Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9381 |
Thalidomide 5-fluoride
2-(2,6-二氧代 - 哌啶-3-基)-5-氟 - 异吲哚-1,3-二酮,H-Isoindole-1,3(2H)-dione, 2-(2,6-dioxo-3-piperidinyl)-5-fluoro- |
Ligand for E3 Ligase | PROTAC |
Thalidomide 5-fluoride (H-Isoindole-1,3(2H)-dione, 2-(2,6-dioxo-3-piperidinyl)-5-fluoro-) 是一种基于沙利度胺的 Cereblon 配体,通过 linker 与 IRAK4 蛋白配体结合形成 PROTACIRAK4 degrader-1。 | |||
T39696 |
Thalidomide-Piperazine 5-fluoride
|
Others | Others |
Thalidomide-Piperazine 5-fluoride is a compound developed by synthesizing an E3 ligase ligand-linker conjugate. It incorporates a cereblon ligand derived from Thalidomide and utilizes a linker commonly employed in PROTAC technology. | |||
T84904 |
Thalidomide-Piperazine 5-fluoride hydrochloride
UUN-14238,Pomalidomide 5'-fluoro-6'-piperazine,UUN14238,UUN 14238 |
Others | Others |
Thalidomide-Piperazine 5-fluoride hydrochloride,作为Thalidomide衍生物,是一种cereblon(CRBN)抑制剂,用作E3 泛素连接酶的配体(Ligands for E3 Ligase),适用于PROTACs合成。 |