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Search Results for " potassium "
Targets Recommended: Potassium Channel Others

513

抑制剂 & 化合物

83

天然产物

3

化合物库

26

重组蛋白

17

同位素标记化合物

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Cat. No. Product Name
L7300 钾通道分子库

152 compounds
152 种钾通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7400 钠通道分子库

118 compounds
118 种钠通道相关化合物的独特集合,可用于高通量筛选和高内涵筛选;
L7110 抗高血压化合物库

678 compounds
678 种高血压相关的小分子,用于高通量和高内涵筛选;

化合物库

钾通道分子库
Cat.No: L7300
Compounds: 152
钠通道分子库
Cat.No: L7400
Compounds: 118
抗高血压化合物库
Cat.No: L7110
Compounds: 678
Cat. No. Product Name Target Signaling Pathways
T5987 Potassium oxonate

Oxonic Acid (potassium salt),氧嗪酸钾,Potassium otastat,Potassium azaorotate

Others Others
Potassium oxonate (Potassium azaorotate) 是用作尿酸酶抑制剂,都5-FU 磷酸化为5-fluorouridine-5'-monophosphate 具有抑制作用。
T68022L Sulotroban potassium

BM 13177 potassium,Sulotroban potassium(72131-33-0 Free base)

PPAR DNA Damage/DNA Repair; Metabolism
Sulotroban potassium 是一种小分子血栓素A2受体(TXA2R)拮抗剂,可用于研究心肌梗塞和血栓形成。
T3096 Canrenoate potassium

坎利酸钾,Potassium aldadiene,Canrenoic acid potassium salt,Potassium canrenoate,Soldactone

Glucocorticoid Receptor Endocrinology/Hormones
Canrenoate potassium (Soldactone) 是一种有效的竞争性盐皮质激素受体 (mineralocorticoid receptor) 拮抗剂,是一种释放 canrenone 的前药。它作为一种利尿剂,用于高血压的研究。
T35381 Aluminum potassium sulfate

Potassium Aluminium Sulfate,APS

Others Others
Aluminum potassium sulfate (Potassium Aluminium Sulfate) 可用于研究严重急性呼吸系统综合症,可用于预防和治疗癌症。
T2239 Raltegravir potassium

MK 0518 potassium salt,Raltegravir potassium salt,雷特格韦钾盐

HIV Protease; Integrase Microbiology/Virology; Proteases/Proteasome
Raltegravir potassium (MK 0518 potassium salt) 是一种整合酶抑制剂,用于研究 HIV 感染。
T8129 Potassium acetate

Diuretic salt,Potassium ethanoate,乙酸钾

Antifungal Microbiology/Virology
Potassium acetate (Diuretic salt) 是一种钾盐,能够用于补充电解质,恢复水电解质平衡,也能用于制备细菌碱性裂解的中和液,以及纯化 DNA 和蛋白质。
T0481 Azilsartan Medoxomil Potassium

TAK-491 Potassium

Azilsartan Medoxomil Potassium (TAK-491 Potassium) 是一种具有口服活性的1型血管紧张素 II 受体拮抗剂(IC50: 0.62 nM)。
T19498 p-Cresyl sulfate potassium

p-Tolyl sulfate potassium salt,p-Cresol sulfate potassium,p-Methylphenyl potassium sulfate,对甲基硫酸钾,Potassium p-tolyl sulfate

Endogenous Metabolite Metabolism
p-Cresyl sulfate potassium (p-Tolyl sulfate potassium salt) 是一种尿毒症毒素,能够与原型蛋白质结合。
T3267 Potassium guaiacolsulfonate hemihydrate

愈创木酚磺酸钾水合物,Potassium guaiacolsulfonate,Potassium 4-guaiacolsulfonate hemihydrate,愈创木酚磺酸钾

Antibacterial; Antibiotic Microbiology/Virology
Potassium guaiacolsulfonate hemihydrate (Potassium guaiacolsulfonate) 是一种芳香族磺酸,在医药中用作祛痰剂,可治疗急性呼吸道感染。它可松弛粘液,与其他药物合用,可治疗普通感冒、感染或过敏引起的咳嗽。
T5580 1-Naphthaleneacetic acid potassium salt

α-萘醋酸钾,α-Naphthaleneacetic acid,Potassium alpha-naphthylacetate,Potassium 1-Naphthaleneacetate,1-NAA Potassium Salt

Phospholipase Metabolism
1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) 是一种合成的植物生长素,能够促进植物生长,也是一种PLA2抑制剂,IC50=13.16 μM。
T22328 Ethyl potassium malonate

Potassium 3-ethoxy-3-oxopropanoate,Malonic Acid Monoethyl Ester Potassium Salt,丙二酸单乙酯钾盐

Others Others
Ethyl potassium malonate 是琥珀酸脱氢酶的竞争性抑制剂,可作为生产丙二酸(三甲基甲硅烷基)乙酯的前体,丙二酸乙酯用于通过酰化制备 β-酮酯,并作为制备丙二酸叔丁酯的中间体。
T0215 Losartan potassium

DuP-753 potassium,洛沙坦钾,氯沙坦钾,MK 954,DuP 753

RAAS Endocrinology/Hormones
Losartan potassium (DuP-753 potassium) 是一种血管紧张素 II 受体 1 型(AT1)拮抗剂,能够与血管紧张素 II 与 AT1 的结合竞争,其 IC50=20 nM。
T36008 Nebentan potassium

YM598

Endothelin Receptor GPCR/G Protein
Nebentan potassium (YM598) 是一种具有口服活性和选择性的非肽类内皮素受体 (ETA receptor) 拮抗剂。Nebentan potassium 抑制肺动脉高压,可用于研究神经系统疾病和心血管疾病。
T4139 D-Luciferin potassium

D-Luciferin K Salt,D-Luciferin Potassium Salt,D-萤光素钾盐,D-荧光素钾盐

Others Others
D-Luciferin potassium (D-Luciferin K Salt) 是一种荧光素酶 (Luc) 的底物,能够催化生物发光昆虫产生典型的黄绿光 (560 nm)。D-Luciferin potassium 可以用于荧光素酶实验。
T0357 Potassium iodide

Tyrosinase Proteases/Proteasome
Potassium iodide 用于治疗过度活跃的甲状腺,并保护甲状腺免受吞咽或吸入放射性碘的辐射影响。可在意外接触放射性碘后或服用含放射性碘的药物前后使用。
T22402 Potassium thioacetate

Others Others
Potassium thioacetate 它已被用于合成聚合物、杂环、纳米颗粒、过渡金属配体、生物活性化合物和大分子包合物。
T68006 Orilotimod potassium

APO805K1

Others Others
Orilotimod potassium (APO805K1)可用于研究斑块状银屑病。
T0940 Acesulfame Potassium

Others Others
Acesulfame potassium 是一种人造甜味剂,长期使用会影响认知功能,可能改变小鼠的神经代谢功能。
T23175 Potassium phosphate monobasic

Others Others
Potassium phosphate monobasic 是生物测定时常用的缓冲液。它是中等浓度至高浓度的磷酸二氢钾水溶液,可用于制备磷酸盐缓冲液以及其他实验试剂。
T6415 Bismuth Subcitrate Potassium

SARS-CoV Microbiology/Virology
Bismuth Subcitrate Potassium 是一种对 12 种幽门螺杆菌有作用的抗生素,抑制组胺H2受体,可用于研究 SARS-CoV-2 感染脆弱患者的腹泻和消化性溃疡病。
T67732 Potassium trimethylsilanolate

Trimethylsiloxypotassium

Others Others
Potassium trimethylsilanolate 是一种催化剂。Potassium trimethylsilanolate 通过(TMSOK)通过硼酸途径促进 Suzuki Miyaura 反应。
T6470 Diclofenac Potassium

双氯芬酸钾,CGP-45840B,Cataflam,Voltfast

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Diclofenac Potassium (CGP-45840B) 是一种非甾体抗炎药,用于减轻炎症并在某些情况下作为镇痛剂减轻疼痛。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的IC50值分别为 5.1 μM 和0.84 μM。
T1425 Pemirolast potassium

BMY 26517,TWT-8152,吡嘧司特钾

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pemirolast potassium (TWT-8152) 是 H1组胺受体拮抗剂和肥大细胞稳定剂,是一种具有抗过敏特性的嘧啶酮衍生物。
T7827 Glycyrrhizinic acid, potassium salt

Others Others
Glycyrrhizinic acid, potassium salt 可减轻藜芦醇引起的室性心律失常。
T22215 1-Naphthyl phosphate potassium salt

Phosphatase Metabolism
1-Naphthyl phosphate potassium salt 是非特异性磷酸酶 (phosphatase) 抑制剂,能够降低剪接校正作用。
T77688 Dipotassium tetrachloroplatinate

Potassium tetrachloroplatinate

Others Others
Dipotassium tetrachloroplatinate (Potassium tetrachloroplatinate) 在实体肿瘤系中表现出抗肿瘤活性,可用于有治疗肿瘤疾病。Dipotassium tetrachloroplatinate 还可充当放射增敏剂,可增强热疗杀伤作用。
T72272 Glibenclamide potassium

Glyburide potassium

Others Others
Glibenclamide (Glyburide) potassium 是 Glibenclamide 的钾盐形式。Glibenclamid potassium 以无水和水合物形式存在,与纯 Glibenclamide 相比具有更高的溶解度。
T10674 Potassium Channel Activator 1

钾离子通道激活剂1,ZINC34634569

Potassium Channel Membrane transporter/Ion channel
Potassium Channel Activator 1 可用于治疗多巴胺能系统被破坏的疾病或病症的研究,例如情绪障碍 ADHD、精神分裂症和其他精神病状态。
T78614 Selnoflast potassium

RO-7486967 potassium

NOD-like Receptor (NLR) Immunology/Inflammation
Selnoflast (potassium) (example 6) 作为NLRP3抑制剂。
T24551 NSC339614 potassium

NSC 339614 potassium,NSC-339614 potassium,NSC339614 potassium salt

Others Others
NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator.
T24630 Phenethicillin potassium

ALPHA-PHENOXYETHYLPENICILLINIC ACID POTASSIUM SALT,PHENETHICILLIN POTASSIUM SALT,Phenethicillin-potassium,Phenethicillinpotassium

Others Others
Phenethicillin potassium is a potassium salt form of phenethicillin with antibacterial activity.
T20365 Monopotassium glutamate

L-谷氨酸钾盐,Potassium glutamate,Potassium L-glutamate

Others Others
Monopotassium glutamate (Potassium glutamate) 可在食品中用作增味剂。
T34116 Potassium caprate

Potassium decanoate

Others Others
Potassium caprate is a biochemical.
T38715 MSDC-0602K

MSDC-0602K,Azemiglitazone potassium

PPAR DNA Damage/DNA Repair; Metabolism
MSDC-0602K (Azemiglitazone potassium) (Azemiglitazone potassium) is a PPARγ-sparing thiazolidinedione (Ps-TZD) compound that binds to PPARγ with an IC50 of 18.25 μM. It also modulates the mitochondrial pyruvate carrier (MPC). This compound, MSDC-0602K, has potential applications in researching fatty liver conditions, including dysfunctional lipid metabolism, inflammation, and insulin resistance. MSDC-0602K acts as an insulin sensitizer, improving insulinemia and fatty liver disease in mice both ...
T39715 MeCY5-NHS ester potassium

Sulfo-Cyanine5 NHS ester potassium,MeCY5-NHS ester potassium

MeCY5-NHS ester (potassium) is a reactive dye designed for labeling proteins and nucleic acids.
T12524 Potassium clavulanate cellulose

Potassium clavulanate:cellulose (1:1)

Others Others
Potassium clavulanate cellulose is a mixture of potassium clavulanate and cellulose, is an inhibitor of beta-lactamase.
T22623 Carboxy-PTIO potassium

Carboxy-PTIO, potassium salt

Others Others
reacts with nitric oxide to form carboxy-PTI derivatives which in turn inhibits nitric oxide synthase
T24900 Troclosene potassium

Fluonon,NSC-251767,NSC 251767,Neochlor 59,Potassium dichloroisocyanurate,NSC251767

Others Others
Troclosene potassium acts as an anti-infective agent on denture cleansers, in hospitals, and in wastewater treatment.
T19948 Grazoprevir potassium salt

MK 5172 potassium,Grazoprevir,Grazoprevir potassium,MK 5172,MK5172,MK-5172

Others Others
Grazoprevir is a drug approved for the treatment of hepatitis C. Grazoprevir is a second-generation hepatitis C virus protease inhibitor acting at the NS3/4a protease targets.
T41058 Nelonemdaz potassium

Neu2000potassium,Salfaprodil

Others Others
Nelonemdaz potassium (also known as Salfaprodil) is a potent NR2B-selective and uncompetitive antagonist of N-methyl-D-aspartate (NMDA). This compound exhibits remarkable neuroprotection against cell death induced by both NMDA and free radicals, in addition to its role as a free radical scavenger.
T68270 Avutometinib potassium

Others Others
Avutometinib potassium is a MEK inhibitor (MEKi) that enhanced the inhibition of pseudovirus infection by GLPG-0187. It Blocks SARS-CoV-2 Delta and Omicron Pseudovirus Infection of Airway Epithelial Cells In Vitro, Which Could Attenuate Disease Severity
T27724 KDT 501 potassium

KDT 501 potassium salt,KDT-501,KDT 501,Tetrahydroisohumulone

Others Others
KDT 501, a PPAR agonist and G protein-coupled receptor (GPR) 120 agonist, is used potentially for the treatment of type 2 diabetes.
T69273 Mexrenoate potassium

Others Others
Mexrenoate potassium is a steroidal aldosterone antagonist and antihypertensive.
T71844 Methyl potassium malonate

Others Others
Methyl potassium malonate is a protein advanced glycosylation inhibitor.
T70589 Saprisartan potassium

Others Others
Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.
T35382 Potassium phosphate dibasic

Dipotassium phosphate

Others Others
Potassium phosphate dibasic (Dipotassium phosphate, K2HPO4)常被用作肥料、食品添加剂和缓冲剂。
T38510 ABT-072 potassium trihydrate

Others Others
ABT-072, also known as potassium trihydrate, is a highly effective non-nucleoside inhibitor of the HCV NS5B polymerase, administered orally. This compound exhibits potent activity against HCV GT1a (with an EC50 of 1 nM) and HCV GT1b (with an EC50 of 0.3 nM).
T33228 MCPA-potassium

Others Others
MCPA-potassium is a bioactive chemical.
T70743 IS-741 potassium

Others Others
IS-741 potassium is a phospholipase A2 inhibitor.
T70203 Galloflavin Potassium

Others Others
Galloflavin Potassium is an inhibitor of lactate dehydrogenase.

化合物

Potassium oxonate
Cat.No: T5987
Synonym: Oxonic Acid (potassium salt),氧嗪酸钾,Potassium otastat,Potassium azaorotate
Target: Others
Sulotroban potassium
Cat.No: T68022L
Synonym: BM 13177 potassium,Sulotroban potassium(72131-33-0 Free base)
Target: PPAR
Canrenoate potassium
Cat.No: T3096
Synonym: 坎利酸钾,Potassium aldadiene,Canrenoic acid potassium salt,Potassium canrenoate,Soldactone
Target: Glucocorticoid Receptor
Aluminum potassium sulfate
Cat.No: T35381
Synonym: Potassium Aluminium Sulfate,APS
Target: Others
Raltegravir potassium
Cat.No: T2239
Synonym: MK 0518 potassium salt,Raltegravir potassium salt,雷特格韦钾盐
Target: HIV Protease, Integrase
Potassium acetate
Cat.No: T8129
Synonym: Diuretic salt,Potassium ethanoate,乙酸钾
Target: Antifungal
Azilsartan Medoxomil Potassium
Cat.No: T0481
Synonym: TAK-491 Potassium
Target:
p-Cresyl sulfate potassium
Cat.No: T19498
Synonym: p-Tolyl sulfate potassium salt,p-Cresol sulfate potassium,p-Methylphenyl potassium sulfate,对甲基硫酸钾,Potassium p-tolyl sulfate
Target: Endogenous Metabolite
Potassium guaiacolsulfonate hemihydrate
Cat.No: T3267
Synonym: 愈创木酚磺酸钾水合物,Potassium guaiacolsulfonate,Potassium 4-guaiacolsulfonate hemihydrate,愈创木酚磺酸钾
Target: Antibacterial, Antibiotic
1-Naphthaleneacetic acid potassium salt
Cat.No: T5580
Synonym: α-萘醋酸钾,α-Naphthaleneacetic acid,Potassium alpha-naphthylacetate,Potassium 1-Naphthaleneacetate,1-NAA Potassium Salt
Target: Phospholipase
Ethyl potassium malonate
Cat.No: T22328
Synonym: Potassium 3-ethoxy-3-oxopropanoate,Malonic Acid Monoethyl Ester Potassium Salt,丙二酸单乙酯钾盐
Target: Others
Losartan potassium
Cat.No: T0215
Synonym: DuP-753 potassium,洛沙坦钾,氯沙坦钾,MK 954,DuP 753
Target: RAAS
Nebentan potassium
Cat.No: T36008
Synonym: YM598
Target: Endothelin Receptor
D-Luciferin potassium
Cat.No: T4139
Synonym: D-Luciferin K Salt,D-Luciferin Potassium Salt,D-萤光素钾盐,D-荧光素钾盐
Target: Others
Potassium iodide
Cat.No: T0357
Synonym:
Target: Tyrosinase
Potassium thioacetate
Cat.No: T22402
Synonym:
Target: Others
Orilotimod potassium
Cat.No: T68006
Synonym: APO805K1
Target: Others
Acesulfame Potassium
Cat.No: T0940
Synonym:
Target: Others
Potassium phosphate monobasic
Cat.No: T23175
Synonym:
Target: Others
Bismuth Subcitrate Potassium
Cat.No: T6415
Synonym:
Target: SARS-CoV
Potassium trimethylsilanolate
Cat.No: T67732
Synonym: Trimethylsiloxypotassium
Target: Others
Diclofenac Potassium
Cat.No: T6470
Synonym: 双氯芬酸钾,CGP-45840B,Cataflam,Voltfast
Target: Apoptosis, Others, COX
Pemirolast potassium
Cat.No: T1425
Synonym: BMY 26517,TWT-8152,吡嘧司特钾
Target: Histamine Receptor
Glycyrrhizinic acid, potassium salt
Cat.No: T7827
Synonym:
Target: Others
1-Naphthyl phosphate potassium salt
Cat.No: T22215
Synonym:
Target: Phosphatase
Dipotassium tetrachloroplatinate
Cat.No: T77688
Synonym: Potassium tetrachloroplatinate
Target: Others
Glibenclamide potassium
Cat.No: T72272
Synonym: Glyburide potassium
Target: Others
Potassium Channel Activator 1
Cat.No: T10674
Synonym: 钾离子通道激活剂1,ZINC34634569
Target: Potassium Channel
Selnoflast potassium
Cat.No: T78614
Synonym: RO-7486967 potassium
Target: NOD-like Receptor (NLR)
NSC339614 potassium
Cat.No: T24551
Synonym: NSC 339614 potassium,NSC-339614 potassium,NSC339614 potassium salt
Target: Others
Phenethicillin potassium
Cat.No: T24630
Synonym: ALPHA-PHENOXYETHYLPENICILLINIC ACID POTASSIUM SALT,PHENETHICILLIN POTASSIUM SALT,Phenethicillin-potassium,Phenethicillinpotassium
Target: Others
Monopotassium glutamate
Cat.No: T20365
Synonym: L-谷氨酸钾盐,Potassium glutamate,Potassium L-glutamate
Target: Others
Potassium caprate
Cat.No: T34116
Synonym: Potassium decanoate
Target: Others
MSDC-0602K
Cat.No: T38715
Synonym: MSDC-0602K,Azemiglitazone potassium
Target: PPAR
MeCY5-NHS ester potassium
Cat.No: T39715
Synonym: Sulfo-Cyanine5 NHS ester potassium,MeCY5-NHS ester potassium
Target:
Potassium clavulanate cellulose
Cat.No: T12524
Synonym: Potassium clavulanate:cellulose (1:1)
Target: Others
Carboxy-PTIO potassium
Cat.No: T22623
Synonym: Carboxy-PTIO, potassium salt
Target: Others
Troclosene potassium
Cat.No: T24900
Synonym: Fluonon,NSC-251767,NSC 251767,Neochlor 59,Potassium dichloroisocyanurate,NSC251767
Target: Others
Grazoprevir potassium salt
Cat.No: T19948
Synonym: MK 5172 potassium,Grazoprevir,Grazoprevir potassium,MK 5172,MK5172,MK-5172
Target: Others
Nelonemdaz potassium
Cat.No: T41058
Synonym: Neu2000potassium,Salfaprodil
Target: Others
Avutometinib potassium
Cat.No: T68270
Synonym:
Target: Others
KDT 501 potassium
Cat.No: T27724
Synonym: KDT 501 potassium salt,KDT-501,KDT 501,Tetrahydroisohumulone
Target: Others
Mexrenoate potassium
Cat.No: T69273
Synonym:
Target: Others
Methyl potassium malonate
Cat.No: T71844
Synonym:
Target: Others
Saprisartan potassium
Cat.No: T70589
Synonym:
Target: Others
Potassium phosphate dibasic
Cat.No: T35382
Synonym: Dipotassium phosphate
Target: Others
ABT-072 potassium trihydrate
Cat.No: T38510
Synonym:
Target: Others
MCPA-potassium
Cat.No: T33228
Synonym:
Target: Others
IS-741 potassium
Cat.No: T70743
Synonym:
Target: Others
Galloflavin Potassium
Cat.No: T70203
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T4807 Potassium sorbate

Sorbic acid potassium salt,山梨酸钾,Potassium 2,4-hexadienoate

Others; Endogenous Metabolite; Antibacterial; Antibiotic; Antifungal Metabolism; Microbiology/Virology; Others
Potassium sorbate (Sorbic acid potassium salt) 是一种高效安全无毒的食品防腐剂,可有效抑制大多数霉菌,酵母和某些细菌。
TN1698 Glucotropaeolin potassium

金莲葡糖硫苷钾盐,Glucotropaeolin,Benzylglucosinolate potassium,Glucotropaeolin Potassium Salt

Others Others
Glucotropaeolin potassium (Benzylglucosinolate potassium) 存在于十字花科蔬菜中,并且 可适度减少动物的自发性DNA 损伤。
T1126 Penicillin V Potassium

青霉素V钾,Penicillin V potassium salt,Phenoxymethylpenicillin potassium salt

Antibacterial; Antibiotic Microbiology/Virology
Penicillin V Potassium (Phenoxymethylpenicillin potassium salt) 是一种有口服活性的抗生素。它可抑制链球菌,艰难梭菌和金黄色葡萄球菌的生长,可研究中耳炎,鼻窦炎,咽炎和扁桃体炎。
T5602 Penicillin G potassium

青霉素钾,Benzylpenicillin potassium

Anti-infection; Antibacterial; Antibiotic Microbiology/Virology
Penicillin G potassium (Benzylpenicillin potassium) 是青霉素家族的一种速效抗生素。
T20198 Potassium gluconate

Kalium-beta,Kalium Gluconate,Kaon elixir,Kaon,Potassium D-gluconate,HSDB 3165,K-Iao

Endogenous Metabolite; Antifungal Metabolism; Microbiology/Virology
Potassium gluconate (Potassium D-gluconate) 是一种具有口服活性和螯合性质的氧化型羧酸,具有杀菌活性。
T4938 Potassium 1H-indol-3-yl sulfate

硫酸吲哚钾盐,Indoxyl sulfate potassium salt,Potassium 3-indoxyl sulfate

AhR; Endogenous Metabolite Immunology/Inflammation; Metabolism
Potassium 1H-indol-3-yl sulfate (Potassium 3-indoxyl sulfate) 是人芳烃受体(AhR)的激动剂。芳烃受体(AhR)最近被发现是免疫炎症条件的病理生理调节剂,Potassium 1H-indol-3-yl sulfate 已被证明是AhR的配体。Potassium 1H-indol-3-yl sulfate 也是膳食蛋白质中色氨酸的代谢物。色氨酸被肠道细菌代谢为吲哚,吲哚被吸收到血液中,然后在肝脏中进一步代谢为硫酸吲哚,通常通过尿液排出体外。在肾功能受损的慢性肾病患者中,Potassium 1H-indol-3-yl sulfate 可作为尿毒症毒素在血清中积累,诱导氧化应激并加速疾病进展。250 μM Potassium 1H-indol-3-yl sulfate 可诱导NF-Κb活化,促进大鼠近端小管细胞TGF-β1和Smad3的表达,与促纤维化活性相关。
T5213 Acetyl phosphate(lithium potassium)

乙酰磷酸锂钾盐,Lithium potassium acetyl phosphate,Acetylphosphoric acid

Others; Endogenous Metabolite Metabolism; Others
Acetyl phosphate lithium potassium (Lithium potassium acetyl phosphate) 是内源性代谢产物的一种。
TN7050 Potassium 7-hydroxy-1-naphthalenesulfona

藏红花酸,2-Naphthol-8-sulfonic Acid Potassium Salt

Others Others
Potassium 7-hydroxy-1-naphthalenesulfona (2-Naphthol-8-sulfonic Acid Potassium Salt) 天然存在于茜草科栀子花的果实、鸢尾科番红花的花和玄参科玄参科的花叶中。
T4916 D-Glucaric acid potassium

D-Saccharic acid potassium salt,Glucosaccharic acid,D-葡萄糖二酸单钾盐,Glucaric Acid

Others; Endogenous Metabolite Metabolism; Others
D-Glucaric acid potassium (D-Saccharic acid potassium salt) 是内源性代谢产物的一种。
T4948 Potassium 2-hydroxy-2-methylsuccinate

(±)-柠苹酸钾 一水合物,(±)-Potassium citramalate monohydrate,(±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt

Others; Endogenous Metabolite Metabolism; Others
Potassium 2-hydroxy-2-methylsuccinate ((±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt) 是内源性代谢产物的一种。
T4898 Potassium 1-carboxyvinyl hydrogenphosphate

PEP-K,磷酸烯醇丙酮酸单钾盐,Phospho(enol)pyruvic acid monopotassium

Others; Endogenous Metabolite Metabolism; Others
Potassium 1-carboxyvinyl hydrogenphosphate (PEP-K) 是内源性代谢产物的一种。
T3S0156 Atractyloside potassium salt

Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐

Others Others
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。
T5069 D-Glucose 6-phosphate potassium salt

Others Others
在细胞中,当葡萄糖被己糖激酶或葡萄糖激酶磷酸化或在糖原分解过程中通过磷酸葡萄糖变位酶转化葡萄糖 1-磷酸时,会产生D-glucose 6-phosphate (G6P)。 G6P 位于糖酵解和戊糖磷酸途径的起点。当血糖水平高时,它也可以作为糖原储存。
T5075 Phytic acid potassium

植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt

Others; BACE; Endogenous Metabolite Metabolism; Neuroscience; Others
Phytic acid dipotassium salt 是内源性代谢产物的一种,抑制 β-分泌酶 1 (BACE1) 。
T82304 Glucobrassicanapin potassium

4-Pentenylglucosinolate potassium

Others Others
Glucobrassicanapin (4-Pentenylglucosinolate) potassium 是脂肪族硫代葡萄糖苷类化合物,主要存在于白菜等蔬菜作物中。
T4942 Galactose 1-phosphate Potassium salt

D-半乳糖 1-磷酸二钾盐五水合物,α-D-Galactose-1-phosphate Dipotassium Pentahydrate

Others; Endogenous Metabolite Metabolism; Others
Galactose 1-phosphate Potassium salt (α-D-Galactose-1-phosphate Dipotassium Pentahydrate) 是一种半乳糖代谢中的中间体和核苷酸糖。
TN2212 Glucosinalbate potassium

白芥子钾盐,Sinalbin potassium salt

Others Others
Sinalbin potassium salt is a natural product
T19457 N-Hydroxypipecolic acid potassium

NHP potassium,1-Hydroxy-2-piperidinecarboxylic acid potassium

Others Others
N-Hydroxypipecolic acid potassium is a metabolite of plant and a systemic acquired resistance (SAR) regulator.
T73772 Estrone sulfate potassium

Endogenous Metabolite Metabolism
Estrone sulfate potassium 是一种雌激素酯和共轭物,是一种天然内源性类固醇。
T65269 L-Aspartic acid potasium salt

Aspartic acid potasium salt,Potassium L-aspartate

Others Others
L-aspartic acid potasium salt(VX-548) 是一种广泛存在于动植物体内的氨基酸。L-aspartic acid potasium salt驱动氮氧化物的产生,从而促进吞噬作用,有助于提高鱼类的成活率。L-aspartic acid potasium salt 可对抗生素产生刺激,刺激作用可能与参与天冬氨酸-4-半醛生物合成的前体有关。
T78471 α,α-Trehalose 6-phosphate potassium

Tre6P potassium

Endogenous Metabolite Metabolism
α,α-Trehalose 6-phosphate (Tre6P) potassium 是一种α,α′-trehalose的6-磷酸衍生物及内源代谢物。在Tre6P磷酸酶 (T6PP) 的催化下,α,α-Trehalose 6-phosphate可被高效转化为α,α′-trehalose。
T11589 Hydroxycitric acid tripotassium hydrate

柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate

ATP Citrate Lyase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) 是一种藤黄果的主要活性成分,也是一种柠檬酸的衍生物。它可竞争性抑制柠檬酸裂解酶 (ATP citrate lyase) ,并具有减肥作用。它有效抑制结石形成,并抑制HIF,具有抗氧化,抗炎和抗肿瘤活性。
T35415 α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)

Others Others
α-D-Glucose-1,6-bisphosphate is abis-phosphorylated derivative of α-D-glucose that has roles in carbohydrate metabolism.1It is the product of the reaction of glucose-1- or 6-phosphate with glucose-1,6-bisphosphate synthase (PGM2LI) in the conversion of 1,3-bisphosphoglycerate to 3-phosphoglycerate.2It is also a cofactor for the bacterial enzyme phosphopentomutase.3,4α-D-Glucose-1,6-bisphosphate has been used in the study of carbohydrate metabolism. 1.Beitner, R.Regulation of carbohydrate metabol...
TN7336 Glucobrassicin potassium

Others Others
Glucobrassicin (potassium) 是一种从野生胡萝卜 (Raphanus raphanistrumL.) 中分离的硫代葡萄糖苷 (GSL),适用于生物熏蒸和化感植物在杂草管理研究中的应用。
T82301 Gluconapin potassium

Gluconapin potassium为萝卜硫素前体,后者为一抗癌效能显著的异硫氰酸酯。
TN7337 Glucoraphenin potassium

Others Others
Glucoraphenin potassium 是一种具口服活性的硫代葡萄糖苷,能通过芥子酶水解产生萝卜硫素,发挥抗癌作用,并可诱导激活异生物质代谢酶(XMEs)。
T78466 Erythronic acid potassium

Endogenous Metabolite Metabolism
Erythronic acid potassium为糖类内源性代谢物,关键作用于高尿酸血症发病及改善过程,并与转醛缩酶缺乏症相关的线粒体功能障碍有关,常用于代谢性疾病研究。
T0690 Quinine

奎宁树

Potassium Channel; Platelet aggregation; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Others
Quinine 是一种从金鸡纳树皮中提取的生物碱,用于预防和治疗疟疾。它也用于特发性肌肉痉挛,可抑制电压脉冲引起的 MT mSlo3 (KCa5.1) 通道 +100 mV 电流, 其IC50值为 169 μM,是一种钾离子通道抑制剂。
T1719 Bufalin

ATPase Membrane transporter/Ion channel
Bufalin 是蟾酥中的一种成分,是Na+/K+-ATPase 抑制剂,具有抗肿瘤活性,可与其基 α1、α2 和 α3 结合,Kd 值分别为 42.5、45 和 40 nM。
T8189 Dihydroberberine

Potassium Channel; HSP; HER Angiogenesis; Cytoskeletal Signaling; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Tyrosine Kinase/Adaptors
Dihydroberberine 可抑制人类 ether-a-go-go 相关基因 (hERG) 通道并显着降低 Hsp90 表达及其与 hERG 的相互作用,具有抗动脉粥样硬化、抗炎、降血脂和抗肿瘤活性。
T37709 2,2,2-Trichloroethanol

Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
2,2,2-Trichloroethanol 是非经典的 K2P 通道 TREK-1和 TRAAK 的激动剂。
TN1092 O-Nornuciferine

Potassium Channel; HER Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
O-Noruciferine 是分离自荷叶的卟啉型生物碱,是有效的 hERG 通道抑制剂。
T0801 Tannic acid

单宁酸,Gallotannic acid

Potassium Channel; HER; CXCR Angiogenesis; Autophagy; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
Tannic acid (Gallotannic acid) 属于多酚类天然产物,是一种 hERG 通道阻塞剂,也是一种 CXCL12/CXCR4 抑制剂。Tannic acid 具有抗菌、抗氧化、抗炎和抗肿瘤等多种生物活性。
T3S1873 Talatisamine

塔拉乌头胺,塔拉萨敏

Potassium Channel Membrane transporter/Ion channel
Talatisamine 是一种乌头生物碱,对K+通道有特异性阻滞作用。它能减弱 beta- 淀粉样低聚物对培养的皮层神经元的毒性。
T3A2467 Allocryptopine

Thalictrimine,Fagarine I,别隐品碱

Potassium Channel Membrane transporter/Ion channel
Allocryptopine (Thalictrimine) 是一种延胡索乙素的衍生物,提取自Corydalis decumbens。Allocryptopine 具有抗心律失常作用,能有效阻断hERG 电流。
T1186 Ifenprodil Tartrate

Potassium Channel; NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
Ifenprodil tartrate 是典型的非竞争性 NMDA 受体拮抗剂,抑制 GIRK (Kir3),通过基底 GIRK 活性减少内向电流,有用做脑血管舒张试剂的潜力。它对 NR1A/NR2B 受体亲和力是 NR1A/NR2A 受体的 400 倍。
T3054 Daurisoline

蝙蝠葛苏林碱,(R,R)-Daurisoline

Others; Potassium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Others
Daurisoline ((R,R)-Daurisoline) 是一种 hERG 抑制剂,也是一种自噬阻滞剂。
TJP2872 Acevaltrate

Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate

ATPase; Others Membrane transporter/Ion channel; Others
Acevaltrate (Acevaltratum) 对人小细胞肺癌细胞系 GLC(4) 和人结肠直肠癌细胞系 COLO 320 具有高细胞毒性,IC50 值为 1-6 uM。它抑制大鼠肾和脑半球中 Na+/K+-ATP 酶活性,IC50分别为 22.8 和 42.3 μM。
T4333 Quinine dihydrochloride

盐酸奎宁,Quinine bimuriate

Others Others
Quinine dihydrochloride (Quinine bimuriate) 是Cinchona(Rubiaceae) 各种物种的主要生物碱。它也是一种抗疟药和肌肉松弛剂(骨骼)。
T3S0081 Oxypeucedanin

(+-)-Oxypeucedanin,氧化前胡素,Oxypeucadanin

Potassium Channel Membrane transporter/Ion channel
Oxypeucedanin ((+-)-Oxypeucedanin) 是呋喃香豆素衍生物,分离自Angelica dahurica。它是选择性开放通道阻滞剂,可抑制hKv1.5通道电流,IC50值为 76 nM。它延长心脏动作电位持续时间,是潜在的抗心律失常试剂。它通过抑制癌细胞迁移来诱导细胞凋亡。
T7938 Quinidine

奎尼丁,奎宁树

Parasite Microbiology/Virology
Quinidine 是一种抗心律失常剂,也是 K+通道的有效阻断剂,其 IC50值为 19.9 μM。它是一种选择性细胞色素 P450db 的有效抑制剂,也可研究疟疾。
TMS2171 (±)-Naringenin

(±)-柚皮素,Salipurpol,柚皮素,Naringenine,Naringenin

Potassium Channel Membrane transporter/Ion channel
(±)-Naringenin (Naringenine) 是一种天然的类黄酮。它通过激活肌细胞中 BKCa 通道发挥对内皮剥脱血管的舒张作用。
T3876 Loureirin B

龙血素B,龙血素 B

PAI-1; ERK; Potassium Channel; JNK MAPK; Membrane transporter/Ion channel; Metabolism
Loureirin B 是从剑叶龙血树中分离到的一种黄酮,是 PAI-1抑制剂,IC50值为 26.10 μM。它抑制 KATP,以及 ERK 和 JNK 的磷酸化,具有抗糖尿病的功效。
T8182 Guanfu base A

Guan-fu base A,关附甲素

P450; Potassium Channel; HER Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Tyrosine Kinase/Adaptors
Guanfu base A 是一种生物碱,分离自 Aconitum coreanum,是非竞争性 CYP2D6抑制剂,对人肝微粒体 (HLM) 的 Ki 为 1.20 μM,对人重组体 (rCYP2D6) 的 Ki 为 0.37 μM。它也是 CYP2D 的有效竞争抑制剂。它还能抑制 HERG 通道电流。Guan-fu base A 具有抗心律失常的作用。
T5S0890 Oleandrin

Neriostene,Folinerin,Foliandrin,欧夹竹桃苷

Apoptosis; ATPase; Potassium Channel; Sodium Channel Apoptosis; Membrane transporter/Ion channel
Oleandrin (Folinerin) 是夹竹桃属中的一种类固醇,可抑制Na+/K+-ATPase 活性,IC50为 620 nM。
T3667 Kalii Dehydrographolidi Succinas

Ddhads,穿琥宁,Dehydroandrographolide Succinate Potasium Salt

Others Others
Kalii Dehydrographolidi Succinas (Dehydroandrographolide Succinate Potasium Salt) 从中药穿心莲中提取得到,具有免疫刺激、抗感染和抗炎作用,对病毒性肺炎和病毒性上呼吸道感染具有潜在的研究价值。
T3092 Nigericin sodium salt

尼日利亚菌素,尼日利亚菌素钠盐

Potassium Channel; NOD-like Receptor (NLR); Antibacterial; Antibiotic; NOD Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Nigericin sodium salt 属于抗生素,是一种 NLRP3 激活剂,也是一种阳离子离子载体。Nigericin sodium 可以触发 NALP3 炎性体的激活,可抑制高尔基体功能并抑制革兰氏阳性菌的生长。
T2850 Bicuculline

荷包牡丹碱,(+)-Bicuculline,d-Bicuculline

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Bicuculline ((+)-Bicuculline) 是从东北延胡索中提取的一种生物碱,能阻断 Ca2+激活钾 (SK) 通道。它是一种竞争性的神经递质 GABAA 受体拮抗剂,IC50为 2 μM。
TN5073 Strophanthidin

毒毛旋花子甙元,Strophanthidine,葡萄球菌素

ATPase; Calcium Channel Membrane transporter/Ion channel; Metabolism
Strophanthidin (Strophanthidine) 是黄花夹竹桃中的一种类固醇,可增加舒张期和收缩期胞内 Ca2+浓度。它在 0.1 和 1 nmol/L 增加Na+/K+-ATPase 活性,1到100 μ mol/L 抑制Na+/K+-ATPase 活性,10 和 100 nmol/L 对Na+/K+-ATPase 活性无影响。
T3S0870 Paederosidic acid methyl ester

鸡屎藤苷酸甲酯,紫草酸甲酯

ATPase; Potassium Channel; NO Synthase Immunology/Inflammation; Membrane transporter/Ion channel
Paederosidic acid methyl ester 是 ATP 敏感的 K+channel 通道激活剂,分离自 P. scandens。它通过激活脑中和脊髓水平中 ATP 敏感型 K+通道提高了痛觉阈值,表现出显著的中枢缓解疼痛活性。
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天然产物

Potassium sorbate
Cat.No: T4807
Synonym: Sorbic acid potassium salt,山梨酸钾,Potassium 2,4-hexadienoate
Target: Others, Endogenous Metabolite, Antibacterial, Antibiotic, Antifungal
Glucotropaeolin potassium
Cat.No: TN1698
Synonym: 金莲葡糖硫苷钾盐,Glucotropaeolin,Benzylglucosinolate potassium,Glucotropaeolin Potassium Salt
Target: Others
Penicillin V Potassium
Cat.No: T1126
Synonym: 青霉素V钾,Penicillin V potassium salt,Phenoxymethylpenicillin potassium salt
Target: Antibacterial, Antibiotic
Penicillin G potassium
Cat.No: T5602
Synonym: 青霉素钾,Benzylpenicillin potassium
Target: Anti-infection, Antibacterial, Antibiotic
Potassium gluconate
Cat.No: T20198
Synonym: Kalium-beta,Kalium Gluconate,Kaon elixir,Kaon,Potassium D-gluconate,HSDB 3165,K-Iao
Target: Endogenous Metabolite, Antifungal
Potassium 1H-indol-3-yl sulfate
Cat.No: T4938
Synonym: 硫酸吲哚钾盐,Indoxyl sulfate potassium salt,Potassium 3-indoxyl sulfate
Target: AhR, Endogenous Metabolite
Acetyl phosphate(lithium potassium)
Cat.No: T5213
Synonym: 乙酰磷酸锂钾盐,Lithium potassium acetyl phosphate,Acetylphosphoric acid
Target: Others, Endogenous Metabolite
Potassium 7-hydroxy-1-naphthalenesulfona
Cat.No: TN7050
Synonym: 藏红花酸,2-Naphthol-8-sulfonic Acid Potassium Salt
Target: Others
D-Glucaric acid potassium
Cat.No: T4916
Synonym: D-Saccharic acid potassium salt,Glucosaccharic acid,D-葡萄糖二酸单钾盐,Glucaric Acid
Target: Others, Endogenous Metabolite
Potassium 2-hydroxy-2-methylsuccinate
Cat.No: T4948
Synonym: (±)-柠苹酸钾 一水合物,(±)-Potassium citramalate monohydrate,(±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt
Target: Others, Endogenous Metabolite
Potassium 1-carboxyvinyl hydrogenphosphate
Cat.No: T4898
Synonym: PEP-K,磷酸烯醇丙酮酸单钾盐,Phospho(enol)pyruvic acid monopotassium
Target: Others, Endogenous Metabolite
Atractyloside potassium salt
Cat.No: T3S0156
Synonym: Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐
Target: Others
D-Glucose 6-phosphate potassium salt
Cat.No: T5069
Synonym:
Target: Others
Phytic acid potassium
Cat.No: T5075
Synonym: 植酸二钾盐,Inositol hexakisphosphate dipotassium salt,Phytic acid dipotassium salt,Fytic Acid dipotassium salt,Inositol polyphosphate dipotassium salt
Target: Others, BACE, Endogenous Metabolite
Glucobrassicanapin potassium
Cat.No: T82304
Synonym: 4-Pentenylglucosinolate potassium
Target: Others
Galactose 1-phosphate Potassium salt
Cat.No: T4942
Synonym: D-半乳糖 1-磷酸二钾盐五水合物,α-D-Galactose-1-phosphate Dipotassium Pentahydrate
Target: Others, Endogenous Metabolite
Glucosinalbate potassium
Cat.No: TN2212
Synonym: 白芥子钾盐,Sinalbin potassium salt
Target: Others
N-Hydroxypipecolic acid potassium
Cat.No: T19457
Synonym: NHP potassium,1-Hydroxy-2-piperidinecarboxylic acid potassium
Target: Others
Estrone sulfate potassium
Cat.No: T73772
Synonym:
Target: Endogenous Metabolite
L-Aspartic acid potasium salt
Cat.No: T65269
Synonym: Aspartic acid potasium salt,Potassium L-aspartate
Target: Others
α,α-Trehalose 6-phosphate potassium
Cat.No: T78471
Synonym: Tre6P potassium
Target: Endogenous Metabolite
Hydroxycitric acid tripotassium hydrate
Cat.No: T11589
Synonym: 柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)
Cat.No: T35415
Synonym:
Target: Others
Glucobrassicin potassium
Cat.No: TN7336
Synonym:
Target: Others
Gluconapin potassium
Cat.No: T82301
Synonym:
Target:
Glucoraphenin potassium
Cat.No: TN7337
Synonym:
Target: Others
Erythronic acid potassium
Cat.No: T78466
Synonym:
Target: Endogenous Metabolite
Quinine
Cat.No: T0690
Synonym: 奎宁树
Target: Potassium Channel, Platelet aggregation, Parasite
Bufalin
Cat.No: T1719
Synonym:
Target: ATPase
Dihydroberberine
Cat.No: T8189
Synonym:
Target: Potassium Channel, HSP, HER
2,2,2-Trichloroethanol
Cat.No: T37709
Synonym:
Target: Potassium Channel, Endogenous Metabolite
O-Nornuciferine
Cat.No: TN1092
Synonym:
Target: Potassium Channel, HER
Tannic acid
Cat.No: T0801
Synonym: 单宁酸,Gallotannic acid
Target: Potassium Channel, HER, CXCR
Talatisamine
Cat.No: T3S1873
Synonym: 塔拉乌头胺,塔拉萨敏
Target: Potassium Channel
Allocryptopine
Cat.No: T3A2467
Synonym: Thalictrimine,Fagarine I,别隐品碱
Target: Potassium Channel
Ifenprodil Tartrate
Cat.No: T1186
Synonym:
Target: Potassium Channel, NMDAR, iGluR
Daurisoline
Cat.No: T3054
Synonym: 蝙蝠葛苏林碱,(R,R)-Daurisoline
Target: Others, Potassium Channel, Autophagy
Acevaltrate
Cat.No: TJP2872
Synonym: Acevaltratum,乙酰缬草三酯,Acetoxyvaltrate
Target: ATPase, Others
Quinine dihydrochloride
Cat.No: T4333
Synonym: 盐酸奎宁,Quinine bimuriate
Target: Others
Oxypeucedanin
Cat.No: T3S0081
Synonym: (+-)-Oxypeucedanin,氧化前胡素,Oxypeucadanin
Target: Potassium Channel
Quinidine
Cat.No: T7938
Synonym: 奎尼丁,奎宁树
Target: Parasite
(±)-Naringenin
Cat.No: TMS2171
Synonym: (±)-柚皮素,Salipurpol,柚皮素,Naringenine,Naringenin
Target: Potassium Channel
Loureirin B
Cat.No: T3876
Synonym: 龙血素B,龙血素 B
Target: PAI-1, ERK, Potassium Channel, JNK
Guanfu base A
Cat.No: T8182
Synonym: Guan-fu base A,关附甲素
Target: P450, Potassium Channel, HER
Oleandrin
Cat.No: T5S0890
Synonym: Neriostene,Folinerin,Foliandrin,欧夹竹桃苷
Target: Apoptosis, ATPase, Potassium Channel, Sodium Channel
Kalii Dehydrographolidi Succinas
Cat.No: T3667
Synonym: Ddhads,穿琥宁,Dehydroandrographolide Succinate Potasium Salt
Target: Others
Nigericin sodium salt
Cat.No: T3092
Synonym: 尼日利亚菌素,尼日利亚菌素钠盐
Target: Potassium Channel, NOD-like Receptor (NLR), Antibacterial, Antibiotic, NOD
Bicuculline
Cat.No: T2850
Synonym: 荷包牡丹碱,(+)-Bicuculline,d-Bicuculline
Target: GABA Receptor
Strophanthidin
Cat.No: TN5073
Synonym: 毒毛旋花子甙元,Strophanthidine,葡萄球菌素
Target: ATPase, Calcium Channel
Paederosidic acid methyl ester
Cat.No: T3S0870
Synonym: 鸡屎藤苷酸甲酯,紫草酸甲酯
Target: ATPase, Potassium Channel, NO Synthase
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Cat. No. Product Name Species Expression System
TMPH-01890 KCNA1 Protein, Human, Recombinant (His)

Voltage-gated potassium channel subunit Kv1.1,Volta...

Human E. coli
KCNA1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 22.2 kDa and the accession number is Q09470.
TMPH-03603 KcsA Protein, S. coelicolor, Recombinant (His)

pH-gated potassium channel KcsA,kcsA

Streptomyces coelicolor E. coli
Acts as a pH-gated potassium ion channel; changing the cytosolic pH from 7 to 4 opens the channel. KcsA Protein, S. coelicolor, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 23.7 kDa and the accession number is P0A333.
TMPH-01891 KCNE2 Protein, Human, Recombinant (His)

MinK-related peptide 1,Potassium voltage-gated chan...

Human E. coli
KCNE2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 17.3 kDa and the accession number is Q9Y6J6.
TMPH-01889 KCNK3 Protein, Human, Recombinant (His & Myc)

Potassium channel subfamily K member 3,TWIK-related...

Human E. coli
pH-dependent, voltage-insensitive, background potassium channel protein. Rectification direction results from potassium ion concentration on either side of the membrane. Acts as an outward rectifier when external potassium concentration is low. When external potassium concentration is high, current is inward. KCNK3 Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 50.5 kDa and the accession number is O...
TMPH-01028 KCNMA1 Protein, Human, Recombinant

K(VCA)alpha,Calcium-activated potassium channel sub...

Human E. coli
KCNMA1 Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 17.2 kDa and the accession number is Q12791.
TMPH-01892 ATP4A Protein, Human, Recombinant (His & Myc)

ATP4A,Gastric H(+)/K(+) ATPase subunit alpha,Potassium

Human E. coli
ATP4A Protein, Human, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 54.6 kDa and the accession number is P20648.
TMPH-01893 ATP4B Protein, Human, Recombinant (GST)

Proton pump beta chain,Gastric H(+)/K(+) ATPase subunit beta...

Human E. coli
ATP4B Protein, Human, Recombinant (GST) is expressed in E. coli expression system with N-GST tag. The predicted molecular weight is 53.6 kDa and the accession number is P51164.
TMPH-01894 ATP4B Protein, Human, Recombinant

Proton pump beta chain,Potassium-transporting ATPas...

Human E. coli
ATP4B Protein, Human, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 26.6 kDa and the accession number is P51164.
TMPH-02309 KCNAB2 Protein, Human, Recombinant (His & SUMO)

Kv-beta-2,K(+) channel subunit beta-2,KCNAB2,Voltage-gated <...

Human E. coli
KCNAB2 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 57.0 kDa and the accession number is Q13303.
TMPH-01358 FXYD3 Protein, Human, Recombinant (His & SUMO)

Phospholemman-like,Chloride conductance inducer protein Mat-...

Human E. coli
FXYD3 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 20.5 kDa and the accession number is Q14802.
TMPH-01714 CHRM1 Protein, Human, Recombinant (His)

Muscarinic acetylcholine receptor M1,CHRM1

Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is Pi turnover. CHRM1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 20.8 kDa and the accession number is P11229.
TMPH-01717 CHRM5 Protein, Human, Recombinant (His)

CHRM5,Muscarinic acetylcholine receptor M5

Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is Pi turnover. CHRM5 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 31.5 kDa and the accession number is P08912.
TMPY-03615 CSEN Protein, Human, Recombinant (His)

Kv channel interacting protein 3, calsenilin,DREAM,KCHIP3,CS...

Human E. coli
KCNIP3 (Potassium Voltage-Gated Channel Interacting Protein 3, also known as CSEN) is a Protein Coding gene. CSEN is a member of the family of voltage-gated potassium (Kv) channel-interacting proteins, which belong to the recoverin branch of the EF-hand superfamily. Members of this family are integral subunit components of native Kv4 channel complexes that may regulate A-type currents, and hence neuronal excitability, in response to changes in intracellular calcium. CSEN also functions as a calc...
TMPH-01716 CHRM3 Protein, Human, Recombinant (B2M & His)

Muscarinic acetylcholine receptor M3,CHRM3

Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is Pi turnover. CHRM3 Protein, Human, Recombinant (B2M & His) is expressed in E. coli expression system with N-6xHis-B2M tag. The predicted molecular weight is 40.7 kDa and the accession number is P20309.
TMPH-03338 CHRM1 Protein, Rat, Recombinant (His)

Muscarinic acetylcholine receptor M1,CHRM1

Rat E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is Pi turnover. CHRM1 Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 21.1 kDa and the accession number is P08482.
TMPJ-00652 PSD-95 Protein, Rat, Recombinant (His)

PSD95,SAP90,Disks large homolog 4,SAP-90,PSD-95,Postsynaptic...

Rat E. coli
Disks large homolog 4(DLG4) is a cell membrane protein and it is a member of the membrane-associated guanylate kinase (MAGUK) family. The protein contains 1 guanylate kinase-like domain,3 PDZ (DHR) domains and 1 SH3 domain. With PSD-93 it is recruited into the same NMDA receptor and potassium channel clusters. These two MAGUK proteins may interact at postsynaptic sites to form a multimeric scaffold for the clustering of receptors, ion channels, and associated signaling proteins. DLG4 is the be...
TMPH-01609 LGI1 Protein, Human, Recombinant (His & Myc)

Leucine-rich glioma-inactivated protein 1,Epitempin-1,LGI1

Human E. coli
Regulates voltage-gated potassium channels assembled from KCNA1, KCNA4 and KCNAB1. It slows down channel inactivation by precluding channel closure mediated by the KCNAB1 subunit. Ligand for ADAM22 that positively regulates synaptic transmission mediated by AMPA-type glutamate receptors. Plays a role in suppressing the production of MMP1/3 through the phosphatidylinositol 3-kinase/ERK pathway. May play a role in the control of neuroblastoma cell survival.
TMPY-01854 DPP10 Protein, Human, Recombinant (His)

DPPY,DPRP3,DPRP-3,DPL2,dipeptidyl-peptidase 10 (non-function...

Human HEK293 Cells
Inactive dipeptidyl peptidase 1, also known as Dipeptidyl peptidase IV-related protein 3, Dipeptidyl peptidase X, Dipeptidyl peptidase-like protein 2, DPRP-3, DPL2 and DPP1, is a single-pass type II membrane protein which belongs to thepeptidase S9B family.DPPIV subfamily. It may modulate cell surface expression and activity of the potassium channels KCND1 and KCND2. DPP1 / DPRP3 has no detectable protease activity, most likely due to the absence of the conserved serine residue normally p...
TMPH-01715 CHRM2 Protein, Human, Recombinant (His)

CHRM2,Muscarinic acetylcholine receptor M2

Human E. coli
The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is adenylate cyclase inhibition. Signaling promotes phospholipase C activity, leading to the release of inositol trisphosphate (IP3); this then triggers calcium ion release into the cytosol. CHRM2 Protein, Human, Recombinant (His) is expressed in E. col...
TMPH-03399 VAMP2 Protein, Rat, Recombinant (His)

Vesicle-associated membrane protein 2,Vamp2,Synaptobrevin-2

Rat E. coli
Involved in the targeting and/or fusion of transport vesicles to their target membrane. Major SNARE protein of synaptic vesicles which mediates fusion of synaptic vesicles to release neurotransmitters. Essential for fast vesicular exocytosis and activity-dependent neurotransmitter release as well as fast endocytosis that mediates rapid reuse of synaptic vesicles. Modulates the gating characteristics of the delayed rectifier voltage-dependent potassium channel KCNB1. VAMP2 Protein, Rat, Recombina...
TMPJ-00988 SEPHS1 Protein, Human, Recombinant (His)

water dikinase 1,SELD,Selenophosphate synthase 1,SEPHS1,SPS1...

Human HEK293 Cells
Selenophosphate synthetase 1 (SEPHS1) belongs to the selenophosphate synthase 1 family, Class II subfamily. It has four different isoforms by alternative splicing. Isoform 1 and isoform 2 are gradually expressed during the cell cycle until G2/M phase and then decreased, which Isoform 3 is gradually expressed during the cell cycle until S phase and then decreased. SEPHS1 can be activated by phosphate ions and by potassium ions. It can synthesize synthesizes selenophosphate from selenide and ATP....
TMPY-03491 Lysozyme 2 Protein, Human, Recombinant (His)

lysozyme like 2,LYZL2

Human Baculovirus Insect Cells
The lysozyme 2 gene is a member of a family of lysozyme-like genes. Lysozymes, especially C-type lysozymes, are well-recognized bacteriolytic factors widely distributed in the animal kingdom and play a mainly protective role in host defense. Lysozymes damage bacterial cell walls by catalyzing the hydrolysis of 1,4-beta-linkages between N-acetylmuramic acid and N-acetyl-D-glucosamine residues in a peptidoglycan and between N-acetyl-D-glucosamine residues in chitodextrins. Lysozyme is part of the ...
TMPY-01695 CASPR2 Protein, Mouse, Recombinant (His)

5430425M22Rik,Caspr2,contactin associated protein-like 2,mKI...

Mouse HEK293 Cells
CNTNAP2/CASPR2 is a member of the neurexin family which functions in the vertebrate nervous system as cell adhesion molecules and receptors. This protein, like other neurexin proteins, contains epidermal growth factor repeats and laminin G domains. In addition, it includes an F5/8 type C domain, discoidin/neuropilin- and fibrinogen-like domains, thrombospondin N-terminal-like domains and a putative PDZ binding site. CNTNAP2/CASPR2 is localized at the juxtaparanodes of myelinated axons, and media...
TMPY-04561 SGK3 Protein, Human, Recombinant (His & GST)

serum/glucocorticoid regulated kinase family, member 3,SGK2,...

Human Baculovirus Insect Cells
Serine / threonine-protein kinase Sgk3, also known as Serum / glucocorticoid-regulated kinase 3, Serum / glucocorticoid-regulated kinase-like and SGK3, is a cytoplasmic vesicle protein that belongs to the protein kinase superfamily and AGC Ser/Thr protein kinase family. SGK3 contains one AGC-kinase C-terminal domain, one protein kinase domain and one PX (phox homology) domain. Two specific sites of SGK3, one in the kinase domain (Thr-32) and the other in the C-terminal regulatory region (Ser-486...
TMPY-06599 ATP1B4 Protein, Human, Recombinant (His)

ATPase, Na+/K+ transporting, β 4 polypeptide,ATPase, Na+/K+ ...

Human E. coli
ATP1B4 is a member of the X(+)/potassium ATPases subunit beta family. It is highly expressed in skeletal muscle and at a lower level in heart. ATP1B4 gene can be found in all vertebrate genomes sequenced to date. However, this gene has undergone a change in function in placental mammals compared to other species. Specifically, in fish, avian, and amphibian species, this gene encodes plasma membrane-bound beta-subunits of Na, K-ATPase. In placental mammals, the encoded protein interacts with the ...
TMPH-02521 PYCARD Protein, Mouse, Recombinant (His & Myc)

Pycard,PYD and CARD domain-containing protein,Apoptosis-asso...

Mouse E. coli
Functions as key mediator in apoptosis and inflammation. Promotes caspase-mediated apoptosis involving predominantly caspase-8 and also caspase-9 in a probable cell type-specific manner. Involved in activation of the mitochondrial apoptotic pathway, promotes caspase-8-dependent proteolytic maturation of BID independently of FADD in certain cell types and also mediates mitochondrial translocation of BAX and activates BAX-dependent apoptosis coupled to activation of caspase-9, -2 and -3. Involved ...

重组蛋白

KCNA1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01890
Species: Human
Expression System: E. coli
KcsA Protein, S. coelicolor, Recombinant (His)
Cat.No: TMPH-03603
Species: Streptomyces coelicolor
Expression System: E. coli
KCNE2 Protein, Human, Recombinant (His)
Cat.No: TMPH-01891
Species: Human
Expression System: E. coli
KCNK3 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01889
Species: Human
Expression System: E. coli
KCNMA1 Protein, Human, Recombinant
Cat.No: TMPH-01028
Species: Human
Expression System: E. coli
ATP4A Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01892
Species: Human
Expression System: E. coli
ATP4B Protein, Human, Recombinant (GST)
Cat.No: TMPH-01893
Species: Human
Expression System: E. coli
ATP4B Protein, Human, Recombinant
Cat.No: TMPH-01894
Species: Human
Expression System: E. coli
KCNAB2 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-02309
Species: Human
Expression System: E. coli
FXYD3 Protein, Human, Recombinant (His & SUMO)
Cat.No: TMPH-01358
Species: Human
Expression System: E. coli
CHRM1 Protein, Human, Recombinant (His)
Cat.No: TMPH-01714
Species: Human
Expression System: E. coli
CHRM5 Protein, Human, Recombinant (His)
Cat.No: TMPH-01717
Species: Human
Expression System: E. coli
CSEN Protein, Human, Recombinant (His)
Cat.No: TMPY-03615
Species: Human
Expression System: E. coli
CHRM3 Protein, Human, Recombinant (B2M & His)
Cat.No: TMPH-01716
Species: Human
Expression System: E. coli
CHRM1 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03338
Species: Rat
Expression System: E. coli
PSD-95 Protein, Rat, Recombinant (His)
Cat.No: TMPJ-00652
Species: Rat
Expression System: E. coli
LGI1 Protein, Human, Recombinant (His & Myc)
Cat.No: TMPH-01609
Species: Human
Expression System: E. coli
DPP10 Protein, Human, Recombinant (His)
Cat.No: TMPY-01854
Species: Human
Expression System: HEK293 Cells
CHRM2 Protein, Human, Recombinant (His)
Cat.No: TMPH-01715
Species: Human
Expression System: E. coli
VAMP2 Protein, Rat, Recombinant (His)
Cat.No: TMPH-03399
Species: Rat
Expression System: E. coli
SEPHS1 Protein, Human, Recombinant (His)
Cat.No: TMPJ-00988
Species: Human
Expression System: HEK293 Cells
Lysozyme 2 Protein, Human, Recombinant (His)
Cat.No: TMPY-03491
Species: Human
Expression System: Baculovirus Insect Cells
CASPR2 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01695
Species: Mouse
Expression System: HEK293 Cells
SGK3 Protein, Human, Recombinant (His & GST)
Cat.No: TMPY-04561
Species: Human
Expression System: Baculovirus Insect Cells
ATP1B4 Protein, Human, Recombinant (His)
Cat.No: TMPY-06599
Species: Human
Expression System: E. coli
PYCARD Protein, Mouse, Recombinant (His & Myc)
Cat.No: TMPH-02521
Species: Mouse
Expression System: E. coli
Cat. No. Product Name Target Signaling Pathways
T70313 Indoxyl Sulfate-d5 potassium salt

Indoxyl sulfate-d5 is intended for use as an internal standard for the quantification of indoxyl sulfate by GC- or LC-MS. Indoxyl sulfate is a uremic toxin and a metabolite of tryptophan. It is formed via sulfation of indole, an intermediate generated from tryptophan by intestinal bacteria, by the sulfotransferase (SULT) isoform 1A1 variant 2 (SULT1A1*2) in the liver. Indoxyl sulfate activates the aryl hydrocarbon receptor (AhR) in HepG2 40/6 hepatoma cells (EC50 = 12.1 nM in a reporter assay). ...
TMID-0234 Penicillin G-d5 potassium salt

Penicillin G-d5 potassium salt 是 Penicillin G potassium salt 的氘代化合物。Penicillin G potassium salt 的 CAS 号为 113-98-4。Benzylpenicillin potassium是青霉素家族的一种速效抗生素。
TMIH-0434 PHPB-d7

(R/S)-2-(1-hydroxy-n-pentyl)benzoic acid potassium salt-d7

PHPB-d7 是 PHPB 的氘代化合物。
TMID-0125 Canrenone-d4

Canrenone-d4 是 Canrenone 的氘代化合物。Canrenone 的 CAS 号为 976-71-6。Canrenone 是一种醛固酮 (aldosterone) 拮抗剂,广泛用作利尿剂。
TMID-0124 Canrenone-d6

Canrenone-d6 是 Canrenone 的氘代化合物。Canrenone 的 CAS 号为 976-71-6。Canrenone 是一种醛固酮 (aldosterone) 拮抗剂,广泛用作利尿剂。
T73713 Flupirtine-d4 hydrochloride

Flupirtine-d4 (D 9998-d4) hydrochloride,Flupirtine (D 9998) hydrochloride的氘代物,为神经元钾通道开放剂,具有拮抗NMDA受体的作用。
TMIH-0601 Vonoprazan-d3

Vonoprazan-d3 是 Vonoprazan 的氘代化合物。Vonoprazan 的 CAS 号为 881681-00-1。Vonoprazan 是一种质子泵抑制剂,是口服活性钾竞争性酸阻断剂,有抗分泌作用。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50值为 19 nM。它可用于研究胃酸相关疾病。
TMIH-0086 Amifampridine-d3 2HCl

Amifampridine-d3 2HCl 是 Amifampridine 2HCl 的氘代化合物。Amifampridine 2HCl 的 CAS 号为 54-96-6。Amifampridine 可用于罕见肌肉疾病的研究。
TMIH-0602 Vonoprazan-d4

Vonoprazan-d4 是 Vonoprazan 的氘代化合物。Vonoprazan 的 CAS 号为 881681-00-1。Vonoprazan 是一种质子泵抑制剂,是口服活性钾竞争性酸阻断剂,有抗分泌作用。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50值为 19 nM。它可用于研究胃酸相关疾病。
TMIJ-0210 Bupivacaine-d9

Bupivacaine-d9 是 Bupivacaine 的氘代化合物。Bupivacaine 的 CAS 号为 38396-39-3。Bupivacaine 是一种 NMDA 受体抑制剂。Bupivacaine 可以阻断钠、L-钙和钾通道。Bupivacaine 有效阻断 SCN5A 通道,IC50 为 69.5 μM。Bupivacaine 可用于慢性疼痛的研究。
T36059 Dichlorphenamide-13C6

Dichlorphenamide-13C6

Dichlorphenamide-13C6is intended for use as an internal standard for the quantification of dichlorphenamide by GC- or LC-MS. Dichlorphenamide is a sulfonamide and an orally bioavailable carbonic anhydrase (CA) inhibitor (Kis = 1.20, 38, 50, and 50 nM for the human CA isoforms CAI, CAII, CAIX, and CAXII, respectively).1It lowers intraocular pressure in rabbits when 50 μl of a 10% solution is applied topically to the eye.2Dichlorphenamide rescues the potassium deficiency and prevents insulin-induc...
TMID-0070 Amiodarone-d10 Hydrochloride

Amiodarone-d10 Hydrochloride 是 Amiodarone Hydrochloride 的氘代化合物。Amiodarone Hydrochloride 的 CAS 号为 19774-82-4。Amiodarone hydrochloride是一种抗心绞痛和 III 类抗心律失常药物,通过抑制钾通道和电压门控钠通道来增加心室和心房肌肉作用的持续时间,可导致心率和血管阻力降低。它通过成纤维细胞中的ERK1/2和p38 MAPK信号传导诱导细胞增殖和肌成纤维细胞分化,可研究室上性和室性心律失常。
TMID-0069 Amiodarone-d4 HCl

Amiodarone-d4 HCl 是 Amiodarone HCl 的氘代化合物。Amiodarone HCl 的 CAS 号为 19774-82-4。Amiodarone hydrochloride是一种抗心绞痛和 III 类抗心律失常药物,通过抑制钾通道和电压门控钠通道来增加心室和心房肌肉作用的持续时间,可导致心率和血管阻力降低。它通过成纤维细胞中的ERK1/2和p38 MAPK信号传导诱导细胞增殖和肌成纤维细胞分化,可研究室上性和室性心律失常。
T69600 Spermidine-d6

Spermidine-d6 is intended for use as an internal standard for the quantification of spermidine by GC- or LC-MS. Spermidine is an endogenous polyamine. It is formed from putrescine by spermidine synthase. Spermidine (25 µM) inhibits the activity of the human inward-rectifying potassium channel Kir2.3 in a patch-clamp assay. It induces autophagy in HeLa cells when used at a concentration of 100 µM and increases the lifespan of D. melanogaster, yeast, and C. elegans. Spermidine (30 mM in the drinki...
T71402 Nicorandil-d4

Nicorandil-d4 is intended for use as an internal standard for the quantification of nicorandil by GC- or LC-MS. Nicorandil is an activator of sulfonylurea receptor 2B (SUR2B) linked to ATP-sensitive potassium channel Kir6.2 (EC50 = ~10 µM) and a nitric oxide (NO) donor. It is selective for SUR2B/Kir6.2 over the SUR2A/Kir6.2 channel (EC50 = >500 µM). Nicorandil activates soluble guanylate cyclase in a cell-free assay and relaxes partially depolarized isolated bovine coronary artery strips (EC50 =...
T71981 Gliclazide-d4

Gliclazide-d4 is intended for use as an internal standard for the quantification of gliclazide by GC- or LC-MS. Gliclazide is a sulfonylurea and an inhibitor of pancreatic β-cell ATP-sensitive potassium (KATP) channels. It is selective for pancreatic β-cell over cardiac and arterial smooth muscle cell KATP channels. Gliclazide (5 μM) increases insulin-induced glucose uptake and glucose transporter 4 (GLUT4) translocation to the plasma membrane in a differentiated 3T3L1 adipocyte model of insulin...
T71303 Flufenamic Acid-d4

Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear...

同位素标记化合物

Indoxyl Sulfate-d5 potassium salt
Cat.No: T70313
Synonym:
Target:
Penicillin G-d5 potassium salt
Cat.No: TMID-0234
Synonym:
Target:
PHPB-d7
Cat.No: TMIH-0434
Synonym: (R/S)-2-(1-hydroxy-n-pentyl)benzoic acid potassium salt-d7
Target:
Canrenone-d4
Cat.No: TMID-0125
Synonym:
Target:
Canrenone-d6
Cat.No: TMID-0124
Synonym:
Target:
Flupirtine-d4 hydrochloride
Cat.No: T73713
Synonym:
Target:
Vonoprazan-d3
Cat.No: TMIH-0601
Synonym:
Target:
Amifampridine-d3 2HCl
Cat.No: TMIH-0086
Synonym:
Target:
Vonoprazan-d4
Cat.No: TMIH-0602
Synonym:
Target:
Bupivacaine-d9
Cat.No: TMIJ-0210
Synonym:
Target:
Dichlorphenamide-13C6
Cat.No: T36059
Synonym: Dichlorphenamide-13C6
Target:
Amiodarone-d10 Hydrochloride
Cat.No: TMID-0070
Synonym:
Target:
Amiodarone-d4 HCl
Cat.No: TMID-0069
Synonym:
Target:
Spermidine-d6
Cat.No: T69600
Synonym:
Target:
Nicorandil-d4
Cat.No: T71402
Synonym:
Target:
Gliclazide-d4
Cat.No: T71981
Synonym:
Target:
Flufenamic Acid-d4
Cat.No: T71303
Synonym:
Target:
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