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Search Results for " xii "
Targets Recommended: Potassium Channel

68

抑制剂 & 化合物

4

天然产物

14

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T80498 Jingzhaotoxin-XII

JzTx-XII

Potassium Channel Membrane transporter/Ion channel
Jingzhaotoxin-XII (JzTx-XII) 作为特异性 Kv4.1 通道抑制剂,表现出 0.363 μM 的 IC50 值,通过改变通道的门控行为来与其相互作用。
T21949 Calpain Inhibitor XII

Others Others
(Rac)-Calpain Inhibitor XII是一种可逆的,选择性抑制钙蛋白酶I(calpain I; μ-calpain)的化合物,具有19 nM的Ki值。其对钙蛋白酶II(calpain II; m-calpain; Ki=120 nM)和组织蛋白酶B(cathepsin B; Ki=750 nM)显示出较低的抑制亲和力。(Rac)-Calpain Inhibitor XII用于研究钙蛋白酶在多种生理过程中的角色,如嗜中性粒细胞趋化性、神经元信号传导和心脏对损伤的响应。
T125110 Eupteleasaponin XII

Others Others
Eupteleasaponin XII 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125110,CAS号为 290809-58-4。
T125868 RA-XII

Others Others
RA-XII 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125868,CAS号为 143343-98-0。
T17281 Z-Ile-Leu-aldehyde

Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII

Others Others
Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.
T79753 hCAIX/XII-IN-8

Carbonic Anhydrase Metabolism
hCAIX/XII-IN-8(compound 3g)是一种对人类(碳酸酐酶)CA IX和XII高效的抑制剂,Ki值分别为8.5和6.7 nM。该化合物对与肿瘤相关的膜结合异构体hCA IX和XII表现出显著的抑制作用,且相对于胞内异构体hCA I和II具有较高的选择性。
T61384 hCAIX/XII-IN-4

Others Others
hCAIX/XII-IN-4 (compound 6c) is a highly potent inhibitor of CAIX/XII. It exhibits Ki values of 4.5 nM, 23.6 nM, >10000 nM, and >10000 nM for CAXII, CAIX, CAI, and CAⅡ, respectively [1].
T72840 hCAIX/XII-IN-6

Others Others
hCAIX/XII-IN-6 是具有口服活性的碳酸酐酶(CA)抑制剂,能够抑制人体 CA 亚型 hCA I、II、IV、IX 及 XII,其 Ki 值分别为 6697 nM、2950 nM、4093 nM、4.1 nM 和 7.7 nM。适用于类风湿关节炎(RA)研究。
T25779 MDK-4683

MDK 4683,CA IX/XII Inhibitor

Others Others
MDK-4683, also known as CA IX/XII Inhibitor, is a hCA IX and hCA XII inhibitor.
T63400 hA2A/hCA XII modulator 1

Others Others
hA2A/hCA XII modulator 1 是 hA2A 腺苷受体 (hA2AAR) 的有效拮抗剂,是一种三唑并吡嗪, 能够作用于hA2AAR (Ki: 6.4 nM)、hA1AR (Ki: 4.819 μM)、hA3AR (Ki>30 μM)。hA2A/hCA XII modulator 1 也人碳酸酐酶 XII (hCA XII) 的有效抑制剂,能够作用于 hCA XII (Ki: 6.2 nM)、hCA II (Ki: 46 nM)、hCA IX (Ki: 466 nM) 和 hCA I (Ki: 8.351 μM)。hA2A/hCA XII modulator 1 表现出研究癌症的潜力。
T79748 hCAIX/XII-IN-7

Carbonic Anhydrase Metabolism
hCAIX/XII-IN-7(compound 3e)为高效的hCA IX与XII抑制剂,对hCA I、II、IX与XII的Ki值分别为3.2 nM、9.2 nM、503.7 nM及59 nM,显示其在缺氧肿瘤研究中的应用潜力。
T60602 hCAIX/XII-IN-5

Others Others
hCAIX/XII-IN-5 (Coumarin 9a) 是一种碳酸酐酶 (CA) 抑制剂,具有出色的 hCA IX/XII 选择性,对 hCA I 和 hCA II 的Ki 值分别为 93.9 和 85.7 nM。hCAIX/XII-IN-5 对癌细胞具有抗增殖活性,可延迟细胞周期并诱导细胞凋亡。
T61015 hCAIX/XII-IN-2

Others Others
hCAIX/XII-IN-2 (compound 6a) 是有效的 hCAIX 和 hCAXII 的选择性抑制剂,其对于hCAI、hCAII、hCAIX 和 hCAXII 的Ki 值分别为 >10000、>10000、30.0、3.6 nM。
T78789 hCA XII-IN-6

Carbonic Anhydrase Metabolism
hCA XII-IN-6(化合物4d)是一种具有84.2 nM Ki值的hCA XII强效抑制剂,显示出抗增殖活性,并可用于癌症的研究。
T61959 hCAIX/XII-IN-3

Others Others
hCAIX/XII-IN-3 (compound 6q) 是一种有效的、选择性的 hCAIX 和 hCAXII 抑制剂。hCAIX/XII-IN-3抑制 hCAI、hCAII、hCAIX 和 hCAXII 的 Ki 值分别为 >10000、>10000、66.2、4.4 nM。
T61873 hCAIX/XII-IN-1

Others Others
hCAIX/XII-IN-1 是一种有效的CAIX/XII 抑制剂,KI 值分别为 0.48 μM 和 0.83 μM。hCAIX/XII-IN-1 显示出体外抗增殖活性。hCAIX/XII-IN-1 诱导 MCF-7 细胞凋亡apoptosis。
T79351 JH-XII-03-02

PROTACs PROTAC
JH-XII-03-02为高效的选择性LRRK2 PROTAC降解剂,适用于帕金森病相关研究。
T63764 hCA XII/II/IX-IN-1

Others Others
hCA XII/II/IX-IN-1 是人碳酸酐酶 (hCA) 的有效抑制剂,能够作用于 hCA I (IC50: 2.6 μM)、 hCA II (IC50: 0.004 μM)、hCA IX (IC50: 0.005 μM) 和 hCA XII (IC50: 0.001 μM)。hCA XII/II/IX-IN-1 表现出抗癌效果。
T4502 BISMUTH SUBGALLATE

次没食子酸铋,Dermatol Puder,Bismuth Gallate

Others Others
Bismuth subgallate (Dermatol Puder) 是一种止血剂,可作用于凝血因子 XII ,促使凝血级联的激活,改善纤维蛋白凝块的早期形成。
T36758 CAIX Inhibitor S4

S4

Carbonic Anhydrase Metabolism
CAIX Inhibitor S4 (S4) 是一种有效的碳酸酐酶 IX/XII 抑制剂,Ki 分别为 7 nM 和 2 nM。 CA II 和 CA I 的 Ki 分别为 546 和 5600 nM。
T78578 GSK-3 Inhibitor XIII

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
GSK-3 Inhibitor XIII,一种ATP竞争性的 GSK-3抑制剂(Ki:24 nM),可用于研究糖尿病和肥胖。
T24111 GSK3i XIII

GSK3 inhibitor XIII,GSK3iXIII,GSK3i-XIII

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
GSK3i XIII (GSK3 inhibitor XIII) 是ATP 竞争性GSK-3抑制剂(Ki: 24 nM)。
T63276 hCAXII-IN-4

Others Others
hCAXII-IN-4 是选择性的、有效的 CA XII 抑制剂,对人CA XII 的Ki 值为 6.4 nM。
T62101 hCAXII-IN-2

Others Others
hCAXII-IN-2 (compound 5i) 是一种人碳酸酐酶 XII (hCA XII) (Ki: 84.2 nM) 和 hCA IX (Ki: 268.5 nM) 的有效抑制剂,对 hCA I 和 hCA II 具有较低的活性。
T79411 hCAXII-IN-7

Carbonic Anhydrase Metabolism
hCAXII-IN-7 (compound 6e)为hCA XII抑制剂,且具备脑屏障通透性。此化合物能够诱导786-0、SF-539和HS 578 T细胞系的凋亡。
T61219 hCAXII-IN-1

Others Others
hCAXII-IN-1 demonstrates selective inhibition of tumor-related subtypes HCA IX and XII, making it potential leading molecules in the development of novel cancer therapeutic drugs with new mechanisms of action.
T60930 CAXII-IN-1

Others Others
CAXII-IN-1 (Compound 17) 具有抗肿瘤活性,它是 CA XII 的选择性抑制剂。CAXII-IN-1 对 hCA XII 和 hCA IX 的 Ki 值分别为 3.8 nM 和 56.0 nM。
T63973 hCAXII-IN-3

Others Others
hCAXII-IN-3 (Compound 6o) 是人碳酸酐酶 XII(hCAXII)的选择性抑制剂 (Ki: 10.0 nM)。
T82361 FXIIa-IN-1

Others Others
XIIa-IN-1-IN-3(Compound 22)作为一种Factor XIIa抑制剂,其Kiapp值为97.8 nM。该化合物主要应用于血栓形成的研究。
T82360 FXIIa-IN-2

Others Others
XIIa-IN-1-IN-2(Compound 21)为一种高效的Factor XIIa抑制剂,具有Kiapp为62.2 nM。该化合物适用于血栓形成的研究领域。
T80485 μ-Conotoxin SxIIIC

Sodium Channel Membrane transporter/Ion channel
μ-Conotoxin SxIIIC是从条纹芋螺(Conus striolatus)提取的不可逆NaV通道(NaV channel)抑制剂,适用于慢性疼痛等神经系统疾病研究。
T82727 Chromoionophore XIII

SNARF-DE

Chromoionophore XIII (SNARF-DE)是一种可用红光激发的pH传感器。其功能质使指示剂分子具有亲脂性而不溶于水,并且能抑制该染料在极性环境下发生内酯化反应。
T61769 hCAXII-IN-5

Others Others
hCAXII-IN-5 (compound 6o) is a highly effective and specific inhibitor of hCAXII. The compound exhibits impressive binding affinities, with Ki values of >10000, >10000, 286.1, and 1.0 nM for hCAI, hCAII, hCAIX, and hCAXII, respectively [1].
T2017 U-104

NSC-213841,MST-104

Carbonic Anhydrase Metabolism
U-104 (NSC-213841) 是 CA IX 和 CA XII 碳酸酐酶 (CA) 抑制剂,其 Ki 分别为 45.1 nM 和 4.5 nM。小鼠模型中,它能够表现出明显的抑制肿瘤生长的作用。
T73177 hCAII-IN-9

Carbonic Anhydrase Metabolism
hCAII-IN-9 是一种强效的碳酸酐酶抑制剂,对hCA II、hCA IX 和hCA XII 有抑制作用,IC50 分别为 1.18 μM 和 0.17 μM , and 2.99 μM 。hCAII-IN-9 没有血脑屏障透过性。
T77018 Garadacimab

CSL312

Factor Xa Metabolism
Garadacimab (CSL312) 是有效的全人 IgG4 单克隆抗体,针对活化因子 XII (FXIIa)。Garadacimab 可用于研究遗传性血管性水肿。 。
T63305 Carbonic anhydrase inhibitor 6

Carbonic Anhydrase Metabolism
Carbonic anhydrase inhibitor 6 是一种高效的人碳酸酐酶 (hCA) 抑制剂,抑制 hCA IX,hCA II,hCA XII和hCA I,可用于研究碳酸酐酶异常引起的疾病。
T77631 Enpp/Carbonic anhydrase-IN-2

Apoptosis; PDE; Carbonic Anhydrase Apoptosis; Metabolism
Enpp/Carbonic anhydrase-IN-2 is a potent dual inhibitor of Enpp and carbonic anhydrase, inhibiting NPP1, NPP2, NPP3, CA-IX, CA-XII, with IC50 values of 1.13, 1.07, 0.74, 0.33, 0.68, respectively.Enpp/Carbonic anhydrase-IN-2 induced apoptosis.Enpp/Carbonic anhydrase-IN-2 has antiproliferative activity against cancer cells and low cytotoxicity against normal cells.
T61745 hCAI/II-IN-6

Carbonic Anhydrase Metabolism
hCAI/II-IN-6 是一种具有选择性和口服活性的human carbonic anhydrase(CA) 抑制剂。hCAI/II-IN-6对 hCA I,hCA II,hCA VII 和 hCA XII 有抑制作用,Ki 值分别为 220,4.9,6.5 和 >50000 nM。hCAI/II-IN-6 在体内显示抗惊厥活性。hCAI/II-IN-6 可以用于研究癫痫。
PDK0269 1-Phenylbiguanide HCl

Phenylbiguanide hydrochloride

Others Others
Compound PDK0269作为5-HT3受体激动剂(3-100 μM, pEC50 5.05±0.06),可急性增加XII(舌下)发作频率和规律性,并降低发作/次。Phenylbiguanide 产生剂量依赖性(10-500 μM)的多巴胺释放增加(280-2000%)。当Ringer 溶液中加入5 μM 的 nomifensine 时,Compound PDK0269对多巴胺释放的影响得到改善或抑制。
T30909 Chromozym PK

Others Others
Chromozym PK is a chromogenic substrate for factor XII assay.
T62026 hCAIX-IN-11

Others Others
hCAIX-IN-11 (Compound 5d) 是选择性的碳酸酐酶 (carbonic anhydrase) IX 和 XII 抑制剂。hCAIX-IN-11抑制 hCA IX 和 hCA XII 的Ki 分别为 32.7 和 623.5 nM。
T63158 hCAIX-IN-10

Others Others
hCAIX-IN-10 (Compound 6i) 是一种选择性碳酸酐酶 IX 和 XII 抑制剂,作用于 hCA IX (Ki: 61.5 nM) 和 hCA XII (Ki: 586.8 nM)。其中 hCA IX 和 hCA XII 是一种跨膜同工型碳酸酐酶,能够作为一些类型肿瘤的生物标志物。hCA XII 有助于正常细胞和肿瘤细胞中酸碱平衡的维持。
T62666 Carbonic anhydrase inhibitor 7

Others Others
Carbonic anhydrase inhibitor 7 是一种人碳酸酐酶 (hCA) 的有效抑制剂,作用于 hCA IX (Ki: 6.5 nM),hCA II (Ki: 7.1 nM),hCA XII (Ki: 72.1 nM) 和 hCA I (Ki: 255.8 nM)。
T79540 hCA/VEGFR-2-IN-1

Carbonic Anhydrase Metabolism
hCA/VEGFR-2-IN-1 是一种高效的双靶点抑制剂,对 hCA IX 和 hCA XII 两种碳酸酐酶(CA)具有极低的Ki值,分别为8.3 nM和4.7 nM。同时,hCA/VEGFR-2-IN-1 也是一种有效的 VEGFR-2 抑制剂,其 IC50 值仅为26.3 nM,并且显示出抗癌活性。
TP1866 β-Amyloid (1-11)

β-amyloid 1-11

Anionic interaction of Beta-amyloid (1-11) with Factor XII is suspected to cause massive activation of the C4 (complement 4) system in the cerebrospinal fluid of Alzheimer’s disease patients.
T62976 Carbonic anhydrase inhibitor 5

Others Others
Carbonic anhydrase inhibitor 5 是一种有效的、选择性的人碳酸酐酶 (hCA) 抑制剂,能够作用于 hCA II (IC50: 42.9 nM)、hCA IX (IC50: 47.6 nM) 和 hCA XII (IC50: 6.7 nM)。
T63005 Carbonic anhydrase inhibitor 11

Others Others
Carbonic anhydrase inhibitor 11 (compound VI) 是一种有效的、选择性碳酸酐酶抑制剂,能够作用于 CA II (Ki: 40 nM)、CA IX (Ki: 39 nM) 和 CA XII (Ki: 900 nM)。
T79588 hCA/VEGFR-2-IN-3

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
hCA/VEGFR-2-IN-3(compound 8j)是一种吲哚酮基苯磺酰胺类化合物,作为hCA IX/XII和VEGFR-2的双重抑制剂,在抗癌领域具有潜在应用。该化合物对VEGFR-2表现出显著的抑制活性(IC50=358 nM),并且与hCAs有较高的亲和力,具体活性为:Ki值分别为4.2 nM(hCA IX),22.9 nM(hCA II),25.1 nM(hCA I)和28.0 nM(hCA XII)。此外,hCA/VEGFR-2-IN-3还对过表达VEGFR-2的乳腺癌细胞显示出抗增殖效果。
T80095 D-Pro-Phe-Arg-Chloromethylketone

Factor Xa Metabolism
D-Pro-Phe-Arg-Chloromethylketone是一种抑制剂,它针对凝血因子XII (coagulation factor XII) 和血浆激肽释放酶 (kallikrein),在血栓形成和炎症过程中具有关键作用。

化合物

Jingzhaotoxin-XII
Cat.No: T80498
Synonym: JzTx-XII
Target: Potassium Channel
Calpain Inhibitor XII
Cat.No: T21949
Synonym:
Target: Others
Eupteleasaponin XII
Cat.No: T125110
Synonym:
Target: Others
RA-XII
Cat.No: T125868
Synonym:
Target: Others
Z-Ile-Leu-aldehyde
Cat.No: T17281
Synonym: Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII
Target: Others
hCAIX/XII-IN-8
Cat.No: T79753
Synonym:
Target: Carbonic Anhydrase
hCAIX/XII-IN-4
Cat.No: T61384
Synonym:
Target: Others
hCAIX/XII-IN-6
Cat.No: T72840
Synonym:
Target: Others
MDK-4683
Cat.No: T25779
Synonym: MDK 4683,CA IX/XII Inhibitor
Target: Others
hA2A/hCA XII modulator 1
Cat.No: T63400
Synonym:
Target: Others
hCAIX/XII-IN-7
Cat.No: T79748
Synonym:
Target: Carbonic Anhydrase
hCAIX/XII-IN-5
Cat.No: T60602
Synonym:
Target: Others
hCAIX/XII-IN-2
Cat.No: T61015
Synonym:
Target: Others
hCA XII-IN-6
Cat.No: T78789
Synonym:
Target: Carbonic Anhydrase
hCAIX/XII-IN-3
Cat.No: T61959
Synonym:
Target: Others
hCAIX/XII-IN-1
Cat.No: T61873
Synonym:
Target: Others
JH-XII-03-02
Cat.No: T79351
Synonym:
Target: PROTACs
hCA XII/II/IX-IN-1
Cat.No: T63764
Synonym:
Target: Others
BISMUTH SUBGALLATE
Cat.No: T4502
Synonym: 次没食子酸铋,Dermatol Puder,Bismuth Gallate
Target: Others
CAIX Inhibitor S4
Cat.No: T36758
Synonym: S4
Target: Carbonic Anhydrase
GSK-3 Inhibitor XIII
Cat.No: T78578
Synonym:
Target: GSK-3
GSK3i XIII
Cat.No: T24111
Synonym: GSK3 inhibitor XIII,GSK3iXIII,GSK3i-XIII
Target: GSK-3
hCAXII-IN-4
Cat.No: T63276
Synonym:
Target: Others
hCAXII-IN-2
Cat.No: T62101
Synonym:
Target: Others
hCAXII-IN-7
Cat.No: T79411
Synonym:
Target: Carbonic Anhydrase
hCAXII-IN-1
Cat.No: T61219
Synonym:
Target: Others
CAXII-IN-1
Cat.No: T60930
Synonym:
Target: Others
hCAXII-IN-3
Cat.No: T63973
Synonym:
Target: Others
FXIIa-IN-1
Cat.No: T82361
Synonym:
Target: Others
FXIIa-IN-2
Cat.No: T82360
Synonym:
Target: Others
μ-Conotoxin SxIIIC
Cat.No: T80485
Synonym:
Target: Sodium Channel
Chromoionophore XIII
Cat.No: T82727
Synonym: SNARF-DE
Target:
hCAXII-IN-5
Cat.No: T61769
Synonym:
Target: Others
U-104
Cat.No: T2017
Synonym: NSC-213841,MST-104
Target: Carbonic Anhydrase
hCAII-IN-9
Cat.No: T73177
Synonym:
Target: Carbonic Anhydrase
Garadacimab
Cat.No: T77018
Synonym: CSL312
Target: Factor Xa
Carbonic anhydrase inhibitor 6
Cat.No: T63305
Synonym:
Target: Carbonic Anhydrase
Enpp/Carbonic anhydrase-IN-2
Cat.No: T77631
Synonym:
Target: Apoptosis, PDE, Carbonic Anhydrase
hCAI/II-IN-6
Cat.No: T61745
Synonym:
Target: Carbonic Anhydrase
1-Phenylbiguanide HCl
Cat.No: PDK0269
Synonym: Phenylbiguanide hydrochloride
Target: Others
Chromozym PK
Cat.No: T30909
Synonym:
Target: Others
hCAIX-IN-11
Cat.No: T62026
Synonym:
Target: Others
hCAIX-IN-10
Cat.No: T63158
Synonym:
Target: Others
Carbonic anhydrase inhibitor 7
Cat.No: T62666
Synonym:
Target: Others
hCA/VEGFR-2-IN-1
Cat.No: T79540
Synonym:
Target: Carbonic Anhydrase
β-Amyloid (1-11)
Cat.No: TP1866
Synonym: β-amyloid 1-11
Target:
Carbonic anhydrase inhibitor 5
Cat.No: T62976
Synonym:
Target: Others
Carbonic anhydrase inhibitor 11
Cat.No: T63005
Synonym:
Target: Others
hCA/VEGFR-2-IN-3
Cat.No: T79588
Synonym:
Target: VEGFR
D-Pro-Phe-Arg-Chloromethylketone
Cat.No: T80095
Synonym:
Target: Factor Xa
Cat. No. Product Name Target Signaling Pathways
T13717 Gypenoside XIII

Others Others
Gypenoside XIII is belonging to the gypenosides. Gypenosides, extracted from Gynostemma pentaphyllum, protect against cardiovascular diseases, especially atherosclerosis.
T82806 Bupleuroside XIII

Bupleuroside XIII为具有肝脏保护作用的天然皂苷。
T0465 Ellagic acid

鞣花酸,Gallogen,Elagostasine

Hedgehog/Smoothened; Casein Kinase; Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; PKA; Syk; PKC; Carbonic Anhydrase Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Ellagic acid (Gallogen) 是从 Eucalyptus maculata Hook 和 E. Hemipholia F. Muell 的 kino 中分离出来的稠合四环天然产物,是一种有效的,ATP 竞争性的CK2抑制剂,IC50和Ki 值分别为 40 nM 和 20 nM。
T40611 (E)-Dehydrodiconiferyl alcohol

Others Others
(E)-Dehydrodiconiferyl alcohol is a potent dual inhibitor of hCA IX and hCA XII, effectively impeding the catalytic activity of both carbonic anhydrase isoforms. Additionally, (E)-Dehydrodiconiferyl alcohol exerts inhibitory effects on the nuclear translocation of NF-κB in the connective tissue of the healing area.

天然产物

Gypenoside XIII
Cat.No: T13717
Synonym:
Target: Others
Bupleuroside XIII
Cat.No: T82806
Synonym:
Target:
Ellagic acid
Cat.No: T0465
Synonym: 鞣花酸,Gallogen,Elagostasine
Target: Hedgehog/Smoothened, Casein Kinase, Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, PKA, Syk, PKC, Carbonic Anhydrase
(E)-Dehydrodiconiferyl alcohol
Cat.No: T40611
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-00694 Carbonic Anhydrase 12 Protein, Human, Recombinant (His)

HsT18816,FLJ20151,carbonic anhydrase XII,CA12,CA

Human HEK293 Cells
Carbonic Anhydrase 12 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 31.6 kDa and the accession number is O43570-1.
TMPH-03106 Coagulation factor XII Protein, Pig, Recombinant (His)

HAF,Hageman factor,F12,Coagulation factor XII

Sus scrofa (Pig) E. coli
Factor XII is a serum glycoprotein that participates in the initiation of blood coagulation, fibrinolysis, and the generation of bradykinin and angiotensin. Prekallikrein is cleaved by factor XII to form kallikrein, which then cleaves factor XII first to alpha-factor XIIa and then trypsin cleaves it to beta-factor XIIa. Alpha-factor XIIa activates factor XI to factor XIa. Coagulation factor XII Protein, Pig, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predic...
TMPY-00688 Carbonic Anhydrase 12 Protein, Mouse, Recombinant (His)

AI314958,Car12,2310047E01Rik,carbonic anhydrase XII

Mouse HEK293 Cells
Carbonic Anhydrase 12 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32.8 kDa and the accession number is Q8CI85.
TMPH-01114 COL12A1 Protein, Human, Recombinant (His)

Collagen alpha-1(XII) chain,COL12A1L,COL12A1

Human E. coli
COL12A1 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPH-03383 Synaptotagmin-12 Protein, Rat, Recombinant (His)

Syt12,Synaptotagmin-12,Synaptotagmin XII,Synaptotag...

Rat E. coli
Synaptic vesicle phosphoprotein that enhances spontaneous neurotransmitter release but does not effect induced neurotransmitter release. Unlike other synaptotagmins, it does not bind Ca(2+) or phospholipids. Essential for mossy-fiber long-term potentiation in the hippocampus. Synaptotagmin-12 Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 50.7 kDa and the accession number is P97610.
TMPH-02588 COL12A1 Protein, Mouse, Recombinant (His)

Collagen alpha-1(XII) chain,COL12A1L,COL12A1

Mouse E. coli
Type XII collagen interacts with type I collagen-containing fibrils, the COL1 domain could be associated with the surface of the fibrils, and the COL2 and NC3 domains may be localized in the perifibrillar matrix.
TMPY-06944 Carbonic Anhydrase 12 Protein, Human, Recombinant (His & Avi), Biotinylated

HsT18816,carbonic anhydrase XII,CAXII,FLJ2...

Human HEK293 Cells
Carbonic Anhydrase 12 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 33.45 kDa and the accession number is NP_001209.1.
TMPK-00478 Carbonic Anhydrase 12 Protein, Cynomolgus, Recombinant (His)

CA12,CAXII,Carbonic anhydrase,CA-XII,Tumor...

Cynomolgus HEK293 Cells
Carbonic anhydrases (CAs) are a family of enzymes involved in the pH regulation of metabolically active cells/tissues. Carbonic anhydrase XII (CA XII) is a key mediator of several signaling pathways that are involved in cancer development.
TMPY-02185 Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)

Coagulation factor 13,coagulation factor XIII, B po...

Human HEK293 Cells
Coagulation factor XIII B chain, also known as Fibrin-stabilizing factor B subunit, Protein-glutamine gamma-glutamyltransferase B chain, Transglutaminase B chain and F13B, is a secreted protein which contains 1 Sushi ( CCP / SCR ) domains. Coagulation factor XIII is the last zymogen to become activated in the blood coagulation cascade. Plasma factor XIII is a heterotetramer composed of 2 A subunits and 2 B subunits. The A subunits have catalytic function, and the B subunits do not have en...
TMPH-00051 Chitin deacetylase Protein, Amylomyces rouxii, Recombinant (His)

Chitin deacetylase,MrCDA,CDA

Amylomyces rouxii E. coli
Hydrolyzes the N-acetamido groups of N-acetyl-D-glucosamine residues in chitin to form chitosan and acetate. Chitin deacetylase Protein, Amylomyces rouxii, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 49.9 kDa and the accession number is P50325.
TMPH-00430 VxXIIC Protein, Conus vexillum, Recombinant (His & Myc & SUMO)

Alpha-conotoxin VxXXC,VxXIIC

Conus vexillum E. coli
Alpha-conotoxins act on postsynaptic membranes, they bind to the nicotinic acetylcholine receptors (nAChR) and thus inhibit them. This toxin specifically blocks mammalian neuronal nAChR of the alpha-7/CHRNA7, alpha-3-beta-2/CHRNA3-CHRNB2 and alpha-4-beta-2/CHRNA4-CHRNB2 subtypes. VxXXA and VxXXB inhibit alpha-7/CHRNA7 and alpha-3-beta-2/CHRNA3-CHRNB2 nAChR more efficiently than VxXXC. VxXXB is the most effective at inhibiting alpha-4-beta-2/CHRNA4-CHRNB2 nAChR, followed by VxXXC and VxXXA. VxXII...
TMPH-03352 KLKB1 Protein, Rat, Recombinant (His)

Fletcher factor,Klkb1,Plasma prekallikrein,Kininogenin,Plasm...

Rat P. pastoris (Yeast)
The enzyme cleaves Lys-Arg and Arg-Ser bonds. It activates, in a reciprocal reaction, factor XII after its binding to a negatively charged surface. It also releases bradykinin from HMW kininogen and may also play a role in the renin-angiotensin system by converting prorenin into renin. KLKB1 Protein, Rat, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 29.8 kDa and the accession number is P14272.
TMPH-03351 KLKB1 Protein, Rat, Recombinant (E. coli, His)

Plasma prekallikrein,Klkb1,Kininogenin,Plasma kallikrein,Fle...

Rat E. coli
The enzyme cleaves Lys-Arg and Arg-Ser bonds. It activates, in a reciprocal reaction, factor XII after its binding to a negatively charged surface. It also releases bradykinin from HMW kininogen and may also play a role in the renin-angiotensin system by converting prorenin into renin. KLKB1 Protein, Rat, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 31.8 kDa and the accession number is P14272.
TMPJ-00734 KNG1 Protein, Human, Recombinant (His)

KNG1,High Molecular Weight Kininogen,BDK,HMWK,KNG,Williams-F...

Human HEK293 Cells
Kininogen-1 is a secreted protein which contains three cystatin domains. There are two alternatively spliced forms, designated as the high molecular weight (HMW) and low MW (LMW) forms. Kininogen-1 plays a critical role in blood coagulation and inflammatory response. Kininogens are inhibitors of thiol proteases. Kininogen-1 participates in blood coagulation by helping to position optimally prekallikrein and factor XI next to factor XII, also inhibits the thrombin- and plasmin-induced aggregation...

重组蛋白

Carbonic Anhydrase 12 Protein, Human, Recombinant (His)
Cat.No: TMPY-00694
Species: Human
Expression System: HEK293 Cells
Coagulation factor XII Protein, Pig, Recombinant (His)
Cat.No: TMPH-03106
Species: Sus scrofa (Pig)
Expression System: E. coli
Carbonic Anhydrase 12 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-00688
Species: Mouse
Expression System: HEK293 Cells
COL12A1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01114
Species: Human
Expression System: E. coli
Synaptotagmin-12 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03383
Species: Rat
Expression System: E. coli
COL12A1 Protein, Mouse, Recombinant (His)
Cat.No: TMPH-02588
Species: Mouse
Expression System: E. coli
Carbonic Anhydrase 12 Protein, Human, Recombinant (His & Avi), Biotinylated
Cat.No: TMPY-06944
Species: Human
Expression System: HEK293 Cells
Carbonic Anhydrase 12 Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPK-00478
Species: Cynomolgus
Expression System: HEK293 Cells
Coagulation factor XIII B/F13B Protein, Human, Recombinant (His)
Cat.No: TMPY-02185
Species: Human
Expression System: HEK293 Cells
Chitin deacetylase Protein, Amylomyces rouxii, Recombinant (His)
Cat.No: TMPH-00051
Species: Amylomyces rouxii
Expression System: E. coli
VxXIIC Protein, Conus vexillum, Recombinant (His & Myc & SUMO)
Cat.No: TMPH-00430
Species: Conus vexillum
Expression System: E. coli
KLKB1 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03352
Species: Rat
Expression System: P. pastoris (Yeast)
KLKB1 Protein, Rat, Recombinant (E. coli, His)
Cat.No: TMPH-03351
Species: Rat
Expression System: E. coli
KNG1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00734
Species: Human
Expression System: HEK293 Cells
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