Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3453 |
WAY-100635 maleate
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM). | |||
T2631 |
WAY-100635 Monomaleate
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
WAY-100635 maleate 是一种选择性的5-hydroxytryptamine 1A 受体拮抗剂,IC50值为 0.91 nM,Ki 值为 0.39 nM。它也是多巴胺 D4受体激动剂,对于5-HT1A 和 α1-肾上腺素的 pIC50值分别为 8.9 和 6.6。 |