185
112
2
11
4
Cat. No. | Product Name | ||
---|---|---|---|
L6500 | 微生物天然产物库 | 685 compounds | |
685 种微生物来源的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选; | |||
L6620 | 抗寄生虫天然产物库 | 253 compounds | |
253 个抗寄生虫相关的天然产物集合,是药物开发、药理研究的有效工具; |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28869 |
Streptomyces A-Factor
A-Factor (Lactone) |
Others | Others |
Streptomyces A-Factor is a microbial hormone found in Streptomyces griseus. A-factor triggers streptomycin biosynthesis and cell differentiation by binding a repressor-type receptor protein (ArpA) and dissociating it from DNA. | |||
T26231 |
Acetyl-pepstatin
Streptomyces pepsin inhibitor,Ac-Pepstatin,乙酰胃泌素 |
||
Streptomyces pepsin inhibitor is used as a pepsin inhibitor. | |||
T8814 |
Nikkomycin Z
尼柯霉素Z,Nikkomycin Z from Streptomyces tendae,尼柯霉素 Z |
Others; Antibiotic; Antifungal | Microbiology/Virology; Others |
Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) 是一种选择性竞争性几丁质合成抑制剂。它是一种核苷肽,可作为几丁质合酶底物 UDP-N-乙酰氨基葡萄糖的竞争性类似物,具有抗真菌作用。 | |||
T1400L |
Demeclocycline
Ledermycin,Bioterciclin,Deteclo,Declostatin,Deganol |
Antibacterial | Microbiology/Virology |
Demeclocycline (Declostatin) 是一种四环素类抗生素,产自金霉素链霉菌(Streptomyces aureofaciens)菌株。Demeclocycline 具有抗菌活性,能抑制血管加压素对肾小管的作用,从而导致利尿。Demeclocycline 可用诱导尿崩症和急性肾衰竭。 | |||
T24243 |
Kanosamine
3-Amino-3-deoxyglucose,3-氨基-3-脱氧-D-葡萄糖 |
Antifungal | Microbiology/Virology |
Kanosamine (3-Amino-3-deoxyglucose) 是一种由链霉菌产生的抗真菌剂。 | |||
T4989 |
Fosfomycin Tromethamine
|
Antibacterial; Antibiotic | Microbiology/Virology |
Fosfomycin tromethamine 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。 | |||
T0788L |
Spectinomycin dihydrochloride pentahydrate
盐酸大观霉素五水合物,Trobicin,Spectogard,Spectinomycin hydrochloride hydrate |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Spectinomycin dihydrochloride pentahydrate (Spectogard) 是一种广谱氨基环糊精抗生素,可以抑制多种革兰氏阳性和革兰氏阴性生物的生长。 | |||
T5435 |
ARV-771
|
Epigenetic Reader Domain; PROTACs | Chromatin/Epigenetic; PROTAC |
ARV-771 是基于 PROTAC 技术的有效 BET 降解剂,对 BRD2(1)、BRD2(2)、BRD3(1)、BRD3(2)、BRD4 (1) 和 BRD4(2)的 Kd 分别为 34、4.7、8.3、7.6、9.6 和 7.6 nM。 | |||
T60020 |
5'-Fluoro-5'-deoxyadenosine
5'-Fluoro-5'-deoxy-adenosine |
Others | Others |
5'-Fluoro-5'-deoxyadenosine (5'-Fluoro-5'-deoxy-adenosine) 常用作研究放线菌卡特链霉菌的工具。 | |||
T19724 |
5NAA
5-NAA,2-氨基-5-硝基苯甲酸,5 NAA |
Others | Others |
5NAA 是一种由疥疮链霉菌分泌的分子,可合成染料和其他硝基芳族化合物的原料。 | |||
T73721 |
Phleomycin D1
PLM D1,PLM-D1 |
Antibacterial; Antibiotic | Microbiology/Virology |
Phleomycin D1 (PLM D1) 是一种由Streptomyces verticillus(轮枝链霉菌)的突变株产生的一种糖肽抗生素,具有抗菌活性,可破坏细菌双螺旋结构的完整性。Phleomycin D1 可用于筛选携带Sh ble基因的转染细胞。 | |||
T16551 |
Pladienolide B
|
Apoptosis | Apoptosis |
Pladienolide B 是一种有效的剪接体抑制剂,是从钝顶链霉菌 Mer-12 中分离出的大环内酯类化合物,其作用靶向剪接体的 SF3B1 亚单位。Pladienolide B 通过抑制前 mRNA 剪接发挥抗肿瘤作用,诱导调亡。Pladienolide B 具有抗肿瘤活性,可用于研究白血病和淋巴肿瘤。 | |||
T19860 |
Clavulanic Acid
BRL 14151,MM-14151,MM 14151,RX-10100,MM14151,BRL14151,BRL-14151 |
Antibacterial; Antifungal | Microbiology/Virology |
Clavulanic Acid(RX-10100) 是一种由生物体克拉维链霉菌产生的主要β-内酰胺类抗生素,是一种强效的细菌 β-内酰胺酶抑制剂,用于研究细菌引起的感染。Clavulanic Acid 具有广谱的生物活性,对多种革兰氏阳性和革兰氏阴性细菌均有活性。 | |||
T30080 |
Ansatrienin A3
|
Others | Others |
Ansatrienin A3 is produced by Streptomyces collinus. | |||
T25422 |
Flambamycin
RP21190,RP-21190,RP 21190 |
Others | Others |
Flambamycin is an antibiotic isolated from Streptomyces hygroscopicus. | |||
T25037 |
Aldecalmycin
|
Others | Others |
Aldecalmycin is a new antimicrobial antibiotic isolated from Streptomyces. | |||
T25504 |
Histargin
|
Others | Others |
Histargin is an enzyme inhibitor separated from Streptomyces roseoviridis. | |||
T26476 |
A28695B
A 28695B,A-28695B |
Others | Others |
A28695B is a polyether antibiotic, it is isolated from Streptomyces albus. | |||
T26116 |
Rokitamycin
|
Others | Others |
Rokitamycin is a macrolide antibiotic produced from strains of Streptomyces kitasatoensis. | |||
T26420 |
A 53868A
Dehydrophos,A-53868A,A53868A |
Others | Others |
A 53868A is an antibiotic, it is isolated from Streptomyces luridus. | |||
T25689 |
Leuseramycin
TM 531,TM531,Antibiotic TM-531,TM-531 |
Others | Others |
Leuseramycin is a polyether antibiotic isolated from Streptomyces hygroscopicus TM-531. | |||
T26416 |
A 33853
A-33853,A33853 |
Others | Others |
A 33853 is an antibiotic isolated from culture broth of Streptomyces sp. | |||
T26178 |
SB-217452
SB217452 |
Others | Others |
SB-217452 is a potent seryl tRNA synthetase inhibitor isolated from Streptomyces. | |||
T25987 |
Probestin
|
Others | Others |
Probestin is an aminopeptidase M inhibitor, isolated from Streptomyces azureus MH663-2F6. | |||
T32122 |
Hydroxypepstatin
|
Others | Others |
Hydroxypepstatin is a new peptatin produced by Streptomyces. | |||
T26275 |
Thrazarine
|
Others | Others |
Thrazarine is a new antitumor antibiotic agent produced by Streptomyces coerulescens MH802-fF5. | |||
T71367 |
OM-4842
|
Others | Others |
OM-4842 is a platelet aggregation inhibitor from Streptomyces. | |||
T33396 |
Misakimycin
|
Others | Others |
Misakimycin is a mammalian cell growth stimulating substance produced by Streptomyces misakiensis BP-3621. | |||
T26176 |
Saphenamycin
Racemic ssaphenamycin |
Others | Others |
Saphenamycin is an antibiotic from a strain of Streptomyces. | |||
T26160 |
Rubomycin H
|
Others | Others |
Rubomycin H is an anthracycline antibiotic from Streptomyces coeruleorubidus. | |||
T38500 |
Enduracidin
Enramycin,恩拉霉素 |
Others | Others |
Enduracidin (Enramycin) is a polypeptide antibiotic produced by Streptomyces fungicides. | |||
T33672 |
Nikkomycin pseudo-J
|
Others | Others |
Nikkomycin pseudo-J is a nikkomycin isolated from Streptomyces tendae. | |||
T32688 |
Leustroducsin C
LSN C |
Others | Others |
Leustroducsin C is an inducer of colony-stimulating factors CSF extracted from Streptomyces platensis SANK 60191. | |||
T25938 |
Pepstanone A
|
Others | Others |
Pepstanone A is a potent aspartyl protease inhibitor, produced by pepstatin-producing Streptomyces. | |||
T69996 |
A-75943
|
Others | Others |
A-75943 is a bone resorption inhibitor from streptomyces. | |||
T28185 |
Nogalamycin
Nogalamycinum,U 15167,Nogalamyicn,U-15167,Nogalamycine,Nogalomycin |
Others | Others |
Nogalamycin is an anthracycline antibiotic with antitumor properties produced by soil bacteria Streptomyces nogalater. | |||
T29419 |
3'-Rhamnopiericidin A(1)
SN-198-C |
Others | Others |
3'-Rhamnopiericidin A(1) is a piericidin rhamnoside from Streptomyces. | |||
T25027 |
Albocycline
TA-2407,Ingramycin |
Others | Others |
Albocycline is a Macrolide antibiotic from Streptomyces bruneogriseus nov. sp. MCRL-0129; specifically anti-staphylococcal, including antibiotic-resistant strains. | |||
T25512 |
Hydroxystreptomycin
Streptomycin C |
Others | Others |
Hydroxystreptomycin is a new antibiotic isolated from Streptomyces Griseocarneus. | |||
T35139 |
WS 1279
WS1279,WS-1279 |
Others | Others |
WS 1279 is an immunoactive lipopeptide that is isolated from Streptomyces. | |||
T25270 |
Conagenin
|
Others | Others |
Conagenin is a small molecular immunomodulator isolated by Streptomyces roseosporus. | |||
T25871 |
Nikkomycin J
|
Others | Others |
Nikkomycin J is used as an insecticide from Streptomyces tendae. | |||
T25762 |
Lucimycin
FI1163,Antibiotic 1163 F.I.,FI 1163,FI-1163,NSC 143257 |
Others | Others |
Lucimycin is a macrolide antibiotic from cultures of Streptomyces lucensis. | |||
T32810 |
LL-C 10037alpha
LLC 10037alpha,LL-c10037alpha |
Others | Others |
LL-C 10037alpha is a gamma-aminoepoxysemiquinone isolated from Streptomyces. | |||
T26088 |
Rimocidin
Rimocidine |
Others | Others |
Rimocidin is a macrolide antifungal compound isolated from Streptomyces rimosus. | |||
T25203 |
Candicidin D
LIA 0704,Candicidin D1,LIA0704,LIA-0704,Levorin A2 |
Others | Others |
Candicidin D is an antifungal agent isolated from Streptomyces griseus. | |||
T24589 |
Paldimycin A
Antibiotic 273 A1-alpha |
Others | Others |
Paldimycin A is a semi-synthetic antibiotic from Streptomyces paulus. | |||
T20706 |
Fosfomycin
Antibiotic 833A,MK-955,Fosfonomycin,MK955,MK 955 |
Others | Others |
Fosfomycin is an antibiotic that is produced by Streptomyces fradiae. | |||
T26333 |
WS 9326A
WS9326A,WS-326A |
Others | Others |
WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger. | |||
T25587 |
Kujimycin A
Desacetyllankamycin |
Others | Others |
Kujimycin A is a macrolide antibiotics agent from various strains of Streptomyces. It has great activity against some Gram-positive bacteria. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15277 |
Fervenulin
|
Parasite | Microbiology/Virology |
Fervenulin 具有杀灭线虫活性,抑制线虫M. incognita 卵孵化和 J2 的校正死亡率,MIC 分别为 30 μg/mL 和 120 μg/mL。 | |||
T1032 |
Erythromycin
红霉素,E-Mycin |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。 | |||
T37009 |
Oxychlororaphine
吩嗪-1-甲酰胺,phenazine-1-carboxamide |
Antibacterial | Microbiology/Virology |
Oxychlororaphine (phenazine-1-carboxamide) 强烈抑制 Streptomyces sp. 411 的生长。 | |||
TN7147 |
6-Hydroxyisatin
6-Hydroxy-1H-indole-2,3-dione,ZINC14455608,6-hydroxyindoline-2,3-dione,6-羟基靛红,6-hydroxy-2,3-dihydro-1H-indole-2,3-dione |
Others | Others |
6-Hydroxyisatin (ZINC14455608) 是一种海洋来源的天然产物,存在于 Streptomyces sp.。 | |||
TN7185 |
7-Cyano-7-deazaguanine
7-CN-7-deazaG |
Others | Others |
7-Cyano-7-deazaguanine (7-CN-7-deazaG) 是一种海洋来源的天然产物,存在于Streptomyces qinglanensis。 | |||
TN6961 |
Heneicosane
N-HENEICOSANE,正二十一烷,henicosane |
Antifungal | Microbiology/Virology |
Heneicosane (henicosane) 是一种信息素,是从 Streptomyces philanthiRL-1-178 或 Serapias cordigera 中分离出来的一种香气成分,可抑制黄曲霉毒素的产生。 | |||
T2762 |
Kasugamycin hydrochloride
Kasumin,盐酸春雷霉素 |
Antibacterial; Antibiotic; Antifungal | Microbiology/Virology |
Kasugamycin hydrochloride (Kasumin) 是一种能结合 30s 和 70s 核糖体,但不能结合 50s 亚基的抗生素。它模拟 mRNA 核苷酸以破坏 tRNA 结合并抑制经典翻译起始。 | |||
T1255 |
Tobramycin
NSC 180514,妥布霉素,Nebramycin Factor 6,Deoxykanamycin B |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Tobramycin (NSC-180514) 是一种胃肠外给药的广谱氨基糖苷类抗生素,可研究由于敏感生物引起的中度至重度细菌感染疾病。 | |||
T1003 |
Tylosin
Fradizine,Tylosin A,泰乐菌素,Tylosine,Tylocine |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylosin (Tylosine) 是一种兽医用大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。 | |||
T13827 |
Pronase E (Activity ≥ 7000 U/g)
Pronase,Pronase E |
Others | Others |
Pronase E 是一种蛋白水解酶混合物,从灰色链霉菌 (Streptomyces griseus) 中获得,能够将蛋白质消化成单个氨基酸。 | |||
T1505 |
Imipenem monohydrate
N-Formimidoyl thienamycin monohydrate,亚胺培南,Imipenem,亚胺培南一水物 |
Antibacterial; Antibiotic | Microbiology/Virology |
Imipenem monohydrate (Imipenem) 是从微生物 Streptomyces cattleya 分离得到的碳青霉烯类抗生素,是一种用于静脉注射的β 内酰胺类抗生素,作用于细菌细胞壁,能广泛有效抑制多种革兰氏阳性和阴性菌。 | |||
T11665 |
Ionomycin calcium
SQ23377 calcium,罗红霉素钙盐(链霉菌属载体) |
Apoptosis; Calcium Channel; Antibacterial; Antibiotic; PKC | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Ionomycin calcium (SQ23377 calcium) 是选择性钙离子载体,也是一种由 Streptomyces conglobatus 产生的抗生素。它对二价阳离子具有高度特异性,还诱导蛋白激酶 C 激活。Ionomycin 促进细胞凋亡。 | |||
T0974 |
Novobiocin Sodium
Albamycinsodium,新生霉素钠,Cathomycin,Albamycin |
Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy | Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology |
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。 | |||
T21430 |
Oxytetracycline Hydrochloride
Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin |
Antiviral; Endogenous Metabolite; Antibacterial; HSV | Immunology/Inflammation; Metabolism; Microbiology/Virology |
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。 | |||
TQ0158 |
Azaserine
CI-337,偶氮丝胺酸,P-165,氮杂丝氨酸,O-Diazoacetyl-L-serine |
Others; Antibiotic | Microbiology/Virology; Others |
Azaserine (CI-337) 是一种从链霉菌属中分离出来的肿瘤抑制抗生素,可作为谷氨酰胺氨基转移酶的抑制剂。 | |||
T15717 |
Lasalocid
Lasalocid-A,Antibiotic X-537A,Ionophore X-537A |
Antibacterial | Microbiology/Virology |
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。 | |||
T0474 |
Erythromycin ethylsuccinate
EES,琥乙红霉素 |
ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology; Proteases/Proteasome |
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。 | |||
T64911 |
Blasticidin S HCl
|
Antibiotic | Microbiology/Virology |
Blasticidin S HCl 是从 Streptomyces griseochromogenes 中分离的肽基核苷类抗生素 (antibiotic),主要通过干扰核糖体中肽键的形成从而抑制原核细胞和真核细胞蛋白的合成。 | |||
T1214 |
Ribostamycin sulfate
Vistamycin sulfate,硫酸核糖霉素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Ribostamycin sulfate (Vistamycin sulfate) 是一种广谱抗菌剂, 在30S 和50S 核糖体亚基结合抑制细菌蛋白质合成, 还抑制蛋白二硫键异构酶分子伴侣活性, 用于药代动力学和肾毒性研究。 | |||
T1679 |
Thiostrepton
Thiactin,Bryamycin,Alaninamide,硫链丝菌素 |
DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Thiostrepton (Alaninamide) 是一种选择性抑制FOXM1的抗生素。FOXM1会与 YAP/TEAD 复合物结合,形成YAP/TEAD/FOXM1 复合物。 | |||
T0788 |
Spectinomycin dihydrochloride
淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。 | |||
T15716 |
Lasalocid sodium
拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。 | |||
TJS0161 |
Eudesmol
β-Eudesmol,桉叶醇,Β-桉叶醇 |
Others | Others |
β-Eudesmol (β-Eudesmol) 是一种倍半萜类化合物,由Streptomyces tendae 产生。 | |||
T67708 |
Thiolutin
Acetopyrrothin |
Antibacterial; Antibiotic | Microbiology/Virology |
Thiolutin (Acetopyrrothin) 是一种内皮细胞粘附抑制剂,由链霉菌产生。 Thiolutin 具有抗生素和抗血管生成特性。 Thiolutin 可快速诱导 Hsp27 的磷酸化。 | |||
T1033 |
Monensin sodium salt
莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt |
Sodium Channel; Antibacterial; Antibiotic | Membrane transporter/Ion channel; Microbiology/Virology |
Monensin sodium salt (Monensin A sodium salt) 是由肉桂链霉菌 分泌的抗生素。它是一种介导Na+/H+交换的离子载体。它引起细胞多泡体 (MVBs) 增大并调节外泌体的分泌。 | |||
T79972 |
Cyclo(L-leucyl-L-valyl)
|
Antifungal | Microbiology/Virology |
Cyclo(L-leucyl-L-valyl) 是从昆明链霉菌 YIM 次级代谢产物中部分离得到的多要化合物,尚未显示出抗菌活性。 | |||
T8373 |
6-Diazo-5-oxo-L-nor-Leucine
DON,L-6-Diazo-5-oxonorleucine,6-重氮-5-氧代-L-正亮氨酸,Diazooxonorleucine |
Influenza Virus; Glutaminase; Antibacterial; Antibiotic | Microbiology/Virology; Proteases/Proteasome |
6-Diazo-5-oxo-L-nor-Leucine (L-6-Diazo-5-oxonorleucine) 是一种谷氨酰胺拮抗剂,具有抗菌、抗病毒和抗癌作用,其Ki 值为 6 μM。它能降低肿瘤细胞的自我更新能力和转移能力 ,在体外表现出遗传毒性。 | |||
T0895 |
Oxytetracycline
土霉素,Terramycin |
ribosome; Endogenous Metabolite; Antibacterial; Antibiotic; HSV | Metabolism; Microbiology/Virology |
Oxytetracycline (Terramycin) 是一种四环素类抗生素。它强力抑制革兰氏阴性和革兰氏阳性细菌。它是一种蛋白质合成抑制剂,可阻止 aminoacil-tRNA 与复杂的核糖体 RNA 结合,具有抗 HSV-1的活性。 | |||
T7285 |
Ionomycin
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Ionomycin 是一种钙离子载体和一种结合钙离子(Ca2+)的抗生素。它是由联合链霉菌(Streptomyces conglobatus)产生的。它在研究中用于提高细胞内钙水平(Ca2+),并作为了解 Ca2+跨生物膜运输的研究工具。Ionomycin 可促进细胞凋亡,诱导蛋白激酶 C (PKC)活化。 | |||
T16340 |
Nosiheptide
RP 9671,Multhiomycin,那西肽 |
Antibacterial; Antibiotic | Microbiology/Virology |
Nosiheptide (Multhiomycin) 是一种由 Streptomyces actuosus 生产的硫肽类抗生素,已被广泛用作动物生长的饲料添加剂。它抑制细菌蛋白质合成,并在特征性大环核心上带有独特的吲哚侧环系统和区域特异性羟基。 | |||
T3607 |
Leucomycin
吉他霉素,Kitasamycin,Leucomycin V,Turimycin |
Antibacterial; Antibiotic | Microbiology/Virology |
Leucomycin (Turimycin) 是一种由 Streptomyces kitasatoensis 产生的大环内酯类抗生素。 | |||
T0819 |
Spiramycin
Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine |
Antibacterial; Antibiotic; Parasite | Microbiology/Virology |
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。 | |||
T1235 |
Lincomycin hydrochloride monohydrate
洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。 | |||
T15091 |
Decoyinine
Decynylene,Angustmycin A |
||
Decoyinine (Decynylene) 是一种选择性的GMP 合成酶抑制剂,是一种新型的潜在微生物杀虫剂,是一种由透明链霉菌产生的次级代谢产物。Decoyinine 诱导水稻对小棕瓢虫Laodelphax striatellus 的抗性。 | |||
T4038 |
Ectoine
THP(B),L-Ectoine,四氢甲基嘧啶羧酸 |
Others; Antibacterial | Microbiology/Virology; Others |
Ectoine (L-Ectoine) 是生活在极其恶劣环境中的细菌所产生的氨基酸衍生物,是一种天然的细胞保护剂。它具有良好的安全性,可研究过敏性鼻炎。它用作渗透调节相容性溶质,可增加皮肤表面的水合作用并稳定脂质层,常用于皮肤护理。 | |||
T8118 |
Bekanamycin
Kanamycin B,卡那霉素,卡那霉素 B |
Antibacterial; Antibiotic | Microbiology/Virology |
Bekanamycin (Kanamycin B) 是一种提取自 Streptomyces kanamyceticus 的氨基糖苷类抗生素,抑制一系列革兰氏阳性和阴性细菌。 | |||
T5352 |
GLYCODEOXYCHOLIC ACID
|
Others; Endogenous Metabolite | Metabolism; Others |
Glycodeoxycholic Acid 是内源性代谢产物的一种,是一种存在于黑链霉菌、布氏锥虫和隐单胞菌中的天然产物,可诱导阻塞性胆汁淤积症患者的肝细胞坏死和自噬。 | |||
T21502 |
Aclacinomycin A
Aclarubicin |
Topoisomerase | DNA Damage/DNA Repair |
Aclacinomycin A (Aclarubicin) 是一种从加利莱链霉菌中分离出的新型蒽环类抗生素,具有抗肿瘤活性。Aclacinomycin A 是拓扑异构酶 I 和 II 的抑制剂,抑制 RNA 活性 。Aclacinomycin A 可用于研究复发性白血病和晚期恶性淋巴瘤。 | |||
T5285 |
3-(Methylthio)propionic acid
3-Methylthiopropionate,3-甲基硫代丙酸,4-Thiapentanoic acid,3-Methylsulfanylpropionic acid |
Others; Endogenous Metabolite; Antifungal | Metabolism; Microbiology/Virology; Others |
3-(Methylthio)propionic acid (4-Thiapentanoic acid) 是methionine 的代谢物,是中间体。 | |||
T1506 |
Vidarabine
Adenine Arabinoside,阿糖腺苷,9-β-D-Arabinofuranosyladenine,Vira-A,Arabinosyladenine,Ara-A |
Nucleoside Antimetabolite/Analog; Tyrosine Kinases; DNA/RNA Synthesis; Antibiotic; HSV | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Vidarabine (Adenine Arabinoside) 是从链霉菌分离的核苷类抗生素,能抗单纯性疱疹和水痘-带状疱疹病毒。它对 HSV-1 和 HSV-2 的 IC50值分别为 9.3 μg/ml 和 11.3 μg/ml。 | |||
T6758 |
Anisomycin
茴香霉素,Flagecidin,NSC 76712,Wuningmeisu C |
Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; JNK | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK; Microbiology/Virology |
Anisomycin (Flagecidin) 属于细菌抗生素,是一种蛋白合成抑制剂和一种 JNK 激活剂。Anisomycin 通过抑制肽基转移酶或 80S 核糖体系统来干扰蛋白质和 DNA 的合成。 | |||
T14329 |
Ascamycin
|
Nucleoside Antimetabolite/Analog; Others; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others |
Ascamycin 是一种由链霉菌属产生的 5'-O-磺酰胺核糖核苷抗生素,对黄单胞菌类显示出选择性的抗菌活性,对柠檬黄单胞菌、口蹄疫黄单胞菌和噬菌体具有抑制作用,MIC 值分别为0.4μg/mL、12.5μg/mL 和12.5μg/mL。 | |||
T0912 |
Tetracycline hydrochloride
NCI-c55561,盐酸四环素,Tetracycline HCl |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。 | |||
T10662L |
Calcimycin
Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187 |
Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal | Apoptosis; Autophagy; Microbiology/Virology |
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。 | |||
T20879 |
Tacrolimus monohydrate
FK-506,FR 900506,Prograf,FR900506,Tacrolimus hydrate,LCP-Tacro,他克莫司一水合物,FK 506 |
Phosphatase; Others; Antibacterial; Antibiotic; Autophagy | Autophagy; Metabolism; Microbiology/Virology; Others |
Tacrolimus monohydrate (LCP-Tacro) 是大环内酯类化合物,它与 FK506 结合蛋白 (FKBP) 结合形成复合物并抑制钙调神经磷酸酶,从而抑制 T 淋巴细胞信号转导和 IL-2 转录。具有强免疫抑制特性。 | |||
T8504 |
Dianemycin
Nanchangmycin (free acid) |
Antibacterial; Antibiotic | Microbiology/Virology |
Dianemycin (Nanchangmycin (free acid)) 由Streptomyces nanchangensis 产生的一种聚醚抗生素,抑制革兰氏阳性菌。它也是一种针对 Zika 病毒的广谱抗病毒药物。 | |||
T0861 |
Tylosin tartrate
酒石酸泰洛星,酒石酸泰乐菌素 |
Antibacterial; Antibiotic | Microbiology/Virology |
Tylosin tartrate 是一种大环内酯类抗生素,是 Streptomyces fradiae 的产物。它对革兰氏阳性菌具有高效的抗菌活性。它作为饲料添加剂可促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。 | |||
T7004 |
Tubercidin
结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine |
Influenza Virus; DNA/RNA Synthesis; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Tubercidin (Sparsomycin A) 是从Streptomyces tubercidicus 得到的抗生素,抑制粪链球菌生长的IC50值为 0.02 μM。它是腺苷磷酸化酶的弱抑制剂,并干扰腺苷和 AMP 的磷酸化。它有抗病毒作用。 | |||
T24729 |
Roseoflavin
|
Antibacterial | Microbiology/Virology |
Roseoflavin 是天然色素,起初分离自Streptomyces davawensis。Roseoflavin 是核黄素和黄素单核苷酸的抗代谢类似物,显示出抗菌活性。 | |||
T26405 |
A 201A
Antibiotic 201A,A201A,A-201A |
Others | Others |
A 201A is a nucleoside antibiotic, it is isolated from Streptomyces capreolus. | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-03605 |
CHOD Protein, Streptomyces sp., Recombinant (GST)
choA,Cholesterol isomerase,CHOD,Cholesterol oxidase |
Streptomyces | E. coli |
Bifunctional enzyme that catalyzes the oxidation of the 3-beta-hydroxy group of cholesterol and the isomerization of the double bond of the resulting product. CHOD Protein, Streptomyces sp., Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 81.9 kDa and the accession number is P12676. | |||
TMPH-00514 |
Endo H Protein, Streptomyces plicatus, Recombinant (His)
Endoglycosidase H,Endo-beta-N-acetylglucosaminidase H,Endo H |
Streptomyces plicatus | P. pastoris (Yeast) |
Cleaves asparagine-linked oligomannose and hybrid, but not complex, oligosaccharides from glycoproteins. | |||
TMPH-03604 |
Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)
Phosphinothricin-resistance protein,Phosphinothricin N-acety... |
Streptomyces hygroscopicus | E. coli |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. Can also acetylate demethylphosphinothricin but not PTT or glutamate. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 24.6 kDa and the accession number is P16426. | |||
TMPH-03607 |
HOE-467A Protein, Streptomyces tendae, Recombinant (His & Myc & SUMO)
Tendamistat,Alpha-amylase inhibitor HOE-467A |
Streptomyces tendae | E. coli |
Inhibits mammalian alpha-amylases specifically but has no action on plant and microbial alpha-amylases. Forms a tight stoichiometric 1:1 complex with alpha-amylase. HOE-467A Protein, Streptomyces tendae, Recombinant (His & Myc & SUMO) is expressed in E. coli expression system with N-10xHis-SUMO and C-Myc tag. The predicted molecular weight is 28.0 kDa and the accession number is P01092. | |||
TMPH-03606 |
P3H 1 Protein, Streptomyces sp., Recombinant (His & Myc)
Proline 3-hydroxylase type I,L-proline cis-3-hydroxylase 1,P... |
Streptomyces | E. coli |
Dioxygenase that catalyzes the 2-oxoglutarate-dependent selective hydroxylation of free L-proline to cis-3-hydroxy-L-proline (cis-3-Hyp). D-proline, trans-4-hydroxy-L-proline, cis-4-hydroxy-L-proline, cis-4-hydroxy-D-proline, and 3,4-dehydro-DL-proline are not substrates. P3H 1 Protein, Streptomyces sp., Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 44.0 kDa and the accession number is P96010. | |||
TMPH-03609 |
Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO)
pat,Phosphinothricin N-acetyltransferase,Phosphinothricin-re... |
Streptomyces viridochromogenes | E. coli |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 36.6 kDa and the accession number is Q57146. | |||
TMPH-03608 |
Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His)
Phosphinothricin N-acetyltransferase,Phosphinothricin-resist... |
Streptomyces viridochromogenes | P. pastoris (Yeast) |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 22.6 kDa and the accession number is Q57146. | |||
TMPH-03603 |
KcsA Protein, S. coelicolor, Recombinant (His)
pH-gated potassium channel KcsA,kcsA |
Streptomyces coelicolor | E. coli |
Acts as a pH-gated potassium ion channel; changing the cytosolic pH from 7 to 4 opens the channel. KcsA Protein, S. coelicolor, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 23.7 kDa and the accession number is P0A333. | |||
TMPH-03602 |
BLIP Protein, S. clavuligerus, Recombinant (His & SUMO)
Beta-lactamase inhibitory protein,BLIP |
Streptomyces clavuligerus | E. coli |
Inhibits a wide variety of beta lactamases. BLIP Protein, S. clavuligerus, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 33.5 kDa and the accession number is P35804. | |||
TMPH-03601 |
Streptavidin Protein, S. avidinii, Recombinant (His)
Streptavidin |
Streptomyces avidinii | P. pastoris (Yeast) |
The biological function of streptavidin is not known. Forms a strong non-covalent specific complex with biotin (one molecule of biotin per subunit of streptavidin). Streptavidin Protein, S. avidinii, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 18.5 kDa and the accession number is P22629. | |||
TMPJ-00871 |
BAR Protein, S. hygroscopicus, Recombinant
bar,PPT N-acetyltransferase,Phosphinothricin-resistance prot... |
Streptomyces hygroscopicus | E. coli |
Phosphinothricin N-acetyltransferase (PAT) is an enzyme that acetylates the free NH2 group of L-phosphinothricin (L-PPT) in the presence of acetyl-CoA as a co-substrate. It is highly specific for L-PPT and does not acetylate other L-amino acids or structurally similar molecules. L-PPT is a glutamate analog that can inhibit glutamine synthetase activity in plants, resulting in the accumulation of ammonia to toxic levels and impairment of photosynthesis. The introduction of a PAT gene into a plant... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMID-0292 |
Tylosin-d3
|
||
Tylosin-d3 是 Tylosin 的氘代化合物。Tylosin 的 CAS 号为 1401-69-0。Tylosin 是一种兽医用大环内酯类抗生素,是Streptomyces fradiae的产物。它对革兰氏阳性菌具有高抗菌活性。它是饲料添加剂用于促进动物生长。它被用于治疗家禽、猪和牛的细菌性痢疾和呼吸道疾病。 | |||
TMIJ-0109 |
Erythromycin Ethylsuccinate-13C-d3
|
||
Erythromycin Ethylsuccinate-13C-d3 是 Erythromycin Ethylsuccinate 的 13C 和氘代化合物。Erythromycin Ethylsuccinate 的 CAS 号为 1264-62-6。Erythromycin Ethylsuccinate是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗HIV-1病毒活性。 | |||
TMIJ-0281 |
Lincomycin-d3
|
||
Lincomycin-d3 是 Lincomycin 的氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。 | |||
TMIJ-0340 |
Lincomycin-13C-d3
|
||
Lincomycin-13C-d3 是 Lincomycin 的 13C 和氘代化合物。Lincomycin 的 CAS 号为 7179-49-9。Lincomycin hydrochloride monohydrate 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。 |