Cat. No. | Product Name | Target | Signaling Pathways |
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TP1955 |
PKC β pseudosubstrate
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Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia pep | |||
TP1955L |
PKC β pseudosubstrate acetate
PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base) |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) 是一种选择性的、细胞渗透的 PKC 抑制剂。 | |||
TP1956L |
PKC ζ pseudosubstrate acetate
PKC ζ pseudosubstrate acetate (799764-07-1 free base) |
PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
PKC ζ pseudosubstrate acetate 是蛋白激酶 C (PKC) ζ 的抑制剂;附着于细胞通透性触角足结构域载体肽。由 PKC ζ 假底物结构域的氨基酸 113-129 组成,通过二硫键连接到触角足结构域载体肽。 Antennapedia 肽在 4 或 37°C 时被完整细胞积极吸收,确保快速有效地吸收抑制肽。一旦进入细胞,二硫键在细胞质中被还原,导致抑制肽的释放。通过 PKC ζ 非依赖性途径诱导肥大细胞脱粒。 | |||
T75885 |
PKC β pseudosubstrate TFA
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PKCβ pseudosubstrate TFA 是一种选择性的、细胞渗透的 PKC 抑制剂。 | |||
T80071 |
PKCζ/ι pseudosubstrate inhibitor
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PKCζ/ι偽基質抑制劑對PKC酶家族表現廣譜抑制作用,並可能促成記憶功能障礙。 | |||
T80508 |
PKCη pseudosubstrate inhibitor,myristoylated
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PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Myristoylated PKCη pseudosubstrate inhibitor 是一种具有细胞渗透性的化合物,它主要应用于研究PKCη的作用机制。 | |||
T80507 |
PKCθ pseudosubstrate peptide inhibitor,myristoylated
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PKC | Chromatin/Epigenetic; Cytoskeletal Signaling |
Myristoylated PKCθ pseudosubstrate peptide inhibitor 是一款合成肽,专门用于研究 PKCθ 的机制。 |