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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T4246L Varenicline

Others Others
Varenicline (CP 526555) 是一种有效的α4β2 nAChR 烟碱乙酰胆碱受体的部分激动剂,EC50值为2.3 μM。Varenicline 是 α3β4 nAChR 和 α7 nAChR 乙酰胆碱受体的完全激动剂,EC50值分别为 55 μM 和 18 μM。Varenicline 是一种基于胞嘧啶结构的烟碱配体,具有戒烟治疗的潜力。
T1657 Varenicline Tartrate

Champix tartrate,酒石酸伐尼克兰,Chantix tartrate,CP 526555-18,酒石酸伐仑克林

AChR Neuroscience
Varenicline Tartrate (CP 526555-18) 是α4β2 烟碱乙酰胆碱受体的部分激动剂,EC50为 2.3 μM。它是 α3β4 和 α7 乙酰胆碱受体完全激动剂,EC50值分别为 55 和 18 μM,用于戒烟方面的研究。
T23502 Varenicline Hydrochloride

Others Others
Varenicline Hydrochloride is a partial agonist of α4β2 nicotinic receptor.
T4246 Varenicline dihydrochloride

AChR Neuroscience
Varenicline dihydrochloride是一种选择性 α4β2 烟碱乙酰胆碱受体部分激动剂。
T85294 Hydroxy Varenicline

2-Hydroxyvarenicline

Others Others
Hydroxy varenicline, a metabolite of the nicotinic acetylcholine receptor (nAChR) agonist varenicline, functions within the biochemical pathway by interacting with nAChR sites.
T36810 uPSEM 792 hydrochloride

Others Others
Ultrapotent PSEM (uPSEM) agonist for PSAM4-GlyR and PSAM4-5HT3 (Ki = 0.7 nM for PSAM4-GlyR and <10 nM for PSAM4-5HT3). Exhibits >10,000-fold agonist selectivity for PSAM4-GlyR over α7-GlyR, α7-5HT3, and 5HT3-R, and 230-fold selectivity over α4β2 nAChR. Also weak partial agonist (~10 %) at α4β2 nAChR. Retains the potency of varenicline (Cat.No. 3754) for PSAM4-GlyR with enhanced chemogenetic selectivity. Does not act as a substrate for P-glycoprotein pumps. Silences neurons in vivo. Brain-penetra...

化合物

Varenicline
Cat.No: T4246L
Synonym:
Target: Others
Varenicline Tartrate
Cat.No: T1657
Synonym: Champix tartrate,酒石酸伐尼克兰,Chantix tartrate,CP 526555-18,酒石酸伐仑克林
Target: AChR
Varenicline Hydrochloride
Cat.No: T23502
Synonym:
Target: Others
Varenicline dihydrochloride
Cat.No: T4246
Synonym:
Target: AChR
Hydroxy Varenicline
Cat.No: T85294
Synonym: 2-Hydroxyvarenicline
Target: Others
uPSEM 792 hydrochloride
Cat.No: T36810
Synonym:
Target: Others
TargetMol Loading
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