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Targets Recommended: Histone Methyltransferase

4

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T17203 UNC0224

Histone Methyltransferase Chromatin/Epigenetic
UNC0224 是 G9a 的特异性抑制剂,Ki 为 2.6 nM,IC50 为 15 nM。 UNC0224 还有效抑制 GLP,IC50 值为 20-58 nM。
T17204 UNC0321

Histone Methyltransferase Chromatin/Epigenetic
UNC0321 是一种有效的组蛋白甲基转移酶 G9a 抑制剂,在 ECSD 和 CLOT 测定中,Ki 为 63 pM,IC50 分别为 9 nM 和 6 nM。 UNC0321 抑制 GLP,在 ECSD 和 CLOT 试验中 IC50 分别为 15 nM 和 23 nM。
T2354 UNC 0631

UNC0631

Histone Methyltransferase Chromatin/Epigenetic
UNC 0631 是一种有效的组蛋白甲基转移酶 G9a 抑制剂,IC50值为 4 nM。它有效降低 MDA-MB-231 细胞中 H3K9me2的水平,IC50为 25 nM。
TQ0232 UNC0646

UNC 0646

Histone Methyltransferase Chromatin/Epigenetic
UNC0646 是一种有效的、选择性的同源蛋白赖氨酸甲基转移酶 G9a 和 GLP 抑制剂,IC50分别为 6 和 15 nM,对 G9a/GLP 的选择性比 SETD7、SUV39H2、SETD8 和 PRMT3 高。它降低 MDA-MB-231 细胞中H3K9me2的水平,IC50为 26 nM。

化合物

UNC0224
Cat.No: T17203
Synonym:
Target: Histone Methyltransferase
UNC0321
Cat.No: T17204
Synonym:
Target: Histone Methyltransferase
UNC 0631
Cat.No: T2354
Synonym: UNC0631
Target: Histone Methyltransferase
UNC0646
Cat.No: TQ0232
Synonym: UNC 0646
Target: Histone Methyltransferase
Cat. No. Product Name Species Expression System
TMPY-01229 SETD7 Protein, Human, Recombinant (His)

SET7/9,SET domain containing (lysine methyltransferase) 7,SE...

Human E. coli
Histone-lysine N-methyltransferase SETD7, also known as SET domain containing (lysine methyltransferase) 7, SET7/9, Histone H3-K4 methyltransferase SETD7, H3-K4-HMTase SETD7, and SETD7, is a member of the histone-lysine methyltransferase family and SET7 subfamily. SETD7 is widely expressed and expressed in pancreatic islets. SETD7 contains three MORN repeats and one SET domain. SETD7 plays a central role in the transcriptional activation of genes such as collagenase or insulin. As a protein lysi...

重组蛋白

SETD7 Protein, Human, Recombinant (His)
Cat.No: TMPY-01229
Species: Human
Expression System: E. coli
TargetMol Loading
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