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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T41005 |
PA-8
|
PACAP | GPCR/G Protein |
PA-8是一种小分子的的 PACAP I 型(PAC1)受体拮抗剂,有 选择性、有效性和口服活性。PA-8抑制PACAP 诱导的CREB 在PAC1-受体上的磷酸化,但对VPAC11或VPAC2受体无抑制作用。PA-8也抑制pacap 诱导的体外cAMP 水平升高(IC50 = 2 nM)和体内鞘内注射后pacap 诱导的厌恶反应和机械异位性痛。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-01427 |
HSPA8 Protein, Human, Recombinant (His)
Lipopolysaccharide-associated protein 1,HSPA8 |
Human | P. pastoris (Yeast) |
HSPA8 Protein, Human, Recombinant (His) is expressed in Yeast. |