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Targets Recommended: Dopamine Receptor

抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
T14767	BP 897 hydrochloride	Dopamine Receptor	GPCR/G Protein; Neuroscience
	BP 897 hydrochloride 是有效的部分多巴胺 D3受体激动剂和弱 D2受体拮抗剂，在多巴胺 D3 受体 (Ki=0.92 nM) 上显示出高亲和力，而在 D2 受体上显示出 70 倍的低亲和力 (Ki=61 nM)。它表现出对可卡因寻求行为的选择性抑制。
T9100	BP 897 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-	Dopamine Receptor	GPCR/G Protein; Neuroscience
	BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) 是一种有效的部分多巴胺D3受体激动剂和弱D2受体拮抗剂，在多巴胺 D3 受体(Ki=0.92 nM) 上显示出高亲和力，而在 D2 受体上显示出 70 倍的低亲和力 (Ki=61 nM)。它表现出对可卡因寻求行为的选择性抑制。
T4385	PF-4840154	TRP/TRPV Channel	Membrane transporter/Ion channel
	PF4840154 是有效的大鼠和人TrpA1通道选择性激动剂，EC50分别为 97 和 23 nM。PF-4840154 可以诱导 TrpA1 介导的小鼠伤害行为。
T38001	LEI-401 LEI 401	Phospholipase	Metabolism
	LEI-401 是一种可穿过血脑屏障且具有选择性和有效性的 NAPE-PLD 抑制剂(IC50：27 nM)。LEI-401 降低自由活动小鼠脑内n -酰基乙醇胺(NAEs)含量，可调节小鼠情绪行为。
T28282	Oxypertine Win-18501,Forit,Win18501,Win 18501	Others	Others
	Oxypertine is an indole-derivative antipsychotic with general properties similar to those of the chlorpromazine and phenothiazine. Oxypertine is used as a treatment for various psychoses including mania, schizophrenia, disturbed behaviour, and severe anx
T26807	Bifeprunox Mesylate Bifeprunox,DU 127090,DU-127090,DU127090	Others	Others
	Bifeprunox is a partial dopamine and serotonin agonist potentially for the treatment of schizophrenia. Bifeprunox suppresses in vivo VTA dopaminergic neuronal activity via D2 and not D3 dopamine autoreceptor activation. Bifeprunox influences nicotine-seek
T27752	KT109 KT-109,KT 109	Others	Others
	KT109 is a selective inhibitor of DAGLβ (IC50 = 42 nM). KT109-treated wild-type mice displayed reductions in LPS-induced allodyni as well as in DAGL-β (-/-) micea. Repeated KT109 administration prevented the expression of LPS-induced allodynia, without ev
T62132	S-777469	Others	Others
	S-777469 是一种选择性的、口服具有活力的大麻素 2 型受体(CB2)激动剂 (Ki: 36 nM)。S-777469 能够剂量依赖性地明显抑制化合物 48/80 诱导的小鼠抓挠行为。S-777469 兴奋 CB2，抑制瘙痒信号的传递，显示出止痒效果。
T38145	Eltoprazine	Others	Others
	Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.IC50 value:Target: 5-HT1A/1B agonist; 5-HT2C antagonistin vitro: The binding of [3H]eltoprazine to whole tissue sections was saturable and revealed an apparent dissociation constant (Kd) of 11 nM. Specific [3H]eltoprazine binding was completely displaced by 5-HT; conversely, unlabelled eltoprazine reduced [3H]5-HT binding to the levels of no...

化合物

BP 897 hydrochloride

Cat.No: T14767

Synonym:

Target: Dopamine Receptor

BP 897

Cat.No: T9100

Synonym: 2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-

Target: Dopamine Receptor

PF-4840154

Cat.No: T4385

Synonym:

Target: TRP/TRPV Channel

LEI-401

Cat.No: T38001

Synonym: LEI 401

Target: Phospholipase

Oxypertine

Cat.No: T28282

Synonym: Win-18501,Forit,Win18501,Win 18501

Target: Others

Bifeprunox Mesylate

Cat.No: T26807

Synonym: Bifeprunox,DU 127090,DU-127090,DU127090

Target: Others

KT109

Cat.No: T27752

Synonym: KT-109,KT 109

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-02393	Thimet Oligopeptidase/THOP1 Protein, Mouse, Recombinant (His) thimet oligopeptidase 1,EP24.15,AI131655,AI327041	Mouse	Baculovirus Insect Cells
	THOP1, also known as Thimet oligopeptidase 1, Thimet oligopeptidase, EC 3.4.24.15, or EP24.15, is a zinc(II) endopeptidase implicated in the processing of numerous physiological peptides. As an intracellular enzyme, highly expressed in the brain, kidneys and neuroendocrine tissue, THOP1 has been proposed to metabolize peptides within cells, thereby affecting antigen presentation and G protein-coupled receptor signal transduction. Its substrates is gonadotrophin-releasing hormone (GnRH), an impor...

重组蛋白

Thimet Oligopeptidase/THOP1 Protein, Mouse, Recombinant (His)

Cat.No: TMPY-02393

Species: Mouse

Expression System: Baculovirus Insect Cells

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