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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T28960 Thaspine HCl

Thaspine,Thaspine HCl, NSC 135784,NSC-135784,NSC135784

Others Others
Thaspine is a potent topoisomerase IB inhibitor. Taspine downregulates VEGF expression and inhibits proliferation of vascular endothelial cells through PI3 kinase and MAP kinase signaling pathways.
T20656 Verapamil

NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil

P450; Calcium Channel; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Verapamil (CP-16533-1) 是一种非二氢吡啶类钙通道阻滞剂,一种 P-gp 抑制剂,也是一种 CYP3A4 抑制剂,具有口服活性。Verapamil 可以用于治疗高血压、心绞痛、心肌梗塞等。

化合物

Thaspine HCl
Cat.No: T28960
Synonym: Thaspine,Thaspine HCl, NSC 135784,NSC-135784,NSC135784
Target: Others
Verapamil
Cat.No: T20656
Synonym: NSC 135784,维拉帕米,NSC-135784,CP-16533-1,(±)-Verapamil
Target: P450, Calcium Channel, P-gp
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