Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T26253 |
Tecastemizole
Norastemizole,R-43512,R43512,R 43512,T 1348 |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Tecastemizole (R 43512) 是 H1 受体的选择性拮抗剂,是阿司咪唑的主要代谢产物,具有抗炎作用。 | |||
T1278 |
Astemizole
Laridal,Histaminos,Paralergin,阿司咪唑 |
Potassium Channel; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience |
Astemizole (Laridal) 是一种长效、非镇静抗组胺药,用于治疗季节性过敏性鼻炎、哮喘、过敏性结膜炎和慢性特发性荨麻疹。它是组胺 H1 受体的拮抗剂,IC50值为 4 nM,还阻断 hERG K+通道,IC50值为 0.9 nM,具有抗胆碱能和止痒作用。 |