, and many more CD34+ cells expressing PADI4 are present in tumour tissues. PADI4 post-translationally converts peptidylarginine to citrulline, a process called citrullination. Studies have demonstrated the high expres...
TMPK-01414 Qa-1b&B2M&Qdm (AMAPRTLLL) Monomer Protein, Mouse, MHC (His & Avi)

Qa-1b,Qdm,MHC,H2-T23

Mouse HEK293 Cells
Qa-1b binds a peptide (AMAPRTLLL), referred to as Qdm (for Qa-1 determinant modifier), derived from the signal sequence of murine class Ia molecules. This peptide binds with high affinity and accounts for almost all of the peptides associated with this molecule. Human histocompatibility leukocyte antigen (HLA)-E, a homologue of Qa-1b, binds similar peptides derived from human class Ia molecules and interacts with CD94/NKG2 receptors on natural killer cells.
TMPK-01074 CD163 Protein, Human, Recombinant (His & Avi)

CD163,HbSR,RM3/1,MM130,CD163 molecule,GHI/61,sCD163,SCARI1,M...

Human HEK293 Cells
The hemoglobin (Hb) scavenger receptor, CD163, is a macrophage-specific protein and the upregulated expression of this receptor is one of the major changes in the macrophage switch to alternative activated phenotypes in inflammation. Accordingly, a high CD163 expression in macrophages is a characteristic of tissues responding to inflammation. CD163 Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 111.4 kDa and th...
TMPY-04722 DcR1/TRAILR3 Protein, Human, Recombinant (His)

TRAILR3,TRID,DCR1,TRAIL-R3,CD263,DCR1-TNFR,tumor necrosis fa...

Human HEK293 Cells
TNFRSF10C CNV in patients with CRC is associated with distant metastatic disease. A high frequency of CGI methylation in the TNFRSF10C promoter results in inactivation of the gene and enhancement of tumor growth in most PC cell lines (except CFPAC-1). Inactivation of TNFRSF10C by CpG island (CGI) hypermethylation can play an important role in PC progression and be potentially useful as a diagnostic marker and a new therapeutic approach for PC.
TMPJ-01099 IL-15RA Protein, Human, Recombinant (hFc, Human Cells)

interleukin-15 receptor subunit α,IL15RA,interleukin-15 rece...

Human HEK293 Cells
Interleukin 15 Receptor alpha (IL-15Rα) is a transmembrane glycoprotein that plays a pleiotropic role in immune development and function, including the positive maintenance of lymphocyte homeostasis. IL-15Rα chain can bind soluble IL-15 and “transpresent” cytokine to the cells, allowing them to respond to IL-15. Soluble IL-15Rα can function as a specific high-affinity IL-15 antagonist. The soluble IL-15/IL-15Rα complexes exhibit a strong agonistic activity which is mediated through membrane-boun...
TMPJ-01461 IL-15RA & IL-15 Protein, Human, Recombinant (hFc)

IL-15 Receptor α & IL-15 Fusion Protein,Interleukin-15,IL15R...

Human HEK293 Cells
IL15RA is a high-affinity receptor for interleukin-15. Il15ra associates as a heterotrimer with the IL-2 receptor beta and gamma subunits to initiate signal transduction. It can signal both in cis and trans where IL15R from one subset of cells presents IL15 to neighboring IL2RG-expressing cells. Il15ra is expressed in special cells including a wide variety of Tand B cells and non-lymphoid cells.IL-15 is a cytokine that regulates T cell and natural killer cell activation and proliferation. IL-15 ...
TMPY-03958 TGF alpha Protein, Human, Recombinant

transforming growth factor α,转化生长因子,transforming growth fact...

Human E. coli
The miR-137 served as a tumor suppressor in non-small cell lung cancer (NSCLC) and its suppressive effect is mediated by repressing TGFA expression. TGFA gene expression was significantly higher in tumor tissues compared to adjacent normal tissue and high TGFA gene expression strongly correlated with poor survival in patients with lung adenocarcinoma, and miR-374a suppresses lung adenocarcinoma cell proliferation and invasion via targeting TGFA gene expression. Transforming growth factor alpha (...
TMPJ-00135 BDNF Protein, Human/Murine/Rat, Recombinant

BDNF,Abrineurin,Brain-Derived Neurotrophic Factor

Human,Mouse,Rat E. coli
Brain-Derived Neurotrophic Factor (BDNF) is a member of the neurotrophin family. Along with other structurally related neurotrophic factors NGF, NT-3 and NT-4, BDNF binds with high affinity to the TrkB kinase receptor. It also binds with the LNGFR (for low-affinity nerve growth factor receptor, also known as p75). BDNF promotes the survival, growth and differentiation of neurons. It serves as a major regulator of synaptic transmission and plasticity at adult synapses in many regions of the CNS. ...
TMPJ-00254 TGF beta 3 Protein, Human/Mouse/Rat, Recombinant

Latency-associated peptide,TGF-beta-3,Transforming growth fa...

Human,Mouse,Rat HEK293 Cells
Transforming growth factor beta 3(TGFB3) is a member of a TGF -β superfamily which is defined by theirstructural and functional similarities. TGFB3 is secreted as a complex with LAP. This latent form of TGFB3becomes active upon cleavage by plasmin, matrix metalloproteases, thrombospondin -1, and a subset ofintegrins. It binds with high affinity to TGF- β RII, a type II serine/threonine kinase receptor. TGFB3 is involved incell differentiation, embryogenesis and development.It is believed to regu...
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重组蛋白

CD64 Protein, Human, Recombinant (His)
Cat.No: TMPY-04261
Species: Human
Expression System: HEK293 Cells
HMGB1 Protein, Human, Recombinant (aa 1-215, His)
Cat.No: TMPY-01848
Species: Human
Expression System: HEK293 Cells
CD64 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01205
Species: Mouse
Expression System: HEK293 Cells
HMGB1 Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-02590
Species: Mouse
Expression System: HEK293 Cells
Fc epsilon RI Protein, Human, Recombinant (His)
Cat.No: TMPY-03054
Species: Human
Expression System: HEK293 Cells
Fc epsilon RI Protein, Human, Recombinant
Cat.No: TMPY-05084
Species: Human
Expression System: HEK293 Cells
HMGB1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02707
Species: Mouse
Expression System: E. coli
HMGB2 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00918
Species: Human
Expression System: HEK293 Cells
HMGB3 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00668
Species: Human
Expression System: HEK293 Cells
FCAMR/CD351 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-05257
Species: Mouse
Expression System: HEK293 Cells
HMGB1 Protein, Human, Recombinant (Truncated)
Cat.No: TMPJ-00095
Species: Human
Expression System: E. coli
HMGB1 Protein, Human, Recombinant (N-teminal)
Cat.No: TMPJ-00094
Species: Human
Expression System: E. coli
CD64 Protein, Rat, Recombinant (His)
Cat.No: TMPY-02015
Species: Rat
Expression System: HEK293 Cells
HMGB1 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03313
Species: Rat
Expression System: E. coli
CD64 Protein, Human, Recombinant (His & Avi), Biotinylated
Cat.No: TMPY-02146
Species: Human
Expression System: HEK293 Cells
PDE9A Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02706
Species: Mouse
Expression System: E. coli
GPIHBP1 Protein, Human, Recombinant (His)
Cat.No: TMPY-00559
Species: Human
Expression System: HEK293 Cells
HMGB1 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00822
Species: Human
Expression System: HEK293 Cells
HDGF Protein, Human, Recombinant (His)
Cat.No: TMPJ-01004
Species: Human
Expression System: E. coli
PDE9A Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01467
Species: Human
Expression System: E. coli
GPIHBP1 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-00557
Species: Human
Expression System: HEK293 Cells
HMGN3 Protein, Human, Recombinant (His)
Cat.No: TMPY-02979
Species: Human
Expression System: E. coli
HMGB1 Protein, Human, Recombinant (aa 57-158, His)
Cat.No: TMPY-03427
Species: Human
Expression System: E. coli
HtpG Protein, Bacteroides fragilis, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00189
Species: Bacteroides fragilis
Expression System: E. coli
TFAM Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02939
Species: Mouse
Expression System: E. coli
HMW1 Protein, Mycoplasma pneumoniae, Recombinant (His & Myc)
Cat.No: TMPH-03027
Species: Mycoplasma pneumoniae
Expression System: E. coli
CD64 Protein, Mouse, Recombinant (His & Avi), Biotinylated
Cat.No: TMPY-01988
Species: Mouse
Expression System: HEK293 Cells
HMW3 Protein, Mycoplasma pneumoniae, Recombinant (His & Myc)
Cat.No: TMPH-03028
Species: Mycoplasma pneumoniae
Expression System: E. coli
HtpG Protein, E. coli, Recombinant (His)
Cat.No: TMPH-00594
Species: E. coli
Expression System: E. coli
HTRA1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02894
Species: Mouse
Expression System: E. coli
HTRA1 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-02081
Species: Human
Expression System: E. coli
HMGN2 Protein, Human, Recombinant (GST)
Cat.No: TMPH-01776
Species: Human
Expression System: E. coli
SLC31A1 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01468
Species: Human
Expression System: E. coli
HtpG Protein, E. coli, Recombinant
Cat.No: TMPH-00595
Species: E. coli
Expression System: E. coli
Fc epsilon RI Protein, Mouse, Recombinant (hFc)
Cat.No: TMPY-03064
Species: Mouse
Expression System: HEK293 Cells
CD122/IL2RB Protein, Human, Recombinant (aa 27-239, His & Avi), Biotinylated
Cat.No: TMPJ-00326
Species: Human
Expression System: HEK293 Cells
KNG1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00734
Species: Human
Expression System: HEK293 Cells
Mucin-5B/MUC5B Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01709
Species: Human
Expression System: E. coli
IL-33 Protein, Rhesus macaque, Recombinant (His)
Cat.No: TMPJ-00617
Species: Rhesus
Expression System: E. coli
NHP2L1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-01019
Species: Human
Expression System: E. coli
5T4/TPBG Protein, Human, Recombinant (aa 60-345, His)
Cat.No: TMPY-05033
Species: Human
Expression System: HEK293 Cells
PADI4 Protein, Human, Recombinant (His)
Cat.No: TMPY-00021
Species: Human
Expression System: Baculovirus Insect Cells
Qa-1b&B2M&Qdm (AMAPRTLLL) Monomer Protein, Mouse, MHC (His & Avi)
Cat.No: TMPK-01414
Species: Mouse
Expression System: HEK293 Cells
CD163 Protein, Human, Recombinant (His & Avi)
Cat.No: TMPK-01074
Species: Human
Expression System: HEK293 Cells
DcR1/TRAILR3 Protein, Human, Recombinant (His)
Cat.No: TMPY-04722
Species: Human
Expression System: HEK293 Cells
IL-15RA Protein, Human, Recombinant (hFc, Human Cells)
Cat.No: TMPJ-01099
Species: Human
Expression System: HEK293 Cells
IL-15RA & IL-15 Protein, Human, Recombinant (hFc)
Cat.No: TMPJ-01461
Species: Human
Expression System: HEK293 Cells
TGF alpha Protein, Human, Recombinant
Cat.No: TMPY-03958
Species: Human
Expression System: E. coli
BDNF Protein, Human/Murine/Rat, Recombinant
Cat.No: TMPJ-00135
Species: Human,Mouse,Rat
Expression System: E. coli
TGF beta 3 Protein, Human/Mouse/Rat, Recombinant
Cat.No: TMPJ-00254
Species: Human,Mouse,Rat
Expression System: HEK293 Cells
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Cat. No. Product Name Target Signaling Pathways
T12300 Olmesartan-d4

RNH-6270 D4,奥美沙坦 D4

Others Others
Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.
T71306 Gemfibrozil-d6

Gemfibrozil-d6 is intended for use as an internal standard for the quantification of gemfibrozil by GC- or LC-MS. Gemfibrozil is a peroxisome proliferator-activated reporter α and PPARγ agonist. In vivo, gemfibrozil reduces serum total cholesterol, triglyceride, and LDL levels in a rat model of high-cholesterol diet-induced hyperlipidemia. Gemfibrozil reduces atherosclerotic plaque area, superoxide production, and expression of the genes encoding the NF-κB subunit p65 and chemokine (C-C) motif l...
T13282 Valsartan-d9

CGP-48933 D9,缬沙坦 D9

Others Others
Valsartan D9 is a deuterium-labeled valsartan. Valsartan is an antagonist of the angiotensin II receptor and for the treatment of high blood pressure and heart failure.
TMIJ-0389 Chrysene-d12

Chrysene-d12 是 Chrysene 的氘代化合物。Chrysene 的 CAS 号为 218-01-9。Chrysene 是高分子量 (HMW) 多环芳烃,有极强的顽固性和致癌性。
TMIJ-0173 Calcipotriol-d4

Calcipotriol-d4 是 Calcipotriol 的氘代化合物。Calcipotriol 的 CAS 号为 112965-21-6。Calcipotriol 是一种合成的 VitD3类似物,对维他命D受体具有高亲和力。
TMIJ-0183 Terazosin-d8

Terazosin-d8 是 Terazosin 的氘代化合物。Terazosin 的 CAS 号为 63590-64-7。
TMIJ-0498 Fluticasone Propionate-d5

Fluticasone Propionate-d5 是 Fluticasone Propionate 的氘代化合物。Fluticasone Propionate 的 CAS 号为 80474-14-2。Fluticasone propionate 是一种选择性糖皮质激素受体激动剂,是一种局部抗炎激素,绝对亲和力KD为 0.5 nM。具有抗病毒活性。
TMIJ-0296 Bezafibrate-d6 (dimethyl-d6)

Bezafibrate-d6 (dimethyl-d6) 是 Bezafibrate 的氘代化合物。Bezafibrate 的 CAS 号为 41859-67-0。Bezafibrate 是一种降血脂剂,是PPAR的激动剂,对人以及鼠PPARα、PPARγ和PPARδ的EC50分别为 50、60和20 μM, 以及 90、55 和110 μM。
T35697 Lauric Acid-13C

Lauric acid-13C is intended for use as an internal standard for the quantification of lauric acid by GC- or LC-MS. Lauric acid is a medium-chain saturated fatty acid. It has been found at high levels in coconut oil.1Lauric acid induces the activation of NF-κB and the expression of COX-2, inducible nitric oxide synthase (iNOS), and IL-1α in RAW 264.7 cells when used at a concentration of 25 μM.2
TMID-0139 17α-Ethynylestradiol-2,4,16,16-d4

17α-Ethynylestradiol-2,4,16,16-d4 是 17α-Ethynylestradiol 的氘代化合物。17α-Ethynylestradiol 的 CAS 号为 57-63-6。Ethynyl Estradiol 是一种高效的生物活性雌激素。
TMIH-0461 Prucalopride-13C-d3

Prucalopride-13C-d3 是 Prucalopride 的 13C 和氘代化合物。Prucalopride 的 CAS 号为 179474-81-8。Prucalopride 是一种选择性、高亲和力的 5-HT4A/4B 受体激动剂,Ki为2.5和 8 nM。它对 5-HT4A/4B 受体的选择性是其他 5-HT 受体亚型的 290 倍以上。
TMIJ-0055 DL-Norepinephrine-d6 HCl

DL-Norepinephrine-d6 HCl 是 DL-NorepinephrineHCl 的氘代化合物。DL-NorepinephrineHCl 的 CAS 号为 55-27-6。DL-Norepinephrine hydrochloride 是一种靶向α1 adrenoceptor和β1 adrenoceptor的神经递质,可降低心内膜下氧分压。它是一种模拟内源性去甲肾上腺素的拟交感神经作用的合成苯乙胺。
TMIJ-0042 Metoprolol-d7 Hydrochloride

Metoprolol-d7 Hydrochloride 是 Metoprolol Hydrochloride 的氘代化合物。Metoprolol Hydrochloride 的 CAS 号为 56392-18-8。Metoprolol 是一种选择性 β1 受体阻滞剂。Metoprolol 用于治疗高血压、因心脏血流不畅而引起的胸痛以及许多心率异常快的疾病。
TMIJ-0371 Coumarin-d4

Coumarin-d4 是 Coumarin 的氘代化合物。Coumarin 的 CAS 号为 91-64-5。Coumarin 是中国北沙参中的一种主要生物活性成分,具有抗癌、抗炎和抗病毒等活性。它作为几种抗凝剂的前体具有临床价值,尤其是华法林。
T70990 ADMA-d6

NG,NG-dimethyl-L-arginine-d6 (ADMA-d6) (hydrochloride) is intended for use as an internal standard for the quantification of NG,NG-dimethyl-L-arginine by GC- or LC-MS. ADMA is an endogenous inhibitor of nitric oxide synthase (NOS). It is formed from arginine by protein arginine methyltransferases (PRMTs) and degraded by dimethylarginine dimethylaminohydrolases (DDAHs) and alanine-glyoxylate aminotransferase 2 (AGXT2). ADMA levels are increased concomitant with an increase in blood pressure in Da...
TMIJ-0050 Butyricacid-d7

Butyricacid-d7 是 Butyricacid 的氘代化合物。Butyricacid 的 CAS 号为 107-92-6。Butyric acid 是一种从许多乳制品中分离出来的脂肪酸,具有抗癌活性。 它抑制组蛋白去乙酰化酶 (HDAC) 并诱导胶质瘤细胞凋亡和 G1 期细胞周期停滞。此外,它在低剂量时刺激上皮细胞增殖,在高剂量时抑制增殖。
TMID-0097 Ethyl-d5-malonic Acid

Ethyl-d5-malonic Acid 是 Ethyl-malonic Acid 的氘代化合物。Ethyl-malonic Acid 的 CAS 号为 601-75-2。Ethylmalonic acid 是潜在有毒物质,非致癌性,与神经性厌食和甲氧基脱羧酶缺乏症有关。
T69600 Spermidine-d6

Spermidine-d6 is intended for use as an internal standard for the quantification of spermidine by GC- or LC-MS. Spermidine is an endogenous polyamine. It is formed from putrescine by spermidine synthase. Spermidine (25 µM) inhibits the activity of the human inward-rectifying potassium channel Kir2.3 in a patch-clamp assay. It induces autophagy in HeLa cells when used at a concentration of 100 µM and increases the lifespan of D. melanogaster, yeast, and C. elegans. Spermidine (30 mM in the drinki...
T35591 Guanfacine-13C,15N3

Guanfacine-13C,15N3

Guanfacine-13C,15N3is intended for us as an internal standard for the quantification of guanfacine by GC- or LC-MS. Guanfacine is an α2-adrenergic receptor (α2-AR) agonist with Kivalues of 93, 1,380, and 3,890 nM for α2A-, α2B-, and α2C-ARs, respectively, in a radioligand binding assay.1It has EC50values of 52, 288, and 602 nM for α2A-, α2B-, and α2C-ARs, respectively, for stimulated [35S]GTPγS binding. It also binds to imidazoline receptor 1 (Ki= 19 nM in a radioligand binding assay).2Guanfacin...
T38297 Ribavirin-13C5

Ribavirin-13C5

Ribavirin-13C5is intended for use as an internal standard for the quantification of ribavirin by GC- or LC-MS. Ribavirin is an antiviral guanosine nucleoside analog.1,2Upon entry into cells, ribavirin is metabolized to an active triphosphate form that induces viral RNA chain termination and inhibits viral polymerases. It reduces replication in a panel of seven RNA and four DNA viruses in Vero cells (EC50s = 2-95 μg/ml).3Ribavirin also reduces replication of severe acute respiratory syndrome coro...

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Synonym: RNH-6270 D4,奥美沙坦 D4
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Target:
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Fluticasone Propionate-d5
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Target:
Lauric Acid-13C
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17α-Ethynylestradiol-2,4,16,16-d4
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Target:
Prucalopride-13C-d3
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Target:
DL-Norepinephrine-d6 HCl
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Target:
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Cat.No: TMIJ-0371
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Cat.No: T70990
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Target:
Butyricacid-d7
Cat.No: TMIJ-0050
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Target:
Ethyl-d5-malonic Acid
Cat.No: TMID-0097
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Target:
Spermidine-d6
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Guanfacine-13C,15N3
Cat.No: T35591
Synonym: Guanfacine-13C,15N3
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Ribavirin-13C5
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Synonym: Ribavirin-13C5
Target:
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