558
152
28
10
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T13318 |
VU0650786
|
GluR | Neuroscience |
VU0650786 是能透过中枢神经系统的,选择性谷氨酸受体亚型 3 的一种负变构调节剂,IC50值为 392 nM,有抗抑郁和抗焦虑活性。 | |||
T9699 |
TAK-615
|
LPA Receptor | GPCR/G Protein |
TAK-615常用于研究肺纤维化,是一种LPA1受体的负变构调节剂。 | |||
T15090 |
Decoglurant
RO4995819 |
GluR | Neuroscience |
Decoglurant (RO4995819) 是 mGluR2和 mGluR3的负变构调制器,有抗抑郁作用。 | |||
T22027 |
AH-7614
AH 7614 |
GPR | Endocrinology/Hormones; GPCR/G Protein |
AH-7614 (AH 7614) 是一种选择性的游离脂肪酸受体 4(FFA4/GPR120) 拮抗剂,对人和大小鼠 FFA4 的pIC50值分别为 7.1、8.1 和 8.1。它能够阻断多不饱和 ω-6 脂肪酸亚油酸和 FFA4 激动剂的作用。 | |||
T19467 |
NADPH tetracyclohexanamine
还原型辅酶II四钠,NADPH (tetracyclohexanamine) |
Ferroptosis | Apoptosis |
NADPH tetracyclohexanamine (NADPH(tetracyclohexanamine)) 是一种辅助因子和生物还原剂。 | |||
T0858 |
Flufenamic acid
Arlef,Nichisedan,氟灭酸,氟芬那酸,Achless |
Potassium Channel; Calcium Channel; Chloride channel; COX; AMPK; Parasite | Chromatin/Epigenetic; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling |
Flufenamic acid (Arlef) 是一种非甾体类抗炎剂,是一种邻氨基苯甲酸衍生物,具有镇痛、抗炎和解热的特性。 它用于肌肉骨骼和关节疾病。 | |||
T3127 |
Glycinamide Hydrochloride
2-Aminoacetamide hydrochloride,甘氨酰胺盐酸盐,Glycine amide hydrochloride |
Others | Others |
Glycinamide Hydrochloride (2-Aminoacetamide hydrochloride) 是一种甘氨酸前药。 | |||
T8627 |
4-Acetamidobenzenesulfonamide
|
Anti-infection | Microbiology/Virology |
4-Acetamidobenzenesulfonamide 用于蛋白质组学研究,是一种抗感染剂。 | |||
T67925 |
Nampt activator-1
|
NAMPT | Metabolism |
NAMPT activator-1 (compound 1) 是一种有效的、专用范围广泛的烟酰胺磷酸基转移酶 (NAMPT) 激活剂(EC50 为3.3-3.7 μM)。NAMPT activator-1能有效保护培养细胞免受 fk866介导的毒性,是神经保护的潜在化合物。 | |||
T7129 |
(E/Z)-Necrosulfonamide
N-[4-[[(3-甲氧基吡嗪基)氨基]磺酰基]苯基]-3-(5-硝基-2-噻吩基)-2-丙烯酰胺 |
MLK | MAPK |
(E/Z)-Necrosulfonamide 是一种新型的 MLKL 抑制剂。 | |||
T50063 |
(2-methyl-2,3-dihydro-1H-inden-2-yl)methanamine HCl
|
Others | Others |
(2-methyl-2,3-dihydro-1H-inden-2-yl)methanamine hydrochloride 是一种环状胺,在结构上与安非他命有关,并已被证明对中枢神经系统具有显著影响。 | |||
T9323 |
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide
4-氨基-6-(三氟甲基)苯-1,3-二磺酰胺,4-Amino-6-(trifluoromethyl)benzene-1,3-d,2,4-Disulfamyl-5-trifluoromethylaniline,2-amino-4-trifluoromethyl-1,5-benzendisulfonamide |
Carbonic Anhydrase | Metabolism |
4-Amino-6-(trifluoromethyl)benzene-1,3-disulfonamide (4-Amino-6-(trifluoromethyl)benzene-1,3-d) 是一种碳酸酐酶抑制剂,用作潜在的抗肿瘤和抗青光眼药物。 | |||
T4226 |
Amenamevir
ASP2151,阿莫奈韦 |
DNA/RNA Synthesis; HSV | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology |
Amenamevir (ASP2151) 是一种新型解旋酶引发酶抑制剂,对水痘带状疱疹病毒和 1 型和 2 型单纯疱疹病毒具有活性,EC50值为 14 ng/mL。 | |||
T33762 |
Fosifloxuridine nafalbenamide
NUC-3373,NUC3373,NUC 3373 |
DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Fosifloxuridine nafalbenamide (NUC 3373) 是一种胸腺嘧啶合酶抑制剂,属于嘧啶核苷酸类似物,具有抗癌活性。它能诱发宿主免疫反应,有潜力增强免疫治疗。 | |||
T0018 |
Procainamide hydrochloride
Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺 |
DNA Methyltransferase; Sodium Channel; AChR; Autophagy | Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Neuroscience |
Procainamide hydrochloride (Procapan) 是一种用于研究心律失常的抗心律失常制剂。 | |||
TPL0388L |
1-[4-(1H-Imidazol-1-yl)phenyl]methanamine dihydrochloride
|
||
1-[4-(1H-Imidazol-1-yl)phenyl]methanamine dihydrochloride 是一种片段分子,在生命科学相关研究中具有广泛的应用。 | |||
T22330 |
Fenamic acid
N-苯基邻氨基苯甲酸,2-Anilinobenzoic acid,Diphenylamine-2-carboxylic acid,2-(Phenylamino)benzoic acid,N-Phenylanthranilic acid |
Chloride channel | Membrane transporter/Ion channel |
Fenamic acid (N-Phenylanthranilic acid) 是氯通道阻滞剂。 | |||
T71708 |
Minamestane
|
Aromatase | Endocrinology/Hormones |
Minamestane 是一种新型不可逆芳香化酶抑制剂。Minamestane 引起人胎盘芳香化酶的时间依赖性抑制,半衰期为4分钟,K 为59nM。Minamestane 具有抗肿瘤活性。 | |||
T20285 |
2-Iodobenzenamine
NSC34544,2-碘苯胺,NSC 34544,NSC-34544 |
Others | Others |
2-Iodobenzenamine (NSC-34544) 是一种生化剂。 | |||
T63290 |
(R,1R)-Tenofovir amibufenamide
(R,1R)-HS-10234 |
Antiviral | Immunology/Inflammation |
(R,1R)-Tenofovir amibufenamide ((R,1R)-HS-10234) 可用于 Tenofovir 前药,可口服,具有抗病毒活性。Tynofovir 是一种核苷酸逆转录酶抑制剂。 | |||
T8590 |
4-(benzyloxy)benzene-1-sulfonamide
|
Others | Others |
4-(benzyloxy)benzene-1-sulfonamide 是人重组 CA-7 的抑制剂。 | |||
T78428 |
X-Gluc cyclohexanamine
|
||
X-Gluc cyclohexanamine是一种用于检测β-葡萄糖醛酸酶(GUS)活性的染料,常用作基因表达的标记,可用于检测目的基因的表达。 | |||
T50061 |
[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine
|
Others | Others |
[4-(4-phenylpiperazin-1-yl)oxan-4-yl]methanamine 是一种哌嗪衍生物,它是血清素和多巴胺受体的部分激动剂,使其成为治疗抑郁症和精神分裂症等精神疾病的候选药物。 | |||
T50040 |
N-(3-methoxyphenyl)prop-2-enamide
|
Others | Others |
N-(3-methoxyphenyl)prop-2-enamide 是一种丙烯酰胺衍生物,被用于制备用于药物递送系统的聚合物材料,如纳米颗粒、微粒和水凝胶。 | |||
T33584 |
Namirotene
CBS 211A,Cbs 211 A |
Others | Others |
Namirotene (CBS 211A) 是一种蛋白质生物合成抑制剂,是一种人工合成的维甲酸类似物,可用于研究角膜疾病、角膜溃疡和干眼综合征。 | |||
T6651 |
Safinamide mesylate
PNU-151774E,FCE28073,PNU-151774E,NW-1015,EMD 1195686 mesylate,沙芬酰胺甲磺酸盐 |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Safinamide mesylate (EMD 1195686 mesylate) 是选择性的、有效的、可逆的单胺氧化酶 B 的抑制剂,对 MAO-A 选择性较低。它能够阻断钠通道和调节谷氨酸释放。它具有神经保护作用,可用于研究帕金森病、缺血脑卒中等疾病。 | |||
T64332 |
Glimepiride sulfonamide
|
Immunology/Inflammation related | Immunology/Inflammation |
Glimepiride sulfonamide 是一种抗炎活性化合物。 | |||
T12171 |
Nampt-IN-5
|
P450; NAMPT | Metabolism |
Nampt-IN-5 是烟酰胺磷酸核糖基转移酶抑制剂。它可抑制 A2780 和 COR-L23 细胞,IC50值分别为 0.7 nM 和 3.9 nM。它还抑制 CYP3A4 活性。 | |||
T0890 |
Mefenamic acid
CN-35355,CI 473,甲芬那酸,甲灭酸 |
COX | Immunology/Inflammation; Neuroscience |
Mefenamic acid (CN-35355) 是一种非甾体抗炎剂,可竞争性抑制hCOX-1和hCOX-2,IC50值分别为 40 nM 和 3 μM。 | |||
T50041 |
N-(4-methoxyphenyl)prop-2-enamide
N-(4-Methoxyphenyl)acrylamide,N-(4-甲氧苯基)丙烯酰基酰胺 |
Others | Others |
N-(4-methoxyphenyl)prop-2-enamide (N-(4-Methoxyphenyl)acrylamide) 是一种用作分子结构单元的丙烯酰胺类化合物。它可以抑制乙酰胆碱酯酶,增加突触间隙中的乙酰胆碱水平;也可以抑制多巴胺的分解,导致大脑中多巴胺水平的升高。 | |||
T7460 |
α-Cyano-4-hydroxycinnamic acid
α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基 |
Monocarboxylate transporter | Membrane transporter/Ion channel |
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) 是非竞争性单羧酸盐转运蛋白 (MCTs) 抑制剂,可抑制线粒体丙酮酸转运蛋白,Ki 值为 6.3 μM。它可作为基质辅助激光解吸电离-飞行时间质谱 (MALDI-TOF) 分析的基质,可以促进肽离子化。 | |||
T21369 |
Mecillinam
Amdinocillin,Mecillinamum,Hexacillin,美西林,Coactin,Penicillin HX |
Antibacterial | Microbiology/Virology |
Mecillinam (Hexacillin) 是一种有抗革兰氏阴性菌活性的 β 内酰胺类广谱抗生素。 | |||
T7560 |
Pivmecillinam hydrochloride
匹美西林盐酸盐,FL-1039 hydrochloride,盐酸匹美西林 |
Antibacterial; Antibiotic | Microbiology/Virology |
Pivmecillinam hydrochloride (FL-1039 hydrochloride) 是Mecillinam 的口服活性前药,是一种广谱青霉素抗生素,对革兰氏阴性菌有活性,可用作氨苄青霉素。 | |||
T1161 |
Prothionamide
1321-TH,Protionamide,丙硫异烟胺 |
Antibacterial; Antibiotic | Microbiology/Virology |
Prothionamide (1321-TH) 是一种具有抗结核活性的硫代酰胺衍生物。它可作用于结核病和麻风病。 | |||
T0249 |
N-Acetylprocainamide
NAPA,Acecainide,乙酰普卡胺,N-乙酰普鲁卡因胺 |
Potassium Channel; Sodium Channel; Drug Metabolite | Membrane transporter/Ion channel; Metabolism |
N-Acetylprocainamide (NAPA) 是K+通道抑制剂,是第三代抗心律失常剂。 | |||
T37906 |
Dibenamine hydrochloride
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Dibenamine hydrochloride 是竞争性的、不可逆的肾上腺素能阻断剂,可以修饰肾上腺素的药理作用。它对小鼠体内肾上腺素的破坏率显著增加。 | |||
T8575 |
ENFENAMIC ACID
|
Platelet aggregation | Others |
Enfenamic acid 是一种能够抑制伤口愈合的非甾体抗炎药。 | |||
T5881 |
Fluazinam
|
Antifungal | Microbiology/Virology |
Fluazinam 是一种具有广谱抗真菌活性的吡啶胺类杀菌剂,对核盘菌群的菌丝生长有很强的抑制作用。 | |||
T64369 |
Dynamin IN-2
|
Dynamin | Cytoskeletal Signaling |
Dynamin IN-2是一种Wiskostatin 类似物。Dynamin IN-2有效抑制 dynamin ,对 dynamin I GTPase 的 IC50 为 1.0 μM。Dynamin IN-2 可阻断网格蛋白介导的内吞作用 (CME),IC50 为 9.5 μM。 | |||
T21798L |
Dynamin inhibitory peptide Acetate
Dynamin inhibitory peptide Acetate(251634-21-6 Free base) |
GTPase | GPCR/G Protein |
Dynamin inhibitory peptide Acetate 是一种具有序列 Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro 的肽,可抑制 GTPase dynamin。 | |||
T67978 |
Cefuzonam
|
Antibiotic | Microbiology/Virology |
Cefuzonam 是一种新型头孢菌素,具有抗炎抗菌活性,可用于研究呼吸道感染、扁桃体炎和肝胆感染。 | |||
T3754 |
Hydrocinnamic alcohol
3-Phenyl-1-Propanol,3-苯丙醇,3-Phenylpropanol |
Others | Others |
Hydrocinnamic alcohol (3-Phenyl-1-Propanol) 存在于 storax 和蕨香脂中,也存在于越橘属水果、番石榴果和果皮、黑莓、其他水果、朗姆酒、白葡萄酒、香菇、松茸和泥煤麦芽中。它是一种调味成分。 | |||
T2553 |
Etofenamate
|
COX | Immunology/Inflammation; Neuroscience |
Etofenamate 是非甾体类抗炎小分子,也是非选择性的 COX 抑制剂,具有抗风湿和解热抗炎作用,可用于缓解疼痛、关节炎等炎症相关疾病的研究。 | |||
T15707 |
Laninamivir
(4S,5R,6R)-5-乙酰氨基-4-胍基-6-((1R,2R)-2,3-二羟基-1-甲氧基丙基)-5,6-二氢-4H-吡喃-2-甲酸,R 125489 |
Influenza Virus | Microbiology/Virology |
Laninamivir (R 125489) 是一种流感神经氨酸酶抑制剂,对流感病毒 H12N5 NA (N5),pH1N1 N1 NA (p09N1) 和 A/RI/5+/1957 H2N2 N2 (p57N2) 的 IC50值分别为 0.90 nM、1.83 nM 和 3.12 nM。 | |||
T7349 |
Ralfinamide
(S)-2-[[4-[(2-氟苄基)氧基]苄基]氨基]丙酰胺,Priralfinamide,FCE-26742A |
Sodium Channel | Membrane transporter/Ion channel |
Ralfinamide (Priralfinamide) 是一种具有口服活性的,来源于 α-aminoamide 的钠离子通道阻滞剂, 在缓解疼痛方面有研究的价值。 | |||
T7185 |
(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
|
Monoamine Oxidase | Neuroscience |
(2-Chloropyridin-4-yl)methanamine hydrochloride 是一种选择性的LOXL2抑制剂,IC50=126 nM。 | |||
T83632 |
Usenamine A
|
||
Usenamine A 是一种从地衣 Usnea longissima中提取到的小分子化合物,具有抗肿瘤活性,可用于研究肿瘤。 | |||
T10319 |
Anamorelin
RC-1291,阿拉莫林,ONO-7643 |
GHSR | GPCR/G Protein |
Anamorelin (ONO-7643) 是新型ghrelin receptor 激动剂,根据FLIPR 检测,得到其EC50=0.74 nM。 | |||
T5454 |
N-(p-amylcinnamoyl) Anthranilic Acid
2-(3-(4-戊基苯基)丙烯酰胺基)苯甲酸,ACA |
Phospholipase; TRP/TRPV Channel | Membrane transporter/Ion channel; Metabolism |
N-(p-amylcinnamoyl) Anthranilic Acid (ACA) 是一种广谱磷脂酶 A2(PLA2) 抑制剂,也是TRP channel 的阻滞剂。ACA 也可逆的抑制钙离子激活氯通道 (calcium-activated chloride channels) ,在心律失常方面具有研究的潜力。 | |||
T6781 |
Benzenesulfonamide
Benzenesulphonamide,苯磺酰胺,Phenyl sulfonamide,Benzosulfonamide |
Carbonic Anhydrase | Metabolism |
Benzenesulfonamide (Benzosulfonamide) 是碳酸酐酶的抑制剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10815 |
Cinnamoylglycine
|
Endogenous Metabolite | Metabolism |
Cinnamoylglycine 是肉桂酸和的甘氨酸结合物,是人体尿液代谢物。它被用作的尿液标志物,能够作为在抗生素研究期之后定殖耐药性的标志物。 | |||
T8145 |
Benzyl cinnamate
肉桂酸苄酯,Benzylcinnamoate,Benzyl 3-phenylpropenoate,Cinnamic acid benzyl ester,Cinnamein |
Immunology/Inflammation related | Immunology/Inflammation |
Benzyl cinnamate (Benzylcinnamoate) 是存在于苏门答腊和槟城的苯甲酸中,是存在于秘鲁香脂和托鲁香脂中,可用作香水和固定剂的成分。 | |||
T32614 |
L-Clausenamide
(-)-Clausenamide |
Microtubule Associated | Cytoskeletal Signaling |
L-Clausenamide 是从黄皮 (Clausena lansium (Lour) skeels) 的树叶中提取出来的生物碱,可用于提高认知功能。L-Clausenamide 对β-淀粉样蛋白 (Aβ) 毒性有抑制作用,通过抑制 tau 蛋白磷酸化阻止神经纤维缠结的形成。L-Clausenamide 具有神经保护活性,可用于调节 Aβ25-35 引发的刺激。L-Clausenamide 可用于研究阿尔兹海默症类的神经系统疾病。 | |||
TN3131 |
5-O-Cinnamoylquinic acid
金银花 |
Others | Others |
5-O-Cinnamoylquinic acid 是一种天然产物。 | |||
T9368 |
3,4-(Methylenedioxy)cinnamic acid
3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid,3,4-(亚甲二氧)肉桂酸 |
Others | Others |
3,4-(Methylenedioxy)cinnamic acid (3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid) 是一种植物衍生化合物,首先从芦笋的根中提取,并进一步表征为一种化感化学物质。 | |||
TN6794 |
N-(3-methoxybenzyl)-octadecanamide
|
Others | Others |
N-(3-methoxybenzyl)-octadecanamide 从玛卡 (Lepidium meyenii Walp.) 转化而来。 | |||
T5875 |
4-Methoxycinnamic acid
|
Endogenous Metabolite | Metabolism |
4-Methoxycinnamic acid 是天然苯丙烷类化合物。 | |||
T5543 |
TriacetonaMine
四甲基哌啶酮,Odoratine,tempidon,tmpone,Vincubine,2,2,6,6-Tetramethyl-4-piperidinone |
Others | Others |
TriacetonaMine (Vincubine) 是一种合成医药产品、农药和聚合物光稳定剂的中间体。它是热解油的主要组分。它是植物和真菌提取物的人工制品,使用丙酮和氢氧化铵,或在分离过程的不同步骤中天然出现铵盐。 | |||
T3006 |
Cinnamylideneacetic acid
Beta-Styrylacrylic acid,5-苯基戊烷-2,4-双酸,5-Phenyl-2,4-pentadienoic acid,5-Phenylpenta-2,4-dienoic acid |
Others; Antibacterial | Microbiology/Virology; Others |
Cinnamylideneacetic acid (Beta-Styrylacrylic acid) 用作合成结构单元、抗疟疾剂。 | |||
T4721 |
β-Nicotinamide mononucleotide
NMN,β-NM,β烟酰胺单核苷酸,烟酰胺单核苷酸 |
Others; Endogenous Metabolite | Metabolism; Others |
β-nicotinamide mononucleotide 是烟酰胺磷酸核糖转移酶 (NAMPT) 反应的产物。β-nicotinamide mononucleotide的作用包括其在细胞生化功能、心脏保护、糖尿病、肥胖相关并发症和阿尔茨海默病中的作用。 | |||
T5653 |
Cinnamyl acetate
3-Phenylallyl acetate,乙酸桂酯 |
Others | Others |
Cinnamyl acetate (3-Phenylallyl acetate) 是一种新型广谱抗菌剂,广泛应用于香料和香料工业。 | |||
T7053 |
p-Hydroxycinnamic acid
p-Coumaric acid,p-Cumaric acid,p-Hydroxy-cinnamic acid,对羟基肉桂酸,NSC 59260 |
Thrombin; Endogenous Metabolite; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Metabolism; Proteases/Proteasome |
p-Hydroxycinnamic acid (NSC-59260) 是常见的食用酚,可抑制血小板活性,对血栓素 B2 和前列腺素 E2 的 IC50值分别为 371 和 126 μM。 | |||
PDK0101 |
4-Methylcinnamic acid
对甲基肉桂酸,对甲基肉桂 |
Antifungal | Microbiology/Virology |
4-Methylcinnamic acid 是一种肉桂酸类似物,可用作克服抗真菌耐受性的干预催化剂。它可提高细胞壁破坏剂的效力。 | |||
T7991 |
2-Hydroxycinnamic acid
邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸 |
Others; SARS-CoV; HIV Protease | Microbiology/Virology; Others; Proteases/Proteasome |
2-Hydroxycinnamic acid 是从肉桂的甲醇提取物中分离出的一种天然产物,具有光氧化活性。它对HIV/SARS-CoV S 假病毒的感染具有抑制作用,IC50为 0.3 mM。 | |||
TN1457 |
Bryonamide B
|
||
Bryonamide B 是一种可从 Bryonia aspera 中提取得到一种葫芦类三萜。 | |||
T66582 |
6-Methylnicotinamide
|
Endogenous Metabolite | Metabolism |
6-Methylnicotinamide 是烟酰胺的衍生物,是一种内源性代谢物。在脑出血 (ICH) 急性期, 6-Methylnicotinamide 突然增加会加剧神经损伤。6-Methylnicotinamide 可用于制作共晶体/盐。 | |||
T6343 |
Geldanamycin
格尔德霉素,NSC 122750 |
HSP; Influenza Virus; Tyrosine Kinases; Antibacterial; Antibiotic | Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Geldanamycin 是一种 HSP90 抑制剂(Kd:1.2 μM),可特异性破坏糖皮质激素受体 (GR)/HSP 的结合。 | |||
TN3048 |
4-Methoxycinnamaldehyde
p-Methoxycinnamaldehyde |
RSV | Microbiology/Virology |
4-Methoxycinnamaldehyde (p-Methoxycinnamaldehyde) 是 Agastache rugosa 的一种活性成分。4-Methoxycinnamaldehyde 对人喉癌细胞系中的呼吸道合胞病毒 (RSV) 具有细胞保护活性,有助于控制 RSV 感染诱发的疾病,IC50 约为 0.055 μg/mL。 | |||
T3759 |
3,4-Dimethoxycinnamic acid
Dimethylcaffeic acid,3,4-二甲氧基肉桂酸,Caffeic acid dimethyl ether,O-Methylferulic acid |
Apoptosis; Virus Protease; Reactive Oxygen Species | Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
3,4-Dimethoxycinnamic acid (O-Methylferulic acid) 是从 Securidaca inappendiculata Hassk 中提取和纯化的单体。 3,4-Dimethoxycinnamic acid 通过 ROS 介导的信号通路对 L-02 细胞发挥抗凋亡作用。抗凋亡作用。 | |||
T13669 |
(E)-Cinnamamide
trans-Cinnamamide,肉桂酰胺 |
Others | Others |
(E)-Cinnamamide (trans-Cinnamamide) 是 Cinnamamide 的活性较低的异构体,Cinnamamide 是一种有效的非致命化学驱虫剂,适用于减少鸟类害虫的损害。 | |||
T2S0973 |
2-Methoxycinnamic acid
AI3-11206,o-Methoxycinnamic acid,2-甲氧基肉桂酸 |
Tyrosinase | Proteases/Proteasome |
2-Methoxycinnamic acid (o-Methoxycinnamic acid) 是非竞争性的酪氨酸酶抑制剂。 | |||
TN1558 |
N-Vanillyldecanamide
癸酸香草酰胺,Decylic acid vanillylamide |
Others | Others |
N-Vanillyldecanamide (Decylic acid vanillylamide) 分离自辣椒果实,以剂量依赖的方式显著减小紫花苜蓿幼苗的自由基长度。 | |||
TN7034 |
N-benzyl-heptadecanamide
N-Benzylheptadecanamide,N-苄基十七烷酰胺 |
Others | Others |
N-benzyl-heptadecanamide (N-Benzylheptadecanamide) 是玛咖中的一种玛卡酰胺。 | |||
T22974 |
Methyl 2,5-dihydroxycinnamate
|
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Methyl 2,5-dihydroxycinnamate 是 erbstatin 类似物,是一种高效、稳定的 EGF 受体相关酪氨酸激酶的抑制剂。 | |||
T25253 |
Cinnamtannin B-1
Cinnamtannin B1 (constituent of cinnamomum verum bark),LDN 0022358,LDN-0022358,LDN0022358,肉桂单宁B-1 |
Antioxidant; COX | Immunology/Inflammation; Neuroscience; oxidation-reduction |
Cinnamtannin B-1 (LDN 0022358) 是一种 A 型原花青素,包含在多种植物中,如越桔、桂树、泽兰肉桂和猪苓。它是一种有效的抗氧化剂和保护剂,可对抗人类血小板的氧化应激和凋亡。它是一种 Cox-2抑制剂。 | |||
TN7061 |
yuanamide
|
Others | Others |
yuanamide 是一种天然化合物,属于生物碱类。 | |||
TN5922 |
3,4-Dimethoxycinnamyl alcohol
(E)-3-(3,4-dimethoxyphenyl)prop-2-en-1-ol,3,4-二甲氧基肉桂醇 |
Others | Others |
3,4-Dimethoxycinnamyl alcohol ((E)-3-(3,4-dimethoxyphenyl)prop-2-en-1-ol) 显示出显着的抗菌和细胞毒性活性。 | |||
T5646 |
Cinnamic acid
3-Phenylacrylic acid,β-Phenylacrylic acid,肉桂酸 |
Endogenous Metabolite | Metabolism |
Cinnamic acid (β-Phenylacrylic acid) 在癌症干预中具有潜在的应用价值,对胶质母细胞瘤,黑色素瘤,前列腺癌,肺癌细胞的IC50=1-4.5 mM。 | |||
T0934 |
Nicotinamide
Nicotinic acid amide,Vitamin B3,Niacinamide,烟酰胺,Vitamin PP |
Sirtuin; Endogenous Metabolite | Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism |
Nicotinamide 是维生素 B3 的吡啶核苷形式,可作为烟酰胺腺嘌呤二核苷酸或 NAD+ 的前体,可通过膳食摄入来补充,能预防或治疗黑舌病和糙皮病。 | |||
TN7036 |
N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide
(9Z,12Z,15Z)-N-[(3-Methoxyphenyl)methyl]-9,12,15-octadecatrienamide,间-甲氧基苄基-亚麻酰胺,Macamide Impurity 14 |
Wnt/beta-catenin | Cytoskeletal Signaling; Stem Cells |
N-(3-Methoxybenzyl)-(9Z,12Z,15Z)-octadecatrienamide (Macamide Impurity 14) 是一种从玛卡中分离得到的玛卡酰胺。它能够激活典型的Wnt/β‐catenin 信号通路,诱导间充质干细胞成骨分化和随后的骨形成,可用于研究骨质疏松症。 | |||
T5552 |
Methyl cinnamate
|
Tyrosinase; Antibacterial; AMPK | Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome |
Methyl cinnamate 是花椒的有效成分,也是一种天然香料。它是一种防止食品褐变的酪氨酸酶抑制剂,具有抗菌活性。它通过由 CaMKK2-AMPK 信号途径介导的机制具有抗脂活性。 | |||
T3208 |
Brevianamide F
Cyclo-L-tryptophyl-L-proline,cyclo-(L-Trp-L-Pro),Cyclo(L-Pro-L-Trp) |
BCRP; PI3K; Antibacterial | Membrane transporter/Ion channel; Microbiology/Virology; PI3K/Akt/mTOR signaling |
Brevianamide F (Cyclo(L-Pro-L-Trp)) 是一种从Colletotrichum gloeosporioides 中分离得到的真菌毒素,属于天然存在的 2,5-二酮哌嗪类,具有抗菌活性。它具有PI3Kα抑制活性,IC50值为 4.8 µM。 | |||
T4S1551 |
Cinnamaldehyde
Cinnamic Aldehyde,肉桂醛 |
HIF | Angiogenesis; Chromatin/Epigenetic |
Cinnamaldehyde (Cinnamic Aldehyde) 具有解热作用。 它是镇静剂。它抑制MDA-MB-435S 细胞的侵袭能力与下调miR-27a 的表达有关。它诱导活性氧的产生,发挥血管扩张和抗癌作用。 它似乎是一种有希望的候选药物,可作为与 5-氟尿嘧啶 (5-FU) 和奥沙利铂 (OXA) 这两种用于 CRC 治疗的化疗药物联合治疗的辅助剂。其作用的可能机制可能涉及药物代谢基因的调节。 它在抑制黑色素瘤的发生和发展方面具有一定的作用,其作用机制可能表现为抑制VEGF 和HIF-α的表达,从而使血管模拟和黑色素瘤细胞新生血管的形成,促进肿瘤的生长。 | |||
TN1352 |
N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide
12顺-亚油酸酰胺,(9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide,n-3-methoxybenzyl-9z-12z-octadecadienamide,玛卡酰胺杂质10 |
Drug Metabolite | Metabolism |
N-(3-Methoxybenzyl-(9z,12z)-octadecadienamide ((9Z,12Z)-N-(3-Methoxybenzyl)octadeca-9,12-dienamide) 是一种 Macamide 杂质,可能用于代谢疾病的研究。 | |||
T10390 |
Asperphenamate
|
Others; Antifungal | Microbiology/Virology; Others |
Asperphenamate 是 Aspergillus flatiipes 的真菌代谢产物。 T47D 细胞、MDA-MB-231 细胞和 HL-60 细胞的 IC50 分别为 92.3 μM、96.5 μM 和 97.9 μM。 Asperphenamate 具有抗癌作用。 | |||
TN1965 |
N-Benzyllinolenamide
N-苄基-(9Z,12Z,15Z)-十八碳三烯酰胺,N-Benzyllinolenamide |
FAAH; Autophagy | Autophagy; Metabolism; Neuroscience |
N-Benzyllinolenamide 是从玛卡中得到的一种生物碱,是脂肪酰胺水解酶抑制剂,IC50 为 41.8 μM。 | |||
T7452 |
2-methoxycinnamaldehyde
2'-甲氧基肉桂醛,O-methoxycinnamaldehyde |
Apoptosis; Others | Apoptosis; Others |
2-methoxycinnamaldehyde 是一种肉桂中的天然产物。它能通过使线粒体膜电位 (ΔΨm) 损失 、激活 caspase-3 和 caspase-9,来抑制细胞增殖和诱导细胞凋亡,具有抗肿瘤活性。它还能抑制血小板衍生生长因子诱导的 HASMC 迁移。 | |||
T12540 |
Pristinamycin IA
Mikamycin IA,普利霉素IA,Mikamycin B |
Others; Antibiotic; P-gp | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Others |
Pristinamycin IA (Mikamycin B) 是 P-糖蛋白的底物,也是一种环肽类大环内酯抗生素。 | |||
T1165 |
Ethionamide
Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide |
Dehydrogenase; CAT; Antibacterial; Antibiotic | Metabolism; Microbiology/Virology; oxidation-reduction |
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。 | |||
T0793 |
Kanamycin sulfate
硫酸卡那霉素,Kanamycin monosulfate,Kanamycin A monosulfate,Ophtalmokalixan |
ribosome; Antibacterial; Antibiotic | Microbiology/Virology |
Kanamycin sulfate (Kanamycin monosulfate) 是氨基糖苷类杀菌抗生素,它通过与细菌30S 核糖体结合起作用。 | |||
TN1500 |
Cinnamyl cinnamate
Phenylallyl cinnamate |
||
Cinnamyl cinnamate (Phenylallyl cinnamate) 是一种天然产物,存在于龙脑丘、白杨中,是可从苏合香脂,白秘鲁香脂中提取出的食用香精。 | |||
T2S1625 |
(E)-Ethyl p-methoxycinnamate
Ethyl para-methoxycinnamate,Ethyl 4-methoxycinnamate,4-Methoxycinnamic Acid Ethyl Ester,对甲氧基肉桂酸乙酯,Ethyl methoxycinnamate,Ethyl p-methoxycinnamate,EPMC |
Others; COX | Immunology/Inflammation; Neuroscience; Others |
(E)-Ethyl p-methoxycinnamate (EPMC) 是从高良姜中提取的一种天然产物,具有抗炎、抗肿瘤和抗微生物作用。它在体外抑制COX-1和COX-2,IC50分别为 1.12 和 0.83 μM。 | |||
TN7126 |
N-Vanillyloctanamide
|
Others | Others |
N-Vanillyloctanamide 是一种来自 Capsicum annuum L. var. 果实的辣椒素。年鉴。 N-Vanillyloctanamide 减少 Lactuca sativa 幼苗的自由基长度,这种抑制是剂量依赖性的。 | |||
T19373 |
Indole-3-methanamine
|
Others | Others |
Indole-3-methanamine 已在大麦、谷物和谷物产品中检测到,但未量化。 | |||
TN7075 |
Linocinnamarin
3-[4-(beta-D-Glucopyranosyloxy)phenyl]acrylic acid methyl ester |
Phospholipase; Syk | Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors |
Linocinnamarin (3-[4-(beta-D-Glucopyranosyloxy)phenyl]acrylic acid methyl ester) 是从 Fragaria ananassa Duch 中分离出来的。 它对抗原刺激脱粒的抑制主要是由于 Syk/磷脂酶 Cgamma (PLCgamma) 途径的失活。 | |||
TN7180 |
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)-
4-(5-溴-1H-吲哚-3-基)嘧啶-2-胺,Meridianin C |
Others | Others |
2-Pyrimidinamine, 4-(5-bromo-1H-indol-3-yl)- (Meridianin C)是一种海洋来源的天然产物,存在于Aplidium meridianum。 | |||
T3731 |
Hydrocinnamic acid
3-Phenylpropanoic acid,氢化肉桂酸,3-Phenylpropionic acid,3-Phenyl-n-propionic acid |
Others; Endogenous Metabolite | Metabolism; Others |
Hydrocinnamic acid 是一种根际化合物,具有生长调控活性。 | |||
T5233 |
N-Methylnicotinamide
N'-Methylnicotinamide,Nicotinic Acid Methylamide,N-Methylpyridine-3-carboxamide,N-甲基烟酰胺 |
Others; Endogenous Metabolite | Metabolism; Others |
N-Methylnicotinamide 是内源性代谢产物的一种,可改善内皮功能障碍。 | |||
T13795 |
Nicotinamide riboside
|
Sirtuin | Chromatin/Epigenetic; DNA Damage/DNA Repair |
Nicotinamide riboside 是维生素 B3 的来源,可以增强氧化代谢并防止高脂肪饮食诱导的代谢异常。它是具有口服活性的 NAD+的前体,增加 NAD+水平并激活SIRT1和SIRT3,可用于研究阿尔茨海默氏病的认知退化。 | |||
TN3049 |
4-Methoxycinnamyl alcohol
|
Others | Others |
4-Methoxycinnamyl alcohol 对MCF-7、HeLa 和DU145癌症细胞系显示出毒性,IC50值分别为14.24、7.82和22.10μg/mL。4-methoxycinnamyl alcohol 是从Foeniculum vulgare 中分离出来的。4-Methoxycinnamyl alcohol 没有显示出凋亡作用,却在10μg/mL DNA 碎片研究显示48小时后发生了坏死。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01129 |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (RERRRKKR to TETR, HA1+HA2, uncleaved, His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (RERRRKKR to TETR, HA1+HA2, uncleaved, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59 kDa and the accession number is Q6DQ34. | |||
TMPY-00744 |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA Protein (His & Fc)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA Protein (His & Fc) is expressed in HEK293 mammalian cells with His and Fc tag. The predicted molecular weight is 85.7 kDa and the accession number is Q5EP31. | |||
TMPY-01152 |
DNAM-1/CD226 Protein, Human, Recombinant (His)
CD226 molecule,DNAM-1,TLiSA1,PTA1,DNAM1 |
Human | HEK293 Cells |
CD226 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.5 kDa and the accession number is Q15762. | |||
TMPY-04028 |
Influenza A H5N1 (A/Vietnam/UT31413II/2008) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Vietnam/UT31413II/2008) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.8 kDa and the accession number is D9I745. | |||
TMPK-00229 |
DNAM-1/CD226 Protein, Human, Recombinant (His & Avi)
PTA1,TLiSA1,DNAM1,CD226,CD226 molecule |
Human | HEK293 Cells |
DNAX accessory molecule-1 (DNAM-1), also known as CD226, is a 65 kDa type I transmembrane glycoprotein in the immunoglobulin superfamily.DNAM-1 mediates cellular adhesion to other cells bearing its ligands, CD112 and CD155, and cross-linking DNAM-1 with antibodies causes cellular activation. Furthermore, DNAM-1 can interact with PVR and PVRL2. DNAM-1/CD226 Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weight is 28.9 kDa... | |||
TMPY-03336 |
Influenza A H5N1 (A/chicken/VietNam/NCVD-016/2008) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | Baculovirus Insect Cells |
Influenza A H5N1 (A/chicken/VietNam/NCVD-016/2008) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60.2 kDa and the accession number is C4P278. | |||
TMPY-05226 |
DNAM-1/CD226 Protein, Human, Recombinant (His), Biotinylated
CD226 molecule,DNAM1,PTA1,TLiSA1,DNAM-1 |
Human | HEK293 Cells |
CD226 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.4 kDa and the accession number is Q15762. | |||
TMPY-05902 |
Influenza A H5N1 (A/Egypt/1394-NAMRU3/2007) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Egypt/1394-NAMRU3/2007) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.7 kDa. | |||
TMPY-05008 |
Influenza A H5N1 (A/Vietnam/UT31413II/2008) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Vietnam/UT31413II/2008) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 59.9 kDa and the accession number is D9I745. | |||
TMPY-00201 |
Influenza A H5N1 (A/chicken/VietNam/NCVD-016/2008) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/chicken/VietNam/NCVD-016/2008) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38.2 kDa and the accession number is C4P278. | |||
TMPH-03450 |
Nicotinamidase/PNC1 Protein, S. cerevisiae, Recombinant
Nicotinamide deamidase,PNC1,Nicotinamidase |
Saccharomyces cerevisiae | E. coli |
Catalyzes the deamidation of nicotinamide, an early step in the NAD(+) salvage pathway. Positively regulates SIR2-mediated silencing and longevity by preventing the accumulation of intracellular nicotinamide, an inhibitor of SIR2, during times of stress. Acts also on nicotinyl hydroxamate. Nicotinamidase/PNC1 Protein, S. cerevisiae, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 25.0 kDa and the accession number is P53184. | |||
TMPY-01504 |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Hemagglutinin/HA Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is A5A5I3. | |||
TMPY-01177 |
DNAM-1/CD226 Protein, Mouse, Recombinant (His)
CD226 molecule,DNAM1,TLiSA1,Pta1,BC051526,DNAM<... |
Mouse | HEK293 Cells |
CD226 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 28.2 kDa and the accession number is Q5DW69. | |||
TMPY-00494 |
Influenza A H5N1 (A/Egypt/3300-NAMRU3/2008) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Egypt/3300-NAMRU3/2008) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is B6ECC1. | |||
TMPY-01130 |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (Native, HA1+HA2, cleaved, His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (Native, HA1+HA2, cleaved, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 60 kDa and the accession number is Q6DQ34. | |||
TMPH-03449 |
Nicotinamidase/PNC1 Protein, S. cerevisiae, Recombinant (His)
Nicotinamidase,PNC1,Nicotinamide deamidase |
Saccharomyces cerevisiae | E. coli |
Catalyzes the deamidation of nicotinamide, an early step in the NAD(+) salvage pathway. Positively regulates SIR2-mediated silencing and longevity by preventing the accumulation of intracellular nicotinamide, an inhibitor of SIR2, during times of stress. Acts also on nicotinyl hydroxamate. Nicotinamidase/PNC1 Protein, S. cerevisiae, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 29.0 kDa and the accession number is P53184. | |||
TMPY-05487 |
DNAM-1/CD226 Protein, Human, Recombinant (hFc)
PTA1,DNAM1,TLiSA1,DNAM-1,CD226 molecule |
Human | HEK293 Cells |
CD226 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 52.7 kDa and the accession number is Q15762. | |||
TMPY-01505 |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 38 kDa and the accession number is A5A5I3. | |||
TMPJ-00968 |
NAMPT Protein, Human, Recombinant (His)
PBEF,PBEF1,Nicotinamide phosphoribosyltransferase,<... |
Human | E. coli |
Pre-B cell colony enhancing factor (PBEF) was originally identified as a cytokine that potentiated the clonal expansion and differentiation of pre-B cells, but it is also acknowledged to be the ubiquitous intracellular enzyme nicotinamide phosphoribosyltranferase (NAMPT) and the adipokine “visfatin”. PBEF is constitutively expressed in the fetal membranes where its greatest expression is in the amnion. It has intracellular and extracellular forms. Most of the intracellular functions of PBEF are ... | |||
TMPH-02810 |
NAMPT Protein, Mouse, Recombinant (His)
Pre-B-cell colony-enhancing factor 1 homolog,Visfatin,Nicoti... |
Mouse | P. pastoris (Yeast) |
NAMPT Protein, Mouse, Recombinant (His) is expressed in yeast with N-10xHis tag. The predicted molecular weight is 57.9 kDa and the accession number is Q99KQ4. | |||
TMPH-03760 |
NAMPT Protein, Mouse, Recombinant
Visfatin,Pre-B-cell colony-enhancing factor 1 homolog,Na... |
Mouse | E. coli |
NAMPT Protein, Mouse, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 55.6 kDa and the accession number is Q99KQ4. | |||
TMPY-00743 |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA1 Protein (His & Fc)
Harvey rat sarcoma viral oncogene homolog |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/VietNam/1203/2004) Hemagglutinin/HA1 Protein (His & Fc) is expressed in HEK293 mammalian cells with His and Fc tag. The predicted molecular weight is 64.4 kDa and the accession number is Q5EP31. | |||
TMPY-05578 |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (His), Biotinylated
Harvey rat sarcoma viral oncogene homolog |
H5N1 | Baculovirus Insect Cells |
Influenza A H5N1 (A/Vietnam/1194/2004) Hemagglutinin/HA Protein (His), Biotinylated is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 60.2 kDa and the accession number is Q6DQ34. | |||
TMPY-00393 |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Neuraminidase/NA Protein
NA Protein |
H5N1 | HEK293 Cells |
Influenza A H5N1 (A/Egypt/2321-NAMRU3/2007) Neuraminidase/NA Protein is expressed in HEK293 mammalian cells. The predicted molecular weight is 49.1 kDa and the accession number is B7U9P3. | |||
TMPY-02577 |
NAMPT Protein, Human, Recombinant (His & GST)
VISFATIN,PBEF,PBEF1,1110035O14Rik,VF,nicotinamide p... |
Human | Baculovirus Insect Cells |
Nicotinamide phosphoribosyltransferase (NAMPT), also known as pre-B-cell colony-enhancing factor 1 (PBEF1) or visfatin, is an enzyme belonging to the family of glycosyltransferases, to be specific, the pentosyltransferases. This enzyme participates in nicotinate and nicotinamide metabolism. This enzyme catalyzes the condensation of nicotinamide with 5- phosphoribosyl-1- pyrophosphate to yield nicotinamide mononucleotide, one step in the biosynthesis of nicotinamide adenine dinucleotide. NAMPT is... | |||
TMPK-00230 |
DNAM-1/CD226 Protein, Human, Recombinant (His & Avi), Biotinylated
CD226,PTA1,CD226 molecule,TLiSA1,DNAM1 |
Human | HEK293 Cells |
DNAX accessory molecule-1 (DNAM-1), also known as CD226, is a 65 kDa type I transmembrane glycoprotein in the immunoglobulin superfamily.DNAM-1 mediates cellular adhesion to other cells bearing its ligands, CD112 and CD155, and cross-linking DNAM-1 with antibodies causes cellular activation. Furthermore, DNAM-1 can interact with PVR and PVRL2. DNAM-1/CD226 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-His-Avi tag. The predicted molecular weig... | |||
TMPH-00930 |
Anamorsin Protein, Human, Recombinant (His & SUMO)
CIAPIN1,Fe-S cluster assembly protein DRE2 homolog,Cytokine-... |
Human | E. coli |
Anamorsin Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 49.6 kDa and the accession number is Q6FI81. | |||
TMPH-03761 |
NAMPT Protein, Mouse, Recombinant (HA & His)
Nicotinamide phosphoribosyltransferase,Visfatin, |
Mouse | E. coli |
NAMPT Protein, Mouse, Recombinant (HA & His) is expressed in E. coli expression system with N-6xHis and C-HA tag. The predicted molecular weight is 60.6 kDa and the accession number is Q99KQ4. |
Cat. No. | Product Name | Target | Signaling Pathways |
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TMIH-0053 |
4-amino-N-(4-nitrophenyl)benzenesulfonamide-d4
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4-amino-N-(4-nitrophenyl)benzenesulfonamide-d4 是 4-amino-N-(4-nitrophenyl)benzenesulfonamide 的氘代化合物。 | |||
T69395 |
Nicotinamide-d4
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Nicotinamide-d4 is intended for use as an internal standard for the quantification of nicotinamide by GC- or LC-MS. Nicotinamide is an amide form of niacin, which is also known as vitamin B3, that can be biosynthesized in vivo or obtained through the diet. It is a precursor in the synthesis of the metabolic cofactor NAD+ and an inhibitor of sirtuin 1 (SIRT1; IC50 = <50 µM). Nicotinamide (10 µM) increases the activity of serine palmitoyltransferase (SPT) and the biosynthesis of ceramide, glucosyl... | |||
T38118 |
Zanamivir-13C,15N2
Zanamivir-13C,15N2 |
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Zanamivir-13C,15N2is intended for use as an internal standard for the quantification of zanamivir by GC- or LC-MS. Zanamivir is a sialic acid analog that inhibits neuraminidase release of newly replicated influenza virus particles.1It has been shown to selectively inhibit the growth of influenza A and B viruses in plaque reduction assays with IC50values ranging from 5 to 14 nM and to directly inhibit influenza A and B virus neuraminidases with IC50values ranging from 0.6 to 7.9 nMin vitro. Intra... | |||
T71303 |
Flufenamic Acid-d4
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Flufenamic acid-d4 is intended for use as an internal standard for the quantification of flufenamic acid by GC- or LC-MS. Flufenamic acid is a non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor (IC50s = 3 and 9.3 µM for human COX-1 and COX-2, respectively). Flufenamic acid inhibits TNF-α-induced increases in COX-2 levels and NF-κB activation in HT-29 colon cancer cells in a concentration-dependent manner. It inhibits calcium influx induced by fMLP or A23187 in human polymorphonuclear... | |||
T36059 |
Dichlorphenamide-13C6
Dichlorphenamide-13C6 |
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Dichlorphenamide-13C6is intended for use as an internal standard for the quantification of dichlorphenamide by GC- or LC-MS. Dichlorphenamide is a sulfonamide and an orally bioavailable carbonic anhydrase (CA) inhibitor (Kis = 1.20, 38, 50, and 50 nM for the human CA isoforms CAI, CAII, CAIX, and CAXII, respectively).1It lowers intraocular pressure in rabbits when 50 μl of a 10% solution is applied topically to the eye.2Dichlorphenamide rescues the potassium deficiency and prevents insulin-induc... | |||
TMIJ-0494 |
Higenamine-d4 HCl
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Higenamine-d4 HCl 是 Higenamine HCl 的氘代化合物。Higenamine HCl 的 CAS 号为 11041-94-4。Higenamine hydrochloride 是一种 β2-AR 激动剂,是用于心力衰竭相关研究的中药乌头的关键成分,具有抗凋亡活性。 | |||
TMID-0192 |
Procainamide-d10
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Procainamide-d10 是 Procainamide 的氘代化合物。Procainamide 的 CAS 号为 51-06-9。Procainamide 是一种特异性强效的 DNA 甲基转移酶 1 (DNMT1) 抑制剂。普鲁卡因胺是一种 1A 类抗心律失常药物。Procainamide 具有研究癌症和心律失常的潜力。 | |||
TMIH-0325 |
MefenaMic Acid-d4
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MefenaMic Acid-d4 是 MefenaMic Acid 的氘代化合物。MefenaMic Acid 的 CAS 号为 61-68-7。Mefenamic acid 是一种非甾体抗炎剂,可竞争性抑制hCOX-1和hCOX-2,IC50值分别为 40 nM 和 3 μM。 | |||
TMIJ-0310 |
Pyrazinamide-d3
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Pyrazinamide-d3 是 Pyrazinamide 的氘代化合物。Pyrazinamide 的 CAS 号为 98-96-4。Pyrazinamide是一种口服抗结核类抗生素。它是一种前药,通过结核分枝杆菌pncA基因编码的 PZase/烟酰胺酶转化为活性吡嗪酸形式。 | |||
TMIH-0034 |
2-Ethyl-2-phenylmalonamide-d5
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2-Ethyl-2-phenylmalonamide-d5 是 2-Ethyl-2-phenylmalonamide 的氘代化合物。 |