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201

抑制剂 & 化合物

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Cat. No. Product Name
L1710 COVID-19化合物库

1133 compounds
1133 种对SARS-CoV-2有抑制作用或潜在抑制作用的化合物集合,可用于高通量和高内涵筛选;

化合物库

COVID-19化合物库
Cat.No: L1710
Compounds: 1133
Cat. No. Product Name Target Signaling Pathways
T12838 SARS-CoV-IN-2

Others Others
SARS-CoV-IN-2 is an effective SARS-CoV replication inhibitor
T79455 SARS-CoV-2 Mpro-IN-9

SARS-CoV-2 Mpro IN 9,SARS-CoV-2 Mpro-IN 9

SARS-CoV Microbiology/Virology
SARS-CoV-2 Mpro-IN-9 (SARS-CoV-2 Mpro IN 9) 是一种高效的 SARS-CoV-2 Mpro 抑制剂,IC50 值为 80 nM。SARS-CoV-2 Mpro-IN-9 具有抗病毒活性,抑制3C样半胱氨酸蛋白酶,可用于研究病毒感染。
T77510 SARS-CoV-2-IN-46

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-46 是一种 SARS-CoV-2 抑制剂。
T77516 SARS-CoV-2-IN-39

Antiviral; SARS-CoV Immunology/Inflammation; Microbiology/Virology
SARS-CoV-2-IN-39是一种 SARS-CoV-2 抑制剂,EC50 为 1 μM。 SARS-CoV-2-IN-39 具有抗病毒活性,通过抑制 SKP2 蛋白并稳定 BECN1 来抑制 SARS-CoV-2
T77652 SARS-CoV-2 3CLpro-IN-20

Antiviral; SARS-CoV Immunology/Inflammation; Microbiology/Virology
SARS-CoV-2 3CLpro-IN-20 是一种共价的 SARS-CoV-2 3CLpro 抑制剂(IC50s: 0.43 μM,)。SARS-CoV-2 3CLpro-IN-20 具有潜在的抗病毒活性。
T60538 SARS-CoV-2-IN-14

3',5-Dichlorosalicylanilide

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-14 是一种有效的、可口服的 SARS-CoV-2 抑制剂(IC50 :0.39 μM),是一种氯硝柳胺类似物。SARS-CoV-2-IN-14在人血浆和肝 S9 酶测定中比氯硝柳胺稳定性更强。SARS-CoV-2-IN-14以口服的方式给药可以提高其生物利用度和半衰期。
T40340 SARS-CoV-2-IN-10

Others Others
SARS-CoV-2-IN-10 is a powerful and non-toxic inhibitor of SARS-CoV-2 3CL protease, with IC50 and EC50 values of 0.13 nM and 1.03 nM, respectively. The SARS-CoV-2 3C-like protease (3CLpro) is a critical enzyme for viral replication and serves as an ideal target for intervention. By targeting the SARS-CoV-2 3CL protease, SARS-CoV-2-IN-10 has the potential to facilitate the development of effective antiviral drugs specific to SARS-CoV-2.
T12836 SARS-CoV-2-IN-1

Others Others
SARS-CoV-2-IN-1 is a potent inhibitor of Mpro(SARS-CoV-2 Mpro, SARS-CoV Mpro and MERS-CoV Mpro with IC50s of 0.67, 0.90 and 0.58 μM, respectively).
T40207 SARS-CoV-2-IN-7

Others Others
SARS-CoV-2-IN-7 demonstrates potent inhibition of viral replication in SARS-CoV-2-infected Vero E6 cells with an IC50 value of 844 nM.
T38942 SARS-CoV-2-IN-9

Others Others
SARS-CoV-2-IN-9 is an inhibitor binding to subsites S1 and S2 in SARS-CoV-2 main protease.
T40341 SARS-CoV-2-IN-11

Others Others
SARS-CoV-2-IN-11 is a highly potent and non-toxic inhibitor of the 3C-like protease (3CLpro) of SARS-CoV-2, demonstrating IC50 and EC50 values of 0.17 nM and 1.45 nM, respectively. This compound targets the essential viral replication enzyme, 3CLpro, making it an attractive candidate for intervention strategies. SARS-CoV-2-IN-11 holds significant promise in the development of specific antivirals against SARS-CoV-2.
T69535 GRL-0820

SARS-CoV-2-IN-6

SARS-CoV Microbiology/Virology
GRL-0820 (SARS-CoV-2-IN-6) 是一种高效的 SARS-CoV-2 3CLpro 抑制剂,可用于研究新型冠状病毒感染。
T60919 SARS-CoV-2-IN-13

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-13 (compound 6) 是氯硝柳胺的类似物。在人血浆和肝S9酶测定中,SARS-CoV-2-IN-13 比氯硝柳胺更稳定。SARS-CoV-2-IN-13 口服给药时可以提高生物利用度和半衰期。SARS-CoV-2-IN-13 是SARS-CoV-2的有效抑制剂,IC50值为 0.057 μM。
T78961 SARS-CoV-2-IN-38

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-38是一种 可口服的 SARS-CoV-2抑制剂,具有潜在的抗病毒活性,可用于研究 SARS 病毒感染。
T63098 SARS-CoV-2 Mpro-IN-2

SARS-CoV Microbiology/Virology
SARS-CoV-2 Mpro-IN-2 是一种选择性的SARS-CoV-2M pro抑制剂,IC50 值为 0.40 μM。SARS-CoV-2 Mpro-IN-2 具有良好的抗病毒活性,可用于研究 COVID-19。
T79659 SARS-CoV-2 3CLpro-IN-16

SARS-CoV Microbiology/Virology
SARS-CoV-2 3CLpro-IN-16为一种共价 SARS-CoV-2 3CLpro 抑制剂,抑制 3CLpro 活性,通过与Cys145形成共价键实现其抑制作用。
T62413 SARS-CoV-2 nsp13-IN-1

Antiviral Immunology/Inflammation
SARS-CoV-2 nsp13-IN-1 是一种选择性 nsp13(非结构蛋白 13) 抑制剂,具有抗病毒活性,抑制nsp13 ssDNA+ATPase, 可用于研究COVID-19病毒感染 。
T79426 SARS-CoV-2-IN-61

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-61(化合物 8i)是SARS-CoV-2 PLpro的抑制剂,其抗病毒活性表现在其IC50值为16 µM。
T80636 SARS-CoV-2-IN-59

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-59(compound E07)为咪唑啉衍生物,其为一种针对SARS-CoV-2的非肽类小分子抑制剂,主要作用于冠状病毒的Mpro。SARS-CoV-2-IN-59于Mpro残基(Met 165, Gln 166,Met165, His 41, Gln 189)处展现出强烈的相互作用。
T78719 SARS-CoV-2-IN-47

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-47(Compound 13)是一种具有针对SARS-CoV-2变体抑制活性的化合物,显示出对Omicron BA.1的IC50值为0.77 μM,以及对Delta病毒株的IC50值为0.93 μM。该化合物可应用于抗病毒研究领域。
T74946 SARS-CoV-2-IN-28

Others Others
SARS-CoV-2-IN-28 是具备双臂二磷酸 C7 烷基酯和延长分子镊子特征的化合物。该化合物展现出针对SARS-CoV-2的抗病毒效能,能以0.4 μM 的 IC50 抑制 SARS-CoV-2 活性及 1.0 μM 的 IC50 抑制病毒尖刺伪粒子转导。此外,SARS-CoV-2-IN-28 在 EC50 为 4.4 μM 的条件下导致脂质体膜破坏。
T62834 SARS-CoV-2-IN-22

Others Others
SARS-CoV-2-IN-22 是一种 SARS-CoV-2 pseudovirus 抑制剂 (IC50: 16.96 μM)。
T60785 SARS-CoV-2-IN-6

Others Others
SARS-CoV-2-IN-6 是IC50值为73 nM 的SARS-CoV-2 3CLpro 抑制剂。
T60962 SARS-CoV-2-IN-18

Others Others
SARS-CoV-2-IN-18 (Compound 26) 是 SARS-CoV-2 3C-样蛋白酶的有效抑制剂 (IC50 = 45 nM)。
T79243 SARS-CoV-2-IN-43

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-43(Compound 8h)是一种有效的抗病毒剂,能够抑制SARS-CoV-2的复制。
T81207 SARS-CoV-2-IN-64

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-64(compound 9)为鹅去氧胆酸衍生物,对SARS-CoV-2刺突糖蛋白具有显著抑制作用。
T61613 SARS-CoV-2-IN-17

Others Others
SARS-CoV-2-IN-17 (Compound 16) is a highly effective inhibitor of SARS-CoV-2 nucleocapsid protein (NPro). It demonstrates potent anti-viral activity, with an EC50 value of 2.18 μM. Furthermore, SARS-CoV-2-IN-17 binds to NPro with a low Kd value of 7.82 μM, highlighting its potency as a NPro ligand [1].
T81209 SARS-CoV-2-IN-62

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-62 (Compound R3b) 为SARS-CoV-2复制抑制剂,细胞毒性较低。在Vero E6细胞和Calu-3细胞中,其抑制病毒复制的EC50值分别为2.97 μM与3.82 μM。
T79570 SARS-CoV-2-IN-55

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-55 (compound 65) 是一种抑制 SARS-CoV-2 的化合物,具有低细胞毒性,IC50 值为 0.3 μM,它通过作用于病毒的刺突蛋白 S 来抑制病毒感染。
T74948 SARS-CoV-2-IN-30

Others Others
SARS-CoV-2-IN-30是含有苯环的双臂二磷酸酯分子镊,展现出对SARS-CoV-2的抗病毒效应,其通过抑制SARS-CoV-2活力与病毒尖刺伪粒子转导,具有IC50值分别为0.6μM和6.9μM。此外,SARS-CoV-2-IN-30能导致脂质体膜破坏,其EC50值为6.9μM。
T79356 SARS-CoV-2-IN-57

Sigma receptor GPCR/G Protein
SARS-CoV-2-IN-57 (化合物(+)-R-26)是一种针对SARS-CoV-2具有高效抑制活性的化合物,其IC50为80 nM。该化合物对Sigma受体表现出高亲和性,与S1R和S2R的Kis值分别为13.6 nM和14.4 nM。
T63292 SARS-CoV-2-IN-24

Others Others
SARS-CoV-2-IN-24 是类木瓜蛋白酶 (PLpro) 的有效抑制剂,能够诱导 SARS-COV-2 木瓜蛋白酶样蛋白酶的构象变化,对 SARS-COV-2 复制具有抑制作用,能够用于研究 SARS-CoV-2
T72718 SARS-CoV-2-IN-36

Others Others
SARS-CoV-2-IN-36 是一种针对SARS-CoV-2 Mpro(SARS-CoV)的有效抑制剂, 其酶测定的IC50值为2.37 μM,Kd值为1.19 μM。在Vero细胞试验中, SARS-CoV-2-IN-36 对UC-1074、RG2674 及NVDBB-2220 SARS-CoV-2变体展现了抗病毒活性。
T64184 SARS-CoV-2-IN-8

Others Others
SARS-CoV-2-IN-8 是一种 SARS-CoV-2 主要的蛋白酶抑制剂 (IC50: 0.75 μM)。
T79328 SARS-CoV-2-IN-54

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-54(Compound 2)为针对SARS-CoV-2的抑制剂,展现出抗病毒活性。它能在Vero E6细胞中抑制SARS-CoV-2,其IC50值为21.4 μM。
T63694 SARS-CoV-2-IN-33

Others Others
SARS-CoV-2-IN-33 是 COVID-19 抑制剂。ARS-CoV-2-IN-3 对 COVID-19 主要蛋白酶 (Mpro) (PDB ID:6LU7) 表现出较好的结合亲和力 (-8.0 Kcal/mole)。SARS-CoV-2-IN-33 对癌细胞表现出较好的抗增殖效果。SSARS-CoV-2-IN-33 能够用于研究癌症和 COVID-19。
T81203 SARS-CoV-2-IN-68

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-68(compound 6C)是共价SARS-CoV-2 PLpro/Mpro抑制剂,展现出有效抗病毒活性,并与PLpro的锌指结构域发生结合。
T78926 SARS-CoV-2-IN-42

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-42(Compound 8q)是一种有效的SARS-CoV-2复制抑制剂,具有较低的半抑制浓度(EC50: 0.4 μM),且对宿主细胞无明显毒性。
T76270 SARS-CoV-2-IN-34

SARS-CoV-2-IN-34 (S-20-1) 是一种可穿透血脑屏障的 pan-coronavirus (CoV) fusion 抑制剂,具有广谱抑制活性。它能有效抑制伪型和真型 SARS-CoV-2 以及其变体 (VOCs) 的感染。SARS-CoV-2-IN-34 对 SARS-CoV-2 的 S1 和 S2 蛋白中的 HR1 和 RBD 结构域显示出高度亲和性,适用于感染研究。
T74947 SARS-CoV-2-IN-29

Others Others
SARS-CoV-2-IN-29为含苯环的双臂二磷酸酯分子镊子,展现出对SARS-CoV-2的抗病毒效果,其抑制SARS-CoV-2活性及病毒尖刺伪粒子转导的IC50值分别为1.5 μM与1.6 μM。此外,SARS-CoV-2-IN-29能破坏脂质体膜,其EC50值为3.0 μM。
T63181 SARS-CoV-2-IN-32

Others Others
SARS-CoV-2-IN-32 是一种 COVID-19 抑制剂。SARS-CoV-2-IN-32COVID-19 主要蛋白酶 (Mpro) (PDB ID:6LU7) 表现出较好的结合亲和力 (-8.8 Kcal/mole),且对癌细胞具有抗增殖作用。SARS-CoV-2-IN-32 能够用于研究癌症和 COVID-19。
T81206 SARS-CoV-2-IN-65

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-65(compound 2f(81))是一种具有口服活性的有效可逆SARS-CoV-2进入抑制剂。它通过抑制Calu-3细胞中RBD:ACE2的相互作用和TMPRSS2的活性,阻断了假病毒通过ACE2依赖性途径的进入。
T74945 SARS-CoV-2-IN-27

Others Others
SARS-CoV-2-IN-27 为具有扩展长度的双臂二磷酸 C6 烷基酯分子镊子,显示出针对 SARS-CoV-2 的抗病毒活性。其抑制 SARS-CoV-2 活力的 IC50 为 1.0 μM,针对病毒尖刺伪粒子转导的 IC50 为 1.7 μM。此外,该化合物能引起脂质体膜破坏,其 EC50 为 6.5 μM。
T81204 SARS-CoV-2-IN-67

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-67 (Compound 16) 是抗SARS-CoV-2的维生素K衍生物,其在VeroE6/TMPRSS2细胞中EC50值为64.8 μM。该化合物能够抑制SARS-CoV-2 RdRp活性。
T78720 SARS-CoV-2-IN-48

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-48 (compound 19)是针对SARS-CoV-2的抑制剂,对Omicron BA.1的IC50值为2.7 μM,展现出了抗病毒活性。
T74943 SARS-CoV-2-IN-25

Others Others
SARS-CoV-2-IN-25 (Compound CP026) 是一种有效的 SARS-CoV-2刺突伪粒子转导抑制剂,IC50为 1.6 μM。SARS-CoV-2-IN-25 抑制包膜病毒和脂质体。
T79245 SARS-CoV-2-IN-45

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-45(Compound 8p)是SARS-CoV-2的有效抑制剂,能够在Calu-3细胞中抑制病毒复制,其EC50值为0.5 μM,同时没有显著的细胞毒性。
T81202 SARS-CoV-2-IN-69

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-69 (Compound 7E)是一种SARS-CoV-2的非共价抑制剂,具有7.4 μM的EC50值。它有效针对SARS-CoV-2的主蛋白酶(Mpro)并作为木瓜蛋白酶(PLpro)的非共价抑制剂。
T78713 SARS-CoV-2-IN-40

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-40(Compound 19)为SARS-CoV-2抑制剂。该化合物在Calu3肺细胞中针对SARS-CoV-2 BA.1及BA.5变体的感染具有抑制作用,其IC50s分别为100 nM与160 nM。
T78765 SARS-CoV-2-IN-51

SARS-CoV Microbiology/Virology
SARS-CoV-2-IN-51(S-10)为针对Omicron的融合抑制剂有效先导化合物,具有抑制Omicron及其他变体的能力,EC50值介于0.82-5.45 μM之间。该化合物通过与SARS-CoV-2病毒S蛋白预融合状态下直接相互作用,从而抑制病毒进入。

化合物

SARS-CoV-IN-2
Cat.No: T12838
Synonym:
Target: Others
SARS-CoV-2 Mpro-IN-9
Cat.No: T79455
Synonym: SARS-CoV-2 Mpro IN 9,SARS-CoV-2 Mpro-IN 9
Target: SARS-CoV
SARS-CoV-2-IN-46
Cat.No: T77510
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-39
Cat.No: T77516
Synonym:
Target: Antiviral, SARS-CoV
SARS-CoV-2 3CLpro-IN-20
Cat.No: T77652
Synonym:
Target: Antiviral, SARS-CoV
SARS-CoV-2-IN-14
Cat.No: T60538
Synonym: 3',5-Dichlorosalicylanilide
Target: SARS-CoV
SARS-CoV-2-IN-10
Cat.No: T40340
Synonym:
Target: Others
SARS-CoV-2-IN-1
Cat.No: T12836
Synonym:
Target: Others
SARS-CoV-2-IN-7
Cat.No: T40207
Synonym:
Target: Others
SARS-CoV-2-IN-9
Cat.No: T38942
Synonym:
Target: Others
SARS-CoV-2-IN-11
Cat.No: T40341
Synonym:
Target: Others
GRL-0820
Cat.No: T69535
Synonym: SARS-CoV-2-IN-6
Target: SARS-CoV
SARS-CoV-2-IN-13
Cat.No: T60919
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-38
Cat.No: T78961
Synonym:
Target: SARS-CoV
SARS-CoV-2 Mpro-IN-2
Cat.No: T63098
Synonym:
Target: SARS-CoV
SARS-CoV-2 3CLpro-IN-16
Cat.No: T79659
Synonym:
Target: SARS-CoV
SARS-CoV-2 nsp13-IN-1
Cat.No: T62413
Synonym:
Target: Antiviral
SARS-CoV-2-IN-61
Cat.No: T79426
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-59
Cat.No: T80636
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-47
Cat.No: T78719
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-28
Cat.No: T74946
Synonym:
Target: Others
SARS-CoV-2-IN-22
Cat.No: T62834
Synonym:
Target: Others
SARS-CoV-2-IN-6
Cat.No: T60785
Synonym:
Target: Others
SARS-CoV-2-IN-18
Cat.No: T60962
Synonym:
Target: Others
SARS-CoV-2-IN-43
Cat.No: T79243
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-64
Cat.No: T81207
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-17
Cat.No: T61613
Synonym:
Target: Others
SARS-CoV-2-IN-62
Cat.No: T81209
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-55
Cat.No: T79570
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-30
Cat.No: T74948
Synonym:
Target: Others
SARS-CoV-2-IN-57
Cat.No: T79356
Synonym:
Target: Sigma receptor
SARS-CoV-2-IN-24
Cat.No: T63292
Synonym:
Target: Others
SARS-CoV-2-IN-36
Cat.No: T72718
Synonym:
Target: Others
SARS-CoV-2-IN-8
Cat.No: T64184
Synonym:
Target: Others
SARS-CoV-2-IN-54
Cat.No: T79328
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-33
Cat.No: T63694
Synonym:
Target: Others
SARS-CoV-2-IN-68
Cat.No: T81203
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-42
Cat.No: T78926
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-34
Cat.No: T76270
Synonym:
Target:
SARS-CoV-2-IN-29
Cat.No: T74947
Synonym:
Target: Others
SARS-CoV-2-IN-32
Cat.No: T63181
Synonym:
Target: Others
SARS-CoV-2-IN-65
Cat.No: T81206
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-27
Cat.No: T74945
Synonym:
Target: Others
SARS-CoV-2-IN-67
Cat.No: T81204
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-48
Cat.No: T78720
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-25
Cat.No: T74943
Synonym:
Target: Others
SARS-CoV-2-IN-45
Cat.No: T79245
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-69
Cat.No: T81202
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-40
Cat.No: T78713
Synonym:
Target: SARS-CoV
SARS-CoV-2-IN-51
Cat.No: T78765
Synonym:
Target: SARS-CoV
Cat. No. Product Name Target Signaling Pathways
T72581 SARS-CoV MPro-IN-2

Others Others
SARS-CoVMPro-IN-2 是一种有效的SARS-CoV-2 Mpro 抑制剂,IC50sub>值为 72.07 nM。病毒的主要蛋白酶 Mpro 作为加工病毒多蛋白的主要酶,有助于 SARS-CoV-2 在宿主细胞中的复制和转录,并已被定性为药物发现的有吸引力的靶点。SARS-CoVMPro-IN-2 具有研究 COVID-19 的潜力。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
TN3651 Cichoriin

Others Others
CichoriinSARS-CoV-2有明显活性,是治疗重症COVID-19的潜在候选物质。
T2869 Emodin

Frangula emodin,大黄素

SARS-CoV; Casein Kinase; Autophagy Autophagy; Metabolism; Microbiology/Virology; Stem Cells
Emodin (Frangula emodin) 是蒽醌衍生物,有抗SARS-CoV 作用。它阻断 SARS 冠状病毒刺突蛋白和血管紧张素转化酶 2 的相互作用。它抑制酪蛋白激酶 2 ,具有抗炎和抗癌作用。它可改善饮食诱导的肥胖小鼠的代谢紊乱。
T2563 Acetyl-L-carnitine hydrochloride

Acetyl L-carnitine hydrochloride,O-Acetylcarnitine,乙酰-L-肉(毒)碱盐酸盐,O-acetyl-L-carnitine,O-Acetyl-L-carnitine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
Acetyl-L-carnitine hydrochloride (Acetyl L-carnitine hydrochloride) 是一种由内源性左旋肉碱的乙酰化形式的盐酸盐组成的营养补充剂,具有潜在的神经保护、认知增强、抗抑郁和免疫调节活性。还可缓解化疗、糖尿病或其他疾病引起的周围神经病变。此外,乙酰左旋肉碱可能通过增加T淋巴细胞成熟来调节免疫反应,并可能下调促炎细胞因子对病毒(如SARS-CoV-2)的反应。它还可能破坏ACE2信号通路并抑制活性氧(ROS)的产生。
T21883 Gedunin

HSP Cytoskeletal Signaling; Metabolism
Gedunin 是从印楝种子中提取的一种重要柠檬苦素,具有抗癌、抗病毒、抗炎和杀虫活性。它可阻断 SARS-CoV-2 病毒进入人宿主细胞,用于 COVID-19 研究。它是Hsp90抑制剂,诱导 Hsp90 依赖的蛋白降解,抑制卵巢癌细胞增殖。
T6670 Silymarin

Silybin B,水飞蓟素

SARS-CoV Microbiology/Virology
Silymarin (Silybin B) 是一种多酚类黄酮,是从水飞蓟或水飞蓟的种子中提取的一种 SARS-CoV-2 主蛋白酶抑制剂。它可降低肿瘤细胞的增殖,血管生成以及胰岛素抵抗,用于预防和治疗肝脏疾病,有潜力研究 COVID-19 。
T79947 10-Hydroxyaloin A

SARS-CoV Microbiology/Virology
10-Hydroxyaloin A有效抑制SARS-CoV-2,与SARS-CoV-2 Mpro活性位点显著结合。
T80010 (25S)-Antcin B

SARS-CoV Microbiology/Virology
Antcin-B是3CLPro的高亲和力有效抑制剂,可用于SARS-CoV-2的研究。
T73900 (±)-Alliin

Others Others
(±)-Alliin 是大蒜的主要活性成分。(±)-Alliin 被认为是SARS-CoV-2 (Mpro)的虚拟抑制剂。

天然产物

SARS-CoV MPro-IN-2
Cat.No: T72581
Synonym:
Target: Others
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Cichoriin
Cat.No: TN3651
Synonym:
Target: Others
Emodin
Cat.No: T2869
Synonym: Frangula emodin,大黄素
Target: SARS-CoV, Casein Kinase, Autophagy
Acetyl-L-carnitine hydrochloride
Cat.No: T2563
Synonym: Acetyl L-carnitine hydrochloride,O-Acetylcarnitine,乙酰-L-肉(毒)碱盐酸盐,O-acetyl-L-carnitine,O-Acetyl-L-carnitine hydrochloride
Target: Others, Endogenous Metabolite
Gedunin
Cat.No: T21883
Synonym:
Target: HSP
Silymarin
Cat.No: T6670
Synonym: Silybin B,水飞蓟素
Target: SARS-CoV
10-Hydroxyaloin A
Cat.No: T79947
Synonym:
Target: SARS-CoV
(25S)-Antcin B
Cat.No: T80010
Synonym:
Target: SARS-CoV
(±)-Alliin
Cat.No: T73900
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPY-05679 SARS-CoV-2 Spike RBD Protein (hFc)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (hFc) is expressed in HEK293 mammalian cells. The predicted molecular weight is 51.8 kDa and the accession number is A0A6G7K2L4.
TMPY-06078 SARS-CoV-2 envelope(CoV-E) protein Protein (C40A & C43A & C44A, His & MBP)

SARS-CoV-2 E. coli
SARS-CoV-2 envelope(CoV-E) protein Protein (C40A & C43A & C44A, His & MBP) is expressed in E. coli expression system. The predicted molecular weight is 52.2 kDa and the accession number is YP_009724392.1.
TMPY-06615 SARS-CoV-2 XBB (Omicron) Spike S1+S2 trimer Protein (His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 XBB (Omicron) Spike S1+S2 trimer Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 136.26 kDa and the accession number is YP_009724390.1.
TMPY-06626 SARS-COV-2 BQ.1/BQ.1.1 (Omicron) Nucleoprotein/NP Protein (His)

SARS-CoV-2 E. coli
SARS-COV-2 BQ.1/BQ.1.1 (Omicron) Nucleoprotein/NP Protein (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 46.36 kDa and the accession number is YP_009724397.2.
TMPY-06071 SARS-CoV-2 RNA-dependent RNA polymerase/RDRP Protein (His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 RNA-dependent RNA polymerase/RDRP Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 108.3 kDa and the accession number is YP_009725307.1.
TMPK-00265 SARS-COV-2 Nucleocapsid Protein (His & Avi), Biotinylated

Nucleocapsid,NC,NP

SARS-CoV-2 E. coli
Nucleocapsid protein (N) is the major viral structural component; its main function is to protect and encapsidate the viral RNA forming viral RNP complex. It is encoded by the S segment vRNA and is abundantly expressed in the cytoplasm of infected cells. SARS-COV-2 Nucleocapsid Protein (His & Avi), Biotinylated is expressed in E. coli expression system with N-His-Avi tag. The predicted molecular weight is 48.9 kDa and the accession number is P0DTC9.
TMPY-05664 SARS-CoV-2 Nucleocapsid Protein (His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Nucleocapsid Protein (His) is expressed in Baculovirus insect cells. The predicted molecular weight is 47.08 kDa and the accession number is P0DTC9.
TMPY-06040 SARS-CoV-2 Spike RBD Protein (G446V, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (G446V, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06044 SARS-CoV-2 Spike RBD Protein (Y505C, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Y505C, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05982 SARS-CoV-2 Spike RBD Protein (A372T, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A372T, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05959 SARS-CoV-2 Spike RBD Protein (V341I, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V341I, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06003 SARS-CoV-2 Spike RBD Protein (P337S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (P337S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05960 SARS-CoV-2 Spike RBD Protein (Y508H, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Y508H, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05681 SARS-CoV-2 Spike RBD Protein (rFc)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (rFc) is expressed in HEK293 mammalian cells. The predicted molecular weight is 50.3 kDa and the accession number is A0A6G7K2L4.
TMPY-05988 SARS-CoV-2 Spike RBD Protein (N370S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (N370S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05962 SARS-CoV-2 Spike RBD Protein (V503F, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V503F, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06004 SARS-CoV-2 Spike RBD Protein (P521R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (P521R, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05983 SARS-CoV-2 Spike RBD Protein (A344S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A344S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05989 SARS-CoV-2 Spike RBD Protein (Q414R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Q414R, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05987 SARS-CoV-2 Spike RBD Protein (K378N, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (K378N, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05967 SARS-CoV-2 Spike RBD Protein (A522S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A522S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05993 SARS-CoV-2 Spike RBD Protein (T393P, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (T393P, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05998 SARS-CoV-2 Spike RBD Protein (N440K, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (N440K, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06049 SARS-CoV-2 Spike RBD Protein (V445F, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V445F, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06098 SARS-CoV-2 Nucleocapsid Protein (I292T, His)

SARS-CoV-2 E. coli
SARS-CoV-2 Nucleocapsid Protein (I292T, His) is expressed in E. coli expression system. The predicted molecular weight is 46.6 kDa and the accession number is P0DTC9.
TMPY-06890 SARS-CoV-2 XBB.1.16 (Omicron) Spike S1 Protein (His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 XBB.1.16 (Omicron) Spike S1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.6 kDa.
TMPY-05991 SARS-CoV-2 Spike RBD Protein (S477N, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (S477N, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05691 SARS-CoV-2 (2019-nCoV) Spike RBD Protein

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 (2019-nCoV) Spike RBD Protein is expressed in HEK293 mammalian cells. The predicted molecular weight is 25.1 kDa and the accession number is A0A6G7K2L4.
TMPY-05995 SARS-CoV-2 Spike RBD Protein (G485S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (G485S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06043 SARS-CoV-2 Spike RBD Protein (F456L, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F456L, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05978 SARS-CoV-2 Spike RBD Protein (S359N, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (S359N, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06086 SARS-CoV-2 Helicase Protein (His)

SARS-CoV-2 E. coli
SARS-CoV-2 Helicase Protein (His) is expressed in E. coli expression system. The predicted molecular weight is 67.8 kDa and the accession number is YP_009725308.1.
TMPY-05723 SARS-CoV-2 Spike S1 Protein (D614G, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike S1 Protein (D614G, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 76.41 kDa and the accession number is A0A6G7K2L4.
TMPY-05977 SARS-CoV-2 Spike RBD Protein (V483I, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V483I, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05751 SARS-CoV-2 Spike RBD Protein (W436R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (W436R, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.51 kDa and the accession number is A0A6G7K2L4.
TMPY-05976 SARS-CoV-2 Spike RBD Protein (T478I, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (T478I, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06065 SARS-CoV-2 Spike RBD Protein (A475V, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A475V, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06070 SARS-CoV-2 Spike RBD Protein (F490L, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F490L, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-06097 SARS-CoV-2 Nucleocapsid Protein (S194L, His)

SARS-CoV-2 E. coli
SARS-CoV-2 Nucleocapsid Protein (S194L, His) is expressed in E. coli expression system. The predicted molecular weight is 46.6 kDa and the accession number is P0DTC9.
TMPY-05974 SARS-CoV-2 Spike RBD Protein (L452R, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (L452R, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-06002 SARS-CoV-2 Spike RBD Protein (K417N, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (K417N, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05984 SARS-CoV-2 Spike RBD Protein (A520V, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A520V, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05663 SARS-CoV-2 Spike RBD Protein (mFc)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (mFc) is expressed in HEK293 mammalian cells. The predicted molecular weight is 51.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05971 SARS-CoV-2 Spike RBD Protein (A348S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A348S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.6 kDa and the accession number is A0A6G7K2L4.
TMPY-05666 SARS-CoV-2 Spike S2 ECD Protein (His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S2 ECD Protein (His) is expressed in Baculovirus insect cells. The predicted molecular weight is 59.37 kDa and the accession number is A0A6G7K2L4.
TMPY-05986 SARS-CoV-2 Spike RBD Protein (F490S, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F490S, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.5 kDa and the accession number is A0A6G7K2L4.
TMPY-05704 SARS-CoV-2 Spike RBD Protein (F342L, His)

SARS-CoV-2 HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F342L, His) is expressed in HEK293 mammalian cells. The predicted molecular weight is 26.51 kDa and the accession number is A0A6G7K2L4.
TMPY-05667 SARS-CoV-2 Spike S1 Protein (His)

SARS-CoV-2 Baculovirus Insect Cells
SARS-CoV-2 Spike S1 Protein (His) is expressed in Baculovirus insect cells. The predicted molecular weight is 76.45 kDa and the accession number is A0A6G7K2L4.
TMPY-05661 SARS-CoV-2 Spike S1 Protein (HEK293, His)

HEK293 Cells
SARS-CoV-2 Spike S1 Protein (HEK293, His) is expressed in HEK293 mammalian cells with His tag. The accession number is A0A6G7K2L4.
TMPH-03491 SARS-CoV-2 Non-structural protein 9/NSP9 Protein (His)

SARS-CoV-2 E. coli
SARS-CoV-2 Non-structural protein 9/NSP9 Protein (His) is expressed in E. coli.
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重组蛋白

SARS-CoV-2 Spike RBD Protein (hFc)
Cat.No: TMPY-05679
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 envelope(CoV-E) protein Protein (C40A & C43A & C44A, His & MBP)
Cat.No: TMPY-06078
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 XBB (Omicron) Spike S1+S2 trimer Protein (His)
Cat.No: TMPY-06615
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-COV-2 BQ.1/BQ.1.1 (Omicron) Nucleoprotein/NP Protein (His)
Cat.No: TMPY-06626
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 RNA-dependent RNA polymerase/RDRP Protein (His)
Cat.No: TMPY-06071
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-COV-2 Nucleocapsid Protein (His & Avi), Biotinylated
Cat.No: TMPK-00265
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 Nucleocapsid Protein (His)
Cat.No: TMPY-05664
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike RBD Protein (G446V, His)
Cat.No: TMPY-06040
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Y505C, His)
Cat.No: TMPY-06044
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A372T, His)
Cat.No: TMPY-05982
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V341I, His)
Cat.No: TMPY-05959
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (P337S, His)
Cat.No: TMPY-06003
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Y508H, His)
Cat.No: TMPY-05960
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (rFc)
Cat.No: TMPY-05681
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (N370S, His)
Cat.No: TMPY-05988
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V503F, His)
Cat.No: TMPY-05962
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (P521R, His)
Cat.No: TMPY-06004
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A344S, His)
Cat.No: TMPY-05983
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (Q414R, His)
Cat.No: TMPY-05989
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (K378N, His)
Cat.No: TMPY-05987
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A522S, His)
Cat.No: TMPY-05967
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (T393P, His)
Cat.No: TMPY-05993
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (N440K, His)
Cat.No: TMPY-05998
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V445F, His)
Cat.No: TMPY-06049
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Nucleocapsid Protein (I292T, His)
Cat.No: TMPY-06098
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 XBB.1.16 (Omicron) Spike S1 Protein (His)
Cat.No: TMPY-06890
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (S477N, His)
Cat.No: TMPY-05991
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 (2019-nCoV) Spike RBD Protein
Cat.No: TMPY-05691
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (G485S, His)
Cat.No: TMPY-05995
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F456L, His)
Cat.No: TMPY-06043
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (S359N, His)
Cat.No: TMPY-05978
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Helicase Protein (His)
Cat.No: TMPY-06086
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 Spike S1 Protein (D614G, His)
Cat.No: TMPY-05723
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (V483I, His)
Cat.No: TMPY-05977
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (W436R, His)
Cat.No: TMPY-05751
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (T478I, His)
Cat.No: TMPY-05976
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A475V, His)
Cat.No: TMPY-06065
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F490L, His)
Cat.No: TMPY-06070
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Nucleocapsid Protein (S194L, His)
Cat.No: TMPY-06097
Species: SARS-CoV-2
Expression System: E. coli
SARS-CoV-2 Spike RBD Protein (L452R, His)
Cat.No: TMPY-05974
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (K417N, His)
Cat.No: TMPY-06002
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A520V, His)
Cat.No: TMPY-05984
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (mFc)
Cat.No: TMPY-05663
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (A348S, His)
Cat.No: TMPY-05971
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S2 ECD Protein (His)
Cat.No: TMPY-05666
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike RBD Protein (F490S, His)
Cat.No: TMPY-05986
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike RBD Protein (F342L, His)
Cat.No: TMPY-05704
Species: SARS-CoV-2
Expression System: HEK293 Cells
SARS-CoV-2 Spike S1 Protein (His)
Cat.No: TMPY-05667
Species: SARS-CoV-2
Expression System: Baculovirus Insect Cells
SARS-CoV-2 Spike S1 Protein (HEK293, His)
Cat.No: TMPY-05661
Species:
Expression System: HEK293 Cells
SARS-CoV-2 Non-structural protein 9/NSP9 Protein (His)
Cat.No: TMPH-03491
Species: SARS-CoV-2
Expression System: E. coli
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Cat. No. Product Name Target Signaling Pathways
TMIH-0146 Chloroquine-d5

Chloroquine-d5 是 Chloroquine 的氘代化合物。Chloroquine 的 CAS 号为 54-05-7。Chloroquine 是一种自噬和 Toll 样受体抑制剂。 氯喹是一种抗疟疾和抗炎剂,广泛用于治疗疟疾和类风湿性关节炎。它在体外控制 SARS-CoV-2 (COVID-19) 感染方面非常有效,EC50 为 1.13 μM。
T38297 Ribavirin-13C5

Ribavirin-13C5

Ribavirin-13C5is intended for use as an internal standard for the quantification of ribavirin by GC- or LC-MS. Ribavirin is an antiviral guanosine nucleoside analog.1,2Upon entry into cells, ribavirin is metabolized to an active triphosphate form that induces viral RNA chain termination and inhibits viral polymerases. It reduces replication in a panel of seven RNA and four DNA viruses in Vero cells (EC50s = 2-95 μg/ml).3Ribavirin also reduces replication of severe acute respiratory syndrome coro...
TMIJ-0339 Bromhexine-d3 HCl

Bromhexine-d3 HCl 是 Bromhexine HCl 的氘代化合物。Bromhexine HCl 的 CAS 号为 611-75-6。Bromhexine hydrochloride 是TMPRSS2蛋白酶的一种特异性有效抑制剂,IC50为 0.75 μM。它可预防和控制SARS-CoV-2感染。它是一种粘液溶解剂,用于治疗与粘稠或过多粘液相关的呼吸系统疾病。
TMID-0208 Hydroxychloroquine-d5

Hydroxychloroquine-d5 是 Hydroxychloroquine 的氘代化合物。Hydroxychloroquine 的 CAS 号为 118-42-3。Hydroxychloroquine 是一种合成抗疟疾剂,有效抑制SARS-CoV-2感染,也抑制 Toll 样受体 7/9 信号传导。

同位素标记化合物

Chloroquine-d5
Cat.No: TMIH-0146
Synonym:
Target:
Ribavirin-13C5
Cat.No: T38297
Synonym: Ribavirin-13C5
Target:
Bromhexine-d3 HCl
Cat.No: TMIJ-0339
Synonym:
Target:
Hydroxychloroquine-d5
Cat.No: TMID-0208
Synonym:
Target:
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