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Targets Recommended: COX

201

抑制剂 & 化合物

56

天然产物

3

化合物库

1

重组蛋白

17

同位素标记化合物

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Cat. No. Product Name
L4710 非甾体类抗炎化合物库

530 compounds
530 种非甾体类的抗炎相关化合物,可用于高通量和高内涵筛选;
L6710 中药抗炎分子库

1246 compounds
1246 种具有抗炎活性或靶向炎症相关靶点的中药单体集合,是药物开发、药理研究的有效工具;
L4700 免疫/炎症分子化合物库

4720 compounds
4720 种具有抗炎症活性的化合物的特有集合,可用于高通量筛选和高内涵筛选;

化合物库

非甾体类抗炎化合物库
Cat.No: L4710
Compounds: 530
中药抗炎分子库
Cat.No: L6710
Compounds: 1246
免疫/炎症分子化合物库
Cat.No: L4700
Compounds: 4720
Cat. No. Product Name Target Signaling Pathways
T2550 Tolmetin

Tolectin,托麦汀

COX Immunology/Inflammation; Neuroscience
Tolmetin (Tolectin) 是非甾体类抗炎药,是可口服的 COX 抑制剂,对人 COX-1 和 COX-2 的 IC50值分别为 0.35 和 0.82 µM。
T11399 Giredestrant

GDC-9545

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Giredestrant (GDC-9545) 是一种口服有效的、选择性的、非甾体的雌激素受体 (ER) 拮抗剂,具有抗肿瘤作用。它可以在 ER 配体结合域内与雌二醇 (Estradiol) 竞争结合并诱导构象变化。
T0380 Bicalutamide

比卡鲁胺,ICI-176334

Androgen Receptor; Autophagy Autophagy; Endocrinology/Hormones
Bicalutamide (ICI-176334) 是一种具有口服活性的非甾体雄激素受体拮抗剂,可研究前列腺癌。
T22371 Mivacurium dichloride

米库氯铵,Mivacurium chloride,二氯美维库铵

AChR Neuroscience
Mivacurium dichloride (Mivacurium chloride) 是苄基异喹啉衍生物,可与 nAChR 偶联,以减少或抑制乙酰胆碱对肌肉细胞末端盘的去极化作用。它也是非去极化短效的神经肌肉阻滞剂和骨骼肌松弛剂。
T6737 Zaltoprofen

CN100,扎托布洛芬,Soleton

COX Immunology/Inflammation; Neuroscience
Zaltoprofen (Soleton) 是一种非甾体类抗炎剂,具有强大的抗炎作用和对炎性疼痛的止痛作用。它是可口服的COX-2抑制剂,对COX-1和COX-2的IC50值分别为 1.3 和 0.34 μM。
T26539 AC-262536

AC262536,4-(3-内型-羟基-8-氮杂双环[3.2.1]辛烷-8-基)萘-1-甲腈

Androgen Receptor Endocrinology/Hormones
AC-262536 是非甾体雄激素受体选择性调节剂,具有有益的合成代谢作用。它可以强效激动雄激素受体,亲和力为1-10 nM。
T0383 Fenspiride hydrochloride

Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利

Adrenergic Receptor; PDE; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Fenspiride hydrochloride (Decaspiride) 是一种口服活性的非甾体抗炎剂,是 H1-组胺受体的拮抗剂,可用于呼吸系统疾病的研究。
T4602 Hydrocortisone hemisuccinate

Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate

Glucocorticoid Receptor; Others; Interleukin Endocrinology/Hormones; Immunology/Inflammation; Others
Hydrocortisone hemisuccinate (hydrocortisone 21-hemisuccinate*free acid) 是糖皮质激素, 是口服有活性的甾体抗炎剂。它能够降低IL-6(IC50:6.7 μM)、IL-3(IC50:21.4 μM)的生物活性,可用于研究溃疡性结肠炎。
T61444 Nonsteroidal aromatase inhibitor 1

Others Others
Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for research in the field of breast cancer [1].
T33414 MK 0434

MK-434,MK0434,MK-0434,MK 434,MK434

Reductase Endocrinology/Hormones; Metabolism
MK 0434 是一种具有口服活性的类固醇 5 α-还原酶抑制剂。
T26109 Robenacoxib

Onsior

COX Immunology/Inflammation; Neuroscience
Robenacoxib (Onsior) 是一种对环氧化酶-2 有很强的选择性的非甾体化合物,具有抗炎活性。
T19679 Benoxaprofen

氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459

COX Immunology/Inflammation; Neuroscience
Benoxaprofen (NSC-299582) 是长效的、强效的抗炎和解热化合物,在体外具有较弱的对环氧合酶的抑制作用,也可以抑制脂氧合酶,在一些炎症动物模型中抑制单核细胞迁移。
T6498 Fenoprofen calcium hydrate

Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate,非诺洛芬钙二水合物

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Fenoprofen calcium hydrate (Progesic dihydrate) 是一非甾体类抗炎症化合物。
T30161 EN3356

AS N001,ASN-001

P450 Metabolism
EN3356 是一种可口服且具有选择性的类固醇 17-α- 羟化酶/C17,20 裂解酶(CYP17A1 或 CYP17)抑制剂,是一种非甾体类裂解酶选择性化合物,具有潜在的抗雄激素和抗肿瘤活性。
T25985 Prifelone

R-830,R830,S-16820,S 16820,R 830

Others Others
Prifelone (R 830) 是一种非甾体抗炎化合物,具有抗氧化活性。
T0321 Indoprofen

吲哚洛芬,(±)-Indoprofe,茚酮苯丙酸

COX Immunology/Inflammation; Neuroscience
Indoprofen ((±)-Indoprofe) 是非甾体类抗炎药, 可用于研究脊髓性肌萎缩。
T30150 AS-601811

AS601811,AS 601811,UNII-LIV8A6AE5F

Androgen Receptor Endocrinology/Hormones
AS-601811 是类固醇 5α还原酶抑制剂和雄激素受体调节剂,可用于研究脱发和痤疮。
T21740 RD162

Androgen Receptor Endocrinology/Hormones
RD162 是一种与雄激素受体 (AR) 特异性结合的非甾体抗雄激素 (NSAA)。
T6540 Ibuprofen Lysine

布洛芬赖氨酸盐,Neoprofen

COX Immunology/Inflammation; Neuroscience
Ibuprofen Lysine (Neoprofen) 是一种非甾体抗炎药。
T14546 Bermoprofen

AD-1590,AJ-1590

Others Others
Bermoprofen (AD-1590) 是一种口服活性非甾体抗炎化合物, 具有抗炎镇痛活性,可用于研究胃溃疡。
T7839 Lasofoxifene Tartrate

CP-336156,酒石酸拉索昔芬

Estrogen Receptor/ERR Endocrinology/Hormones
Lasofoxifene Tartrate (CP-336156) 是一种非甾体类的雌激素受体选择性调节剂 (SERM)。
T22307 Diclofenac Epolamine

diclofenac hydroxyethylpyrrolidine,DHEP,2-((2,6-二氯苯基)氨基)苯乙酸 1-吡咯烷乙醇盐,DIEP

Others Others
Diclofenac Epolamine (DHEP) 是一种非甾体抗炎药 (NSAID),具有镇痛和解热作用。
T11340 Furprofen

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Furprofen 是一种非甾体类抗炎剂,抑制前列腺 (PGE) 合成,可用于研究类风湿关节炎和骨关节炎。
T0184 Fenoprofen calcium dihydrate

COX Immunology/Inflammation; Neuroscience
Fenoprofen calcium dihydrate 是一种丙酸衍生物,用作非甾体抗炎剂。
T27209 Droxicam

Droxicamum,屈昔康

Others Others
Droxicam (Droxicamum) 是一种非甾体抗炎化合物,可用于缓解肌肉骨骼疾病的炎症和疼痛的研究。
T27635 Isoxepac

伊索克酸,Olopatadine USP Related Compound C

Others Others
Isoxepac (Olopatadine USP Related Compound C) 是非甾体抗炎剂,显示出抗炎、镇痛和解热活性,已在多种动物模型中进行了相关研究。
T19694 Hydronidone

F351,F-351,F 351

Others Others
Hydronidone (F-351) 是一种 pyridine 衍生物。Hydronidone 对肝纤维化具有潜在的治疗作用。
T1720 Amfenac Sodium Hydrate

一水氨芬酸钠,Amfenac Sodium Monohydrate,氨芬酸钠水合物

COX Immunology/Inflammation; Neuroscience
Amfenac Sodium Hydrate 是一种含有乙酸部分的非甾体镇痛抗炎药,是 COX-2抑制剂。
T15246 Esaxerenone

艾沙利酮,XL-550,CS-3150

Glucocorticoid Receptor Endocrinology/Hormones
Esaxerenone (XL-550) 是高效的、选择性的非类固醇盐皮质激素受体拮抗剂。
T14666 BL-1249

Potassium Channel Membrane transporter/Ion channel
BL-1249 是一种具有选择性和有效性的非甾体钾通道激活剂,具有抗炎活性,可激活 K2P2.1 (TREK-1) 和 K2P10.1 (TREK-2)。
T7313 Enclomiphene citrate

恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate

Estrogen Receptor/ERR Endocrinology/Hormones
Enclomiphene citrate (trans-Clomiphene citrate) 是口服具有活力的 oestrogen receptor 拮抗剂,具有抗雌激素活性。
T7389 G15

Estrogen Receptor/ERR Endocrinology/Hormones
G15 是一种高亲和力的、选择性的 G 蛋白偶联雌激素受体(GPER/GPR30)拮抗剂(Ki:20 nM)。
T7293 EC330

Others Others
EC330 是一种白血病抑制因子抑制剂。
T0448 (S)-(+)-Ibuprofen

左旋布洛芬,Dexibuprofen,(S)-Ibuprofen,(S)-(+)-布洛芬

BCL; Thrombin; Cysteine Protease; COX; PPAR Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; Proteases/Proteasome
(S)-(+)-Ibuprofen (Dexibuprofen) 是 Ibuprofen 的 S(+)-对映异构体,能够有效的抑制COX-1(IC50:2.1 μM)和COX-2(IC50:1.6 μM),。它具有抗癌、退热、止痛,抗炎的效果。
T27798 Lapisteride

CS891B,CS-891,CS-891B,CS891

Others Others
Lapisteride (CS-891) 一种类固醇5α-还原酶抑制剂,可用于治疗良性前列腺增生(BPH)和雄激素性脱发,可有效预防或治疗AGA 。
T1258 Nabumetone

BRL14777,萘丁美酮

COX; Glutathione Peroxidase Immunology/Inflammation; Metabolism; Neuroscience
Nabumetone (BRL14777) 是一种非甾体抗炎药,是选择性COX-2抑制剂,其活性代谢物 6MNA 可抑制环加氧酶 I 和 II。
T0285 Isoxicam

伊索昔康,Isoxicamum,Isoxicamo,Maxicam

COX Immunology/Inflammation; Neuroscience
Isoxicam (Isoxicamum) 是可口服的非甾体抗炎剂,可通过抑制环氧合酶 1 和 2 来阻断前列腺素的合成,可用于关节炎的研究。
T17217 Vamorolone

地塞米松EP杂质E,VBP15

Glucocorticoid Receptor; NF-κB Endocrinology/Hormones; NF-κB
Vamorolone (VBP15) 是一种首创的,具有口服活性的解离性类固醇 (dissociative steroidal) 抗炎药和膜稳定剂。它抑制 (NF-κB) 抑制作用,并降低了激素的影响。它改善肌营养不良,无副作用。
T0637 2-Acetyl-6-methoxynaphthalene

Others Others
2-Acetyl-6-methoxynaphthalene 是naphthalene tome 和naproxen 的关键中间体,用于合成非甾体抗炎镇痛药。
T1421 Aceclofenac

醋氯芬酸,Preservex,Airtal

COX Immunology/Inflammation; Neuroscience
Aceclofenac (Preservex) 是一种可口服的非甾体抗炎药,可用于缓解疼痛、骨关节炎、强直性脊柱炎、类风湿性关节炎的研究。
T4561 Tiaprofenic acid

Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam

Others; COX Immunology/Inflammation; Neuroscience; Others
Tiaprofenic acid (Acido tiaprofenico) 是可口服的非甾体抗炎药,通过抑制环氧化酶抑制前列腺素合成,可用于风湿性疾病的研究。
T0319 Suxibuzone

琥布宗,Calibene,Suxibuzonum,Suxibuzona

COX Immunology/Inflammation; Neuroscience
Suxibuzone (Suxibuzona) 是非甾体类抗炎药 Phenylbutazone 的前药,可用于关节和肌肉疼痛研究。
T4542 Clonixin

Clonixic acid,氯尼辛

Others Others
Clonixin (Clonixic acid) 是一种非甾体抗炎药,具有口服活性。
T19967 Fendosal

芬度柳,HP 129,P 71-0129,P71-0129,P-71-0129,HP129,HP-129

Immunology/Inflammation related Immunology/Inflammation
Fendosal (HP-129) 是一种非甾体抗炎药。在预防性和治疗性辅助诱导的慢性炎症多关节炎模型中,它的活性是阿司匹林的 6.9 至 9.5 倍。
T12361 Parcetasal

MR-897

Others Others
Parcetasal (MR-897) 是一种非甾类体抗炎剂,在缓解疼痛方面具有研究价值。
T5843 Tarenflurbil

MPC7869,(R)-Flurbiprofen,R-flurbiprofen,氟比洛芬,R-氟比洛芬

Retinoid Receptor; Autophagy Autophagy; Metabolism
Tarenflurbil ((R)-Flurbiprofen) 是 Flurbiprofen 的 R 型对映体,可抑制 [3H]9-cis-RA 结合到 RXRαLBD,IC50为 75 μM。它可研究阿尔兹海默症。
T26926 Butibufen

FF 105,FF-106,FF 106,FF106

Lipoxygenase Metabolism
Butibufen (FF-106) 是一种具有口服活性的非甾体抗炎化合物,是潜在的环氧合酶抑制剂,具有止痛和解热活性,抑制尿素合成。Butibufen 可用于研究风湿性疾病。
T27254 Eltenac

B78820,B 78820,B-78820,BY-820,BY820,BY 820

COX Immunology/Inflammation; Neuroscience
Eltenac (B78820) 是一种非甾体抗炎剂,是 COX 抑制剂,具有镇痛活性。Eltenac 抑制 COX-1 和 COX-2 ,可用于研究急性呼吸窘迫综合征(ARDS)。
T1582 Naproxen

萘普生,(S)-Naproxen

COX; Autophagy Autophagy; Immunology/Inflammation; Neuroscience
Naproxen ((S)-Naproxen) 是COX-1和COX-2的抑制剂,在细胞试验中IC50值分别为8.72 和5.15 μM。它是丙酸衍生物和非甾体抗炎药,具有抗炎、解热和镇痛活性。
T0463 Loxoprofen

Loxoprofene,洛索洛芬,Loxoprofeno,Koloxo

COX Immunology/Inflammation; Neuroscience
Loxoprofen (Koloxo) 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX 抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。

化合物

Tolmetin
Cat.No: T2550
Synonym: Tolectin,托麦汀
Target: COX
Giredestrant
Cat.No: T11399
Synonym: GDC-9545
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Bicalutamide
Cat.No: T0380
Synonym: 比卡鲁胺,ICI-176334
Target: Androgen Receptor, Autophagy
Mivacurium dichloride
Cat.No: T22371
Synonym: 米库氯铵,Mivacurium chloride,二氯美维库铵
Target: AChR
Zaltoprofen
Cat.No: T6737
Synonym: CN100,扎托布洛芬,Soleton
Target: COX
AC-262536
Cat.No: T26539
Synonym: AC262536,4-(3-内型-羟基-8-氮杂双环[3.2.1]辛烷-8-基)萘-1-甲腈
Target: Androgen Receptor
Fenspiride hydrochloride
Cat.No: T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利
Target: Adrenergic Receptor, PDE, Histamine Receptor
Hydrocortisone hemisuccinate
Cat.No: T4602
Synonym: Hydrocortisone 21-he,氢化可的松琥珀酸酯,hydrocortisone 21-hemisuccinate*free acid,Hydrocortisone 21-hemisuccinate
Target: Glucocorticoid Receptor, Others, Interleukin
Nonsteroidal aromatase inhibitor 1
Cat.No: T61444
Synonym:
Target: Others
MK 0434
Cat.No: T33414
Synonym: MK-434,MK0434,MK-0434,MK 434,MK434
Target: Reductase
Robenacoxib
Cat.No: T26109
Synonym: Onsior
Target: COX
Benoxaprofen
Cat.No: T19679
Synonym: 氧苯恶唑丙酸,NSC 299582,LY-90459,Benoxaphen. Compound 90459
Target: COX
Fenoprofen calcium hydrate
Cat.No: T6498
Synonym: Feprona dihydrate,Fenoprofen calcium salt dihydrate,Progesic dihydrate,非诺洛芬钙二水合物
Target: Apoptosis, Others, COX
EN3356
Cat.No: T30161
Synonym: AS N001,ASN-001
Target: P450
Prifelone
Cat.No: T25985
Synonym: R-830,R830,S-16820,S 16820,R 830
Target: Others
Indoprofen
Cat.No: T0321
Synonym: 吲哚洛芬,(±)-Indoprofe,茚酮苯丙酸
Target: COX
AS-601811
Cat.No: T30150
Synonym: AS601811,AS 601811,UNII-LIV8A6AE5F
Target: Androgen Receptor
RD162
Cat.No: T21740
Synonym:
Target: Androgen Receptor
Ibuprofen Lysine
Cat.No: T6540
Synonym: 布洛芬赖氨酸盐,Neoprofen
Target: COX
Bermoprofen
Cat.No: T14546
Synonym: AD-1590,AJ-1590
Target: Others
Lasofoxifene Tartrate
Cat.No: T7839
Synonym: CP-336156,酒石酸拉索昔芬
Target: Estrogen Receptor/ERR
Diclofenac Epolamine
Cat.No: T22307
Synonym: diclofenac hydroxyethylpyrrolidine,DHEP,2-((2,6-二氯苯基)氨基)苯乙酸 1-吡咯烷乙醇盐,DIEP
Target: Others
Furprofen
Cat.No: T11340
Synonym:
Target: Prostaglandin Receptor
Fenoprofen calcium dihydrate
Cat.No: T0184
Synonym:
Target: COX
Droxicam
Cat.No: T27209
Synonym: Droxicamum,屈昔康
Target: Others
Isoxepac
Cat.No: T27635
Synonym: 伊索克酸,Olopatadine USP Related Compound C
Target: Others
Hydronidone
Cat.No: T19694
Synonym: F351,F-351,F 351
Target: Others
Amfenac Sodium Hydrate
Cat.No: T1720
Synonym: 一水氨芬酸钠,Amfenac Sodium Monohydrate,氨芬酸钠水合物
Target: COX
Esaxerenone
Cat.No: T15246
Synonym: 艾沙利酮,XL-550,CS-3150
Target: Glucocorticoid Receptor
BL-1249
Cat.No: T14666
Synonym:
Target: Potassium Channel
Enclomiphene citrate
Cat.No: T7313
Synonym: 恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate
Target: Estrogen Receptor/ERR
G15
Cat.No: T7389
Synonym:
Target: Estrogen Receptor/ERR
EC330
Cat.No: T7293
Synonym:
Target: Others
(S)-(+)-Ibuprofen
Cat.No: T0448
Synonym: 左旋布洛芬,Dexibuprofen,(S)-Ibuprofen,(S)-(+)-布洛芬
Target: BCL, Thrombin, Cysteine Protease, COX, PPAR
Lapisteride
Cat.No: T27798
Synonym: CS891B,CS-891,CS-891B,CS891
Target: Others
Nabumetone
Cat.No: T1258
Synonym: BRL14777,萘丁美酮
Target: COX, Glutathione Peroxidase
Isoxicam
Cat.No: T0285
Synonym: 伊索昔康,Isoxicamum,Isoxicamo,Maxicam
Target: COX
Vamorolone
Cat.No: T17217
Synonym: 地塞米松EP杂质E,VBP15
Target: Glucocorticoid Receptor, NF-κB
2-Acetyl-6-methoxynaphthalene
Cat.No: T0637
Synonym:
Target: Others
Aceclofenac
Cat.No: T1421
Synonym: 醋氯芬酸,Preservex,Airtal
Target: COX
Tiaprofenic acid
Cat.No: T4561
Synonym: Tiaprofensaeure,噻洛芬酸,Acido tiaprofenico,Surgam
Target: Others, COX
Suxibuzone
Cat.No: T0319
Synonym: 琥布宗,Calibene,Suxibuzonum,Suxibuzona
Target: COX
Clonixin
Cat.No: T4542
Synonym: Clonixic acid,氯尼辛
Target: Others
Fendosal
Cat.No: T19967
Synonym: 芬度柳,HP 129,P 71-0129,P71-0129,P-71-0129,HP129,HP-129
Target: Immunology/Inflammation related
Parcetasal
Cat.No: T12361
Synonym: MR-897
Target: Others
Tarenflurbil
Cat.No: T5843
Synonym: MPC7869,(R)-Flurbiprofen,R-flurbiprofen,氟比洛芬,R-氟比洛芬
Target: Retinoid Receptor, Autophagy
Butibufen
Cat.No: T26926
Synonym: FF 105,FF-106,FF 106,FF106
Target: Lipoxygenase
Eltenac
Cat.No: T27254
Synonym: B78820,B 78820,B-78820,BY-820,BY820,BY 820
Target: COX
Naproxen
Cat.No: T1582
Synonym: 萘普生,(S)-Naproxen
Target: COX, Autophagy
Loxoprofen
Cat.No: T0463
Synonym: Loxoprofene,洛索洛芬,Loxoprofeno,Koloxo
Target: COX
Cat. No. Product Name Target Signaling Pathways
T3901 Solasonine

Others Others
Solasonine 是一种甾体糖苷生物碱,从龙葵中分离获得,对人胃癌细胞有细胞毒性。
T4035 Khasianine

Others Others
Khasianine 是一种从茄属植物Solanum Nigrum L 中提取的甾体糖生物碱,具有抗肿瘤作用。
T3S1251 Neoruscogenin

ROR Metabolism
Neoruscogenin 是甾体 sapogenin 家族的成员,是一种可生物利用且具有高亲和力的核受体RORα (NR1F1)激动剂。
T3S0509 Gaultherin

COX Immunology/Inflammation; Neuroscience
Gaultherin 是一种分离自 Gaultheria yunnanensis 中的天然水杨酸酯衍生物。它是一种非甾体类抗炎药,具有止痛和抗炎作用,与 Aspirin 相比没有胃溃疡作用。
T3S1265 Liriopesides B

山麦冬皂苷B,Nolinospiroside F

Others Others
Liriopesides B (Nolinospiroside F) 是一种甾体皂苷,分离自 Ophiopogon japonicas 中,具有抗氧化和抗衰老活性。
T7024 Qingyangshengenin

青阳参甙元,Qingyangshengenin A,Cynanchagenin

Others Others
Qingyangshengenin (Cynanchagenin) 是一种孕烷糖苷,是一种分离自Cychuchumot ophyllum(Asclepiadaceae) 的根中的 C21 类固醇糖苷配基。它具有抗癌作用。
T0301 Ethisterone

炔孕酮,17α-Ethynyltestosterone,Pregneninolone

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Ethisterone (17α-Ethynyltestosterone) 是一种口服活性类固醇避孕药,是一种合成类固醇雌激素。据报道,它具有雄激素活性,用于妇科疾病的研究。
T4036 Solasodine

Solancarpidine,Purapuridine,澳洲茄铵,Solasodin

Apoptosis; Others; E1/E2/E3 Enzyme; Antifungal Apoptosis; Microbiology/Virology; Others; Ubiquitination
Solasodine (Purapuridine) 是存在于茄科植物中的一种类固醇生物碱。它具有神经保护、降压、抗真菌、抗癌、抗动脉粥样硬化、抗雄激素和抗炎活性。
T2S0250 Pseudoprotogracillin

伪原纤细薯蓣皂苷

Others Others
Pseudoprotogracillin 是一种从薯蓣科中提取的甾体皂苷类天然产物。
T10233 Acetylarenobufagin

HIF Angiogenesis; Chromatin/Epigenetic
Acetylarenobufagin 是一种类固醇缺氧诱导因子-1 (HIF-I) 调节剂。
T8094 16-​Dehydroprogesterone

16-Dehydroprogesterone,16-去氢黄体酮

Endogenous Metabolite Metabolism
16-​Dehydroprogesterone 是甾体孕激素。
T2S2295 Timosaponin A1

知母皂苷A1

Others Others
Timosaponin A1 是一种黄酮类甾体皂苷,分离自知母中。
TN2329 Zingiberen newsaponin

Zingiberensis saponin I,盾叶新苷

PARP; PAFR; Caspase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Proteases/Proteasome
Zingiberen newsaponin 是分离自盾叶薯 (Dioscorea zingiberensis) 中。 它能够诱导血小板聚集。
T2S1749 Protogracillin

原纤细薯蓣皂甙

Others Others
Protogracillin 是一种甾体皂苷,分离自Dioscorea zingiberensisWright (DZW) 中。从 DZW 根状茎中获得的甾体皂苷具有抗血栓作用,同时由降低心血管疾病风险的潜力。
T2962 5α-Cholestan-3β-ol

Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇

Others; Endogenous Metabolite Metabolism; Others
Dihydrocholesterol 是衍生化的类固醇化合物的一种,抑制胆固醇吸收。
TN6712 yibeissine

Others Others
Yibeissine 是一种甾体生物碱,分离自贝母球茎中。
T2825 Cyclopamine

环巴胺,11-Deoxojervine

Hedgehog/Smoothened; Endogenous Metabolite; Smo GPCR/G Protein; Metabolism; Stem Cells
Cyclopamine (11-Deoxojervine) 是Hedgehog 通路的拮抗剂,细胞实验中IC50=46 nM。它还是选择性Smo 抑制剂。
T2321 Protodioscin

Furostanol I,原薯蓣皂苷

Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Protodioscin (Furostanol I) 是一种山药根茎中的主要甾体皂苷,具有抗高血脂、抗癌活性。
TN2282 trans-Stilbene

反式-1,2二苯乙烯,1,2-Diphenylethylene (trans),(E)-Stilbene

Others Others
trans-Stilbene (1,2-Diphenylethylene (trans)) 可用于制备荧光增白剂、染料激光器、非甾体合成雌激素。
T20712 Conessine

Conessinum,Wrightine,地麻素,Roquessine,Neriine,Konessin

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Conessine (Conessinum) 是一种具有抗疟活性的甾体生物碱,是高效选择性H3 受体拮抗剂,对于人、狗、豚鼠和大鼠 H3受体的Ki 分别为 5.4、6.0、5.7 和 25 nM。
T3150 Caudatin

告达亭苷元,告达庭

Apoptosis; Others Apoptosis; Others
Caudatin 是白首乌中的一种甾体类天然产物,具有抗肿瘤和抗血管生成作用。它是一种 C-21 甾体糖苷,可使细胞周期停滞,诱导细胞凋亡。
T5751 Tigogenin

Others Others
Tigogenin 是甾体皂甙元,普遍用于甾体类药物的合成。它能够阻碍小鼠骨髓基质细胞脂肪细胞分化,促使成骨细胞的分化。
T16338 Norgestimate metabolite Norelgestromin

17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮

Drug Metabolite Metabolism
Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) 是norgestimate 的一种活性代谢物。它是用于避孕贴片的甾体孕激素,与雌激素乙炔雌二醇结合使用。
TN1383 Timosaponin B III

Anemarsaponin BIII,知母皂苷B3,知母皂苷BIII

Others; Platelet aggregation Others
Timosaponin B III (Anemarsaponin BIII) 是一种具有生物活性的甾体皂苷,从知母中分离出来。Timosaponin B III 具有抗炎、抗血小板聚集和抗抑郁作用。
T1048 Estradiol

雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estradiol (E2) 是一种天然的类固醇性激素,对于女性生育能力和第二性征的维持至关重要。Estradiol 通过雌激素受体 β (ERβ) 上调 IL-6 表达。
T2733 Sarsasapogenin

Parigenin,知母皂苷元,Sarsagenin

Apoptosis; NF-κB; Endogenous Metabolite Apoptosis; Metabolism; NF-κB
Sarsasapogenin (Parigenin) 是一种甾体皂苷元,从中草药知母中分离到,具有抗糖尿病、抗氧化、抗癌、抗炎等作用。
T4034 Solamargine

Solamargin,δ-Solanigrine,澳洲茄边碱

Apoptosis; p38 MAPK; P-gp; STAT Apoptosis; JAK/STAT signaling; MAPK; Membrane transporter/Ion channel; Neuroscience; Stem Cells
Solamargine (δ-Solanigrine) 是一种来源于茄属植物的类固醇 Solasodine 的衍生物,诱导非选择性细胞毒性和 P-gp 抑制作用。它通过下调 MMP-2 和 MMP-9 的表达和活性来显著抑制 HepG2 细胞的迁移和侵袭,在多种癌症中均表现出抗癌活性。
TMS1461 Qingyangshengenin B

青阳参甙元B,青阳参苷元B,Otophylloside B

Beta Amyloid Neuroscience
Qingyangshengenin B (Otophylloside B) 是一种分离自 Qingyangshen 的 C-21 甾体苷。它能够在 mRNA 水平上抑制 Aβ 的表达来减少 Aβ 的沉积,对 Aβ 的毒性有保护作用。它具有抗癫痫作用。
T4000 (±)-Equol

Equol,(±)-雌马酚,(R,S)-Equol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Drug Metabolite Endocrinology/Hormones; Metabolism
(±)-Equol ((R,S)-Equol) 是 equol 的外消旋体。它对 ERα 和 ERβ 的 EC50s of 分别为 200 和 74 nM。Equol 是大豆异黄酮黄豆苷和大豆黄素的代谢产物。
T6491 (-)-(S)-Equol

(−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
(-)-(S)-Equol (4',7-Dihydroxyisoflavan) 是雌激素受体β的高亲和力配体。
T34584 Scillaren A

Transvaalin,Scillaglykosid A

Others Others
Scillaren A is a a crystalline steroidal glycoside from Scilla maritima.
T33926 Penupogenin

Penupogenin is a steroidal aglycone isolated from the roots of Cynanchum auriculatum.
T2S2321 Pennogenin

Others Others
Pennogenin steroidal saponins could be utilized to develop anticancer medicines.
T32610 Laxogenin

6-Oxotigogenin

Laxogenin is a new steroidal sapogenin extracted from Smilax sieboldi Miq.
T13757 Lirioprolioside B

Others Others
Lirioprolioside B is a steroidal glycoside isolated from the underground organs of Liriope spicata var. prolifera.
T40890 Proprotogracillin

Others Others
Proprotogracillin is a steroidal glycoside isolated from the bulbs of lilium speciosum.
T30170 Aspafilioside A

Aspafilioside A is a steroidal saponin isolated from the root of Asparagus filicinus.
T13577 β-Zearalenol

Others Others
β-Zearalenol, a non-steroidal estrogenic mycotoxin synthesized by Fusarium species, potentially influences transcription and affects gene expression on the translational level.
T39854 Cycloposine

Others Others
Cycloposine, a steroidal alkaloid present in the roots and rhizomes of Veratrum californicum, is known to possess teratogenic properties.
T13641 Dehydrotomatine

Others Others
Dehydrolycopene is a major steroidal sugar alkaloid (SGAs), which is mainly found in mature green fruits, leaves and flowers of tomatoes. Dehydrotomato is targeted at bacteria, fungi, insects and animals.
T82544 Disporoside C

Disporoside C, 分子式为C41H66O12, 是一种甾体皂苷,可从植物Disporopsis pernyi中提取。
T10913 Cyclobuxine D

Others Others
Cyclobuxine D is a steroidal alkaloid extracted from Buxus microphylla. Cyclostatin D has obvious bradycardia effect on rat heart, and inhibits acetylcholine and Ba ++ induced longitudinal muscle contraction isolated from rabbit jejunum.
T40193 Ebeiedinone

Others Others
Ebeiedinone, a steroidal alkaloid derived from Fritillaria species, effectively inhibits the activity of human whole blood cholinesterase (ChE) at a concentration of 0.1 mM, resulting in a significant inhibitory effect of 69.0%.
T81545 Parisyunnanoside H

Parisyunnanoside H,一种甾体皂苷,可从Paris polyphylla Smith var. yunnanensis分离提取。
T13805 Ophiopogonin C

Ophiopogonin C,麦冬胶原蛋白 C

Others Others
Ophiopogonin C is a natural product isolated from the tubers of Ophiopogon japonicus, is a rare naturally occurring C29 steroidal glycoside.
T81093 Sterebin F

Sterebin F, 一种甾类化合物,来源于Stevia rebaudiana叶的分离提取,表现出降血糖的活性。
T83259 6β-Hydroxystigmasta-4,22-dien-3-one

6β-Hydroxystigmasta-4,22-dien-3-one为一类固醇化合物,可从Hedychium coronarium中提取。
T81097 Stauntoside M

Stauntoside M是一种从Cynanchum stauntonii的根中分离得到的类固醇糖苷。
T82480 Elephanoside D

Elephanoside D(化合物8)是从丝兰(Yucca elephantipes Regel)茎部分离出的一种甾体皂苷。
T82549 Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside

Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside (compound 9) 为甾体皂甙类化合物,源自Paris polyphylla var. yunnanensis,具有特定的结构特征。
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天然产物

Solasonine
Cat.No: T3901
Synonym:
Target: Others
Khasianine
Cat.No: T4035
Synonym:
Target: Others
Neoruscogenin
Cat.No: T3S1251
Synonym:
Target: ROR
Gaultherin
Cat.No: T3S0509
Synonym:
Target: COX
Liriopesides B
Cat.No: T3S1265
Synonym: 山麦冬皂苷B,Nolinospiroside F
Target: Others
Qingyangshengenin
Cat.No: T7024
Synonym: 青阳参甙元,Qingyangshengenin A,Cynanchagenin
Target: Others
Ethisterone
Cat.No: T0301
Synonym: 炔孕酮,17α-Ethynyltestosterone,Pregneninolone
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Solasodine
Cat.No: T4036
Synonym: Solancarpidine,Purapuridine,澳洲茄铵,Solasodin
Target: Apoptosis, Others, E1/E2/E3 Enzyme, Antifungal
Pseudoprotogracillin
Cat.No: T2S0250
Synonym: 伪原纤细薯蓣皂苷
Target: Others
Acetylarenobufagin
Cat.No: T10233
Synonym:
Target: HIF
16-​Dehydroprogesterone
Cat.No: T8094
Synonym: 16-Dehydroprogesterone,16-去氢黄体酮
Target: Endogenous Metabolite
Timosaponin A1
Cat.No: T2S2295
Synonym: 知母皂苷A1
Target: Others
Zingiberen newsaponin
Cat.No: TN2329
Synonym: Zingiberensis saponin I,盾叶新苷
Target: PARP, PAFR, Caspase
Protogracillin
Cat.No: T2S1749
Synonym: 原纤细薯蓣皂甙
Target: Others
5α-Cholestan-3β-ol
Cat.No: T2962
Synonym: Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇
Target: Others, Endogenous Metabolite
yibeissine
Cat.No: TN6712
Synonym:
Target: Others
Cyclopamine
Cat.No: T2825
Synonym: 环巴胺,11-Deoxojervine
Target: Hedgehog/Smoothened, Endogenous Metabolite, Smo
Protodioscin
Cat.No: T2321
Synonym: Furostanol I,原薯蓣皂苷
Target: Androgen Receptor, Endogenous Metabolite
trans-Stilbene
Cat.No: TN2282
Synonym: 反式-1,2二苯乙烯,1,2-Diphenylethylene (trans),(E)-Stilbene
Target: Others
Conessine
Cat.No: T20712
Synonym: Conessinum,Wrightine,地麻素,Roquessine,Neriine,Konessin
Target: Histamine Receptor
Caudatin
Cat.No: T3150
Synonym: 告达亭苷元,告达庭
Target: Apoptosis, Others
Tigogenin
Cat.No: T5751
Synonym:
Target: Others
Norgestimate metabolite Norelgestromin
Cat.No: T16338
Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮
Target: Drug Metabolite
Timosaponin B III
Cat.No: TN1383
Synonym: Anemarsaponin BIII,知母皂苷B3,知母皂苷BIII
Target: Others, Platelet aggregation
Estradiol
Cat.No: T1048
Synonym: 雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Sarsasapogenin
Cat.No: T2733
Synonym: Parigenin,知母皂苷元,Sarsagenin
Target: Apoptosis, NF-κB, Endogenous Metabolite
Solamargine
Cat.No: T4034
Synonym: Solamargin,δ-Solanigrine,澳洲茄边碱
Target: Apoptosis, p38 MAPK, P-gp, STAT
Qingyangshengenin B
Cat.No: TMS1461
Synonym: 青阳参甙元B,青阳参苷元B,Otophylloside B
Target: Beta Amyloid
(±)-Equol
Cat.No: T4000
Synonym: Equol,(±)-雌马酚,(R,S)-Equol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite
(-)-(S)-Equol
Cat.No: T6491
Synonym: (−)-Equol,Equol,4',7-Dihydroxyisoflavan,4',7-Isoflavandiol,雌马酚
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Scillaren A
Cat.No: T34584
Synonym: Transvaalin,Scillaglykosid A
Target: Others
Penupogenin
Cat.No: T33926
Synonym:
Target:
Pennogenin
Cat.No: T2S2321
Synonym:
Target: Others
Laxogenin
Cat.No: T32610
Synonym: 6-Oxotigogenin
Target:
Lirioprolioside B
Cat.No: T13757
Synonym:
Target: Others
Proprotogracillin
Cat.No: T40890
Synonym:
Target: Others
Aspafilioside A
Cat.No: T30170
Synonym:
Target:
β-Zearalenol
Cat.No: T13577
Synonym:
Target: Others
Cycloposine
Cat.No: T39854
Synonym:
Target: Others
Dehydrotomatine
Cat.No: T13641
Synonym:
Target: Others
Disporoside C
Cat.No: T82544
Synonym:
Target:
Cyclobuxine D
Cat.No: T10913
Synonym:
Target: Others
Ebeiedinone
Cat.No: T40193
Synonym:
Target: Others
Parisyunnanoside H
Cat.No: T81545
Synonym:
Target:
Ophiopogonin C
Cat.No: T13805
Synonym: Ophiopogonin C,麦冬胶原蛋白 C
Target: Others
Sterebin F
Cat.No: T81093
Synonym:
Target:
6β-Hydroxystigmasta-4,22-dien-3-one
Cat.No: T83259
Synonym:
Target:
Stauntoside M
Cat.No: T81097
Synonym:
Target:
Elephanoside D
Cat.No: T82480
Synonym:
Target:
Diosgenin-3-O-rhamnosyl(1→2)[glucosyl(1→6)]glucoside
Cat.No: T82549
Synonym:
Target:
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Cat. No. Product Name Species Expression System
TMPH-01640 MRGPRX2 Protein, Human, Recombinant (His)

Mas-related G-protein coupled receptor member X2,MRGPRX2

Human E. coli
Mast cell-specific receptor for basic secretagogues, i.e. cationic amphiphilic drugs, as well as endo- or exogenous peptides, consisting of a basic head group and a hydrophobic core. Recognizes and binds small molecules containing a cyclized tetrahydroisoquinoline (THIQ), such as non-steroidal neuromuscular blocking drugs (NMBDs), including tubocurarine and atracurium. In response to these compounds, mediates pseudo-allergic reactions characterized by histamine release, inflammation and airway c...

重组蛋白

MRGPRX2 Protein, Human, Recombinant (His)
Cat.No: TMPH-01640
Species: Human
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
T12336 Oxaprozin D4

Wy-21743 D4

Others Others
Oxaprozin D4 is the deuterium labeled Oxaprozin, is a non-steroidal anti-inflammatory drug (NSAID).
T11998 Meloxicam-d3

Meloxicam D4

Others Others
Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 μM ;(Target:COX-2; IC50: 0.49 μM).
T11754 Ketorolac-d5

Ketorolac D5

PPAR DNA Damage/DNA Repair; Metabolism
Ketorolac D5, a deuterium-labeled version of Ketorolac, is a non-steroidal anti-inflammatory agent that functions as a nonselective COX inhibitor. It exhibits IC50 values of 20 nM for COX-1 and 120 nM for COX-2.
T27210 DRX-065

DRX 065,DRX065,deuterated R-enantiomer of pioglitazone

DRX-065 is a stabilized and deuterated R-enantiomer of pioglitazone. DRX-065 has pharmacological properties desirable for the treatment of NASH (mitochondrial function modulation, non-steroidal anti-inflammatory effects, and glucose lowering effects) with
T11246 Etoricoxib-d4

MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4

Others Others
Etoricoxib D4 is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 and COX-1 in human whole blood.Etoricoxib D4 is a deuterium labeled Etoricoxib.
TMIH-0472 Rac Loxoprofen sodium-d3

Rac Loxoprofen sodium-d3 是 Rac Loxoprofen sodium 的氘代化合物。Rac Loxoprofen sodium 的 CAS 号为 68767-14-6。Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
TMIH-0325 MefenaMic Acid-d4

MefenaMic Acid-d4 是 MefenaMic Acid 的氘代化合物。MefenaMic Acid 的 CAS 号为 61-68-7。Mefenamic acid 是一种非甾体抗炎剂,可竞争性抑制hCOX-1和hCOX-2,IC50值分别为 40 nM 和 3 μM。
TMIJ-0211 Loxoprofen-d4

Loxoprofen-d4 是 Loxoprofen 的氘代化合物。Loxoprofen 的 CAS 号为 68767-14-6。Loxoprofen 是一种非甾体类抗炎药,具有解热作用,可用于缓解疼痛的研究。它是非选择性COX抑制剂,对 COX-1 和 COX-2 的IC50分别为 6.5 和 13.5 μM。
TMIH-0290 Ketorolac-d5-P1

Ketorolac-d5-P1 是 Ketorolac 的氘代化合物。Ketorolac 的 CAS 号为 74103-06-3。Ketorolac 是非甾体抗炎剂,是非选择性的COX抑制剂,对 COX-1 和 COX-2 的IC50值分别为 20 和 120 nM。
TMIH-0291 Ketorolac-d5-P2

Ketorolac-d5-P2 是 Ketorolac 的氘代化合物。Ketorolac 的 CAS 号为 74103-06-3。Ketorolac 是非甾体抗炎剂,是非选择性的COX抑制剂,对 COX-1 和 COX-2 的IC50值分别为 20 和 120 nM。
TMID-0276 MAA-d3

MAA-d3 是 MAA 的氘代化合物。MAA 的 CAS 号为 519-98-2。4-Methylamino antipyrine 是 Metamizole 的活性代谢产物,可用于疼痛和发烧的研究。Metamizole 是吡唑啉酮类非甾体抗炎药,可抑制COX。
TMIJ-0135 Abiraterone-d4

Abiraterone-d4 是 Abiraterone 的氘代化合物。Abiraterone 的 CAS 号为 154229-19-3。Abiraterone 是不可逆的CYP17A1抑制剂,具有抗雄激素作用,抑制细胞色素 p450 酶 CYP17 的 17α-羟化酶 (IC50:2.5 nM) 和 17,20-裂合酶 (IC50:15 nM) 活性。
T71288 Phenylbutazone-d9

Phenylbutazone-d9 is intended for use as an internal standard for the quantification of phenylbutazone by GC- or LC-MS. Phenylbutazone is a non-steroidal anti-inflammatory drug and an inhibitor of the peroxidase activity of COX (IC50 = ~100 µM in the presence of hydrogen peroxide). It also inhibits prostaglandin I synthase (IC50 = ~25 µM in the presence of hydrogen peroxide). Phenylbutazone (2 mg/kg) reduces increases in type II collagen levels in the inflamed joints of an equine model of LPS-in...
TMIJ-0207 (S)-Ketoprofen-d3

(S)-Ketoprofen-d3 是 (S)-Ketoprofen 的氘代化合物。(S)-Ketoprofen 的 CAS 号为 22161-81-5。S-(+)-Ketoprofen 抑制COX-1和COX-2的IC50值分别为 1.9 和 27 nM。
T71212 Lornoxicam-d4

Lornoxicam-d4 is intended for use as an internal standard for the quantification of lornoxicam by GC- or LC-MS. Lornoxicam is a COX inhibitor and non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory and analgesic properties. It inhibits production of thromboxane B2 from arachidonic acid in HEL human erythroleukemic cells, which endogenously express COX-1, as well as inhibits LPS-induced formation of prostaglandin F1α from arachidonic acid in Mono-Mac-6 cells, which endogenously e...
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...
T71141 Fenspiride-d5

Fenspiride-d5 is intended for use as an internal standard for the quantification of fenspiride by GC- or LC-MS. Fenspiride is an antagonist of histamine H1 receptors and a non-steroidal anti-inflammatory drug (NSAID). It inhibits histamine-induced contraction of isolated guinea pig trachea but not histamine-induced inotropy of isolated guinea pig heart. It also inhibits phosphodiesterase 4 (PDE4), PDE5, and PDE3 (IC50s = 69, ~158, and 363 µM, respectively, in isolated human bronchi derived from ...

同位素标记化合物

Oxaprozin D4
Cat.No: T12336
Synonym: Wy-21743 D4
Target: Others
Meloxicam-d3
Cat.No: T11998
Synonym: Meloxicam D4
Target: Others
Ketorolac-d5
Cat.No: T11754
Synonym: Ketorolac D5
Target: PPAR
DRX-065
Cat.No: T27210
Synonym: DRX 065,DRX065,deuterated R-enantiomer of pioglitazone
Target:
Etoricoxib-d4
Cat.No: T11246
Synonym: MK-0663 D4,依托考昔 D4,L-791456 D4,Etoricoxib D4
Target: Others
Rac Loxoprofen sodium-d3
Cat.No: TMIH-0472
Synonym:
Target:
MefenaMic Acid-d4
Cat.No: TMIH-0325
Synonym:
Target:
Loxoprofen-d4
Cat.No: TMIJ-0211
Synonym:
Target:
Ketorolac-d5-P1
Cat.No: TMIH-0290
Synonym:
Target:
Ketorolac-d5-P2
Cat.No: TMIH-0291
Synonym:
Target:
MAA-d3
Cat.No: TMID-0276
Synonym:
Target:
Abiraterone-d4
Cat.No: TMIJ-0135
Synonym:
Target:
Phenylbutazone-d9
Cat.No: T71288
Synonym:
Target:
(S)-Ketoprofen-d3
Cat.No: TMIJ-0207
Synonym:
Target:
Lornoxicam-d4
Cat.No: T71212
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
Fenspiride-d5
Cat.No: T71141
Synonym:
Target:
TargetMol Loading
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