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Search Results for " parasite "
Targets Recommended: Parasite Parasite

242

抑制剂 & 化合物

115

天然产物

3

化合物库

12

重组蛋白

1

同位素标记化合物

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Cat. No. Product Name
L4510 抗寄生虫库

419 compounds
419 种具有抗寄生虫活性的小分子化合物;
L1800 抗感染化合物库

2938 compounds
2938 种具有抗感染活性的化合物的特有集合,包括抗细菌、抗真菌、抗巨细胞病毒、抗HIV、抗SARS、抗流感等活性;
L6500 微生物天然产物库

550 compounds
550 种微生物来源的生物活性小分子化合物的特有集合,用于高通量、高内涵筛选;

化合物库

抗寄生虫库
Cat.No: L4510
Compounds: 419
抗感染化合物库
Cat.No: L1800
Compounds: 2938
微生物天然产物库
Cat.No: L6500
Compounds: 550
Cat. No. Product Name Target Signaling Pathways
T15272 Febantel

Parasite Microbiology/Virology
Febantel 是一种用于家禽和家畜的蛔虫、绦虫感染的驱虫剂。
T5114 Pyridaben

Calcium Channel; Parasite Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Pyridaben 是一种METI 杀螨剂,可抑制复合物 I 处的线粒体电子转运。它对多种螨虫具有活性,通过滤纸接触给药,在 25 mg/mL、100 mg/mL 和 200 mg/mL 的剂量下,分别诱导 100% 的C. malaccensis,D. farina 和T. putrescentia 死亡率。
T5839 Phosalone

Parasite Microbiology/Virology
Phosalone 是一种有机磷酸盐化学品,通常用作杀虫剂和杀螨剂。
T22415 Resorantel

Parasite Microbiology/Virology
Resorantel 是一种驱虫剂,用于研究牛和羊的寄生虫病,也被用于研究G. aegypticus。
T19714 Fenpyroximate

Others Others
Fenpyroximate 是一种有效的杀螨剂。
T7146 Piperazine adipate

Parasite Microbiology/Virology
Piperazine adipate 是一种广谱驱虫剂,可抵抗哺乳动物中很多常见的寄生虫感染。
T21727 Ivermectin B1a

SARS-CoV; Parasite Microbiology/Virology
Ivermectin B1a 是 Avermectin B1a 的一种衍生物,是 Ivermectin 的主要成分。Ivermectin 是广谱的抗寄生虫剂。Ivermectin 也是抗 SARS-CoV-2/COVID-19 的候选药物。
T6623 Oxibendazole

Apoptosis; Parasite Apoptosis; Microbiology/Virology
Oxibendazole 是一种苯并咪唑驱虫药,用于防止马和一些家养宠物的蛔虫、圆线虫、线虫、蛲虫和肺虫感染。。它可诱导细胞凋亡,具有抗癌和抗炎活性。
T38272 Thiacloprid

AChR; Parasite Microbiology/Virology; Neuroscience
Thiacloprid 属于氯烟碱类杀虫剂,主要用于防治蔬菜和果园中的蚜虫。它会破坏 DNA 的稳定性,通过疏水或氢相互作用,结合到小沟槽中,改变 DNA 的结构和稳定性。
T0873 Dinitolmide

二硝托胺,Zoalene

Antibiotic; Parasite Microbiology/Virology
Dinitolmide (Zoalene) 是一种家禽饲料添加剂,是家禽的抗球虫剂。
T15409 GNF179

Parasite Microbiology/Virology
GNF179 是8,8-二甲基 IP 类似物。 它表现出对多药耐药菌株 W2 的效力,具有良好的体外代谢稳定性和体内口服生物相容性。
T14766 BPH-715

Others; Parasite Microbiology/Virology; Others
BPH-715 抑制恶性疟原虫的肝脏阶段生长,对 HepG2 细胞中的恶性疟原虫外红细胞的形成的 IC50 为 10 μM。
T39849 Propargite

Parasite Microbiology/Virology
Propropgite 通过诱导 DNA 损伤来诱导 β 细胞坏死。它诱导 MIN6 细胞死亡的 IC50为 1 μM.。它可用于杀死螨虫。
T38845 Dodecamethylpentasiloxane

Parasite Microbiology/Virology
Dodecamethylpentasiloxane 可用作臭虫杀虫剂。 Dodecamethylpentasiloxane 是硅氧烷的一种成分,可用作硅油。
T7901 Emodepside

Bay 44-4400

Parasite Microbiology/Virology
Emodepside (Bay 44-4400) 是一种对多种胃肠道线虫有效的驱虫药,具有广谱驱虫活性。
T3188 RE-640

CCR; Parasite Immunology/Inflammation; Microbiology/Virology
NSC-5844 (RE-640) 是 4-氨基喹啉衍生物,起抗肿瘤和抗疟疾作用。
T0997 Temephos

双硫磷,Temefos

AChR; Parasite Microbiology/Virology; Neuroscience
Temephos (Temefos) 是一种胆碱酯酶抑制剂,是一种有机硫代磷酸盐杀虫剂,用于治疗被携带疾病的昆虫侵染的水。
T4218 Broxaldine

Brobenzoxaldine,溴沙定

Antibacterial; Antibiotic; Parasite; Antifungal Microbiology/Virology
Broxaldine (Brobenzoxaldine) 是一种具有抗原生动物活性的小分子药物。它抑制艰难梭菌的 MIC 值为 4 µM,并具有抗真菌作用。
T2180 Hexythiazox

Parasite Microbiology/Virology
Hexythiazox 是一种螨类生长调节剂和噻唑烷类杀螨剂,对多种螨类具有长效杀虫作用,适用于植物从萌芽到结果的任何生长阶段。
T0066 Dichlorophen

双氯酚,DDM,Dichlorophene

Antibacterial; Parasite; Antifungal Microbiology/Virology
Dichlorophen (DDM) 是一种抗微生物剂,对绦虫,原生动物,真菌和细菌具有活性,通过增加肠道内容物的清除,消除肠道中的绦虫感染。
T15775 Lotilaner

GABA Receptor; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Lotilaner 是杀寄生虫剂,是非竞争性的昆虫GABACl 受体拮抗剂,对果蝇 GABA 受体的IC50值为 23.84 nM。对家犬的 GABAA 无明显作用。
T5639 lufenuron

Fluphenacur,虱螨脲

Parasite Microbiology/Virology
Lufenuron (Fluphenacur) 和几丁质合成抑制剂,可抑制节肢动物的蜕皮,控制蚤和鱼虱。
T9741 INE963

Others Others
INE963 是快速有效的血液阶段抗疟剂,EC50为 3-6 nM。INE963 有单纯性疟疾的研究潜力。
T7400 RRX-001

Apoptosis; Dehydrogenase; Parasite Apoptosis; Metabolism; Microbiology/Virology
RRx-001 是一种低氧选择性的表观遗传因子,被用作放射或化疗敏感剂,能诱发凋亡,克服骨髓瘤的耐药性。它是G6PD 的有效抑制剂,具有抗疟、抗癌活性。它是免疫检查点的抑制剂,可下调CD47和SIRP-α。
T0998 Diazinon

二嗪磷,Dimpylate,二嗪农

AChE; Parasite Microbiology/Virology; Neuroscience
Diazinon (Dimpylate) 是一种硫磷酸酯,是非内吸性有机磷杀虫剂,有效抑制,包括蟑螂、蠹虫、蚂蚁和跳蚤在内的多种害虫。
T1145 Diminazene Aceturate

Others; Serine Protease; Parasite Microbiology/Virology; Others; Proteases/Proteasome
Diminazene aceturate 是血管紧张素转化酶 2 的激活剂,具有强效抗炎特性。它还是一种抗锥虫药物,适用于牲畜。它主要生化机理是通过与富含腺嘌呤-胸腺嘧啶碱基对的位点发生特异性相互作用,以非插入方式与锥虫动子体 DNA 结合。
T5471 GUANABENZ

Adrenergic Receptor GPCR/G Protein; Neuroscience
GUANABENZ 是一种中枢 alpha-2 肾上腺素能激动剂。它的作用机制是作为肾上腺素能 α2-激动剂。
T13928 Tioxazafen

Others; Parasite Microbiology/Virology; Others
Tioxazafen 是一种二取代的恶二唑,是一种广谱种子处理杀线虫剂,对玉米,大豆和棉花中的线虫有效。
T6532 Hesperadin

Influenza Virus; Parasite; Aurora Kinase; Autophagy Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Microbiology/Virology
Hesperadin 是 Aurora A 和 B 的 ATP 竞争性吲哚酮抑制剂,抑制 Aurora B 的 IC50值为250nM。它通过阻断核分裂和胞质分裂而抑制布鲁氏锥虫的生长。它也是一种广谱流感抗病毒剂。
T10336 Antimalarial agent 1

Parasite Microbiology/Virology
Antimalarial agent 1 是一种抗疟药。
T0471 Decoquinate

Decoxy,Deccox,癸氧喹酯

Parasite Microbiology/Virology
Decoquinate (Deccox) 是一种喹诺酮衍生物,抑制疟原虫肝发育和红细胞复制,可研究家庭反刍动物的球虫病。
T8337 Nequinate

Xanthine Oxidase; Parasite Metabolism; Microbiology/Virology
Nequinate 是一种喹啉化合物,是一种抗球虫剂,可预防球虫病。它抑制黄嘌呤氧化还原酶活性。
T3266 Lumefantrine

Benflumetol,dl-Benflumelol,苯芴醇

Others; Parasite; Autophagy Autophagy; Microbiology/Virology; Others
Lumefantrine (dl-Benflumelol) 是一种抗疟药,用于治疗急性单纯性疟疾。与Artemether 联用,可提高疗效。
T0376 Crotamiton

Eurax,Crotamitone,克罗米通,Veteusan

Parasite Microbiology/Virology
Crotamiton (Eurax) 既是杀疥螨剂 ,可研究疥疮,也是止痒剂, 可除去疥疮寄生虫。
T1172 Diclazuril

地克珠利,R-64433

Antibiotic; Parasite Microbiology/Virology
Diclazuril (R-64433) 是一种具有口服活性的抗球虫剂,是苯乙腈衍生物。它可用于某些传染病和寄生虫病的相关研究。
T3493 Clofentezine

Bisclofentazin,Acaristop,Apollo,四螨嗪

Others Others
Clofentezine (Apollo) 是生长抑制剂,对螨虫具有显著的致死作用。
T21687 Conoidin A

Parasite Microbiology/Virology
Conoidin A 是刚地弓形虫过氧化物酶 II 的细胞通透性抑制剂,有杀线虫特性。它共价结合 TgPrxII 的过氧化物催化位点 Cys47,不可逆地抑制其过氧化物活性,IC50为 23 µM。它也抑制哺乳动物 PrxI 和 PrxII 的氧化。它具有抗氧化、神经保护作用,可研究缺血性心脏病。
T3202 Fluensulfone

MCW-2

Parasite Microbiology/Virology
Fluensulfone (MCW-2) 是一种新型杀线虫剂,可化学防治植物寄生线虫。
T6452 Closantel Sodium

Antibacterial; Parasite Microbiology/Virology
Closantel sodium 是抗寄生虫活性的卤化水杨酰苯胺。它是高度特异性的盘尾丝虫几丁质酶抑制剂。
T0930 Sulfadiazine

Sulphadiazine,磺胺嘧啶

Antibacterial; Antibiotic; Parasite; Autophagy Autophagy; Microbiology/Virology
Sulfadiazine (Sulphadiazine) 是一种磺胺类抗生素具有抗疟活性,可研究弓形虫病。
T8767 PfDHODH-IN-2

Dehydrogenase; Parasite Metabolism; Microbiology/Virology
PfDHODH-IN-2 是一种二氢噻吩酮衍生物,是一种有效的恶性疟原虫二氢乳清酸脱氢酶抑制剂,其IC50值为 1.11 µM。它具有抗疟作用,可研究疟疾。
T1435 Praziquantel

吡喹酮,Pyquiton,Droncit,Biltricide

Calcium Channel; Antibiotic; Parasite Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Praziquantel (Droncit) 是一种外消旋混合物,由 (R)-Praziquantel 和 (S)-Praziquantel 组成。它可研究血吸虫病。
T8381 Amodiaquine

Others; Histone Methyltransferase; Parasite Chromatin/Epigenetic; Microbiology/Virology; Others
Amodiaquine 是一种合成的4-氨基喹啉类抗疟剂,是一种有口服活性的组胺 N-甲基转移酶抑制剂。它也是一种Nurr1激动剂,有抗炎活性,可特异性结合Nurr1的配体结合域,EC50约为20 μM。
T16125 MMV390048

Parasite; PI4K Microbiology/Virology; PI3K/Akt/mTOR signaling
MMV390048 是一种抗疟药,是一种新型化学疟原虫 PI4K 抑制剂。它与疟原虫 PI4K 的 ATP 结合位点结合,不与除人类 PIP4K2C 外的其他恶性疟原虫和人类激酶结合。
T0286 Bephenium (hydroxynaphthoate)

羟萘酸苄酚宁,Bephenium Hydroxynaphthoate

Parasite Microbiology/Virology
Bephenium hydroxynaphthoate 是一种灭虫剂,可研究蛔虫感染,也是B 型AChR 激动剂。
T5477 ELQ-300

Parasite Microbiology/Virology
ELQ-300 是一种有口服生物活性的抗疟疾剂,可作为细胞色素 bc1 复合物的还原位点的抑制剂
T6309 AZ960

AZ 960

Apoptosis; Virus Protease; JAK; Parasite Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Microbiology/Virology; Stem Cells
AZ960 是一种高效选择性的 JAK2激酶抑制剂,Ki 值为0.45 nM。
T7182 Metaflumizone

BAS-320I,氰氟虫腙

Sodium Channel; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Metaflumizone (BAS-320I) 是一种缩氨基脲杀虫剂,是钠离子通道阻滞剂。
T64320 ML251

Glucokinase; Parasite Metabolism; Microbiology/Virology
ML251 是一种有效的新型纳摩尔 T. brucei 和 T. cruzi 磷酸果糖激酶抑制剂,对 T. brucei PFK 和 T. cruzi PFK 的 IC50值为 0.37和 0.13 μM,可研究寄生虫。
T4269 Buparvaquone

布帕伐醌,Butalex,BW 720C

Antibiotic; Parasite Microbiology/Virology
Buparvaquone (BW 720C) 是与parvaquone 和atovaquone 有关的一种羟基萘醌类抗原虫药。

化合物

Febantel
Cat.No: T15272
Synonym:
Target: Parasite
Pyridaben
Cat.No: T5114
Synonym:
Target: Calcium Channel, Parasite
Phosalone
Cat.No: T5839
Synonym:
Target: Parasite
Resorantel
Cat.No: T22415
Synonym:
Target: Parasite
Fenpyroximate
Cat.No: T19714
Synonym:
Target: Others
Piperazine adipate
Cat.No: T7146
Synonym:
Target: Parasite
Ivermectin B1a
Cat.No: T21727
Synonym:
Target: SARS-CoV, Parasite
Oxibendazole
Cat.No: T6623
Synonym:
Target: Apoptosis, Parasite
Thiacloprid
Cat.No: T38272
Synonym:
Target: AChR, Parasite
Dinitolmide
Cat.No: T0873
Synonym: 二硝托胺,Zoalene
Target: Antibiotic, Parasite
GNF179
Cat.No: T15409
Synonym:
Target: Parasite
BPH-715
Cat.No: T14766
Synonym:
Target: Others, Parasite
Propargite
Cat.No: T39849
Synonym:
Target: Parasite
Dodecamethylpentasiloxane
Cat.No: T38845
Synonym:
Target: Parasite
Emodepside
Cat.No: T7901
Synonym: Bay 44-4400
Target: Parasite
RE-640
Cat.No: T3188
Synonym:
Target: CCR, Parasite
Temephos
Cat.No: T0997
Synonym: 双硫磷,Temefos
Target: AChR, Parasite
Broxaldine
Cat.No: T4218
Synonym: Brobenzoxaldine,溴沙定
Target: Antibacterial, Antibiotic, Parasite, Antifungal
Hexythiazox
Cat.No: T2180
Synonym:
Target: Parasite
Dichlorophen
Cat.No: T0066
Synonym: 双氯酚,DDM,Dichlorophene
Target: Antibacterial, Parasite, Antifungal
Lotilaner
Cat.No: T15775
Synonym:
Target: GABA Receptor, Parasite
lufenuron
Cat.No: T5639
Synonym: Fluphenacur,虱螨脲
Target: Parasite
INE963
Cat.No: T9741
Synonym:
Target: Others
RRX-001
Cat.No: T7400
Synonym:
Target: Apoptosis, Dehydrogenase, Parasite
Diazinon
Cat.No: T0998
Synonym: 二嗪磷,Dimpylate,二嗪农
Target: AChE, Parasite
Diminazene Aceturate
Cat.No: T1145
Synonym:
Target: Others, Serine Protease, Parasite
GUANABENZ
Cat.No: T5471
Synonym:
Target: Adrenergic Receptor
Tioxazafen
Cat.No: T13928
Synonym:
Target: Others, Parasite
Hesperadin
Cat.No: T6532
Synonym:
Target: Influenza Virus, Parasite, Aurora Kinase, Autophagy
Antimalarial agent 1
Cat.No: T10336
Synonym:
Target: Parasite
Decoquinate
Cat.No: T0471
Synonym: Decoxy,Deccox,癸氧喹酯
Target: Parasite
Nequinate
Cat.No: T8337
Synonym:
Target: Xanthine Oxidase, Parasite
Lumefantrine
Cat.No: T3266
Synonym: Benflumetol,dl-Benflumelol,苯芴醇
Target: Others, Parasite, Autophagy
Crotamiton
Cat.No: T0376
Synonym: Eurax,Crotamitone,克罗米通,Veteusan
Target: Parasite
Diclazuril
Cat.No: T1172
Synonym: 地克珠利,R-64433
Target: Antibiotic, Parasite
Clofentezine
Cat.No: T3493
Synonym: Bisclofentazin,Acaristop,Apollo,四螨嗪
Target: Others
Conoidin A
Cat.No: T21687
Synonym:
Target: Parasite
Fluensulfone
Cat.No: T3202
Synonym: MCW-2
Target: Parasite
Closantel Sodium
Cat.No: T6452
Synonym:
Target: Antibacterial, Parasite
Sulfadiazine
Cat.No: T0930
Synonym: Sulphadiazine,磺胺嘧啶
Target: Antibacterial, Antibiotic, Parasite, Autophagy
PfDHODH-IN-2
Cat.No: T8767
Synonym:
Target: Dehydrogenase, Parasite
Praziquantel
Cat.No: T1435
Synonym: 吡喹酮,Pyquiton,Droncit,Biltricide
Target: Calcium Channel, Antibiotic, Parasite
Amodiaquine
Cat.No: T8381
Synonym:
Target: Others, Histone Methyltransferase, Parasite
MMV390048
Cat.No: T16125
Synonym:
Target: Parasite, PI4K
Bephenium (hydroxynaphthoate)
Cat.No: T0286
Synonym: 羟萘酸苄酚宁,Bephenium Hydroxynaphthoate
Target: Parasite
ELQ-300
Cat.No: T5477
Synonym:
Target: Parasite
AZ960
Cat.No: T6309
Synonym: AZ 960
Target: Apoptosis, Virus Protease, JAK, Parasite
Metaflumizone
Cat.No: T7182
Synonym: BAS-320I,氰氟虫腙
Target: Sodium Channel, Parasite
ML251
Cat.No: T64320
Synonym:
Target: Glucokinase, Parasite
Buparvaquone
Cat.No: T4269
Synonym: 布帕伐醌,Butalex,BW 720C
Target: Antibiotic, Parasite
Cat. No. Product Name Target Signaling Pathways
T5708 LUPENONE

Phosphatase; Parasite Metabolism; Microbiology/Virology
Lupenone 是从Rhizoma Musae 中分离出的 lupine 型三萜类天然产物。它有如抗炎,抗病毒,抗糖尿病,抗癌,改善南美锥虫病的药理活性。
TN1016 Kukoamine A

NF-κB; Lipoxygenase; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB
Kukoamine A 是一种天然的精胺衍生物,具有抗癌、抗高血压、细胞保护、抗氧化和抗炎活性。它是锥虫硫磷还原酶抑制剂,Ki 值为 1.8 μM。
T11811 Laetanine

Parasite Microbiology/Virology
Laetanine 是从Litsea laeta 提取到的一种去甲马飞生物碱,有抗疟原虫活性。
T6S2024 Harpagide

Antibacterial; Parasite Microbiology/Virology
Harpagide 是从Scrophularia cryptophila 中分离出来的一种鸢尾糖苷,具有抗炎和抗寄生虫活性,对T.b. rhodesiense 具有体外锥虫杀虫活性,IC50为 21 μg/mL,它对L. donovani 的IC50值为 2.0 μg/mL。
TN1012 Febrifugine

IL Receptor; Anti-infection; Parasite Immunology/Inflammation; Microbiology/Virology
Febrifugine 是存在于常山的根和叶中的一种喹唑啉酮类生物碱,有抗疟活性。它是一种有效的抗球虫药,具有杀灭裂殖体的作用。
T5889 Kojic acid

Tyrosinase; Parasite Microbiology/Virology; Proteases/Proteasome
Kojic acid 是 Aspergillus oryzae 产生的一种真菌代谢物,用作抗氧化剂和防辐射剂,可抑制酪氨酸酶。
T5660 Menthone

IL Receptor; TNF; NF-κB; Parasite Apoptosis; Immunology/Inflammation; Microbiology/Virology; NF-κB
Menthone 是一种从植物和薄荷油中提取的单萜,是精油的主要挥发性成分,具有抗炎和抗氧化特性。
T1381 Milbemycin oxime

Others; Antibiotic; Parasite Microbiology/Virology; Others
Milbemycin oxime 是一种大环内酯,具有广谱抗寄生虫活性。它由 Milbemycin A4 和 A3 组成。它可结合谷氨酸门控的氯离子通道,可作用于肠道线虫,肺和心脏蠕虫。
TN6730 Epoxyazadiradione

NF-κB NF-κB
Epoxyazadiradione 是从印楝果实中得到的柠檬苦素。它能够可逆的、非竞争性的抑制人类、约氏疟原虫、疟原虫的互变异构酶活性。它具有抗疟原虫和人类 MIF 诱导的促炎反应的潜力。
T5771 Hypocrellin A

Antibacterial; PKC; Parasite Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
Hypocrellin A 是一种天然的PKC 抑制剂,具有光诱导的抗肿瘤、抗真菌和抗病毒活性,还对 MHC 限制性抗原呈递发挥免疫调节作用。
TN1610 Epimagnolin A

Parasite Microbiology/Virology
Epimagnolin A 是一种糠醛木脂素,具有中等的抗疟原虫活性,IC50值为5.7 μg/mL。
TN3466 Atherosperminine

cAMP; Calcium Channel; AChR; Parasite GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Atherosperminine 是一种天然生物碱,在体外表现出抗疟原虫活性,IC50为 5.80 μM。它具有DPPH 自由基清除活性,其IC50值为 29.56 µg/mL。它对气管有非特异性的弛缓作用。它是一种良好的还原剂,具有螯合金属的能力。
T5800 Allosecurinine

Allosecurinin

Antifungal Microbiology/Virology
Allosecurinine 是一种从 M.indica 和 M.discoidea 中分离出的 Securinega 生物碱,具有抗真菌活性。
T15277 Fervenulin

Parasite Microbiology/Virology
Fervenulin 具有杀灭线虫活性,抑制线虫M. incognita 卵孵化和 J2 的校正死亡率,MIC 分别为 30 μg/mL 和 120 μg/mL。
TN1100 Nepodin

transporter; COX; AMPK; Parasite Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
Nepodin 是从Rumex crispus 中分离的一种醌氧化还原酶抑制剂,具有抗糖尿病和抗疟疾的作用。。它通过激活 AMPK 刺激 GLUT4 向质膜的转运。
T13539 Allopurinol riboside

Others; Endogenous Metabolite; Parasite; Drug Metabolite Metabolism; Microbiology/Virology; Others
Allopurinol riboside 是别嘌醇的代谢产物,具有抗寄生虫作用。 Allopurinol riboside 竞争性抑制嘌呤核苷磷酸化酶对肌苷的作用,Ki 为 277 μM。
TN4660 Niranthin

Anti-infection; HBV; PAFR; Topoisomerase DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology
Niranthin 是一种木脂素,具有广泛的药理活性。它是L. donovaniIB 拓扑异构酶的非竞争性抑制剂,可用于研究耐药利什曼病的治疗。
TN6512 Tectol

Transferase; Parasite Metabolism; Microbiology/Virology
Tectol 是从Lippia sidoides 中分离的,对人白血病细胞株 HL60 和 CEM 具有显著的抑制作用。它是法尼基转移酶抑制剂,在人和布氏锥虫的IC50分别为 2.09 和 1.73 μM。它具有抗疟原虫活性,是一种中等活性的生长抑制剂,IC50 为 3.44±0.20μM。
T0690 Quinine

奎宁树

Potassium Channel; Platelet aggregation; Parasite Membrane transporter/Ion channel; Microbiology/Virology; Others
Quinine 是一种从金鸡纳树皮中提取的生物碱,用于预防和治疗疟疾。它也用于特发性肌肉痉挛,可抑制电压脉冲引起的 MT mSlo3 (KCa5.1) 通道 +100 mV 电流, 其IC50值为 169 μM,是一种钾离子通道抑制剂。
T2S2172 nerolidol

(±)-Nerolidol,Peruviol,橙花叔醇

Others; Endogenous Metabolite; Antibacterial; Parasite; Antifungal Metabolism; Microbiology/Virology; Others
Nerolidol (Peruviol) 是天然膜活性倍半萜,有抗肿瘤、抗细菌、抗真菌和抗寄生虫活性。它对动物有镇静作用,氧化过程对神经元病理后果起关键作用。
TN2239 Strictosamide

异长春花苷内酰胺

ATPase; Potassium Channel; Sodium Channel; Parasite; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Strictosamide 具有抗炎、抗疟原虫和抗真菌活性。
T4S0590 Columbin

Phospholipase; COX; Parasite Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Columbin 是有口服活性的二萜呋喃内酯,选择性抑制COX-1和COX-2,EC50值为 327 μM 和 53.1 μM,具有抗炎和抗锥虫体作用。
T6S0084 Tuberostemonine

对叶百部碱,Tuberstemonine

Parasite Microbiology/Virology
Tuberostemonine (Tuberstemonine) 是一种生物碱,可作为抗疟疾剂,有较高的肠道通透性。
T5780 HYPOCRELLIN B

Apoptosis; Parasite; Antifungal Apoptosis; Microbiology/Virology
Hypocrellin B 是从真菌Hypocrella bambusae 和Shiraia bambusicola 中分离得到的一种感光颜料,可用于癌症光动力研究。它是一个凋亡诱导剂,还拥有抗菌和抗利什曼活性。
T8275 (+)-Isopulegol

异苏木精,異洋薄[荷]醇

Parasite Microbiology/Virology
(+)-Isopulegol 是加拿大薄荷树中发现的一种萜类,是T. confusum 成虫和T. granarium 幼虫的摄食引诱剂,对S. granarius 和T. confusum 的成虫具有刺激作用。
TN1860 Licoflavone B

甘草黄酮 B,甘草黄酮B

ATPase; Anti-infection; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Licoflavone B 是从甘草中得到的一种类黄酮,抑制曼氏血吸虫 ATPase 和 ADPase 的活性,IC50值分别为 23.78 µM 和 31.50 µM。
T0969 Doramectin

Dectomax,Cyclohexylavermectin B1,多拉菌素

Others; Antibiotic; Parasite Microbiology/Virology; Others
Doramectin (Dectomax) 是 Ivermectin 的衍生物。它是一种抗寄生虫抗生素。它具有在 NMRI 小鼠感染模型中抗曼氏链球菌作用。
T10835 Cletoquine

Desethylhydroxychloroquine

Parasite; Antifection Microbiology/Virology
Cletoquine 是 Hydroxychloroquine 的主要活性代谢物。 Cletoquine 具有对抗基孔肯雅病毒 (CHIKV) 的能力。 Cletoquine 具有抗疟作用,并具有治疗自身免疫性疾病的潜力。
T0433 Artesunate

WR-256283,青蒿琥酯

Virus Protease; Ferroptosis; STAT; Parasite Apoptosis; JAK/STAT signaling; Microbiology/Virology; Stem Cells
Artesunate (WR-256283) 是治疗疟疾的青蒿素组药物的一部分。 它是青蒿素的半合成衍生物,具有水溶性。
T0938 Thiabendazole

2-(4-Thiazolyl)benzimidazole,噻菌灵

Microtubule Associated; Mitochondrial Metabolism; Parasite Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Thiabendazole (2-(4-Thiazolyl)benzimidazole) 是具有驱虫特性的苯并咪唑衍生物。
T2827 Asiatic acid

Asiantic acid,Dammarolic acid,积雪草酸

Apoptosis; p38 MAPK; Parasite Apoptosis; MAPK; Microbiology/Virology
Asiatic acid (Dammarolic acid) 是在Centella asiatica 中发现的一种五环三萜,有抗炎活性,可诱导黑色素瘤细胞的凋亡,有可能治疗皮肤癌。
TN7103 13,21-Dihydroeurycomanone

Pasakbumin C

Anti-infection; Parasite Microbiology/Virology
13,21-Dihydroeurycomanone (Pasakbumin C) 是从 Eurycoma longifolia 根部分离得到的一种天然产物,有抗寄生虫活性。
TWS2045 Bruceine D

鸦胆子素D,鸦胆子苦素D

Apoptosis; Antiviral; Gamma-secretase; Parasite Apoptosis; Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome; Stem Cells
Bruceine D 是Notch 抑制剂,有抗癌活性,诱导几种人癌细胞调亡。它是一种有效的植物性昆虫拒食剂,有显著的系统特性和抑制害虫生长的作用。它具有较强的驱虫活性,抑制D. intermedius 的 EC50值为 0.57 mg/L。
TN1432 Bacopasaponin C

(-)-假马齿苋皂苷 C,假马齿苋皂苷C

Anti-infection; GABA Receptor; NMDAR Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷,具有抗肿瘤和抗利什曼原虫作用。
TN2027 Oxysanguinarine

8-Oxosanguinarine,氧化血根碱,Hydroxysanguinarine

Parasite Microbiology/Virology
Oxysanguinarine (Hydroxysanguinarine) 是一种来自Meconopsis simplicifolia 的小檗生物碱,具有抗疟和抗血小板聚集活性,对登革热病毒具有潜在的抑制作用。
T6447 Clindamycin

Clinimycin,Sobelin,Chlolincocin,克林霉素

Antibacterial; Antibiotic Microbiology/Virology
Clindamycin (Sobelin) 从细菌核糖体中解离肽基-tRNA,破坏细菌蛋白质合成。 它是一种半合成广谱抗生素,由母体化合物林可霉素化学修饰而成。
T4593 ISOPIMPINELLIN

5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen

Antiviral; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology
Isopimpinellin (4,9-Dimethoxypsoralen) 是从 Pimpinella saxifrage 根部分离得到的一种天然产物,具有抗病毒和抗利什曼病活性。
T7938 Quinidine

奎尼丁,奎宁树

Parasite Microbiology/Virology
Quinidine 是一种抗心律失常剂,也是 K+通道的有效阻断剂,其 IC50值为 19.9 μM。它是一种选择性细胞色素 P450db 的有效抑制剂,也可研究疟疾。
T3254 PHYTOL

植醇,trans-Phytol,(E)-Phytol

Antibacterial; PPAR; Parasite DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
PHYTOL (trans-Phytol) 是一种从叶绿素中提取的二萜醇,广泛应用于食品添加剂和医药领域,具有很好的抗血吸虫特性。它具有抗伤害、抗氧化、抗炎、抗过敏等作用。它对结核分枝杆菌和金黄色葡萄球菌具有抗菌活性。
T1155 Mebendazole

甲苯达唑,甲苯咪唑,Telmin,Mebenvet,Vermox,Pantelmin

Apoptosis; Microtubule Associated; Parasite Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Mebendazole (Mebenvet) 是一种 hedgehog 抑制剂,用作驱虫药。
T0819 Spiramycin

Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Spiramycin (Rovamycin) 是一种由安博链霉菌产生的大环内酯类抗生素,具有抗细菌和弓形虫活性,并具有抗寄生虫作用。它由 16 个内酯环组成,其上附着 mycaminose,forosamine 和 mycarose 三种糖。
T6S0214 dl-Maackiain

(+)-Maackiain,高丽槐素,Demethylpterocarpin

Apoptosis; Parasite Apoptosis; Microbiology/Virology
dl-Maackiain (Demethylpterocarpin) 是分离自Maackia amurensis Rupr.et Maxim 的一种杀幼虫剂,针对埃及伊蚊,其LD50为 21.95 μg/ ml。
T10388 Asparagusic acid

1,2-二噻戊环-4-羧酸,芦笋酸

Parasite Microbiology/Virology
Asparagusic acid 是芦笋植物中的一种含硫气味成分,是植物生长抑制剂,具有抗寄生虫作用。
T0896 Furaltadone hydrochloride

Furaltadone HCl,盐酸呋喃它酮

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Furaltadone hydrochloride (Furaltadone HCl) 是硝基呋喃药,可研究肠沙门氏菌感染,治疗球虫病。Furaltadone 具有体外抑制葡萄球菌作用。
T3792 Ajugol

益母草苷,益母草苷A,Leonuride

Parasite Microbiology/Virology
Ajugol (Leonuride) 是从Sideritis germanicopolitana 分离得到的一种环烯醚糖苷。它有抗原生动物活性,对Trypanosoma b. rhodesiense 锥虫的 IC50为 31.8 μg/mL。
T8259 Doxycycline monohydrate

水合强力霉素,强力霉素一水物

MMP; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline monohydrate 是一种四环素抗生素,是广谱金属蛋白酶抑制剂,具有抗菌活性。
T2S2046 Bruceine A

Dihydrobrusatol,鸦胆子素 A,NSC31616

Antibiotic; Parasite Microbiology/Virology
Bruceine A (NSC-31616) 是一种从鸦胆子 (L.) 的干果中提取的天然类苦素化合物,有治疗犬巴贝斯虫病的潜力。
TN1341 8-Deoxygartanin

8-脱氧藤黄苷

Beta Amyloid; NF-κB; Parasite Microbiology/Virology; Neuroscience; NF-κB
8-Deoxygartanin 是山竹果中的异戊烯化呫吨酮。它是丁基胆碱酯酶选择性抑制剂,对阿尔茨海默病 (AD) 具有多功能活性,可能是有希望治疗 AD 的化合物。
THS1455 DihydroarteMisinic acid

双氢青蒿酸,Dihydro-Artmisinic Acid,二氢青蒿酸

Ferroptosis; Parasite Apoptosis; Microbiology/Virology
DihydroarteMisinic acid (Dihydro-Artmisinic Acid) 是青蒿的天然产物,是青蒿素的主要直接前体,青蒿素是一种广泛用于治疗疟疾的药草。
T0012 Cinchonine

LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁

Apoptosis; P-gp; Parasite Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Cinchonine (LA40221) 是金鸡纳树皮中的一种天然产物。它可激活内质网应激诱导的人肝癌细胞凋亡。它是一种酰胺类局部麻醉剂。
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天然产物

LUPENONE
Cat.No: T5708
Synonym:
Target: Phosphatase, Parasite
Kukoamine A
Cat.No: TN1016
Synonym:
Target: NF-κB, Lipoxygenase, DNA/RNA Synthesis, Parasite
Laetanine
Cat.No: T11811
Synonym:
Target: Parasite
Harpagide
Cat.No: T6S2024
Synonym:
Target: Antibacterial, Parasite
Febrifugine
Cat.No: TN1012
Synonym:
Target: IL Receptor, Anti-infection, Parasite
Kojic acid
Cat.No: T5889
Synonym:
Target: Tyrosinase, Parasite
Menthone
Cat.No: T5660
Synonym:
Target: IL Receptor, TNF, NF-κB, Parasite
Milbemycin oxime
Cat.No: T1381
Synonym:
Target: Others, Antibiotic, Parasite
Epoxyazadiradione
Cat.No: TN6730
Synonym:
Target: NF-κB
Hypocrellin A
Cat.No: T5771
Synonym:
Target: Antibacterial, PKC, Parasite
Epimagnolin A
Cat.No: TN1610
Synonym:
Target: Parasite
Atherosperminine
Cat.No: TN3466
Synonym:
Target: cAMP, Calcium Channel, AChR, Parasite
Allosecurinine
Cat.No: T5800
Synonym: Allosecurinin
Target: Antifungal
Fervenulin
Cat.No: T15277
Synonym:
Target: Parasite
Nepodin
Cat.No: TN1100
Synonym:
Target: transporter, COX, AMPK, Parasite
Allopurinol riboside
Cat.No: T13539
Synonym:
Target: Others, Endogenous Metabolite, Parasite, Drug Metabolite
Niranthin
Cat.No: TN4660
Synonym:
Target: Anti-infection, HBV, PAFR, Topoisomerase
Tectol
Cat.No: TN6512
Synonym:
Target: Transferase, Parasite
Quinine
Cat.No: T0690
Synonym: 奎宁树
Target: Potassium Channel, Platelet aggregation, Parasite
nerolidol
Cat.No: T2S2172
Synonym: (±)-Nerolidol,Peruviol,橙花叔醇
Target: Others, Endogenous Metabolite, Antibacterial, Parasite, Antifungal
Strictosamide
Cat.No: TN2239
Synonym: 异长春花苷内酰胺
Target: ATPase, Potassium Channel, Sodium Channel, Parasite, Antifungal
Columbin
Cat.No: T4S0590
Synonym:
Target: Phospholipase, COX, Parasite
Tuberostemonine
Cat.No: T6S0084
Synonym: 对叶百部碱,Tuberstemonine
Target: Parasite
HYPOCRELLIN B
Cat.No: T5780
Synonym:
Target: Apoptosis, Parasite, Antifungal
(+)-Isopulegol
Cat.No: T8275
Synonym: 异苏木精,異洋薄[荷]醇
Target: Parasite
Licoflavone B
Cat.No: TN1860
Synonym: 甘草黄酮 B,甘草黄酮B
Target: ATPase, Anti-infection, Parasite
Doramectin
Cat.No: T0969
Synonym: Dectomax,Cyclohexylavermectin B1,多拉菌素
Target: Others, Antibiotic, Parasite
Cletoquine
Cat.No: T10835
Synonym: Desethylhydroxychloroquine
Target: Parasite, Antifection
Artesunate
Cat.No: T0433
Synonym: WR-256283,青蒿琥酯
Target: Virus Protease, Ferroptosis, STAT, Parasite
Thiabendazole
Cat.No: T0938
Synonym: 2-(4-Thiazolyl)benzimidazole,噻菌灵
Target: Microtubule Associated, Mitochondrial Metabolism, Parasite
Asiatic acid
Cat.No: T2827
Synonym: Asiantic acid,Dammarolic acid,积雪草酸
Target: Apoptosis, p38 MAPK, Parasite
13,21-Dihydroeurycomanone
Cat.No: TN7103
Synonym: Pasakbumin C
Target: Anti-infection, Parasite
Bruceine D
Cat.No: TWS2045
Synonym: 鸦胆子素D,鸦胆子苦素D
Target: Apoptosis, Antiviral, Gamma-secretase, Parasite
Bacopasaponin C
Cat.No: TN1432
Synonym: (-)-假马齿苋皂苷 C,假马齿苋皂苷C
Target: Anti-infection, GABA Receptor, NMDAR
Oxysanguinarine
Cat.No: TN2027
Synonym: 8-Oxosanguinarine,氧化血根碱,Hydroxysanguinarine
Target: Parasite
Clindamycin
Cat.No: T6447
Synonym: Clinimycin,Sobelin,Chlolincocin,克林霉素
Target: Antibacterial, Antibiotic
ISOPIMPINELLIN
Cat.No: T4593
Synonym: 5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen
Target: Antiviral, DNA/RNA Synthesis, Parasite
Quinidine
Cat.No: T7938
Synonym: 奎尼丁,奎宁树
Target: Parasite
PHYTOL
Cat.No: T3254
Synonym: 植醇,trans-Phytol,(E)-Phytol
Target: Antibacterial, PPAR, Parasite
Mebendazole
Cat.No: T1155
Synonym: 甲苯达唑,甲苯咪唑,Telmin,Mebenvet,Vermox,Pantelmin
Target: Apoptosis, Microtubule Associated, Parasite
Spiramycin
Cat.No: T0819
Synonym: Espiramicin,螺旋霉素,Sequamycin,Rovamycin,Provamycin,Formacidine
Target: Antibacterial, Antibiotic, Parasite
dl-Maackiain
Cat.No: T6S0214
Synonym: (+)-Maackiain,高丽槐素,Demethylpterocarpin
Target: Apoptosis, Parasite
Asparagusic acid
Cat.No: T10388
Synonym: 1,2-二噻戊环-4-羧酸,芦笋酸
Target: Parasite
Furaltadone hydrochloride
Cat.No: T0896
Synonym: Furaltadone HCl,盐酸呋喃它酮
Target: Antibacterial, Antibiotic, Parasite
Ajugol
Cat.No: T3792
Synonym: 益母草苷,益母草苷A,Leonuride
Target: Parasite
Doxycycline monohydrate
Cat.No: T8259
Synonym: 水合强力霉素,强力霉素一水物
Target: MMP, Antibacterial, Antibiotic, Parasite
Bruceine A
Cat.No: T2S2046
Synonym: Dihydrobrusatol,鸦胆子素 A,NSC31616
Target: Antibiotic, Parasite
8-Deoxygartanin
Cat.No: TN1341
Synonym: 8-脱氧藤黄苷
Target: Beta Amyloid, NF-κB, Parasite
DihydroarteMisinic acid
Cat.No: THS1455
Synonym: 双氢青蒿酸,Dihydro-Artmisinic Acid,二氢青蒿酸
Target: Ferroptosis, Parasite
Cinchonine
Cat.No: T0012
Synonym: LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁
Target: Apoptosis, P-gp, Parasite
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Cat. No. Product Name Species Expression System
TMPY-04180 PfLDH Protein, P. falciparum, Recombinant (His)

PfLDH,L-lactate dehydrogenase

P. falciparum E. coli
Plasmodium falciparum lactate dehydrogenase (PfLDH) is a key enzyme for energy generation of malarial parasites and is considered to be a potential antimalarial target. The ability of PfLDH- or PfIDEh-based immuno-PCR assays to detect <1 parasite/microL suggests that improvements of bound antibody sensor technology may greatly increase the sensitivity of malaria rapid diagnostic tests. The PfLDH test could be used to detect failures and, therefore, to assess anti-malarial efficacy.
TMPH-03140 Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His)

Plasmepsin I,Aspartic hemoglobinase I,Plasmepsin 1,PMI

Plasmodium falciparum E. coli
During the asexual blood stage, catalyzes the initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation; specifically cleaves between Phe-33 and Leu-34 of Hb alpha-chain. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 41.0 k...
TMPK-00827 CD43 Protein, Mouse, Recombinant (His)

SPN,GPL115,Galgp,Ly-48,CD43,Leukosialin,Sialophorin,A630014B...

Mouse HEK293 Cells
CD43 is a large transmembrane protein involved in T cell activation. Previous studies of CD43-/- mice in viral models have demonstrated a role for CD43 in Th1/Th2 skewing, activation of Foxp3 Treg, and T cell apoptosis. CD43 (leukosialin) is a large sialoglycoprotein abundantly expressed on the surface of most cells from the hematopoietic lineage. CD43 is directly involved in the contact between cells participating in a series of events such as signaling, adherence and host parasite interactions...
TMPH-03141 Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc)

Plasmepsin II,Aspartic hemoglobinase II,PMII,Plasmepsin 2,Pf...

Plasmodium falciparum Baculovirus Insect Cells
During the asexual blood stage, participates in initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation. May cleave preferentially denatured hemoglobin that has been cleaved by PMI. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predict...
TMPH-03142 Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc)

PMII,PfAPD,Plasmepsin 2,PfPM1,Aspartic hemoglobinase II,Plas...

Plasmodium falciparum E. coli
During the asexual blood stage, participates in initial cleavage of native host hemoglobin (Hb) resulting in Hb denaturation. May cleave preferentially denatured hemoglobin that has been cleaved by PMI. Digestion of host Hb is an essential step which provides the parasite with amino acids for protein synthesis, and regulates osmolarity (Probable). Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. T...
TMPH-03634 GRA3 Protein, Toxoplasma gondii, Recombinant (His)

P30,GRA3,Dense granule protein 3

Toxoplasma gondii E. coli
Direct host-parasite interaction occurs at the cytoplasmic faces of the parasitophorous vacuole membrane (PVM) and the host endoplasmic reticulum (ER) membrane via GRA3 and host CAMLG association. Direct insertion of GRA3 ER retrieval motif into the host ER membrane contributes to the host ER recruitment to the PVM. GRA3 Protein, Toxoplasma gondii, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 10.8 kDa and the accession number is ...
TMPK-00832 CD43 Protein, Human, Recombinant (His)

Galgp,SPN,LSN,Sialophorin,CD43,A630014B01Rik,GPL115,Ly-48,Le...

Human HEK293 Cells
CD43 (leukosialin) is a large sialoglycoprotein abundantly expressed on the surface of most cells from the hematopoietic lineage. CD43 is directly involved in the contact between cells participating in a series of events such as signaling, adherence and host parasite interactions. The induction of acute myocarditis involves the engagement of CD43 cytoplasmic tripeptide sequence KRR to ezrin-radixin-moiesin cytoskeletal proteins. CD43 Protein, Human, Recombinant (His) is expressed in HEK293 mamma...
TMPK-01305 CD43 Protein, Cynomolgus, Recombinant (His)

CD43,A630014B01Rik,LSN,GPL115,Galgp,SPN,Ly-48,Leukosialin,Si...

Cynomolgus HEK293 Cells
CD43 (leukosialin) is a large sialoglycoprotein abundantly expressed on the surface of most cells from the hematopoietic lineage. CD43 is directly involved in the contact between cells participating in a series of events such as signaling, adherence and host parasite interactions. The induction of acute myocarditis involves the engagement of CD43 cytoplasmic tripeptide sequence KRR to ezrin-radixin-moiesin cytoskeletal proteins. CD43 Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 ...
TMPJ-01217 Mgl2 Protein, Mouse, Recombinant (His)

Macrophage Galactose-type C-lectin 2,Mgl2,CD301b,Macrophage ...

Mouse HEK293 Cells
Macrophage galactose N-acetyl-galactosamine-specific lectin 2(Mgl2), also known as CD301b, is a 38 kDa member that belongs to the C-type lectin family. Two MGL proteins are encoded by separate genes in the mouse, but share 91% amino acid (aa) identity in the extracellular domain (ECD). Only one MGL occurs in human and rat and this MGL is structurally more similar to mouse MGL1 than MGL2. However, human MGL and mouse MGL2 both bind specifically to terminal GalNAc residues, in contrast with mouse...
TMPY-01771 Latexin Protein, Mouse, Recombinant (His)

latexin

Mouse E. coli
Latexin, also known as endogenous carboxypeptidase inhibitor, tissue carboxypeptidase inhibitor, TCI, ECI, and LXN, is a cytoplasm protein that belongs to the protease inhibitor I47 (latexin) family. It is highly expressed in the heart, prostate, ovary, kidney, pancreas, and colon. Latexin / LXN is the only known endogenous specific inhibitor of zinc-dependent metallocarboxypeptidases (MCPs) present in mammalians so far. Latexin is originally identified as a molecular marker for the regional spe...
TMPY-03968 Secretogranin II Protein, Human, Recombinant (His)

EM66,SgII,SN,CHGC,secretogranin II

Human HEK293 Cells
Kit ligand, also known as Hematopoietic growth factor KL, Mast cell growth factor, Steel factor, Stem cell factor, c-Kit ligand, Kitlg and KITL, is a single-pass type I membrane protein that belongs to the SCF family. KITL / kit ligand also belongs to the family of dimeric transmembrane growth factors. The soluble form of KIT ligand is a secreted protein. Mast cells are thought to participate in a variety of immune responses, such as parasite resistance and the allergic reaction. Mast cell devel...
TMPY-01027 Mast Cell Protease-1/MCPT-1 Protein, Mouse, Recombinant (His)

carnitine palmitoyltransferase 1B (muscle),AV080368,Mcp-1

Mouse HEK293 Cells
Mast Cell Protease 1 (MMCP-1), also known as MCP-1, MCPT-1 and β-chymase, is a member of the Chymase family of chymotrypsin-like serine proteases. MCPT-1 is a 26 kDa β-chymase that is a component of mast cell granules. It is a 226 amino acid (aa) protein that has a conserved pattern of six cysteines and one potential glycosylation site. The granule-derived mouse mast cell proteases-1 and -2 (mMCP-1 and -2) colocalize in similar quantities in mucosal mast cells but micrograms of mMCP-1 compared w...

重组蛋白

PfLDH Protein, P. falciparum, Recombinant (His)
Cat.No: TMPY-04180
Species: P. falciparum
Expression System: E. coli
Plasmepsin-1 Protein, Plasmodium falciparum, Recombinant (His)
Cat.No: TMPH-03140
Species: Plasmodium falciparum
Expression System: E. coli
CD43 Protein, Mouse, Recombinant (His)
Cat.No: TMPK-00827
Species: Mouse
Expression System: HEK293 Cells
Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (His & Myc)
Cat.No: TMPH-03141
Species: Plasmodium falciparum
Expression System: Baculovirus Insect Cells
Plasmepsin-2 Protein, Plasmodium falciparum, Recombinant (E. coli, His & Myc)
Cat.No: TMPH-03142
Species: Plasmodium falciparum
Expression System: E. coli
GRA3 Protein, Toxoplasma gondii, Recombinant (His)
Cat.No: TMPH-03634
Species: Toxoplasma gondii
Expression System: E. coli
CD43 Protein, Human, Recombinant (His)
Cat.No: TMPK-00832
Species: Human
Expression System: HEK293 Cells
CD43 Protein, Cynomolgus, Recombinant (His)
Cat.No: TMPK-01305
Species: Cynomolgus
Expression System: HEK293 Cells
Mgl2 Protein, Mouse, Recombinant (His)
Cat.No: TMPJ-01217
Species: Mouse
Expression System: HEK293 Cells
Latexin Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01771
Species: Mouse
Expression System: E. coli
Secretogranin II Protein, Human, Recombinant (His)
Cat.No: TMPY-03968
Species: Human
Expression System: HEK293 Cells
Mast Cell Protease-1/MCPT-1 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01027
Species: Mouse
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
TMIH-0457 Proguanil-d6 HCl

Proguanil-d6 HCl 是 Proguanil HCl 的氘代化合物。Proguanil HCl 的 CAS 号为 637-32-1。Proguanil hydrochloride 是一种双胍类抗疟疾剂,在体内代谢形成环胍。它还是一种二氢叶酸还原酶抑制剂。

同位素标记化合物

Proguanil-d6 HCl
Cat.No: TMIH-0457
Synonym:
Target:
TargetMol Loading
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