Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12675L |
PT2399
|
HIF/HIF Prolyl-Hydroxylase; HIF | Angiogenesis; Chromatin/Epigenetic; Metabolism |
PT2399 是高选择性的HIF-2α拮抗剂,能直接结合 HIF-2α PAS B 结构域,IC50=6 nM,具有显著的体内抗肿瘤特性。 | |||
T12675 |
(Rac)-PT2399
|
HIF | Angiogenesis; Chromatin/Epigenetic |
(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM). |