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Search Results for " silibinin-d3 "

2

抑制剂 & 化合物

1

天然产物

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T35536 Tpl2 Kinase Inhibitor (hydrochloride)

Others Others
Tpl2 kinase inhibitor is an inhibitor of tumor progression locus 2 (Tpl2; IC50= 0.05 μM).1It is selective for Tpl2 over MEK, p38 MAPK, Src, MK2, and PKC (IC50s = >40, 180, >400, 110, and >400 μM, respectively). Tpl2 kinase inhibitor inhibits LPS-induced TNF-α production in isolated human monocytes and whole blood (IC50s = 0.7 and 8.5 μM, respectively). It enhances differentiation induced by calcitriol in HL-60 and U937 leukemia cells when used at a concentration of 5 μM.2Tpl2 kinase inhibitor (5...
T26284 Tpl2-IN-I

Tpl2 inhibitor I,Tpl2-inhibitor-I,Tpl2 IN I,Tpl2 kinase inhibitor

Others Others
Tpl2-IN-I is an inhibitor of tumour progression locus 2 (Tpl2) kinase.

化合物

Tpl2 Kinase Inhibitor (hydrochloride)
Cat.No: T35536
Synonym:
Target: Others
Tpl2-IN-I
Cat.No: T26284
Synonym: Tpl2 inhibitor I,Tpl2-inhibitor-I,Tpl2 IN I,Tpl2 kinase inhibitor
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1660 Silibinin

水飞蓟宾 A,水飞蓟宾,Silibinin A,Silybin,Silymarin I

Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Silibinin (Silybin) 是水飞蓟的主要活性成分,具有抗癌和化疗预防作用,能抑制细胞增殖和迁移。

天然产物

Silibinin
Cat.No: T1660
Synonym: 水飞蓟宾 A,水飞蓟宾,Silibinin A,Silybin,Silymarin I
Target: Reactive Oxygen Species, Autophagy
Cat. No. Product Name Target Signaling Pathways
TMIH-0521 Silibinin-d3

Silibinin-d3Silibinin 的氘代化合物。Silibinin 的 CAS 号为 22888-70-6。Silibinin 是水飞蓟的主要活性成分,具有抗癌和化疗预防作用,能抑制细胞增殖和迁移。

同位素标记化合物

Silibinin-d3
Cat.No: TMIH-0521
Synonym:
Target:
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