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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T21459 |
Splenopentin diacetate
Thymopoietin III pentapeptide (32-36),SP5,Splenopentin Acetate,醋酸脾脏五肽,Splenin pentapeptide (32-36),Arg-lys-glu-val-tyr |
Others | Others |
Splenopentin diacetate (Splenin pentapeptide (32-36)) 是一种合成的免疫调节肽,可以再现脾和胸腺激素胸腺生成素的生物活性。 | |||
T5473 |
ASP5878
ASP-5878 |
FGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
ASP5878 是一种 FGFR 1 (IC50:0.47 nM)、FGFR 2 (IC50:0.6 nM)、FGFR 3 (IC50:0.74 nM)、和 FGFR 4 (IC50:3.5 nM)的抑制剂,具有口服活性,具有潜在的抗肿瘤作用。 | |||
T60130 |
USP5-IN-1
|
DUB | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination |
USP5-IN-1 (compound 64) 是一种有效的去泛素酶USP5抑制剂,与 USP5 ZnF UBD 结合,KD 值为 2.8 μM。USP5-IN-1对九种含有结构相似的 ZnF UBD 结构域的蛋白质具有选择性。USP5-IN-1 抑制 USP5 对双泛素底物的催化裂解。 | |||
T76228 |
ASP5286
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ASP5286 是一种新型的非免疫 cyclophilin 抑制剂,用于研究 HCV。 | |||
T30168 |
ASP5878 HCl
ASP 5878,ASP5878,ASP-5878 |
Others | Others |
ASP5878 is an oral bioavailable fibroblast growth factor receptor (FGFR) inhibitor with potential anti-tumor activity. | |||
T40756 |
[Asp5]-Oxytocin
[Asp5]-Oxytocin |
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[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity. | |||
T76211 |
[Asp5]-Oxytocin acetate
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[Asp5]-Oxytocin acetate 是一款功能强大的5位 (5-position) 神经垂体激素类似物,能引发体外大鼠子宫收缩,其效果可被 Mg2+ 增强。此化合物展现出在大鼠子宫收缩、禽血管抑制及大鼠抗利尿作用方面的活性。 | |||
T22884 |
JW 67
|
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
JW 67 是典型 Wnt 信号通路的抑制剂,IC50为 1.17 μM。它影响由 β- 连环蛋白/GSK-3β/AXIN/APC/CK1 组成的多蛋白复合物,快速降低活性 β- 连环蛋白,随后下调Wnt 靶基因。它也抑制结直肠癌细胞生长。 |
Cat. No. | Product Name | Species | Expression System |
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TMPH-01980 |
SFTPC Protein, Human, Recombinant (GST)
Pulmonary surfactant-associated proteolipid SPL(Val... |
Human | E. coli |
SFTPC Protein, Human, Recombinant (GST) is expressed in E. coli. | |||
TMPY-02211 |
USP5 Protein, Human, Recombinant (His)
ISOT,ubiquitin specific peptidase 5 (isope... |
Human | Baculovirus Insect Cells |
Ubiquitin carboxyl-terminal hydrolase 5, also known as Deubiquitinating enzyme 5, Isopeptidase T, Ubiquitin thiolesterase 5, Ubiquitin-specific-processing protease 5, ISOT and USP5, is a member of the peptidase C19 family. USP5 contains 2 UBA domains and one UBP-type zinc finger. The UBP-type zinc finger domain interacts selectively with an unmodified C-terminus of the proximal ubiquitin. Both UBA domains are involved in polyubiquitin recognition. The UBP-type zinc finger domain crystallizes as ... | |||
TMPH-03489 |
SARS-CoV-2 3C-like proteinase NSP5 Protein (His)
|
SARS-CoV-2 | E. coli |
SARS-CoV-2 3C-like proteinase NSP5 Protein (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 39.8 kDa and the accession number is YP_009725301.1. |