33
3
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T72024 |
ZIM
|
Others | Others |
ZIM,一种从4-Aminoantipyrine衍生的降冰片烯,有效诱导DNA损伤,造成基因组及染色体损害,进而引发细胞死亡和激活吞噬。其化疗潜力适用于癌症研究。 | |||
T4239 |
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde
1,3-DIMETHYL-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOLE-5-CARBALDEHYDE |
Others | Others |
1,3-dimethyl-2-oxobenzimidazole-5-carbaldehyde 是中间体。 | |||
T10672 |
Capzimin
|
Others | Others |
Capzimin 是蛋白酶体异肽酶 Rpn11 的选择性抑制剂。 | |||
T7505 |
Azimilide Dihydrochloride
NE-10064 Dihydrochloride,盐酸阿齐利特 |
Potassium Channel | Membrane transporter/Ion channel |
Azimilide Dihydrochloride (NE-10064 Dihydrochloride) 是 I(Ks) 和 I(Kr) 抑制剂,具有抗心律失常活性。 | |||
T68054 |
Denzimol
|
Others | Others |
Denzimol 是一种新型抗惊厥化合物。Denzimol 对强直性癫痫发作具有选择性。 | |||
T9152 |
2-(2-Hydroxyphenyl)-1H-benzimidazole
|
Others | Others |
2-(2-Hydroxyphenyl)-1H-benzimidazole 已被用于合成聚合物和其他材料的催化剂。 | |||
Fr12535 |
2-(Trifluoromethyl)benzimidazole
|
Others | Others |
Compound Fr12535 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12535,CAS号为 312-73-2。 | |||
T19749 |
Azimsulfuron
A 8947,A8947,A-8947 |
Others | Others |
Azimsulfuron 是一种除草剂,可用于控制稻田杂草。 | |||
T0377 |
Clofazimine
NSC-141046,氯法齐明,氯苯吩嗪 |
DNA; Antibacterial; Antibiotic | DNA Damage/DNA Repair; Microbiology/Virology |
Clofazimine (NSC-141046) 是一种具有显著的抗炎效果的亚氨基酚嗪类染料,与其它抗分支杆菌药物联用来治疗AIDS 和克罗恩病。 | |||
T8311 |
Obefazimod
ABX-464,ABX464 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Obefazimod (ABX-464) 是一种抗HIV 剂。它抑制受刺激的外周血单核细胞中的 HIV-1 复制,IC50值为 0.1 μM 至 0.5 μM。 | |||
T68168L |
(2E,2'E)-Upenazime
|
Others | Others |
Upenazime 是诊断成像的非放射性的前体试剂。 | |||
TQ0167 |
Zimlovisertib
PF-06650833,PF06650833 |
IRAK | Immunology/Inflammation; NF-κB |
Zimlovisertib (PF-06650833) 是口服有活性的、可生物利用的白介素-1 受体相关激酶 4 (IRAK4) 选择性抑制剂,其IC50=0.2 nM,在 PBMC 分析中,IC50=2.4 nM。它具有研究类淋巴瘤、风湿性关节炎、狼疮等疾病的潜力。 | |||
T3124 |
Carbendazim
Bavistin,Carbendazole,多菌灵,Mercarzole |
Antifungal | Microbiology/Virology |
Carbendazim (Mercarzole) 是一种具有抗肿瘤活性的苯并咪唑衍生物,可用于癌症研究。它是一种口服广谱苯并咪唑杀菌剂,可作为真菌疾病研究的杀虫剂。 | |||
T7478 |
2-Chloro-1-(4-fluorobenzyl)benzimidazole
|
Reductase | Endocrinology/Hormones; Metabolism |
2-Chloro-1-(4-fluorobenzyl)benzimidazole 是醛糖还原酶 (ALR2) 的抑制剂。 | |||
T14922 |
Cefodizime
|
Antibacterial; Antibiotic | Microbiology/Virology |
Cefodizime 是一种新型头孢菌素抗生素,具有广泛的生物活性。Cefodizime 对肾脏没有毒性且具有良好的耐受性和免疫调节活性,具有抗菌活性,可用于研究呼吸系统和泌尿系统的严重感染。 | |||
T0662 |
2-Hydroxybenzimidazole
2-Benzimidazolinone,2-羟基苯并咪唑 |
Others | Others |
2-Hydroxybenzimidazole (2-Benzimidazolinone) 在工业上用作中间体。 | |||
T31810 |
Flubenzimine
Cropotex,BAY slj 0312,EINECS 253-703-1,BRN 2403690 |
Others | Others |
Flubenzimine is a bio-active chemical. Detailed information has not been published. | |||
T21642 |
4,5,6,7-Tetrabromobenzimidazole
|
Others | Others |
4,5,6,7-Tetrabromo-1H-benzimidazole 是一种酪蛋白激酶 2(CK2)的选择性和 ATP 竞争性抑制剂。 | |||
T69002 |
Zimeldine hydrochloride hydrate
|
Others | Others |
Zimeldine hydrochloride hydrate is a serotonin uptake inhibitor that was formerly used for depression but was withdrawn worldwide in September 1983 because of the risk of Guillain-Barre Syndrome associated with its use. | |||
T26072 |
Rhazimine
|
Others | Others |
Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation. | |||
T74747 |
Tamuzimod
|
Others | Others |
Tamuzimod 是一个强大的免疫调节剂.Tamuzimod 具有S1P 受体调节活性乙C50小于 1μ米。 | |||
T67503 |
5-Methoxy-2-benzimidazolethiol
|
Others | Others |
5-Methoxy-2-benzimidazolethiol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T67503,CAS号为 37052-78-1。 | |||
T29216 |
Zimelidine
A23140,A 23140,A-23140 |
Others | Others |
Zimelidine is a serotonin uptake inhibitor formerly used for depression, but was withdrawn worldwide because of the risk of Gullain-Barre syndrome associated with its use. | |||
T76709 | Zimberelimab | ||
Zimberelimab 是一种全人源IgG4抗PD-1单克隆抗体,具有很高的亲和力和选择性。 Zimberelimab 具有抗肿瘤活性,可用于各种癌症研究,包括宫颈癌、非小细胞肺癌和霍奇金淋巴瘤。 | |||
T30739 |
Carbendazim mixture with flusilazole
|
Others | Others |
Carbendazim mixture with flusilazole is a bioactive chemical. | |||
T24713 |
Zimet 38-74
Zimet 38-74,Zimet 38-74;Z 38-74,Z 38-74 |
Others | Others |
Zimet 38-74 is an agent of antiviral. | |||
T64402 |
4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide hydrochloride
|
Others | Others |
4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide hydrochloride 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T64402,CAS号为 2331268-15-4。 | |||
T81718 |
N-[4-(2-Benzimidazolyl)phenyl]maleimide
|
||
N-[4-(2-Benzimidazolyl)phenyl]maleimide,作为荧光探针,具有315 nm的最大激发波长和360 nm的最大发射波长。该化合物适用于对硫醇类化合物进行荧光检测。 | |||
T23560 |
Zimelidine dihydrochloride
|
Others | Others |
5-HT re-uptake inhibitor | |||
T3124L |
Carbendazim HCl
Lignasan,Carbendazim hydrochloride,Sandomil P |
Others | Others |
Carbendazim HCl is a widely used, broad-spectrum benzimidazole fungicide and a metabolite of benomyl. | |||
T68168 |
upenazime
|
Others | Others |
upenazime 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T68168,CAS号为 95268-62-5。 | |||
T25307 |
Denzimol hydrochloride
REC 15-1533 |
Others | Others |
Denzimol hydrochloride 是一种新型抗惊厥药物,能抑制电性和化学性诱发的强直性癫痫发作,但不能阻止阵挛性癫痫发作。其表现与苯妥英和卡马西平相似,但与巴比妥类和苯二氮卓类不同。 | |||
T22594 |
Azimilide
|
Others | Others |
class III anti-arrhythmic drug |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8126 |
Cefodizime Sodium
|
Others; Antibacterial; Antibiotic | Microbiology/Virology; Others |
Cefodizime sodium 是一种头孢菌素抗生素,具有抗菌活性。它对肾脏没有毒性,具有良好的耐受性和免疫调节活性,可研究呼吸道和泌尿道的严重感染。 | |||
T38675 |
Hikizimycin
Anthelmycin |
Others | Others |
Hikizimycin is a potent anthelmintic and antibacterial natural product. | |||
TN4652 |
Niazimicin
|
NF-κB; PI3K; AChR; Antifection | Microbiology/Virology; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling |
Niazimicin are NF-B and PI3K inhibitors, which shows antimicrobial, hypotensive and spasmolytic activities. Niazimicin has potent antitumor promoting activity in the two-stage carcinogenesis in mouse skin using 7,12-dimethylbenz(a)anthracene (DMBA) as ini |