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Targets Recommended: Others

33

抑制剂 & 化合物

3

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Cat. No. Product Name Target Signaling Pathways
T72024 ZIM

Others Others
ZIM,一种从4-Aminoantipyrine衍生的降冰片烯,有效诱导DNA损伤,造成基因组及染色体损害,进而引发细胞死亡和激活吞噬。其化疗潜力适用于癌症研究。
T4239 1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde

1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOLE-5-CARBALDEHYDE

Others Others
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde 是中间体。
T10672 Capzimin

Others Others
Capzimin 是蛋白酶体异肽酶 Rpn11 的选择性抑制剂。
T7505 Azimilide Dihydrochloride

NE-10064 Dihydrochloride,盐酸阿齐利特

Potassium Channel Membrane transporter/Ion channel
Azimilide Dihydrochloride (NE-10064 Dihydrochloride) 是 I(Ks) 和 I(Kr) 抑制剂,具有抗心律失常活性。
T68054 Denzimol

Others Others
Denzimol 是一种新型抗惊厥化合物。Denzimol 对强直性癫痫发作具有选择性。
T9152 2-(2-Hydroxyphenyl)-1H-benzimidazole

Others Others
2-(2-Hydroxyphenyl)-1H-benzimidazole 已被用于合成聚合物和其他材料的催化剂。
Fr12535 2-(Trifluoromethyl)benzimidazole

Others Others
Compound Fr12535 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12535,CAS号为 312-73-2。
T19749 Azimsulfuron

A 8947,A8947,A-8947

Others Others
Azimsulfuron 是一种除草剂,可用于控制稻田杂草。
T0377 Clofazimine

NSC-141046,氯法齐明,氯苯吩嗪

DNA; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料,与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。
T8311 Obefazimod

ABX-464,ABX464

HIV Protease Microbiology/Virology; Proteases/Proteasome
Obefazimod (ABX-464) 是一种抗HIV 剂。它抑制受刺激的外周血单核细胞中的 HIV-1 复制,IC50值为 0.1 μM 至 0.5 μM。
T68168L (2E,2'E)-Upenazime

Others Others
Upenazime 是诊断成像的非放射性的前体试剂。
TQ0167 Zimlovisertib

PF-06650833,PF06650833

IRAK Immunology/Inflammation; NF-κB
Zimlovisertib (PF-06650833) 是口服有活性的、可生物利用的白介素-1 受体相关激酶 4 (IRAK4) 选择性抑制剂,其IC50=0.2 nM,在 PBMC 分析中,IC50=2.4 nM。它具有研究类淋巴瘤、风湿性关节炎、狼疮等疾病的潜力。
T3124 Carbendazim

Bavistin,Carbendazole,多菌灵,Mercarzole

Antifungal Microbiology/Virology
Carbendazim (Mercarzole) 是一种具有抗肿瘤活性的苯并咪唑衍生物,可用于癌症研究。它是一种口服广谱苯并咪唑杀菌剂,可作为真菌疾病研究的杀虫剂。
T7478 2-Chloro-1-(4-fluorobenzyl)benzimidazole

Reductase Endocrinology/Hormones; Metabolism
2-Chloro-1-(4-fluorobenzyl)benzimidazole 是醛糖还原酶 (ALR2) 的抑制剂。
T14922 Cefodizime

Antibacterial; Antibiotic Microbiology/Virology
Cefodizime 是一种新型头孢菌素抗生素,具有广泛的生物活性。Cefodizime 对肾脏没有毒性且具有良好的耐受性和免疫调节活性,具有抗菌活性,可用于研究呼吸系统和泌尿系统的严重感染。
T0662 2-Hydroxybenzimidazole

2-Benzimidazolinone,2-羟基苯并咪唑

Others Others
2-Hydroxybenzimidazole (2-Benzimidazolinone) 在工业上用作中间体。
T31810 Flubenzimine

Cropotex,BAY slj 0312,EINECS 253-703-1,BRN 2403690

Others Others
Flubenzimine is a bio-active chemical. Detailed information has not been published.
T21642 4,5,6,7-Tetrabromobenzimidazole

Others Others
4,5,6,7-Tetrabromo-1H-benzimidazole 是一种酪蛋白激酶 2(CK2)的选择性和 ATP 竞争性抑制剂。
T69002 Zimeldine hydrochloride hydrate

Others Others
Zimeldine hydrochloride hydrate is a serotonin uptake inhibitor that was formerly used for depression but was withdrawn worldwide in September 1983 because of the risk of Guillain-Barre Syndrome associated with its use.
T26072 Rhazimine

Others Others
Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation.
T74747 Tamuzimod

Others Others
Tamuzimod 是一个强大的免疫调节剂.Tamuzimod 具有S1P 受体调节活性乙C50小于 1μ米。
T67503 5-Methoxy-2-benzimidazolethiol

Others Others
5-Methoxy-2-benzimidazolethiol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67503,CAS号为 37052-78-1。
T29216 Zimelidine

A23140,A 23140,A-23140

Others Others
Zimelidine is a serotonin uptake inhibitor formerly used for depression, but was withdrawn worldwide because of the risk of Gullain-Barre syndrome associated with its use.
T76709 Zimberelimab

Zimberelimab 是一种全人源IgG4抗PD-1单克隆抗体,具有很高的亲和力和选择性。 Zimberelimab 具有抗肿瘤活性,可用于各种癌症研究,包括宫颈癌、非小细胞肺癌和霍奇金淋巴瘤。
T30739 Carbendazim mixture with flusilazole

Others Others
Carbendazim mixture with flusilazole is a bioactive chemical.
T24713 Zimet 38-74

Zimet 38-74,Zimet 38-74;Z 38-74,Z 38-74

Others Others
Zimet 38-74 is an agent of antiviral.
T64402 4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide hydrochloride

Others Others
4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64402,CAS号为 2331268-15-4。
T81718 N-[4-(2-Benzimidazolyl)phenyl]maleimide

N-[4-(2-Benzimidazolyl)phenyl]maleimide,作为荧光探针,具有315 nm的最大激发波长和360 nm的最大发射波长。该化合物适用于对硫醇类化合物进行荧光检测。
T23560 Zimelidine dihydrochloride

Others Others
5-HT re-uptake inhibitor
T3124L Carbendazim HCl

Lignasan,Carbendazim hydrochloride,Sandomil P

Others Others
Carbendazim HCl is a widely used, broad-spectrum benzimidazole fungicide and a metabolite of benomyl.
T68168 upenazime

Others Others
upenazime 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T68168,CAS号为 95268-62-5。
T25307 Denzimol hydrochloride

REC 15-1533

Others Others
Denzimol hydrochloride 是一种新型抗惊厥药物,能抑制电性和化学性诱发的强直性癫痫发作,但不能阻止阵挛性癫痫发作。其表现与苯妥英和卡马西平相似,但与巴比妥类和苯二氮卓类不同。
T22594 Azimilide

Others Others
class III anti-arrhythmic drug

化合物

ZIM
Cat.No: T72024
Synonym:
Target: Others
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde
Cat.No: T4239
Synonym: 1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOLE-5-CARBALDEHYDE
Target: Others
Capzimin
Cat.No: T10672
Synonym:
Target: Others
Azimilide Dihydrochloride
Cat.No: T7505
Synonym: NE-10064 Dihydrochloride,盐酸阿齐利特
Target: Potassium Channel
Denzimol
Cat.No: T68054
Synonym:
Target: Others
2-(2-Hydroxyphenyl)-1H-benzimidazole
Cat.No: T9152
Synonym:
Target: Others
2-(Trifluoromethyl)benzimidazole
Cat.No: Fr12535
Synonym:
Target: Others
Azimsulfuron
Cat.No: T19749
Synonym: A 8947,A8947,A-8947
Target: Others
Clofazimine
Cat.No: T0377
Synonym: NSC-141046,氯法齐明,氯苯吩嗪
Target: DNA, Antibacterial, Antibiotic
Obefazimod
Cat.No: T8311
Synonym: ABX-464,ABX464
Target: HIV Protease
(2E,2'E)-Upenazime
Cat.No: T68168L
Synonym:
Target: Others
Zimlovisertib
Cat.No: TQ0167
Synonym: PF-06650833,PF06650833
Target: IRAK
Carbendazim
Cat.No: T3124
Synonym: Bavistin,Carbendazole,多菌灵,Mercarzole
Target: Antifungal
2-Chloro-1-(4-fluorobenzyl)benzimidazole
Cat.No: T7478
Synonym:
Target: Reductase
Cefodizime
Cat.No: T14922
Synonym:
Target: Antibacterial, Antibiotic
2-Hydroxybenzimidazole
Cat.No: T0662
Synonym: 2-Benzimidazolinone,2-羟基苯并咪唑
Target: Others
Flubenzimine
Cat.No: T31810
Synonym: Cropotex,BAY slj 0312,EINECS 253-703-1,BRN 2403690
Target: Others
4,5,6,7-Tetrabromobenzimidazole
Cat.No: T21642
Synonym:
Target: Others
Zimeldine hydrochloride hydrate
Cat.No: T69002
Synonym:
Target: Others
Rhazimine
Cat.No: T26072
Synonym:
Target: Others
Tamuzimod
Cat.No: T74747
Synonym:
Target: Others
5-Methoxy-2-benzimidazolethiol
Cat.No: T67503
Synonym:
Target: Others
Zimelidine
Cat.No: T29216
Synonym: A23140,A 23140,A-23140
Target: Others
Zimberelimab
Cat.No: T76709
Synonym:
Target:
Carbendazim mixture with flusilazole
Cat.No: T30739
Synonym:
Target: Others
Zimet 38-74
Cat.No: T24713
Synonym: Zimet 38-74,Zimet 38-74;Z 38-74,Z 38-74
Target: Others
4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide hydrochloride
Cat.No: T64402
Synonym:
Target: Others
N-[4-(2-Benzimidazolyl)phenyl]maleimide
Cat.No: T81718
Synonym:
Target:
Zimelidine dihydrochloride
Cat.No: T23560
Synonym:
Target: Others
Carbendazim HCl
Cat.No: T3124L
Synonym: Lignasan,Carbendazim hydrochloride,Sandomil P
Target: Others
upenazime
Cat.No: T68168
Synonym:
Target: Others
Denzimol hydrochloride
Cat.No: T25307
Synonym: REC 15-1533
Target: Others
Azimilide
Cat.No: T22594
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T8126 Cefodizime Sodium

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefodizime sodium 是一种头孢菌素抗生素,具有抗菌活性。它对肾脏没有毒性,具有良好的耐受性和免疫调节活性,可研究呼吸道和泌尿道的严重感染。
T38675 Hikizimycin

Anthelmycin

Others Others
Hikizimycin is a potent anthelmintic and antibacterial natural product.
TN4652 Niazimicin

NF-κB; PI3K; AChR; Antifection Microbiology/Virology; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in the two-stage carcinogenesis in mouse skin using 7,12-dimethylbenz(a)anthracene (DMBA) as ini

天然产物

Cefodizime Sodium
Cat.No: T8126
Synonym:
Target: Others, Antibacterial, Antibiotic
Hikizimycin
Cat.No: T38675
Synonym: Anthelmycin
Target: Others
Niazimicin
Cat.No: TN4652
Synonym:
Target: NF-κB, PI3K, AChR, Antifection
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