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Search Results for " yap "
Targets Recommended: YAP YAP

37

抑制剂 & 化合物

10

天然产物

6

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T13364 YAP/TAZ inhibitor-1

YAP Stem Cells
YAP/TAZ inhibitor-1 是一种 YAP/TAZ 抑制剂(IC50 <0.100 μΜ),可用于研究免疫功能异常和癌症。
TP2160L1 YAP-TEAD-IN-1 acetate

YAP-TEAD-IN-1 acetate (1659305-78-8 Free base)

YAP Stem Cells
YAP-TEAD-IN-1 acetate 是一种有效的、竞争性的 YAP-TEAD 相互作用抑制剂,IC50 为 25 nM。
T60218 YAP/TAZ inhibitor-2 

YAP Stem Cells
YAP/TAZ inhibitor-2 是一种有效的具有口服活性的TEAD-YAP/TAZ 抑制剂,EC50值为 3 nM。YAP/TAZ inhibitor-2 具有抗增殖和抗肿瘤活性。
T77725 YAP-TEAD-IN-3

IAG933

YAP Stem Cells
YAP-TEAD-IN-3 是 YAP/TAZ-TEAD 相互作用的抑制剂,对于 Avi-人 TEAD4217-434 的 IC50 为 9 nM。 YAP-TEAD-IN-3 抑制 YAP 报告基因表达 (IC50 = 0.048 μM) 和 NCI-H2052 细胞增殖 (IC50 = 0.048 μM)。
TP2160 YAP-TEAD-IN-1

Others Others
YAP-TEAD-IN-1 is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TEAD1 (Kd: 15 nM) than YAP (50-171) (Kd: 40 nM).
TP2160L YAP-TEAD-IN-1 TFA

Others Others
YAP-TEAD-IN-1 TFA is a competitive inhibitor of YAP–TEAD interaction (IC50: 25 nM). It shows a higher binding affinity to TEAD1 (Kd: 15 nM) than YAP (50-171) (Kd: 40 nM).
T72888 YAP-TEAD-IN-2

YAP Stem Cells
YAP-TEAD-IN-2 (化合物6)作为一种YAP-TEAD PPI抑制剂,表现出高效性,其半抑制浓度(IC50)仅为2.7 nM。
T9053 Lats-IN-1

Others; YAP Others; Stem Cells
Lats-IN-1 是一种 ATP 竞争性的、高效的Lats1和Lats2激酶抑制剂,能促进有丝分裂后哺乳动物组织的 Yap 依赖性增殖。
T22372 MYF-01-37

1-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one

Others; YAP Others; Stem Cells
MYF-01-37 (1-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one) 是共价TEAD 抑制剂,靶向 Cys380,能够可逆地抑制 YAP/TEAD 相互作用。
T8421 TED-347

YAP Stem Cells
TED-347 是不可逆的、共价的 YAP-TEAD 蛋白质-蛋白质相互作用变构抑制剂,对 TEAD4•Yap1 蛋白质-蛋白质相互作用的 EC50为 5.9 μM。它与 TEAD4 中央口袋内的 Cys-367 特异性共价结合(Ki:10.3 μM)。它可以抑制 TEAD 的转录活性,并且具有抗肿瘤作用。
T9954 K-975

Others Others
K-975是一种高选择性的具有口服活性的TEAD 抑制剂,可有效抑制TEAD 和YAP1/TAZ 之间的蛋白质-蛋白质相互作用。
T3050 ML-7 hydrochloride

ML-7 HCl,ML-7盐酸盐

Serine/threonin kinase; Myosin; YAP; PKA; PKC Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
ML-7 hydrochloride (ML-7 HCl) 是一种可渗透细胞的、可逆的、有效的、ATP 竞争性的肌球蛋白轻链激酶(MLCK) 特异性抑制剂,IC50为300 nM。它还抑制平滑肌肌球蛋白轻链激酶、PKA 和 PKC。
T3112 Verteporfin

维替泊芬,BPD-MA,CL 318952

Apoptosis; YAP; VDA; Autophagy Angiogenesis; Apoptosis; Autophagy; Stem Cells
Verteporfin (BPD-MA) 是一种 YAP 抑制剂,抑制 YAP-TEAD 相互作用。Verteporfin 也是一种光敏剂,用于光动力疗法。Verteporfin 还可以诱导细胞凋亡,抑制自噬。
T1477 AICAR

NSC105823,AICA Riboside,Acadesine,阿卡地新,AICAR (Acadesine)

Mitophagy; YAP; AMPK; Autophagy Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
AICAR (NSC105823) 是一种腺苷类似物,是一种 AMP 激活的蛋白激酶激活剂,可用于治疗急性淋巴细胞白血病和糖尿病。
T2008 LY294002

LY 294002,NSC 697286,SF 1101

Apoptosis; DNA-PK; Casein Kinase; PI3K; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
LY294002 (SF 1101) 是一种 PI3K 的广谱抑制剂,抑制 PI3Kα、PI3Kδ 和 PI3Kβ (IC50=0.5/0.57/0.97 μM)。LY294002 也是 DNA-PK 抑制剂 (IC50=1.4 μM) 和 CK2 抑制剂 (IC50=98 nM)。LY294002 可以激活凋亡和自噬。
T7038 4-Methylayapin

4-甲基-6,7-亚甲基二氧代香豆素,4-METHYL-6,7-METHYLENEDIOXYCOUMARIN

Others Others
4-Methylayapin 用作中间体。
T9566 PY-60

Annexin A; YAP GPCR/G Protein; Stem Cells
PY-60 有效激活针对膜联蛋白 A2 (Kd = 1.4 µM) 的 YAP 转录活性。 PY-60 在能够通过增殖重塑表皮的成年动物中激活促增殖、依赖于 YAP 的转录程序。
T77729 MY-1076

Apoptosis; YAP Apoptosis; Stem Cells
MY-1076 是一种高效的 YAP 抑制剂,具有抗胃癌活性。MY-1076 剂量依赖性诱导G2/M期阻滞,诱导 YAP 降解和细胞凋亡,抑制微管蛋白聚合。MY-1076 抑制 MGC-803、SGC-7901、HCT-116 和 KYSE450 细胞增殖。
T62077 VT103

VT-103,VT 103

YAP Stem Cells
VT103 是一种具有口服活性和选择性的 TEAD1 蛋白棕榈酰化抑制剂,是 VT101 的类似物。 VT103 有潜在的抗肿瘤活性,可抑制 YAP/TAZ-TEAD 促进的基因转录,阻断 TEAD auto-palmitoylation,阻断 YAP/TAZ和TEAD 之间的相互作用。VT103 可用于研究HER2阳性乳腺癌、前列腺癌和三阴性乳腺癌。
T78558 GNE-7883

GNE 7883,GNE7883

YAP Stem Cells
GNE-7883是一种靶向 TEAD 转录因子的抑制剂,抑制细胞增殖,抑制YAP/TAZ的激活,可用于研究YAP/TAZ依赖型肿瘤。
T67872 VT104

YAP Stem Cells
VT104是一种有效的YAP/TAZ 抑制剂,具有口服活性,可用于癌症研究。VT104阻止内源性TEAD1和TEAD3蛋白棕榈酰化。
T69760 TT-10

TAZ-K

YAP Stem Cells
TT-10 (TAZ-K) 作为YES相关蛋白(YAP)-转录增强因子结构域(TEAD)活性的激活剂,适用于心肌细胞丢失伴随心脏病研究。
T60144 TDI-011536

Others Others
TDI-011536 是一种有效的 Lats 激酶抑制剂,能中断 Hippo-Yap 的信号传导,并可启动受损心肌细胞的增殖。TDI-011536 可用于研究器官的保护和再生。
T14997 Conteltinib

SY-707,CT-707

FAK; PYK2; ALK Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Conteltinib (CT-707) 是一种靶向FAK、ALK 和 Pyk2 的酶抑制剂,具有抗肿瘤活性。Conteltinib 对 FAK 有明显的抑制作用,通过抑制 YAP 信号传导来克服肝细胞癌中缺氧介导的索拉非尼耐药性,可用于晚期 ALK 阳性非小细胞肺癌和淋巴癌。
T60148 MSC-4106

YAP Stem Cells
MSC-4106 是一种有效的、具有口服活性的 YAP/TAZ-TEAD 抑制剂。 MSC-4106 阻断 TEAD1 和 TEAD3 的自棕榈酰化,并且对 NCI-H226 异种移植瘤模型显示抑制作用。
T60013 GA-017

Others Others
GA-017是一种有效的选择性 LATS1和 LATS2(大型肿瘤抑制激酶 1/2) 抑制剂,其 IC50值分别为 4.10 和 3.92 nM。GA-017 是细胞增殖的激活剂。GA-017 促进 YAP/TAZ 激活和核转位。GA-017 在 3D 培养条件下促进细胞生长。GA-017 增强小鼠肠道类器官的离体形成。
T6108 Ki16425

Debio 0719

LPA Receptor; LPL Receptor GPCR/G Protein
Ki16425 (Debio 0719) 是一种竞争性、有效和可逆的 LPA1、LPA2 和 LPA3 拮抗剂,Ki 分别为 0.34、6.5 和 0.93 μM。它可抑制LPA 诱导的 HEK293A 细胞中 YAP/TAZ 的去磷酸化,降低LPA 诱导的 p42/p44 MAPK 激活。
T76004 Super-TDU TFA

Super-TDU TFA 是一种特异性的 YAP 拮抗剂,可以靶向 YAP-TEAD 相互作用。Super-TDU TFA 可以抑制胃癌小鼠模型的肿瘤生长。
TP1569 Super-TDU (TFA) (1599441-71-0 free base)

Super-TDU (TFA)

uper-TDU is an inhibitory peptide targeting YAP-TEADs interaction.
T22434 Super-TDU

Others Others
Super-TDU, an inhibitory peptide, targets YAP-TEADs interaction.
T83951 TM2 TEAD inhibitor

Others Others
TM2 TEAD抑制剂是一种有效并且可逆的TEA领域转录因子抑制剂(IC50为TEAD4自动棕榈酰化和TEAD2棕榈酰化分别为38 nM和156 nM)。它抑制TEAD-YAP的结合和转录活性。TM2 TEAD抑制剂在YAP依赖型癌症细胞中,无论是单独使用还是与MEK抑制剂联合使用,都显示出强大的抗增殖效果。同时抑制体外YAP依赖的肝脏类器官生长。
T81056 SWTX-143

YAP Stem Cells
SWTX-143,一新型共价YAP/TAZ-TEAD 抑制剂,能结合四种TEAD亚型的棕榈酰化口袋。SWTX-143特异性、不可逆地抑制YAP/TAZ-TEAD转录活性,表现出抗肿瘤活性。
TP1383 Super-TDU 1-31

Super-TDU (1-31) is a peptide of Super-TDU, which is an inhibitor of YAP-TEADs, shows potent anti-tumor activity.
T82165 HTH-02-006

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
HTH-02-006,一种NUAK2抑制剂(IC50 = 126 nM),能够降低HuCCT-1细胞中磷酸化MYPT1水平,并抑制YAP驱动的细胞增殖、肝肿大和肿瘤发生,同时具备抗纤维化保护效果。
T76005 Super-TDU (1-31)

Super-TDU (1-31) 是 Super-TDU 的肽片段。Super-TDU (1-31) 是 YAP-TEAD 复合物的抑制剂。Super-TDU 在胃癌小鼠模型中显示出有效的抗肿瘤活性并抑制肿瘤生长。
T83938 TAT-PDHPS1

Others Others
TAT-PDHPS1是一种针对Yes-associated protein (YAP) 信号的肽抑制剂。它由内源性肽PDHPS1和能穿透细胞的肽序列TAT组成。PDHPS1与蛋白磷酸酶2磷酸酶激活因子(PTPA)结合, 激活蛋白磷酸酶2A (PP2A)。该激活促进YAP的磷酸化和抑制YAP靶向基因的表达。TAT-PDHPS1能够抑制体外卵巢癌细胞的增殖和小鼠皮下异种移植肿瘤模型中的卵巢肿瘤生长。
T76005L Super-TDU (1-31) (TFA)

Super-TDU (1-31) TFA 是 Super-TDU 的肽片段。Super-TDU (1-31) TFA 是YAP-TEAD 复合物的抑制剂。Super-TDU TFA 在胃癌小鼠模型中显示出有效的抗肿瘤活性并抑制肿瘤生长。

化合物

YAP/TAZ inhibitor-1
Cat.No: T13364
Synonym:
Target: YAP
YAP-TEAD-IN-1 acetate
Cat.No: TP2160L1
Synonym: YAP-TEAD-IN-1 acetate (1659305-78-8 Free base)
Target: YAP
YAP/TAZ inhibitor-2 
Cat.No: T60218
Synonym:
Target: YAP
YAP-TEAD-IN-3
Cat.No: T77725
Synonym: IAG933
Target: YAP
YAP-TEAD-IN-1
Cat.No: TP2160
Synonym:
Target: Others
YAP-TEAD-IN-1 TFA
Cat.No: TP2160L
Synonym:
Target: Others
YAP-TEAD-IN-2
Cat.No: T72888
Synonym:
Target: YAP
Lats-IN-1
Cat.No: T9053
Synonym:
Target: Others, YAP
MYF-01-37
Cat.No: T22372
Synonym: 1-[3-Methyl-3-[3-(trifluoromethyl)anilino]pyrrolidin-1-yl]prop-2-en-1-one
Target: Others, YAP
TED-347
Cat.No: T8421
Synonym:
Target: YAP
K-975
Cat.No: T9954
Synonym:
Target: Others
ML-7 hydrochloride
Cat.No: T3050
Synonym: ML-7 HCl,ML-7盐酸盐
Target: Serine/threonin kinase, Myosin, YAP, PKA, PKC
Verteporfin
Cat.No: T3112
Synonym: 维替泊芬,BPD-MA,CL 318952
Target: Apoptosis, YAP, VDA, Autophagy
AICAR
Cat.No: T1477
Synonym: NSC105823,AICA Riboside,Acadesine,阿卡地新,AICAR (Acadesine)
Target: Mitophagy, YAP, AMPK, Autophagy
LY294002
Cat.No: T2008
Synonym: LY 294002,NSC 697286,SF 1101
Target: Apoptosis, DNA-PK, Casein Kinase, PI3K, Autophagy
4-Methylayapin
Cat.No: T7038
Synonym: 4-甲基-6,7-亚甲基二氧代香豆素,4-METHYL-6,7-METHYLENEDIOXYCOUMARIN
Target: Others
PY-60
Cat.No: T9566
Synonym:
Target: Annexin A, YAP
MY-1076
Cat.No: T77729
Synonym:
Target: Apoptosis, YAP
VT103
Cat.No: T62077
Synonym: VT-103,VT 103
Target: YAP
GNE-7883
Cat.No: T78558
Synonym: GNE 7883,GNE7883
Target: YAP
VT104
Cat.No: T67872
Synonym:
Target: YAP
TT-10
Cat.No: T69760
Synonym: TAZ-K
Target: YAP
TDI-011536
Cat.No: T60144
Synonym:
Target: Others
Conteltinib
Cat.No: T14997
Synonym: SY-707,CT-707
Target: FAK, PYK2, ALK
MSC-4106
Cat.No: T60148
Synonym:
Target: YAP
GA-017
Cat.No: T60013
Synonym:
Target: Others
Ki16425
Cat.No: T6108
Synonym: Debio 0719
Target: LPA Receptor, LPL Receptor
Super-TDU TFA
Cat.No: T76004
Synonym:
Target:
Super-TDU (TFA) (1599441-71-0 free base)
Cat.No: TP1569
Synonym: Super-TDU (TFA)
Target:
Super-TDU
Cat.No: T22434
Synonym:
Target: Others
TM2 TEAD inhibitor
Cat.No: T83951
Synonym:
Target: Others
SWTX-143
Cat.No: T81056
Synonym:
Target: YAP
Super-TDU 1-31
Cat.No: TP1383
Synonym:
Target:
HTH-02-006
Cat.No: T82165
Synonym:
Target: AMPK
Super-TDU (1-31)
Cat.No: T76005
Synonym:
Target:
TAT-PDHPS1
Cat.No: T83938
Synonym:
Target: Others
Super-TDU (1-31) (TFA)
Cat.No: T76005L
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2353 8-Hydroxyapigenin

Isoscutellarein

Antioxidant; Influenza Virus Microbiology/Virology; oxidation-reduction
8-Hydroxyapigenin (Isoscutellarein) 是从植物黄芩中提取的黄铜类化合物,具有抗炎抗氧和抗流感病毒的活性。
TN1489 3'-Methoxyapiin

Graveobioside B,3'-Methoxy apiin,Chrysoeriol 7-apiosylglucoside,3'-甲氧基芹菜苷

Others Others
3'-Methoxyapiin (Graveobioside B) 是一种来自 Eminium spiculatum 植物的类黄酮。
TN2422 6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide

Others Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide is a natural product from Carthamus tinctorius Linn.
TN2907 3,6-Dimethoxyapigenin

Others Others
3,6-Dimethoxyapigenin是一种天然产物,属于无患子科车桑子属,其产品编号为 TN2907,CAS号为 22697-65-0。3,6-Dimethoxyapigenin可用作对照参考。
TN1210 2-Hydroxy-1-Methoxyaporphine

P450 Metabolism
2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosiglitazone.
T79933 (−)-N-Hydroxyapiosporamide

NHAP

NF-κB NF-κB
(−)-N-Hydroxyapiosporamide (NHAP)为生物碱类NF-κB抑制剂,表现出体外及体内抗肿瘤活性,常用于结直肠癌(CRC)研究。
T83410 2,3,5,6-Tetramethoxyaporphine

2,3,5,6-Tetramethoxyaporphine 是阿扑啡碱类化合物,具有止咳作用并具药用价值,可从黄角罂粟(Glaucium flavum Cr.,罂粟科)中提取。
T14149 AICAR phosphate

AICA Riboside phosphate,Acadesine phosphate

Mitophagy; NOS; YAP; AMPK Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; PI3K/Akt/mTOR signaling; Stem Cells
AICAR phosphate (Acadesine phosphate) 是 AMPK 激活剂且是自噬、YAP 和 mitophagy 抑制剂,也是一种腺苷类似物, 可调节糖代谢和脂代谢,抑制促炎细胞因子和 iNOS 的产生。
T1679 Thiostrepton

Thiactin,Bryamycin,Alaninamide,硫链丝菌素

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。
T3S1416 Decursin

Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素

Apoptosis; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
Decursin (Decursinol angelate) 是一种细胞毒性剂,是一种来自朝鲜当归根的有效蛋白激酶 C 激活剂。它通过 Hippo/YAP 信号通路抑制 HepG2 细胞的生长。它通过下调 CXCR7 表达来抑制胃癌中的肿瘤生长,迁移和侵袭。

天然产物

8-Hydroxyapigenin
Cat.No: TN2353
Synonym: Isoscutellarein
Target: Antioxidant, Influenza Virus
3'-Methoxyapiin
Cat.No: TN1489
Synonym: Graveobioside B,3'-Methoxy apiin,Chrysoeriol 7-apiosylglucoside,3'-甲氧基芹菜苷
Target: Others
6-hydroxyapigenin-6-O-β-D-glucoside-7-O-β-D-glucuronide
Cat.No: TN2422
Synonym:
Target: Others
3,6-Dimethoxyapigenin
Cat.No: TN2907
Synonym:
Target: Others
2-Hydroxy-1-Methoxyaporphine
Cat.No: TN1210
Synonym:
Target: P450
(−)-N-Hydroxyapiosporamide
Cat.No: T79933
Synonym: NHAP
Target: NF-κB
2,3,5,6-Tetramethoxyaporphine
Cat.No: T83410
Synonym:
Target:
AICAR phosphate
Cat.No: T14149
Synonym: AICA Riboside phosphate,Acadesine phosphate
Target: Mitophagy, NOS, YAP, AMPK
Thiostrepton
Cat.No: T1679
Synonym: Thiactin,Bryamycin,Alaninamide,硫链丝菌素
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Decursin
Cat.No: T3S1416
Synonym: Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素
Target: Apoptosis, PKC
Cat. No. Product Name Species Expression System
TMPH-03764 YAP1 Protein, Human, Recombinant (His)

YAP1-2gamma,YAP2L,YAP65

Human P. pastoris (Yeast)
Transcriptional regulator which can act both as a coactivator and a corepressor and is the critical downstream regulatory target in the Hippo signaling pathway that plays a pivotal role in organ size control and tumor suppression by restricting proliferation and promoting apoptosis. The core of this pathway is composed of a kinase cascade wherein STK3/MST2 and STK4/MST1, in complex with its regulatory protein SAV1, phosphorylates and activates LATS1/2 in complex with its regulatory protein MOB1,...
TMPH-00005 YAP1 Protein, Human, Recombinant (Isoform 9, His)

Protein yorkie homolog,YAP1,Yes-associated protein ...

Human P. pastoris (Yeast)
YAP1 Protein, Human, Recombinant (Isoform 9, His) is expressed in yeast with C-6xHis tag. The predicted molecular weight is 56.4 kDa; 80 kDa, reducing conditions and the accession number is P46937-9.
TMPY-02648 PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)

adenylate cyclase activating polypeptide 1 (pituitary) recep...

Human HEK293 Cells
Pituitary adenylate cyclase activating polypeptide (PACAP, Adcyap1) activation of PAC1 receptors ( Adcyap1r1) significantly increases excitability of guinea pig cardiac neurons. This modulation of excitability is mediated in part by plasma membrane G protein-dependent activation of adenylyl cyclase and downstream signaling cascades. Studies point to the potential role of the (pituitary) adenylate cyclase activating polypeptide receptor 1 (ADCYAP1R1) gene, which has been implicated in stress resp...
TMPY-06815 SYAP1 Protein, Human, Recombinant (His)

PRO3113,synapse associated protein 1

Human Baculovirus Insect Cells
Synapse-associated protein 1 (SYAP1), also known as PRO3113 and BSTA, belongs to the synapse-associated BSD domain family, featuring three α-helices and two conserved tryptophan and phenylalanine residues located at the C-terminus. Expressed near neuronal Golgi and synaptic regions of cerebellar Purkinje cells, SYAP1 has been linked to intact sensorimotor control and general vesicular trafficking in neurons. SYAP1-deficient mice display impaired locomotor activity. In cultured adipocytes, SYAP1 ...
TMPY-04398 MST1 Protein, Human, Recombinant (His)

serine/threonine kinase 4,KRS2,MST1,TIIAC,YSK3

Human Baculovirus Insect Cells
Dysregulation of MST1/STK4, a key kinase component of the Hippo-YAP pathway, is linked to the etiology of many cancers with poor prognosis. STK4/Hippo pathway may have important therapeutic implications for cancer. The tumor suppressor serine/threonine-protein kinase 4 (STK4) differentially regulates TLR3/4/9-mediated inflammatory responses in macrophages and thereby is protective against chronic inflammation-associated Hepatocellular carcinoma (HCC). STK4 has potential as a diagnostic biomarker...
TMPH-01689 PLD6 Protein, Human, Recombinant (His)

Mitochondrial phospholipase,Choline phosphatase 6,Protein zu...

Human E. coli
Presents phospholipase and nuclease activities, depending on the different physiological conditions. Interaction with Mitoguardin (MIGA1 or MIGA2) affects the dimer conformation, facilitating the lipase activity over the nuclease activity. Plays a key role in mitochondrial fusion and fission via its phospholipase activity. In its phospholipase role, it uses the mitochondrial lipid cardiolipin as substrate to generate phosphatidate (PA or 1,2-diacyl-sn-glycero-3-phosphate), a second messenger sig...

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YAP1 Protein, Human, Recombinant (His)
Cat.No: TMPH-03764
Species: Human
Expression System: P. pastoris (Yeast)
YAP1 Protein, Human, Recombinant (Isoform 9, His)
Cat.No: TMPH-00005
Species: Human
Expression System: P. pastoris (Yeast)
PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)
Cat.No: TMPY-02648
Species: Human
Expression System: HEK293 Cells
SYAP1 Protein, Human, Recombinant (His)
Cat.No: TMPY-06815
Species: Human
Expression System: Baculovirus Insect Cells
MST1 Protein, Human, Recombinant (His)
Cat.No: TMPY-04398
Species: Human
Expression System: Baculovirus Insect Cells
PLD6 Protein, Human, Recombinant (His)
Cat.No: TMPH-01689
Species: Human
Expression System: E. coli
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