1
7
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T125460 |
N-Acetylnornuciferine
|
Others | Others |
N-Acetylnornuciferine 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T125460。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3369 |
Nuciferine
(-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Nuciferine ((-)-Nuciferine) 是一种在埃及蓝睡莲和水芙蓉中发现的生物碱,是5-HT2A、5-HT2B 和5-HT2C 拮抗剂,IC50分别为 478 nM、1 μM 和 131 nM。它也是5-HT7的反向激动剂,IC50为 150 nM。 | |||
TN1091 |
Dehydronuciferine
|
AChE | Neuroscience |
Dehydronuciferine 是一种乙酰胆碱酯酶抑制剂,其 IC50=25 μg/mL,是从 Nelumbo nucifera Gaertn 的叶子中分离得到。 | |||
TQ0296L |
N-Nornuciferine hydrochloride(4846-19-9 free base)
N-Nornuciferine hydrochloride |
P450 | Metabolism |
N-Nornuciferine hydrochloride(4846-19-9 free base) (N-Nornuciferine hydrochloride) 是荷叶中的一种 aporphine 生物碱,显着抑制 CYP2D6(IC50:3.76 μM,Ki:2.34 μM)。 | |||
TWS0704 |
N-Methylnuciferine
|
Others | Others |
N-Methylnuciferine 是一种从Lotus Plumule提取的生物碱,可改善脂多糖诱导的抑郁样行为。 | |||
TN1092 |
O-Nornuciferine
|
Potassium Channel; HER | Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors |
O-Noruciferine 是分离自荷叶的卟啉型生物碱,是有效的 hERG 通道抑制剂。 | |||
TQ0296 |
N-Nornuciferine
|
P450 | Metabolism |
N-Nornuciferine, an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 μM). | |||
T34143 |
Pronuciferine
(+)-Pronuciferine |
||
Pronuciferine ameliorate the glucose and lipid metabolism in insulin-resistant 3T3-L1 adipocytes. |