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Search Results for " smyd2 "

Targets Recommended: Histone Methyltransferase

抑制剂 & 化合物

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T12939	SMYD2-IN-1	Histone Methyltransferase	Chromatin/Epigenetic
	SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM).
T6879	LLY-507 LLY507,LLY 507	Histone Methyltransferase	Chromatin/Epigenetic
	LLY-507 是一种有效的、细胞活性的、特异性的蛋白质赖氨酸甲基转移酶 SMYD2 抑制剂。它是一种化学探针，用于解析 SMYD2 在癌症和其他生物过程中的功能。它有抑制 SMYD2 甲基化 p53 肽的能力，IC50小于 15 nM。
TQ0100	AZ505	Histone Methyltransferase	Chromatin/Epigenetic
	AZ505 是一种选择性SMYD2抑制剂，IC50值为 0.12 μM。
T7403	BAY-598	Histone Methyltransferase	Chromatin/Epigenetic
	BAY-598 是SMYD2的选择性抑制剂，IC50值为 27 nM。
T70087	EPZ032597	Histone Methyltransferase	Chromatin/Epigenetic
	EPZ032597 是一种新型 SMYD2 选择性抑制剂，IC50 值为16 nM。EPZ032597 具有抗癌活性，可用于预防和治疗胰腺癌。
T10427	AZ505 ditrifluoroacetate	Histone Methyltransferase	Chromatin/Epigenetic
	AZ505 ditrifluoroacetate is an effective and selective SMYD2 inhibitor (IC50: 0.12 μM).
T63783	AZ506	Others	Others
	AZ506 是一种 SMYD2 的有效抑制剂 (IC50: 17 nM)。AZ506 能够抑制细胞中 SMYD2 甲基转移酶的活性，减少 SMYD2 介导的甲基化信号。
T5381	A-893	Others	Others
	A-893 是一个具有细胞活性的，甲基转移酶SMYD2的抑制剂，IC50值为 2.8 nM。
T26744	BAY-598 R-isomer BAY598 R-isomer,BAY 598 R-isomer	Others	Others
	BAY-598 R-异构体是BAY589的R-异构体，它可用作参考化合物。它是是赖氨酸N-甲基转移酶（SMYD2）的抑制剂，对SMYD2比蛋白酶激活的受体1（PAR1）具有选择性。

化合物

SMYD2-IN-1

Cat.No: T12939

Synonym:

Target: Histone Methyltransferase

LLY-507

Cat.No: T6879

Synonym: LLY507,LLY 507

Target: Histone Methyltransferase

AZ505

Cat.No: TQ0100

Synonym:

Target: Histone Methyltransferase

BAY-598

Cat.No: T7403

Synonym:

Target: Histone Methyltransferase

EPZ032597

Cat.No: T70087

Synonym:

Target: Histone Methyltransferase

AZ505 ditrifluoroacetate

Cat.No: T10427

Synonym:

Target: Histone Methyltransferase

Synonym: BAY598 R-isomer,BAY 598 R-isomer

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-01204	SMYD2 Protein, Human, Recombinant (His) ZMYND14,SET and MYND domain containing 2,HSKM-B,KMT...	Human	Baculovirus Insect Cells
	SET and MYND domain-containing protein 2, also known as HSKM-B, SMYD2, and KMT3C, is a member of the SMYD protein family. It contains one MYND-type zinc finger and one SET domain. Not much is known about SMYD2. However, the interest in better understanding the roles of SMYD2 has grown because of reports indicating that SMYD2 methylates p53 and histone H3. In Xenopus, SMYD1 and SMYD2 were expressed in various muscle tissues and related to muscle cell differentiation. SMYD2 mRNA is most highly exp...