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Search Results for " riluzole hydrochloride "
Targets Recommended: GABA Receptor

2

抑制剂 & 化合物

1

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T41265 Riluzole hydrochloride

AQST-117 hydrochloride,PK 26124 hydrochloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Riluzole hydrochloride (PK 26124 hydrochloride) 是一种抗惊厥化合物,属于钠通道阻滞剂家族,抑制 GABA 摄取。Riluzole hydrochloride是钠-谷氨酸拮抗剂,具有抗癌和神经保护活性,可用于研究肌萎缩侧索硬化症和神经系统疾病。
T0349 Riluzole

PK 26124,RP-54274,利鲁唑

GABA Receptor; Sodium Channel; NMDAR Membrane transporter/Ion channel; Neuroscience
Riluzole (RP-54274) 是一种谷氨酸拮抗剂,用作抗惊厥药并延长肌萎缩侧索硬化症患者的生存期。它还抑制 GABA 摄取,IC50值为 43 μM。

化合物

Riluzole hydrochloride
Cat.No: T41265
Synonym: AQST-117 hydrochloride,PK 26124 hydrochloride
Target: GABA Receptor
Riluzole
Cat.No: T0349
Synonym: PK 26124,RP-54274,利鲁唑
Target: GABA Receptor, Sodium Channel, NMDAR
Cat. No. Product Name Target Signaling Pathways
T37608 Riluzole-13C,15N2

Riluzole-13C,15N2

Riluzole-13C,15N2 is intended for use as an internal standard for the quantification of riluzole by GC- or LC-MS. Riluzole is a benzothiazole derivative with anti-excitotoxic effects that acts by blocking the presynaptic release of glutamate, indirectly antagonizing glutamate receptors, and inactivating neuronal voltage-gated Na+ channels (ED50 = 2.3 μM). Riluzole suppresses glutamate-induced seizures in rats at an ED50 value of 3.2 mg/kg and displays neuroprotective effects in hypoxic animals a...

同位素标记化合物

Riluzole-13C,15N2
Cat.No: T37608
Synonym: Riluzole-13C,15N2
Target:
TargetMol Loading
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